4,5,6,7-Tetrahydroisoindole-1,3-diones
    33.
    发明授权
    4,5,6,7-Tetrahydroisoindole-1,3-diones 失效
    4,5,6,7-四氢异吲哚-1,3-二酮

    公开(公告)号:US4919704A

    公开(公告)日:1990-04-24

    申请号:US226701

    申请日:1988-08-01

    摘要: There are disclosed novel herbicidally active pyrrolidine-2,5-diones and 4,5,6,7-tetrahydroisoindolel,3-diones of formula ##STR1## wherein R.sup.1 is hydrogen; or C.sub.1 -C.sub.4 alkyl;R.sup.2 is C.sub.1 -C.sub.4 alkyl; orR.sup.1 and R.sup.2, when taken together, are a (CH.sub.2).sub.4 group which may be substituted by one or two C.sub.1 -C.sub.4 alkyl groups;X is hydrogen; or halogen;A is ##STR2## or O--R.sup.4 ; R.sup.3 is hydroxy; (C.sub.1 -C.sub.8)-alkoxy; (C.sub.1 -C.sub.4)-alkoxy-(C.sub.1 -C.sub.4)-alkoxy-(C.sub.1 -C.sub.4)-akoxy; (C.sub.1 -C.sub.4)-alkylthio-(C.sub.1 -C.sub.4)-alkoxy; mono- or di(C.sub.1 -C.sub.4)-alkylamino-(C.sub.1 -C.sub.4)-alkoxy; (C.sub.1 -C.sub.8)-cyanoalkoxy; (C.sub.3 -C.sub.8)-alkenyloxy; (C.sub.3 -C.sub.8)-haloalkenyloxy; (C.sub.3 -C.sub.8)-alkynyloxy; (C.sub.3 -C.sub.7)-cycloalkoxy; (C.sub.3 -C.sub.7)-cycloalkyl-(C.sub.1 -C.sub.4)-alkoxy; halo(C.sub.3 -C.sub.7)-cycloalkoxy; unsubstituted or substituted benzyloxy, phenoxy or phenylthio; the salt groups --O--Na, --O--K, --O--(Ca).sub.0.5, --O--(Mg).sub.0.5 or --O--NH.sub.4 ; amino; unsubstituted or substituted (C.sub.1 -C.sub.4)-alkylamino or di(C.sub.1 -C.sub.4)-alkylamino; (C.sub.3 -C.sub.4)-alkenylamino; diallylamino; N-pyrrolidino; N-piperidino; N-morpholino; N-thiomorpholino; N-piperidazino; (C.sub.1 -C.sub.8)-alkylthio; (C.sub.3 -C.sub.8)-alkenylthio; benzylthio; unsubstituted or substituted (C.sub.1 -C.sub.4)-alkylthio or (C.sub.1 -C.sub.4)-alkoxy;R.sup.4 is (C.sub.1 -C.sub.8)-alkyl; (C.sub.3 -C.sub.7)-cycloalkyl; (C.sub.3 -C.sub.7)-cycloalkyl-(C.sub.1 -C.sub.4)-alkyl; (C.sub.3 -C.sub.7)-halocycloalkyl; (C.sub.1 -C.sub.8)-alkylcarbonyl; allylcarbonyl; unsubstituted or substituted benzylcarbonyl, benzoyl or dioxolanyl; furoyl; thienoyl; unsubstituted or substituted C.sub.1 -C.sub.4 alkyl.The invention further relates to the preparation of the compounds of formula I, to herbicidal compositions containing them and to the use thereof as herbicides and plant growth regulators, and to novel intermediates for the preparation of these compounds.

    摘要翻译: 公开了新颖的除草活性吡咯烷-2,5-二酮和4,5,6,7-四氢异吲哚,其中R 1是氢的式(I)的3-二酮; 或C 1 -C 4烷基; R2是C1-C4烷基; 当R 1和R 2一起时,可以被一个或两个C 1 -C 4烷基取代的(CH 2)4基团; X是氢; 或卤素; A是或O-R4; R3是羟基; (C1-C8) - 烷氧基; (C 1 -C 4) - 烷氧基 - (C 1 -C 4) - 烷氧基 - (C 1 -C 4) - 烷氧基; (C 1 -C 4) - 烷硫基 - (C 1 -C 4) - 烷氧基; 单或二(C 1 -C 4) - 烷基氨基 - (C 1 -C 4) - 烷氧基; (C 1 -C 8) - 氰基烷氧基; (C 3 -C 8) - 烯氧基; (C3-C8) - 卤代烯氧基; (C 3 -C 8) - 炔氧基; (C 3 -C 7) - 环烷氧基; (C 3 -C 7) - 环烷基 - (C 1 -C 4) - 烷氧基; 卤代(C 3 -C 7) - 环烷氧基; 未取代或取代的苄氧基,苯氧基或苯硫基; 盐基-O-Na,-O-K,-O-(Ca)0.5,-O-(Mg)0.5或-O-NH 4; 氨基; 未取代或取代的(C 1 -C 4) - 烷基氨基或二(C 1 -C 4) - 烷基氨基; (C 3 -C 4) - 烯基氨基; 二烯丙基氨基 N-吡咯烷子; N-哌啶子基 N-吗啉代; N-硫代吗啉代 N-哌嗪基; (C 1 -C 8) - 烷硫基; (C 3 -C 8) - 烯基硫基; 苄硫基; 未取代或取代的(C 1 -C 4) - 烷硫基或(C 1 -C 4) - 烷氧基; R4是(C1-C8) - 烷基; (C 3 -C 7) - 环烷基; (C 3 -C 7) - 环烷基 - (C 1 -C 4) - 烷基; (C 3 -C 7) - 卤素环烷基; (C 1 -C 8) - 烷基羰基; 烯丙基羰基; 未取代或取代的苄基羰基,苯甲酰基或二氧戊环基; 糠基 噻吩甲酰 未取代或取代的C 1 -C 4烷基。 本发明还涉及式I化合物,含有它们的除草组合物及其作为除草剂和植物生长调节剂的用途以及用于制备这些化合物的新型中间体的制备。

    Weapon system with a carrier vehicle and a preferably vehicle dependent mortar
    35.
    发明授权
    Weapon system with a carrier vehicle and a preferably vehicle dependent mortar 有权
    具有载体车辆和优选车辆依赖砂浆的武器系统

    公开(公告)号:US08534180B2

    公开(公告)日:2013-09-17

    申请号:US13089040

    申请日:2011-04-18

    IPC分类号: F41F1/06

    CPC分类号: F42B30/12 F41H7/02

    摘要: A weapon system includes a carrier vehicle and a vehicle dependent mortar, wherein the carrier vehicle has a crew space and a weaponry space to house the mortar, and the mortar is charged in an index position with mortar grenades, with several sheddable propellant modules on the tail shaft thereof. The weapon system avoids manual loading of the mortar with mortar grenades because an automatic loader is arranged in a weapon space separated from the crew space by a separating wall. The loader transports the mortar grenade from a magazine in the weapon space into the index position of the barrel of the mortar and axially inserts it into the mouth of the barrel, and an automatic shedding device is arranged in the weapon space to automatically remove unnecessary propellant modules from the mortar grenade after fixing target parameters and before insertion of the mortar grenade into the barrel.

    摘要翻译: 武器系统包括载体车辆和车辆依赖砂浆,其中运载工具具有船员空间和用于容纳迫击炮的武器空间,并且将砂浆以灰浆手榴弹装载在索引位置,并在其上安装若干可喷洒的推进剂模块 尾轴。 武器系统避免用砂浆手榴弹手动装载砂浆,因为将自动装载机布置在与船员空间分离的武器空间中。 装载机将迫击炮手榴弹从武器空间的杂志运送到砂浆桶的索引位置,并将其轴向插入枪管的口中,并在武器空间内设置自动卸载装置,以自动移除不必要的推进剂 在固定目标参数后,将砂浆手榴弹插入枪管之前,从迫击炮手榴弹模块。

    Combat vehicle having an observation system
    36.
    发明授权
    Combat vehicle having an observation system 失效
    具有观察系统的战车

    公开(公告)号:US07032495B2

    公开(公告)日:2006-04-25

    申请号:US10349936

    申请日:2003-01-24

    IPC分类号: F41G5/24

    摘要: A combat tank is converted into an artillery observation tank without requiring removal of the main gun. The combat tank is converted by integrating retrofitted equipment necessary for the artillery observation, especially the navigation system (12), into the vehicle turret (4) such that it does not collide with the main gun. The navigation system (12) is installed with an arbitrary orientation at an arbitrary location in the vehicle turret (4), and adjusted at this location, without requiring a complicated adjustment mechanism for the observation system, or attachment to the elevating mass. The necessary elevation values for the line of sight (21) are obtained through the evaluation of the angular values of a mirror in the mirror head, such as of a primary-target telescope (20), or through evaluation of gun-position angles.

    摘要翻译: 战斗坦克被转换成炮兵观察坦克,而不需要拆除主炮。 战斗坦克是通过将炮兵观察所必需的改装设备,特别是导航系统(12)集成到车辆炮塔(4)中,使其不与主炮冲突而进行转换。 导航系统(12)在车辆转塔(4)中的任意位置处以任意方向安装,并且在该位置处被调整,而不需要用于观察系统的复杂的调节机构或附接到升降体。 通过评估诸如主目标望远镜(20)的镜头中的反射镜的角度值,或通过评估枪位置角度来获得视线(21)的必要仰角值。

    Herbicidally active thiadiazabicyclononanes and nonenes

    公开(公告)号:US5180418A

    公开(公告)日:1993-01-19

    申请号:US732988

    申请日:1991-07-19

    摘要: Cycloalkanecarboxylic acid derivatives of formula I ##STR1## wherein W is ##STR2## and A is CO--R.sub.3 or CN; R.sub.1 is hydrogen or fluorine; R.sub.2 is halogen or cyano; R.sub.3 is chlorine, X--R.sub.5, amino, C.sub.1 -C.sub.4 alkylamino, d-C.sub.1 -C.sub.4 alkylamino, C.sub.2 -C.sub.4 haloalkylamino, di-C.sub.2 -C.sub.4 haloalkylamino, C.sub.1 -C.sub.4 hydroxyalkylamino, di-C.sub.1 -C.sub.4 hydroxyalkylamino, C.sub.3 -C.sub.4 alkenylamino, diallylamino, --N-pyrrolidino, --N-piperidino, --N-morpholino, --N-thiomorpholino, --N-piperidazino, the group --O--N.dbd.C--(R.sub.9)R.sub.10 or the group --N--R.sub.6 (OR.sub.6); each of R.sub.4 and R.sub.14, independently of the other, is hydrogen, fluorine, chlorine, bromine, C.sub.1 -C.sub.4 alkyl or trifluoromethyl; R.sub.5 is hydrogen, C.sub.1 -C.sub.10 alkyl, C.sub.1 -C.sub.4 alkoxy-C.sub.1 -C.sub.4 alkyl, halo-C.sub.1 -C.sub.8 alkyl, C.sub.1 -C.sub.10 alkylthio-C.sub.1 -C.sub.4 alkyl, di-C.sub.1 -C.sub.4 alkylamino-C.sub.1 -C.sub.4 alkyl, cyano-C.sub.1 -C.sub.8 alkyl, C.sub.3 -C.sub.8 alkenyl, halo-C.sub.3 -C.sub. 8 alkenyl, C.sub.3 -C.sub.8 alkynyl, C.sub.3 -C.sub.7 cycloalkyl, C.sub.3 -C.sub.7 cycloalkyl-C.sub.1 -C.sub.4 alkyl or halo-C.sub.3 -C.sub.7 cycloalkyl, or benzyl which is unsubstituted or substituted at the phenyl ring by up to three identical or different substituents selected from halogen, C.sub.1 -C.sub.4 alkyl, halo-C.sub.1 -C.sub.4 alkyl, halo-C.sub.1 -C.sub.4 alkoxy or C.sub.1 -C.sub.4 alkoxy, or is an alkali metal ion, an alkaline earth metal ion or an ammonium ion, the group --[CHR.sub.6 --(CH.sub.2).sub.m ]--COOR.sub.7, or the group [CHR.sub.6 --(CH.sub.2).sub.t --Si(R.sub.8).sub.3 ]; R.sub.6 is hydrogen or C.sub.1 -C.sub.4 alkyl; R.sub.7 is hydrogen, C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.8 alkenyl, C.sub.3 -C.sub.8 alkynyl, C.sub.1 -C.sub.8 alkoxy-C.sub.2 -C.sub.8 alkyl, C.sub.1 -C.sub.8 alkylthio-C.sub.2 -C.sub.8 alkyl or C.sub.3 -C.sub.7 cycloalkyl; R.sub.8 is C.sub.1 - C.sub.4 alkyl; R.sub.9 is C.sub.1 -C.sub.4 alkyl; R.sub.10 is C.sub.1 -C.sub.4 alkyl or phenyl; or R.sub.9 and R.sub.10, together with the carbon atom to which they are bonded, form a cyclohexane ring; R.sub.11 is C.sub.1 -C.sub.8 alkyl; R.sub.12 is hydrogen or C.sub.1 -C.sub.8 alkyl; R.sub.13 is hydrogen, C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.7 cycloalkyl, C.sub.1 -C.sub.4 alkoxy-C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkylthio-C.sub.1 -C.sub.4 alkyl, halo-C.sub.1 -C.sub.7 alkyl, C.sub.3 -C.sub.7 alkenyl or C.sub.3 -C.sub.7 alkynyl; X, Y, Y.sub.1, Y.sub.2, Y.sub.3, Y.sub.4, Z.sub.1 and Z.sub.2 are each independently oxygen or sulfur; n is 0, 1, 2, 3 or 4; m is 0, 1, 2, 3 or 4; q is 1 or 2; and t is 0, 1, 2, 3 or 4, have good pre- and post-emergence selective herbicidal and growth regulating properties.

    Composition for protecting cultivated plants from the phytotoxic action
of herbicides
    40.
    发明授权
    Composition for protecting cultivated plants from the phytotoxic action of herbicides 失效
    用于保护栽培植物免受除草剂植物毒性作用的组合物

    公开(公告)号:US4676823A

    公开(公告)日:1987-06-30

    申请号:US817216

    申请日:1986-01-08

    摘要: When applied as safeners, the haloacylaminoalkylphosphinates, haloacylaminoalkylphosphinates and haloacylaminoalkylphosphine oxides of the formula I below are able to protect cultivated plants from the phytotoxic effects of herbicides. Suitable crops are preferably sorghum, cereals, rice, maize and soya beans and the herbicides employed are chloroacetanilides and thiocarbamates.The haloacylaminoalkylphosphonates, haloacylaminoalkylphosphinates and haloacylaminoalkylphosphine oxides have the formula I ##STR1## wherein R.sub.1 is C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.2 -C.sub.4 alkenyloxy, C.sub.2 -C.sub.4 alkynyloxy, C.sub.1 -C.sub.4 haloalkyl, C.sub.2 -C.sub.8 alkoxyalkoxy or C.sub.1 -C.sub.4 cyanoalkoxy,R.sub.2 is hydrogen or a substitutent as defined for R.sub.1,R.sub.3 and R.sub.4 are each independently hydrogen, C.sub.1 -C.sub.4 alkyl or one of R.sub.3 and R.sub.4 is also a radical ##STR2## or both taken together with the carbon atom to which they are attached are also a C.sub.3 -C.sub.11 cycloalkyl radical,R.sub.5 is hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.3 -C.sub.7 cycloalkyl, C.sub.2 -C.sub.4 alkenyl, C.sub.2 -C.sub.4 -alkynyl, C.sub.2 -C.sub.8 alkoxyalkyl, C.sub.1 -C.sub.4 haloalkyl or aralkyl,R.sub.6 is hydrogen or C.sub.1 -C.sub.4 alkyl,X.sub.1 and X.sub.2 are each independently halogen or one of X.sub.1 and X.sub.2 is also hydrogen, andn is 1, 2 or 3.

    摘要翻译: 当作为安全剂使用时,下式I的卤代酰基氨基烷基次膦酸酯,卤代酰基氨基烷基次膦酸酯和卤代酰基氨基烷基氧化膦能够保护栽培植物免受除草剂的植物毒性作用。 合适的作物优选是高粱,谷类,水稻,玉米和大豆,所用的除草剂是氯乙酰苯胺和硫代氨基甲酸盐。 卤代酰基氨基烷基膦酸酯,卤代酰基氨基烷基次膦酸酯和卤代酰基氨基烷基氧化膦具有式I(I)其中R1是C1-C4烷基,C1-C4烷氧基,C2-C4链烯氧基,C2-C4炔基氧基,C1-C4卤代烷基,C2-C8烷氧基烷氧基或C1-C4氰基烷氧基,R2是 氢或R 1,R 3和R 4所定义的取代基各自独立地为氢,C 1 -C 4烷基或R 3和R 4中的一个也是基团,或者它们与它们所连接的碳原子一起也是C3 -C 11环烷基,R 5是氢,C 1 -C 4烷基,C 3 -C 7环烷基,C 2 -C 4烯基,C 2 -C 4炔基,C 2 -C 8烷氧基烷基,C 1 -C 4卤代烷基或芳烷基,R 6是氢或C 1 -C 4烷基, 卤素或X1和X2之一也是氢,n是1,2或3。