Thiazolidine-2,4-dione derivatives, salts and preparation processes
thereof
    31.
    发明授权
    Thiazolidine-2,4-dione derivatives, salts and preparation processes thereof 失效
    噻唑烷-2,4-二酮衍生物,其盐及其制备方法

    公开(公告)号:US5308856A

    公开(公告)日:1994-05-03

    申请号:US938228

    申请日:1992-10-26

    CPC分类号: C07D417/10

    摘要: The present invention provides novel thiazolidine-2,4-dione derivatives possessing blood sugar-lowering action and aldose reductase-inhibitory action, their salts, their preparation processes and drugs containing them, and relates to thiazolidine-2,4-dione derivatives represented by a general formula (1) ##STR1## [wherein R.sup.1 and R.sup.2 denote identically or differently hydrogen atoms, halogens, lower alkyl groups, hydroxyl groups, lower alkoxy groups, nitro groups or amino groups (said amino group may be substituted with lower alkyl group or lower alkanoyl group, R.sup.3 denotes a hydrogen atom or lower alkyl group, A denotes a lower alkylene or carbonyl group, and B and W denote differently lower alkylenes, carbonyl groups or bonding hands], or their salts.

    摘要翻译: PCT No.PCT / JP92 / 00190 Sec。 371日期:1992年10月26日 102(e)日期1992年10月26日PCT提交1992年2月24日PCT公布。 出版物WO92 / 14730 本发明提供具有降血糖作用和醛糖还原酶抑制作用的新型噻唑烷-2,4-二酮衍生物及其盐,其制备方法和含有它们的药物,涉及噻唑烷-2 由通式(1)表示的4-二酮衍生物(Ⅰ)[其中R1和R2表示相同或不同的氢原子,卤素,低级烷基,羟基,低级烷氧基,硝基或氨基( 所述氨基可以被低级烷基或低级烷酰基取代,R3表示氢原子或低级烷基,A表示低级亚烷基或羰基,B和W表示不同的低级亚烷基,羰基或键合键], 或其盐。

    Production process of phenylglycosides
    33.
    发明授权
    Production process of phenylglycosides 失效
    苯基糖苷的生产工艺

    公开(公告)号:US4889927A

    公开(公告)日:1989-12-26

    申请号:US163839

    申请日:1988-03-03

    IPC分类号: C07H1/00 C07H15/203

    CPC分类号: C07H15/203

    摘要: This invention concerns a process for producing phenolic substances with beneficial biological activities in a high yield, which comprises: subjecting a glycose of which an OH group at the 1 position is substituted for a halogen atom and of which other groups are substituted for acyl groups, and a phenol of which at least one of the ortho-positions in regard to phenolic OH groups is substituted to reaction with an alkali metal hydride in dimethylsulfoxide or dimethylformamide in the presence of or non-presence of a quat-ammonium salt and then hydrolyzing said acyl groups with an alkaline substance.

    摘要翻译: 本发明涉及以高产率生产具有有益生物活性的酚类物质的方法,该方法包括:使1位上的OH基团的糖取代卤素原子,其它基团取代酰基, 以及苯酚,其中酚基OH基团的至少一个邻位被取代为与二价亚砜或二甲基甲酰胺中的碱金属氢化物反应,在或不存在季铵盐,然后水解所述 具有碱性物质的酰基。

    Fibrosis inhibitor
    36.
    发明授权
    Fibrosis inhibitor 有权
    纤维化抑制剂

    公开(公告)号:US08729086B2

    公开(公告)日:2014-05-20

    申请号:US12919885

    申请日:2009-02-26

    IPC分类号: A61K31/4965 C07D241/02

    CPC分类号: C07D241/20 A61K31/4965

    摘要: [Object] The main object of the present invention is to provide a fibrosis inhibitor.[Solving Means] The present invention relates to a fibrosis inhibitor containing the heterocyclic derivative represented by the following general formula (1) or a pharmaceutically acceptable salt thereof as an active ingredient; In the formula (1), R1 and R2 are the same or different and each represents an optionally substituted aryl; R3 and R4 are the same or different and each represents hydrogen atom or alkyl; R5 represents hydrogen atom, alkyl or halogen atom; Y represents N or N→O; A represents NR6, and R6 represents hydrogen atom, alkyl, etc.; D represents alkylene or alkenylene which is optionally substituted with hydroxy; E represents phenylene or a single bond; G represents O, S, etc.; and Q represents carboxy, alkoxycarbonyl, etc.

    摘要翻译: 本发明的主要目的在于提供纤维化抑制剂。 本发明涉及含有下述通式(1)表示的杂环衍生物或其药学上可接受的盐作为有效成分的纤维化抑制剂。 在式(1)中,R 1和R 2相同或不同,表示任选取代的芳基; R3和R4相同或不同,各自表示氢原子或烷基; R5代表氢原子,烷基或卤素原子; Y表示N或N→O; A表示NR6,R6表示氢原子,烷基等。 D表示任选被羟基取代的亚烷基或亚烯基; E表示亚苯基或单键; G代表O,S等; Q表示羧基,烷氧基羰基等。

    Communication control system, communication control method, call control server device, and call control program
    37.
    发明授权
    Communication control system, communication control method, call control server device, and call control program 有权
    通信控制系统,通信控制方式,呼叫控制服务器设备和呼叫控制程序

    公开(公告)号:US08700783B2

    公开(公告)日:2014-04-15

    申请号:US12996807

    申请日:2009-06-15

    IPC分类号: G06F15/16

    摘要: Upon receipt of an access request from a Web terminal, a service providing server transmits a shop ID stored in an external information database to the Web terminal. When the shop ID is selected by the Web terminal, the service providing server acquires external connection destination information, and notifies a SIP proxy server of the information via the Web terminal. When notified of the information, the SIP proxy server identifies internal connection destination information in an internal information database, based on an IP address added at the time of the notification of the external connection destination information. After making a call to a telephone device with the use of the identified internal connection destination information, the SIP proxy server makes a call to the shop with the use of the external connection destination information. After that, the SIP proxy server establishes a connection between the telephone device and the shop.

    摘要翻译: 在从Web终端接收到访问请求时,服务提供服务器将存储在外部信息数据库中的商店ID发送到Web终端。 当由Web终端选择商店ID时,服务提供服务器获取外部连接目的地信息,并通过Web终端向SIP代理服务器通知该信息。 SIP代理服务器在通知该信息时,根据在通知外部连接目的地信息时添加的IP地址,在内部信息数据库中识别内部连接目的地信息。 在通过使用所识别的内部连接目的地信息对电话设备进行呼叫之后,SIP代理服务器通过使用外部连接目的地信息来呼叫商店。 之后,SIP代理服务器建立电话设备和商店之间的连接。

    Vehicle driving apparatus
    39.
    发明授权
    Vehicle driving apparatus 有权
    车辆驾驶装置

    公开(公告)号:US08170760B2

    公开(公告)日:2012-05-01

    申请号:US12746437

    申请日:2009-03-23

    IPC分类号: G06F19/00

    摘要: A vehicle driving apparatus that can execute cranking of an internal combustion engine by transmitting a mechanical power from a rotor of a motor to an engine output shaft without executing an engaging/disengaging operation of a clutch. A driving apparatus of a hybrid vehicle includes a first speed change mechanism capable of receiving mechanical power from an engine output shaft by a first input shaft and transmitting the mechanical power to drive wheels, a second speed change mechanism capable of receiving the mechanical power from the engine output shaft and a rotor by a second input shaft engaged with the rotor and transmitting the mechanical power to the drive wheels, a first clutch capable of engaging the engine output shaft with the first input shaft, and a second clutch capable of engaging the engine output shaft with the second input shaft.

    摘要翻译: 一种车辆驾驶装置,其能够通过将来自电动机的转子的机械动力传递到发动机输出轴而不执行离合器的接合/分离操作来执行内燃机的起动。 混合动力车辆的驱动装置包括能够通过第一输入轴从发动机输出轴接收机械动力并将机械动力传递到驱动轮的第一变速机构,能够从所述第二变速机构接收来自所述第二变速机构的机械动力的第二变速机构, 发动机输出轴和转子通过与转子接合并将机械动力传递到驱动轮的第二输入轴,能够将发动机输出轴与第一输入轴接合的第一离合器和能够接合发动机的第二离合器 输出轴与第二输入轴。

    Wheel for vehicle
    40.
    发明授权
    Wheel for vehicle 有权
    车轮

    公开(公告)号:US08020945B2

    公开(公告)日:2011-09-20

    申请号:US12155246

    申请日:2008-05-30

    IPC分类号: B60B7/06

    CPC分类号: B60B7/14

    摘要: A wheel for vehicle includes a wheel body, a decorated member, and a visible space. The wheel body has a rim, a hub, and a plurality of spokes connecting the hub and the rim. The decorated member is made from resin, is disposed on a surface of at least one of the spokes, and is retained to the wheel body. The visible space is disposed between the decorated member and the one of the spokes at least, exhibits a height in an axial direction of the wheel body, and is visible from an axial outer side of the wheel body.

    摘要翻译: 用于车辆的车轮包括轮体,装饰构件和可见空间。 轮体具有轮辋,轮毂和连接轮毂和轮辋的多个辐条。 装饰构件由树脂制成,设置在至少一个辐条的表面上,并被保持在轮体上。 所述可视空间至少设置在所述装饰构件和所述一个所述辐条之间,在所述车轮主体的轴向方向上具有高度,并且从所述车轮主体的轴向外侧可见。