Substituted quinoline compounds and their use as safeners
    44.
    发明授权
    Substituted quinoline compounds and their use as safeners 失效
    取代的喹啉化合物及其作为安全剂的用途

    公开(公告)号:US5756422A

    公开(公告)日:1998-05-26

    申请号:US535028

    申请日:1995-10-18

    摘要: Substituted quinoline compounds, processes for their preparation, composition containing them, and their use as safeners Compounds of the formula I and salts thereof ##STR1## in which R.sup.1 �lacuna! CN, C(.dbd.Z)--Q(A.sub.i X.sub.i).sub.q --R, --C(.dbd.Z)--QR*, 1,2,3,4-tetrazol-5-yl, 1,3,4-triazol-2-yl, 1,3-oxazol-2-yl, and the remaining radicals are as defined in claim 1, are suitable for use as safeners for protecting crop plants such as, for example, cereals, rice and maize, against herbicide damage. Some of the compounds are known and some are novel and they can be prepared from quinolin-8-oxy derivatives by the processes of claim 7.

    摘要翻译: PCT No.PCT / EP94 / 01396 Sec。 371 1995年10月18日第 102(e)日期1995年10月18日PCT 1994年5月2日PCT PCT。 第WO94 / 26716号公报 日期:1994年11月24日取代喹啉化合物,其制备方法,含有它们的组合物及其作为安全剂的用途式I化合物及其盐其中R1 [lacuna] CN,C(= Z) -Q(AiXi)qR,-C(= Z)-QR *,1,2,3,4-四唑-5-基,1,3,4-三唑-2-基,1,3-恶唑-2 并且剩余的基团如权利要求1中所定义,适合用作安全剂,用于保护作物植物,例如谷物,水稻和玉米,以防止除草剂损害。 一些化合物是已知的,一些是新的,它们可以通过权利要求7的方法由喹啉-8-氧基衍生物制备。

    Acylated aminophenylsulfonylureas; preparation and use as herbicides and
plant growth regulators
    46.
    发明授权
    Acylated aminophenylsulfonylureas; preparation and use as herbicides and plant growth regulators 失效
    酰化氨基苯基磺酰脲 作为除草剂和植物生长调节剂的制备和使用

    公开(公告)号:US5658854A

    公开(公告)日:1997-08-19

    申请号:US268274

    申请日:1994-06-30

    摘要: Acylated aminophenylureas, preparation and use as herbicides and plant growth regulatorsThe compounds of the formula I or their salts ##STR1## in which G is a radical G1, G2 or G3 ##STR2## R.sup.1 is H or alkyl, R.sup.2 is COOH, CSOH or a derivative of the carboxyl or thiocarboxyl group, of 1 to 20 carbon atoms, or acyl of the type CO-R.degree. of 1-12 carbon atoms, or an imino, hydrazone or oxime derivative of the group CO-R.degree., and R.degree. , R.sup.3a, R.sup.4a, R.sup.3b, R.sup.4b, W, X, Y and Z are as defined in claim 1, are suitable as selective herbicides and plant growth regulators in crops.The preparation is carried out in analogy to known processes (see claim 5) by way of intermediates, some of which are new, from the group consisting of benzene-sulfonamides (II), benzenesulfonyl isocyanates (IV) and benzesulfonyl chlorides (VI) and heterocyclically substituted carbamates (III), amines (V) and/or (thio)-isocyanates (XIX).

    摘要翻译: 酰化氨基苯基脲,作为除草剂和植物生长调节剂的制备和用途式I化合物或其盐,其中G是基团G1,G2或G3(G1)(图像)(G2) (G3)R1为H或烷基,R2为COOH,CSOH或含1-20个碳原子的羧基或硫代羧基的衍生物,或碳原子数为1〜12的CO-R DEG型酰基, 或CO-R DEG基团的亚氨基,腙或肟衍生物,R DEG,R3a,R4a,R3b,R4b,W,X,Y和Z如权利要求1所定义,适合作为选择性除草剂和植物生长 农作物的监管者。 类似于已知方法(参见权利要求5),通过中间体(其中一些是新的),由苯磺酰胺(II),苯磺酰基异氰酸酯(IV)和苯磺酰氯(VI)和苯磺酰基异氰酸酯 杂环取代的氨基甲酸酯(III),胺(V)和/或(硫代) - 异氰酸酯(XIX)。

    Substituted isoxazolines, process for their preparation, composition
containing them, and their use of safeners
    48.
    发明授权
    Substituted isoxazolines, process for their preparation, composition containing them, and their use of safeners 失效
    取代的异恶唑啉,其制备方法,含有它们的组合物及其使用安全剂

    公开(公告)号:US5516750A

    公开(公告)日:1996-05-14

    申请号:US306110

    申请日:1994-09-14

    CPC分类号: A01N25/32 A01N43/80

    摘要: Substituted isoxazolines, process for their preparation, compositions containing them, and their use as safeners.Compounds of the formula (I) and salts thereof, ##STR1## in which R.sup.1 is carboxyl, formyl or another acyl radical or a derivative of the last-mentioned 3 groups,R.sup.2 is hydrogen, halogen, C.sub.1 -C.sub.18 -alkyl, C.sub.3 -C.sub.8 -cycloalkyl, C.sub.2 -C.sub.8 -alkenyl, C.sub.2 -C.sub.8 -alkynyl, C.sub.1 -C.sub.18 -alkoxy, C.sub.2 -C.sub.8 -alkenyloxy, C.sub.2 -C.sub.8 -alkynyloxy, C.sub.1 -C.sub.18 -alkylthio, C.sub.2 -C.sub.8 -alkenylthio, each of the last-mentioned 9 radicals in each case being unsubstituted or substituted, or (C.sub.1 -C.sub.8 -alkoxy)carbonyl, andR.sup.3 and R.sup.4 independently of one another are an aliphatic, araliphatic or heteroaraliphatic radical having 1 to 30 carbon atoms which is unsubstituted or substituted by one or more functional groups, oran aromatic or heteroaromatic radical which is unsubstituted or substituted,are suitable as safenets for pesticides, preferably herbicides, in crop plants. The compounds can be prepared from alkenes (II) and nitrile oxides (III) by the process of claim 6.

    摘要翻译: 取代的异恶唑啉,其制备方法,含有它们的组合物及其作为安全剂的用途。 式(I)化合物及其盐,其中R1是羧基,甲酰基或另一个酰基或最后提到的3个基团的衍生物,其中R 2是氢,卤素,C 1 -C 18 - 烷基 ,C 3 -C 8 - 环烷基,C 2 -C 8 - 烯基,C 2 -C 8 - 炔基,C 1 -C 18 - 烷氧基,C 2 -C 8 - 烯氧基,C 2 -C 8 - 炔氧基,C 1 -C 18烷硫基, 在每种情况下最后提及的9个基团是未取代的或取代的,或(C 1 -C 8 - 烷氧基)羰基,且R 3和R 4彼此独立地是具有1至30个碳原子的脂族,芳脂族或杂脂族基团,其是未取代的 或被一个或多个官能团取代,或未取代或取代的芳族或杂芳族基团适合作为农作物的保藏剂,优选除草剂在作物植物中。 化合物可以通过权利要求6的方法由烯烃(II)和氧化腈(III)制备。

    Process for the preparation of N-alkylsulfonylaminosulfonylureas
    49.
    发明授权
    Process for the preparation of N-alkylsulfonylaminosulfonylureas 失效
    制备N-烷基磺酰氨基脲的方法

    公开(公告)号:US5155222A

    公开(公告)日:1992-10-13

    申请号:US731518

    申请日:1991-07-17

    CPC分类号: C07D521/00

    摘要: Known herbicides of the formula (I) ##STR1## in which R.sup.1 is alkyl, alkenyl or alkynyl, which are optionally substituted by halogen, alkoxy or alkoxycarbonyl,R.sup.2 is H, alkyl, alkenyl, alkynyl or cycloalkyl,R.sup.3 and R.sup.4 are H or alkyl,R.sup.5 and R.sup.6 are H, alkyl or alkoxy, each of which can be substituted by halogen, alkoxy or alkylthio, or are halogen, alkylthio, alkylamino or dialkylamino,or, if R.sup.2 or R.sup.3 is H, their salts with bases, can be obtained when compounds of the formula IIR.sup.1 -SO.sub.2 -NR.sup.2 -SO.sub.2 -NHR.sup.3 (II)in whichR.sup.1, R.sup.2 and R.sup.3 are as defined above,are reacted with compounds of the formula III ##STR2## in which R.sup.4, R.sup.5 and R.sup.6 are as defined above andR.sup.7 is alkyl, haloalkyl or optionally substituted phenyl,in an inert organic solvent, to give the compounds of the formula I.

    摘要翻译: 式(I)的已知除草剂其中R 1为任选被卤素,烷氧基或烷氧基羰基取代的烷基,烯基或炔基,R 2为H,烷基,烯基,炔基或环烷基,R 3和R 4 卤素,烷硫基,烷基氨基或二烷基氨基,或者如果R2或R3是H,则它们的盐与 当其中R 1,R 2和R 3如上所定义的式IIR 1 -SO 2 -NR 2 -SO 2 -NHR 3(II)的化合物与式III的化合物(III)反应时,可以获得碱, 其中R4,R5和R6如上定义,R7是烷基,卤代烷基或任选取代的苯基,在惰性有机溶剂中,得到式I化合物。