公开(公告)号：US20080248952A1

公开(公告)日：2008-10-09

申请号：US11631004

申请日：2005-07-06

申请人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： C07D487/04 ,  A01N43/90 ,  A01N25/00

CPC分类号： A01N43/90 ,  C07D487/04

摘要： Substituted triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or a group R1, R1 and R2 together with the nitrogen atom, to which they are attached, may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and which may comprise one to three further heteroatoms from the groups consisting of O, N and S as ring member and/or may be substituted according to the description; L is fluorine, chlorine or methyl; X is cyano, C1-C4-alkyl, C1-C4-alkoxy or C1-C2-haloalkoxy, where X is not methyl if R1 and R2 together are n-pentylene or 3-methyl-n-pentylene and L is fluorine, or R1 and R2 together are 3-methyl-n-pentylene and L is chlorine; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 取代基如下定义：式I的取代三唑并嘧啶：R 1是烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，卤代环烯基，炔基， 包含一至四个由O，N和S组成的组的杂原子的五或六元饱和的部分不饱和或芳族杂环，R 2是氢或基团R 1， R 1，R 2和R 2与它们所连接的氮原子一起也可以形成五元或六元杂环基或杂芳基，它们是 通过N连接并且其可以包含一个至三个由O，N和S组成的基团的另外的杂原子作为环成员和/或可以根据描述被取代; L是氟，氯或甲基; X是氰基，C 1 -C 4 - 烷基，C 1 -C 4 - 烷氧基或C 1 -C 4 - 如果R 1和R 2一起都是正 - 亚戊基，其中X不是甲基，其中X不是甲基 或3-甲基 - 正戊烯，L是氟，R 1和R 2一起是3-甲基 - 正戊烯，L是氯; 制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20080227795A1

公开(公告)日：2008-09-18

申请号：US10585992

申请日：2005-01-15

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04 ,  A01P3/00

CPC分类号： C07D487/04 ,  A01N43/90

摘要： The invention relates to substituted triazolopyrimidines of formula (I), with the substituents as follows: R1, R2=H, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkinyl, haloalkinyl, phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle, comprising one to four heteroatoms of the group O, N or S, R1 and R2 can, together with the nitrogen atom to which it is attached, form a five- or six-membered heterocycle or heteroaryl, bonded via N and containing one to three further heteroatoms from the group O, N and S as ring members, substituted as per the description, L1=fluorine, chlorine or bromine, L2=H, alkyl or alkoxy and X=halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy. The invention further relates to methods and intermediates for production of said compounds, agents comprising the same and use thereof for controlling fungal pests harmful to plants.

摘要翻译： 本发明涉及式（I）的取代三唑并嘧啶，其取代基如下：R 1，R 2 = H，烷基，卤代烷基，环烷基，卤代环烷基，烯基， 卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基，苯基，萘基或五元或六元饱和的部分不饱和或芳族杂环，其包含一至四个O，N或S的杂原子， / SUP>和R 2可以与其所连接的氮原子一起形成五元或六元杂环或杂芳基，其通过N键合并含有一至三个其它杂原子 基团O，N和S作为环成员，根据描述被取代，L 1 =氟，氯或溴，L 2 = H，烷基或烷氧基，X = 卤素，氰基，烷基，卤代烷基，烷氧基或卤代烷氧基。 本发明还涉及用于生产所述化合物的方法和中间体，包含该化合物的试剂和用于控制对植物有害的真菌害虫的用途。

公开(公告)号：US20070129380A1

公开(公告)日：2007-06-07

申请号：US10565656

申请日：2004-07-03

申请人： Frank Schieweck ,  Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Oliver Wagner ,  Siegfried Strathmann ,  Ulrich Scholf ,  Maria Scherer ,  Reinhard Stierl

发明人： Frank Schieweck ,  Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Oliver Wagner ,  Siegfried Strathmann ,  Ulrich Scholf ,  Maria Scherer ,  Reinhard Stierl

IPC分类号： A61K31/505 ,  C07D239/42

CPC分类号： C07D239/42

摘要： The invention relates to 2-substituted pyrimidines of the formula I in which the index n and these substituents R1, R2 and R3 are as defined in the description and R4 is as defined below: R4 corresponds to one of the formulae where Ra is hydrogen, C1-C6-alkyl, C2-C8-alkenyl, C2-C8-alkynyl, C3-C6-cycloalkyl or C1-C4-alkoxy and R5 is hydrogen, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C1-C4-alkyloxy-C1-C2-alkyl, phenyl-C1-C2-alkyl or phenyloxy-C1-C2-alkyl, to processes for preparing these compounds, to compositions comprising these compounds and to their use as pesticides.

摘要翻译： 本发明涉及式I的2-取代嘧啶，其中指数n和这些取代基R 1，R 2和R 3是 如在说明书中所定义的，R 4是如下定义的：R 4对应于下式之一其中R a a是氢，C 1〜 C 1 -C 6烷基，C 2 -C 8 - 烯基，C 2 - 亚烷基，C 2 -C 6 - C 1 -C 8 - 炔基，C 3 -C 6 - 环烷基或C 1 -C 6 - 4 - 烷氧基和R 5是氢，C 1 -C 6 - 烷基，C 2〜 C 1 -C 6 - 烯基，C 2 -C 6 - 炔基，C 1 -C 6 - 4 - 烷氧基-C 1 -C 2 - 烷基，苯基-C 1 -C 2 - 亚烷基 烷基或苯氧基-C 1 -C 2 - 烷基，用于制备这些化合物的方法，包含这些化合物的组合物及其作为农药的用途。

公开(公告)号：US20050107619A1

公开(公告)日：2005-05-19

申请号：US10507605

申请日：2003-03-12

申请人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Jordi Blasco ,  Norbert Gotz ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Reinhard Stierl

发明人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Jordi Blasco ,  Norbert Gotz ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Reinhard Stierl

IPC分类号： A01N37/18 ,  A01N37/36 ,  A01N37/38 ,  C07B61/00 ,  C07C231/12 ,  C07C233/22 ,  C07C235/34 ,  C07C233/73

CPC分类号： C07C235/34 ,  A01N37/18 ,  A01N37/36 ,  A01N37/38 ,  C07C233/22 ,  C07C2601/02 ,  C07C2601/08 ,  C07C2601/14

摘要： Z-substituted acrylamides of formula (I), where the substituents have the following meanings: X=H, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, with X in the 3- or 4-position, n=1 or 2, where X can be different if n=2, R1=alkyl, haloalkyl, cycloalkyl, alkoxy, haloalkoxy, aziridine and oxirane and R2=H, alkyl, haloalkyl, allyl, propargyl or CH2C≡C-alkyl. Methods for production thereof, agents comprising the above and the use thereof for the treatment of plant-pathogenic fungal pests.

摘要翻译： 式（I）的Z-取代的丙烯酰胺，其中取代基具有以下含义：X = H，卤素，烷基，卤代烷基，烷氧基，卤代烷氧基，其中X为3-或4-位，n = 1或2，其中 如果n = 2，则X可以不同，R 1 =烷基，卤代烷基，环烷基，烷氧基，卤代烷氧基，氮丙啶和环氧乙烷，R 2 = H，烷基，卤代烷基，烯丙基 炔丙基或CH 2C≡C-烷基。 其制备方法，包含上述物质及其用于治疗植物致病性真菌害虫的用途。

公开(公告)号：US20050181948A1

公开(公告)日：2005-08-18

申请号：US10509112

申请日：2003-03-27

申请人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Jordi Blasco ,  Norbert Gotz ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Reinhard Stierl

发明人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Jordi Blasco ,  Norbert Gotz ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Reinhard Stierl

IPC分类号： C07D213/56 ,  C07D213/61 ,  C07D263/10 ,  A01N43/60 ,  A01N43/40 ,  A01N43/54

CPC分类号： C07D263/10 ,  C07D213/56 ,  C07D213/61

摘要： The present invention relates to novel phenethylacrylamides of the formula I in which the substituents R1, R2, R3 and R4 have the following meanings: R1 is hydrogen, halogen, C1-C4-alkyl, C1-C4-alkoxy, C3-C8-cycloalkyl, C1-C4-haloalkoxy or C1-C4-haloalkyl; R2 is hydrogen, halogen, C1-C4-alkyl, C1-C4-alkoxy, C3-C10-cycloalkyl, C1-C4-haloalkoxy or C1-C4-haloalkyl; R3 is C1-C4-alkyl, C1-C4-haloalkyl, propargyl, C3-C4-alkenyl or a radical of the formula —H2C—C≡C—C(Ra, Ra)—Rc, wherein Ra, Rb independently of one another are hydrogen or methyl and Rc is hydrogen or C1-C4-alkyl; R4 is methyl or C1-haloalkyl; and Het is a 5- or 6-membered heteroaromatic ring, to processes for their preparation, and to the use of phenethylacrylamides of the formula I for controlling phytopathogenic harmful fungi.

摘要翻译： 本发明涉及式I的新的苯乙基丙烯酰胺，其中取代基R 1，R 2，R 3和R 4 具有以下含义：R 1是氢，卤素，C 1 -C 4 - 烷基，C 1 C 1 -C 4 - 烷氧基，C 3 -C 8 - 环烷基，C 1 -C 4 - 卤代烷氧基或C 1 -C 4 - 卤代烷基; R 2是氢，卤素，C 1 -C 4 - 烷基，C 1 -C 3 - 4 - 烷氧基，C 3 -C 10 - 环烷基，C 1 -C 4 - 卤代烷氧基或C 1 -C 4 - 卤代烷基; R 3是C 1 -C 4 - 烷基，C 1 -C 4烷基，C 1 -C 4烷基，C 1 -C 4 - 烷基，炔丙基，C 3 -C 4 - 烯基或式-H 2C≡CC（R 0）的基团 其中R a，R b，R b独立地为C 1 -C 4，其中R a，R b， 另一个是氢或甲基，R c是氢或C 1 -C 4 - 烷基; R 4是甲基或C 1 - 卤代烷基; 并且Het是5或6元杂芳环，用于其制备方法，以及使用式I的苯乙基丙烯酰胺来控制植物病原性有害真菌。

公开(公告)号：US20070117852A1

公开(公告)日：2007-05-24

申请号：US10582040

申请日：2004-12-22

申请人： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Anja Schwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  John-Bryan Speakman ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl

发明人： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Anja Schwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  John-Bryan Speakman ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl

IPC分类号： A01N43/56 ,  A01N43/40 ,  A01N43/78 ,  C07D213/24

CPC分类号： C07D213/82 ,  A01N43/40 ,  A01N43/56 ,  A01N43/78 ,  A01N47/48 ,  C07C251/38 ,  C07D207/34 ,  C07D231/14 ,  C07D263/34 ,  C07D277/56 ,  C07D279/12 ,  C07D307/30 ,  C07D307/54 ,  C07D307/71 ,  C07D333/38

摘要： The present invention relates to (hetero)cyclylcarboxanilides of the formula I, in which n is 0, 1, 2, 3 or 4; and m is 1, 2 or 3, Y is oxygen or sulfur; A is unsubstituted or substituted phenyl or is an at least monounsaturated, unsubstituted or substituted 5- or 6-membered heterocycle, R1, R2, R3m, R4m, R5 and R6 are as defined in claim 1, and their agriculturally useful salts. Moreover, the present invention relates to the use of the (hetero)cyclylcarboxanilides of the formula I and their agriculturally useful salts as fungicides, and to crop protection compositions comprising these compounds.

摘要翻译： 本发明涉及式（I）的（杂）环己基甲酰苯胺，其中n为0,1,2,3或4; m为1,2或3，Y为氧或硫; A是未取代或取代的苯基，或至少是一个不饱和的，未取代的或取代的5元或6元杂环，R 1，R 2，R 3， R 4，R 5，R 5和R 6如权利要求1所定义，及其农业上有用的盐。 此外，本发明涉及式I的（杂）环己基甲酰苯胺及其农业上有用的盐作为杀真菌剂，以及包含这些化合物的作物保护组合物的用途。

公开(公告)号：US20050272749A1

公开(公告)日：2005-12-08

申请号：US10531981

申请日：2003-11-04

申请人： Jordi Tormo Blasco ,  Carsten Bletner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo Blasco ,  Carsten Bletner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： C07D487/04 ,  A61K31/519

CPC分类号： C07D487/04

摘要： 5-Alkyl-7-aminotriazolopyrimidines of the formula I, where: R1, R2 are hydrogen, alkyl, alkenyl, alkynyl, haloalkyl, cycloalkyl, phenyl, naphthyl; 5- or 6-membered saturated, unsaturated or aromatic heterocyclyl which contains one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or R1 and R2 together with the bridging nitrogen atom can form a 5- or 6-membered ring which contains one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; R3 is cycloalkyl or bicycloalkyl; where R1, R2 and R3 may be substituted as outlined in the description; X is alkyl or haloalkyl; and their salts; processes and intermediates for their preparation, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

摘要翻译： 式I的5-烷基-7-氨基三唑并嘧啶，其中：R 1，R 2是氢，烷基，烯基，炔基，卤代烷基，环烷基，苯基，萘基; 含有1-4个氮原子或一至三个氮原子和一个硫或氧原子的5-或6-元饱和，不饱和或芳族杂环基; 或R 1和R 2与桥连氮原子一起可以形成含有1-4个氮原子或一至三个氮原子的5-或6-元环，并且 一个硫或氧原子; R 3是环烷基或双环烷基; 其中R 1，R 2和R 3可以如说明书中概述的那样被取代; X是烷基或卤代烷基; 和它们的盐; 描述了其制备方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20080249113A1

公开(公告)日：2008-10-09

申请号：US11659192

申请日：2005-07-28

申请人： Carsten Blettner ,  Jochen Dietz ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Carsten Blettner ,  Jochen Dietz ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04 ,  A01N25/26 ,  A01P3/00

CPC分类号： A01N43/90 ,  A01N43/653 ,  A01N47/14 ,  A01N43/50 ,  A01N57/12 ,  A01N47/04 ,  A01N37/34 ,  A01N43/40 ,  A01N37/50 ,  A01N37/46 ,  A01N43/84 ,  A01N37/38 ,  A01N43/28 ,  A01N47/38 ,  A01N43/54 ,  A01N43/32 ,  A01N59/20 ,  A01N2300/00

摘要： Fungicidal mixtures, comprising as active components 1) a 5-chloro-6-phenyl-7-heterocyclylaminotriazolopyrimidine of the formula I, in which D together with the nitrogen atom forms a pyrrolidine, piperidine or azepine ring, which rings are unsubstituted or substituted by one or two methyl groups or by an ethyl, propyl or butyl group; and L is methyl, fluorine or chlorine; and 2) at least one active compound II selected from the following groups: A) azoles; B) strobilurins; C) acylalanines; D) amine derivatives; E) anilinopyrimidines; F) dicarboximides; G) cinnamides and analogs; H) antibiotics; K) dithiocarbamates; L) heterocyclic compounds according to the description; M) sulfur and copper fungicides; N) nitrophenyl derivatives; O) phenylpyrroles; P) sulfenic acid derivatives; Q) other fungicides according to the description; or R) growth retardants; in a synergistically effective amount, novel triazolopyrimidines, methods for controlling harmful fungi using compounds or mixtures of a compound I with an active compound of groups A) to R) and the use of the compounds I with the active compounds of groups A) to R) for preparing such mixtures, and also compositions comprising these compounds or mixtures.

摘要翻译： 包含作为活性组分的杀真菌混合物1）式I的5-氯-6-苯基-7-杂环基氨基三唑并嘧啶，其中D与氮原子一起形成吡咯烷，哌啶或氮杂环，该环是未取代的或被 一个或两个甲基或乙基，丙基或丁基; L为甲基，氟或氯; 和2）至少一种选自以下组的活性化合物II：A）唑类; B）嗜球果伞素 C）酰基丙氨酸; D）胺衍生物; E）苯胺嘧啶嘧啶; F）二羧酰亚胺; G）肉桂酸酯类似物; H）抗生素; K）二硫代氨基甲酸盐; L）杂环化合物; M）硫和铜杀菌剂; N）硝基苯基衍生物; O）苯基吡咯; P）亚磺酸衍生物; Q）其他杀菌剂根据说明; 或R）生长阻滞剂; 协同有效量的新型三唑并嘧啶，使用化合物或化合物I与A）至R）的活性化合物的混合物来控制有害真菌的方法以及将化合物I与基团A）至R的活性化合物 ），以及包含这些化合物或混合物的组合物。

公开(公告)号：US20090036509A1

公开(公告)日：2009-02-05

申请号：US11628324

申请日：2005-06-11

申请人： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Anja Schwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Frank Werner ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl ,  Maria Scherer

发明人： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Anja Schwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Frank Werner ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl ,  Maria Scherer

IPC分类号： A01N43/56 ,  C07D231/14 ,  A01P3/00

CPC分类号： C07D231/14

摘要： The present invention relates to N-(ortho-phenyl)-1-methyl-3-trifluoromethylpyrazole-4-carboxanilides of the formula I in which the substituents are as defined below: R1 and R2 independently of one another are halogen, C1-C6-alkyl, C1-C6-haloalkyl, cyano, nitro, methoxy, trifluoromethoxy or difluoromethoxy; with the proviso that when R2 is chlorine in position 4, R1 is not trifluoromethyl in position 3.

摘要翻译： 本发明涉及式I的N-（邻 - 苯基）-1-甲基-3-三氟甲基吡唑-4-甲酰苯胺，其中取代基如下所定义：R 1和R 2彼此独立地为卤素，C 1 -C 6 烷基，C 1 -C 6卤代烷基，氰基，硝基，甲氧基，三氟甲氧基或二氟甲氧基; 条件是当R2在4位是氯时，R1不在3位是三氟甲基。

公开(公告)号：US20070149400A1

公开(公告)日：2007-06-28

申请号：US10582934

申请日：2004-12-15

申请人： Jordi Tormo i Blasco ,  Carsten Biettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Biettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Substituted triazolopyrimidines of the formula I in which the substituents are as defined below: L is hydrogen, chlorine or bromine; R1, R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain a further heteroatom from the group consisting of O, N and S as ring member and/or may be substituted as defined in the description; R3 is alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl, cycloalkyl, halocycloalkyl or phenylalkyl; R1, R2 and/or R3 may be substituted as defined in the description; X is halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 取代基如下定义的式I的取代三唑并嘧啶：L是氢，氯或溴; R 1，R 2是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或苯基，萘基或五或 含有一至四个由O，N和S杂原子组成的组的六元饱和，部分不饱和或芳族杂环，R 1和R 2连同氮 它们所连接的原子也可以形成通过N连接的五元或六元杂环基或杂芳基，并且可以含有作为环成员的O，N和S中的另外的杂原子和/或可被取代为 在说明书中定义; R 3是烷基，卤代烷基，烯基，卤代烯基，炔基，卤代炔基，环烷基，卤代环烷基或苯基烷基; R 1，R 2和/或R 3可以如说明书中所定义的取代; X是卤素，氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; 制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。