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64 条记录 (耗时 0.02 秒)

    Disubstituted triphenylmethylimidazoles
    51.
    发明授权
    Disubstituted triphenylmethylimidazoles 失效
    分离的三苯基甲基咪唑

    公开(公告)号：US4052409A

    公开(公告)日：1977-10-04

    申请号：US339430

    申请日：1973-03-08

    申请人： Karl Heinz Buchel ,  Erik Regel ,  Manfred Plempel

    发明人： Karl Heinz Buchel ,  Erik Regel ,  Manfred Plempel

    IPC分类号： C07D233/62 ,  C07D521/00

    CPC分类号： C07D231/12 ,  C07D233/56 ,  C07D249/08

    摘要： Imidazoles of the formula ##STR1## and pharmaceutically acceptable nontoxic salts thereof, wherein X is methyl or chloro,Y is methyl or chloro, or, when Z is methyl or chloro, Y is hydrogen, andZ is methyl or chloro, or, when Y is methyl or chloro, Z is hydrogen,Are useful as antimycotics for the treatment of mycotic infections in humans and animals. The imidazoles may be produced by reacting the corresponding triphenylmethylcarbinol with a brominating or chlorinating agent and thereafter reacting the resultant triphenylmethyl halide, either with or without isolation, with imidazole in the presence or absence of an acid-binding agent, or they may be prepared by reacting a triphenylmethyl halide with imidazole, either in the presence or absence of an acid-binding agent.

    N-Methyl-imidazole derivatives for treating mycotic infections
    53.
    发明授权
    N-Methyl-imidazole derivatives for treating mycotic infections 失效
    用于治疗真菌感染的N-甲基 - 咪唑衍生物

    公开(公告)号：US3980780A

    公开(公告)日：1976-09-14

    申请号：US554203

    申请日：1975-02-28

    申请人： Wilfried Draber ,  Karl Heinz Buchel ,  Erik Regel ,  Manfred Plempel

    发明人： Wilfried Draber ,  Karl Heinz Buchel ,  Erik Regel ,  Manfred Plempel

    IPC分类号： A61K31/495 ,  A61K31/505 ,  C07D241/12 ,  C07D403/06

    CPC分类号： C07D403/06 ,  A61K31/495 ,  A61K31/505 ,  C07D241/12

    摘要： N-methyl-imidazole derivatives of the formula: ##EQU1## or a pharmaceutically acceptable non-toxic salt thereof, wherein X is an unsubstituted or substituted 6-membered heteroaromatic moiety having two nitro heteroatoms,Y is an unsubstituted or substituted aliphatic moiety, an unsubstituted or substituted cycloaliphatic moiety, an unsubstituted or substituted aralkyl moiety or an unsubstituted or substituted aryl moiety, andZ is an unsubstituted or substituted aliphatic moiety, an unsubstituted or substituted cycloaliphatic moiety, an unsubstituted or substituted aralkyl moiety, an unsubstituted or substituted aryl moiety, an unsubstituted or substituted pyridyl moiety or an alkoxycarbonyl moiety,Are useful as antimycotic agents.

    摘要翻译： 其中X是具有两个硝基杂原子的未取代或取代的6元杂芳族部分，Y是未取代的或未取代的或未取代的 取代的脂族部分，未取代或取代的脂环族部分，未取代或取代的芳烷基部分或未取代或取代的芳基部分，Z是未取代或取代的脂族部分，未取代或取代的脂环族部分，未取代或取代的芳烷基部分， 未取代或取代的芳基部分，未取代或取代的吡啶基部分或烷氧基羰基部分，作为抗菌剂有用。

    Substituted triazolylmethyl-oxiranes and their use as intermediates for fungicides
    55.
    发明授权
    Substituted triazolylmethyl-oxiranes and their use as intermediates for fungicides 失效
    取代的三唑基甲基 - 环氧乙烷及其作为杀真菌剂的中间体

    公开(公告)号：US4499281A

    公开(公告)日：1985-02-12

    申请号：US352689

    申请日：1982-02-26

    申请人： Graham Holmwood ,  Erik Regel

    发明人： Graham Holmwood ,  Erik Regel

    IPC分类号： C07D405/06 ,  A01N43/653 ,  C07D249/08 ,  C07D521/00 ,  A01N43/64

    CPC分类号： C07D231/12 ,  C07D233/56 ,  C07D249/08

    摘要： A substituted triazolylmethyl-oxirane of the formula ##STR1## in which R is optionally substituted alkyl, aryl or cycloalkyl is prepared by reacting a triazolyl-ketone of the formula ##STR2## with (a) dimethyloxosulphonium methylide of the formula ##STR3## or (b) trimethylsulphonium methylsulphate of the formula[(CH.sub.3).sub.3 S].sup..sym. CH.sub.3 SO.sub.4.sup..crclbar.in the presence of a diluent.The end product can then be reacted with a phenol of the formulaR"--OHto produce known fungicidally active compounds of the formula ##STR4## in which R" is optionally substituted phenyl.

    摘要翻译： 其中R为任选取代的烷基，芳基或环烷基的取代三唑基甲基 - 环氧乙烷通过使式（IMAGE）的三唑基酮与（a）式（IMAGE）的二甲基氧基锍甲基化物或（ b）在稀释剂存在下，式[（CH3）3S]（+）CH3SO4（ - ）的三甲基锍甲基硫酸盐。 然后可以使最终产物与式R“-OH的酚反应以产生已知的具有式”IMAGE“的杀真菌活性化合物，其中R”为任选取代的苯基。

    Azolylamidine compounds and herbicidal compositions
    58.
    发明授权
    Azolylamidine compounds and herbicidal compositions 失效
    唑基脒化合物和除草组合物

    公开(公告)号：US4073636A

    公开(公告)日：1978-02-14

    申请号：US607986

    申请日：1975-08-26

    申请人： Erik Regel ,  Ludwig Eue ,  Robert R. Schmidt

    发明人： Erik Regel ,  Ludwig Eue ,  Robert R. Schmidt

    IPC分类号： C07D207/34 ,  C07D231/12 ,  C07D231/56 ,  C07D233/68 ,  C07D233/92 ,  C07D249/04 ,  C07D249/08 ,  C07D249/10 ,  A01N9/22

    CPC分类号： C07D249/08 ,  C07D207/34 ,  C07D231/12 ,  C07D231/56 ,  C07D233/68 ,  C07D233/92 ,  C07D249/04

    摘要： New azolylamidines of the formula ##STR1## WHEREIN N IS AN INTEGER FROM 0 TO 5,R.sup.1 is halogen, alkyl, alkoxy, alkylthio, haloalkoxy, haloalkylthio, halophenoxy or haloalkyl;R.sup.2 and R.sup.3, independently of one another, are each hydrogen, alkyl, alkoxyalkyl, cycloalkyl, alkoxy or alkoxycarbonylalkyl, of, preferably not more than 7 carbon atoms; or taken together, represent a lower alkylene bridge which can be interrupted by one or more hetero-atoms; andAz represents an azolyl radical selected from imidazol-1-yl, pyrrol-1-yl, pyrazol-1-yl,1,2,4-triazol-1-yl, 1,2,4-triazol-4-yl or 1,2,3-triazol-1-yl,And their salts are outstandingly effective herbicides showing particularly selective action.

    摘要翻译： 式（I）的新的吡唑基脒，其中N为0至5的整数，R 1为卤素，烷基，烷氧基，烷硫基，卤代烷氧基，卤代烷硫基，卤代苯氧基或卤代烷基; R 2和R 3彼此独立地为氢，烷基，烷氧基烷基，环烷基，烷氧基或烷氧基羰基烷基，优选不超过7个碳原子; 或一起代表可被一个或多个杂原子中断的低级亚烷基桥; 并且Az表示选自咪唑-1-基，吡咯-1-基，吡唑-1-基，1,2,4-三唑-1-基，1,2,4-三唑-4-基或 1,2,3-三唑-1-基，它们的盐是非常有效的除草剂，显示出特别的选择性作用。