Compositions containing N-amino- and N-hydroxy-quinazolinones and methods for preparing libraries thereof
    56.
    发明授权
    Compositions containing N-amino- and N-hydroxy-quinazolinones and methods for preparing libraries thereof 失效
    含有N-氨基和N-羟基 - 喹唑啉酮的组合物及其制备方法

    公开(公告)号:US06184377B2

    公开(公告)日:2001-02-06

    申请号:US08990855

    申请日:1997-12-15

    申请人: Yun Gao

    发明人: Yun Gao

    IPC分类号: C07D23992

    CPC分类号: C07D239/92

    摘要: The present invention is directed to certain N-amino- and N-hydroxy-quinazolinone compounds and synthetic methods for synthesis thereof, which compounds may find use in combinatorial libraries. More specifically, the invention is directed to the synthesis of 3-hydroxy- and 3-amino-4(1H)-quinazolinones via the reaction of an appropriate 2-aminobenzamide compound with a carboxylic acid or acyl halide at ambient temperature performed on a solid support or in solution.

    摘要翻译: 本发明涉及某些N-氨基 - 和N-羟基 - 喹唑啉酮化合物及其合成方法,该化合物可用于组合文库。 更具体地,本发明涉及通过适当的2-氨基苯甲酰胺化合物与羧酸或酰基卤在环境温度下对固体进行的反应合成3-羟基 - 和3-氨基-4(1H) - 喹唑啉酮 支持或解决方案。

    Ruthenium-catalyzed production of cyclic sulfates
    57.
    发明授权
    Ruthenium-catalyzed production of cyclic sulfates 失效
    钌催化的环状硫酸盐生产

    公开(公告)号:US5321143A

    公开(公告)日:1994-06-14

    申请号:US712199

    申请日:1991-06-07

    摘要: A ruthenium catalyzed method to synthesize cyclic sulfate compounds from the corresponding cyclic sulfites, and the cyclic sulfate reaction products obtained by this method. These cyclic sulfates further react with selected nucleophiles to give various substituted products. The method is an efficient means for the synthesis of chiral building blocks from tartaric acid enantiomers in high yields using an overall two-stage, one-pot reaction procedure. The chiral compounds can be transformed by nucleophilic reactions into chiral building blocks useful for the synthesis of natural biologically active products, such as antibiotics and pheromones.

    摘要翻译: 从相应的环状亚硫酸盐合成环状硫酸盐化合物的钌催化方法和通过该方法得到的环状硫酸盐反应产物。 这些环状硫酸盐与选择的亲核试剂进一步反应,得到各种取代的产物。 该方法是使用总体两步一锅反应方法以高产率从酒石酸对映异构体合成手性结构单元的有效手段。 手性化合物可以通过亲核反应转化成用于合成天然生物活性产物(如抗生素和信息素)的手性结构单元。

    Electrocatalytic oxidation method for the production of cyclic sulfates
and sulfamidates
    58.
    发明授权
    Electrocatalytic oxidation method for the production of cyclic sulfates and sulfamidates 失效
    用于生产环状硫酸盐和氨磺酸盐的电催化氧化法

    公开(公告)号:US5271812A

    公开(公告)日:1993-12-21

    申请号:US717432

    申请日:1991-06-19

    摘要: The invention relates to a process for the production of cyclic sulfates and cyclic sulfamidates from the corresponding cyclic sulfite and cyclic sulfamidite substrate, respectively. The method involves the electrolysis of a solvent mixture containing active metal species, non-metal oxidant species and substrate.

    摘要翻译: 本发明涉及分别从相应的环状亚硫酸盐和环状亚磺酰胺基质制备环状硫酸盐和环状磺酰胺酸盐的方法。 该方法涉及电解含有活性金属物质,非金属氧化剂物质和底物的溶剂混合物。

    Radio frequency identification tag having diversion-proof function and manufacturing method thereof
    60.
    发明授权
    Radio frequency identification tag having diversion-proof function and manufacturing method thereof 有权
    具有防转移功能的射频识别标签及其制造方法

    公开(公告)号:US09292783B2

    公开(公告)日:2016-03-22

    申请号:US14342531

    申请日:2012-03-20

    摘要: The present invention provides a radio frequency identification electronic tag with diversion-proof function and a process for making the same. The radio frequency identification electronic tag with diversion-proof function is formed of a supporting layer, a release liner, an antenna and a chip, wherein the release liner is bonded to one side of the supporting layer to form an entity, the antenna is bonded to the other side of the release liner, or, the antenna is bonded to the two sides of the entity formed by the supporting layer and the release liner, and is connected via overbridge points on the antenna, the overbridge points run through the supporting layer and the release liner so that antennas at the two sides are switched into conduction; the chip is bonded to the antenna. Once the RFID tag with diversion-proof function is peeled off or transferred, its physical structure will be destroyed and the information contained therein cannot be read, achieving the object of incapable of being reused. At the same time, the thermosetting resins are bonded organically according to the processing technology of the RFID tag, then the bonding points and the overbridge points of the chip have higher bonding fastness with the supporting layer, it is not easy for the chip to peel off with the release liner and better overbridge effect is achieved, which can greatly improve the yield of the finished RFID tag with diversion-proof function.

    摘要翻译: 本发明提供一种具有防分离功能的射频识别电子标签及其制造方法。 具有防转移功能的射频识别电子标签由支撑层,释放衬垫,天线和芯片形成,其中释放衬垫结合到支撑层的一侧以形成实体,天线被结合 或者天线结合到由支撑层和释放衬垫形成的实体的两侧,并且通过天线上的超桥点连接,跨桥点穿过支撑层 和释放衬垫,使得两侧的天线被切换成导通; 该芯片与天线结合。 一旦具有防转移功能的RFID标签被剥离或转移,其物理结构将被破坏,并且其中包含的信息不能被读取,从而达到无法再次使用的目的。 同时,根据RFID标签的加工工艺,热固性树脂有机结合,芯片的接合点和跨桥点与支撑层具有较高的粘接牢度,芯片不易剥离 脱离衬垫,实现更好的超桥效应,可以大大提高成品RFID标签的带防拆功能的产量。