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公开(公告)号:US5189063A
公开(公告)日:1993-02-23
申请号:US570099
申请日:1990-08-17
申请人: Alexander Klausener , Herbert Gayer , Wolfgang Kramer , Dieter Berg , Wilhelm Brandes , Gerd Hanssler , Ulrike Wachendorff-Neumann
发明人: Alexander Klausener , Herbert Gayer , Wolfgang Kramer , Dieter Berg , Wilhelm Brandes , Gerd Hanssler , Ulrike Wachendorff-Neumann
IPC分类号: C07D317/60 , A01N37/06 , A01N37/36 , A01N37/38 , A01N37/44 , A01N37/48 , A01N43/16 , A01N43/18 , A01N43/30 , A01N43/40 , A01N43/74 , A01N43/80 , C07C67/31 , C07C69/73 , C07C69/732 , C07C69/734 , C07C229/32 , C07C229/44 , C07C251/42 , C07C251/52 , C07C251/60 , C07C323/55 , C07C323/56 , C07C323/57 , C07D211/70 , C07D213/55 , C07D213/61 , C07D213/64 , C07D261/08 , C07D263/32 , C07D277/20 , C07D277/24 , C07D277/30 , C07D307/54 , C07D309/20 , C07D309/22 , C07D317/54 , C07D333/24 , C07D335/02 , C07D401/06 , C07D401/12 , C07D403/06 , C07D403/12 , C07D405/06 , C07D409/06 , C07D413/06 , C07D417/06 , C07D521/00
CPC分类号: A01N43/74 , A01N37/36 , A01N37/38 , A01N37/44 , A01N37/48 , A01N43/30 , A01N43/40 , A01N43/80 , C07C229/44 , C07C323/56 , C07C69/734 , C07D213/61 , C07D261/08 , C07D263/32 , C07D277/24 , C07D309/22 , C07D317/54 , C07D335/02
摘要: Pesticidal substituted acrylic esters of the formula ##STR1## in which R.sup.1 represents alkyl, or represents unsubstituted or substituted aralkyl,R.sup.2 represents dialkylamino, or represents a radical --Z--R.sup.3,R.sup.3 represents alkyl, or represents unsubstituted or substituted aralkyl,Z represents oxygen or sulphur,A represents ##STR2## where n represents a number from 0 to 6,R.sup.4 and R.sup.5 in each case independently of one another represent alkyl, or together represent an alkylene chain having 2 to 7 carbon atoms, andR.sup.6 represents alkyl, or represents a radical ##STR3## where R.sup.7 represents alkyl, alkoxy or dialkylamino,B represents the group CH--R.sup.8 or, whereR.sup.9 represents unsubstituted or substituted alkyl, alkenyl, alkynyl, aralkyl, aryl or hetaryl, and R and Q independently of one another represent hydrogen, alkyl, halogenoalkyl or alkoxy.
摘要翻译: 式(I)的杀虫取代的丙烯酸酯,其中R 1表示烷基,或表示未取代或取代的芳烷基,R 2表示二烷基氨基,或表示基团-Z-R 3,R 3表示烷基,或表示未取代或取代的芳烷基, Z表示氧或硫,A表示
其中n表示0至6的数,R4和R5各自独立地表示烷基,或一起表示具有2至7个碳原子的亚烷基链,R6表示 烷基,或表示基团,其中R 7表示烷基,烷氧基或二烷基氨基,B表示基团CH-R 8,或其中R 9表示未取代或取代的烷基,烯基,炔基,芳烷基,芳基或杂芳基,R和Q独立地 彼此表示氢,烷基,卤代烷基或烷氧基。 -
公开(公告)号:US5149859A
公开(公告)日:1992-09-22
申请号:US582443
申请日:1990-09-14
申请人: Atsuo Hazato , Takumi Takeyasu , Koji Tomimori , Yoshinori Kato
发明人: Atsuo Hazato , Takumi Takeyasu , Koji Tomimori , Yoshinori Kato
IPC分类号: C07C69/612 , C07C69/738 , C07C251/38 , C07C251/40 , C07C251/48 , C07C259/06 , C07C259/10 , C07C323/22 , C07C323/52 , C07C323/57
CPC分类号: C07C323/22 , C07C251/40 , C07C251/48 , C07C259/06 , C07C259/10 , C07C323/52 , C07C323/57 , C07C69/738
摘要: A naphthalene derivative having the formula (I): ##STR1## wherein R.sup.1 represents a hydrogen atom, a C.sub.1 -C.sub.5 alkyl group or a non-toxic salt moiety; R.sup.2 and R.sup.3 independently represent a hydrogen atom or --OR.sup.4 where R.sup.4 represents a hydrogen atom or a C.sub.1 -C.sub.3 alkyl group;A represents a group: ##STR2## [where X.sup.1 and X.sup.2 represents an oxygen atom or N--OR.sup.5 (where R.sup.5 represents a hydrogen atom or a C.sub.1 -C.sub.3 alkyl group)], a group: ##STR3## [where Y.sup.1 and Y.sup.2 independently an oxygen atom or a group N--OR.sup.6 (where R.sup.6 represents a hydrogen atom or a C.sub.1 -C.sub.3 alkyl group)], or a group: ##STR4## (where n is 0 or 1); and B represents --(CH.sub.2).sub.m -- wherein m is an integer of 1, to 8,--(CH.sub.2).sub.m.sbsb.1 --O--(CH.sub.2).sub.m.sbsb.2 -- wherein m.sub.1 and m.sub.2 are independently 1 or 2, or ##STR5## wherein m.sub.3 is 0 or 1.
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公开(公告)号:US4624962A
公开(公告)日:1986-11-25
申请号:US697340
申请日:1985-02-01
IPC分类号: C07C275/16 , C07C67/00 , C07C239/00 , C07C275/24 , C07C279/14 , C07C301/00 , C07C303/40 , C07C311/30 , C07C313/00 , C07C315/04 , C07C317/50 , C07C323/44 , C07C323/57 , C07C323/59 , C07D207/16 , C07D207/22 , C07D209/20 , C07D209/42 , C07D209/52 , C07D211/60 , C07D213/55 , C07D217/12 , C07D217/26 , C07D223/06 , C07D231/12 , C07D233/54 , C07D277/06 , C07D333/24 , C07D333/60 , C07D401/12 , C07D403/12 , C07D409/12 , C07D471/04 , C07D495/04 , A61K31/40
CPC分类号: C07D231/12 , C07C275/24 , C07C323/44 , C07D207/16 , C07D207/22 , C07D209/20 , C07D209/42 , C07D209/52 , C07D211/60 , C07D213/55 , C07D217/26 , C07D223/06 , C07D233/64 , C07D277/06 , C07D333/24 , C07D333/60 , C07D401/12 , C07D403/12 , C07D409/12 , C07D471/04 , C07D495/04 , C07C2101/04 , C07C2101/08
摘要: Compounds of the formula I ##STR1## in which n denotes 0-3,R.sup.1 and R.sup.1' are the same or different and denote hydrogen, alkyl or alkenyl, phenyl or benzyl, each substituted as desired;R.sup.2 denotes hydrogen, alkyl or alkenyl;R.sup.3 denotes hydrogen, alkyl, hydroxyalkyl, alkoxyalkyl or aminoalkyl, alkanoylaminoalkyl, guanidinoalkyl, imidazolylalkyl, indolylalkyl, mercaptoalkyl or alkylthioalkyl, phenylalkyl, hydroxphenylalkyl, phenoxyalkyl or phenylthioalkyl, or R.sup.2 and R.sup.3, together with the C and N atoms carrying them, denote a saturated or unsaturated 4- to 8-membered monocyclic or 8- to 10-membered bicyclic isocycle or heterocycle, optionally monosubstituted or disubstituted by hydroxyl, alkoxy having 1 to 3 C atoms or alkyl,R.sup.4 denotes hydrogen, alkyl, alkenyl, alkadienyl, alkinyl, alkeninyl or alkadiinyl, cycloalkyl, phenyl, benzyl, phenethyl or phenylpropyl, each of which can be optionally monosubstituted or disubstituted;R.sup.5 denotes hydrogen or alkyl, hydroxyl or alkoxy andR.sup.6 denotes hydrogen, optionally substituted alkyl, cycloalkyl, alkenyl, optionally monosubstituted or disubstituted phenyl or naphthyl, their salts, a process for their preparation and their use as medicaments.
摘要翻译: 式I的化合物其中n表示0-3,R1和R1'相同或不同,表示氢,烷基或链烯基,苯基或苄基,各自根据需要取代; R2表示氢,烷基或烯基; R3表示氢,烷基,羟基烷基,烷氧基烷基或氨基烷基,烷酰基氨基烷基,胍基烷基,咪唑基烷基,吲哚基烷基,巯基烷基或烷硫基烷基,苯基烷基,羟基苯基烷基,苯氧基烷基或苯硫基烷基,或R2和R3与携带它们的C和N原子一起表示饱和 或不饱和的4至8元单环或8至10元双环的单环或杂环,任选被羟基,具有1至3个C原子的烷氧基或烷基单取代或二取代,R4表示氢,烷基,烯基,链烯基,炔基, 链烯基或烷撑基,环烷基,苯基,苄基,苯乙基或苯基丙基,它们各自可以任选被单取代或二取代; R5表示氢或烷基,羟基或烷氧基,R6表示氢,任选取代的烷基,环烷基,烯基,任选单取代或二取代的苯基或萘基,它们的盐,其制备方法及其作为药物的用途。
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公开(公告)号:US4515803A
公开(公告)日:1985-05-07
申请号:US413663
申请日:1982-09-01
IPC分类号: C07C275/16 , C07C67/00 , C07C239/00 , C07C275/24 , C07C279/14 , C07C301/00 , C07C303/40 , C07C311/30 , C07C313/00 , C07C315/04 , C07C317/50 , C07C323/44 , C07C323/57 , C07C323/59 , C07D207/16 , C07D207/22 , C07D209/20 , C07D209/42 , C07D209/52 , C07D211/60 , C07D213/55 , C07D217/12 , C07D217/26 , C07D223/06 , C07D231/12 , C07D233/54 , C07D277/06 , C07D333/24 , C07D333/60 , C07D401/12 , C07D403/12 , C07D409/12 , C07D471/04 , C07D495/04 , C07D209/12
CPC分类号: C07D231/12 , C07C275/24 , C07C323/44 , C07D207/16 , C07D207/22 , C07D209/20 , C07D209/42 , C07D209/52 , C07D211/60 , C07D213/55 , C07D217/26 , C07D223/06 , C07D233/64 , C07D277/06 , C07D333/24 , C07D333/60 , C07D401/12 , C07D403/12 , C07D409/12 , C07D471/04 , C07D495/04 , C07C2101/04 , C07C2101/08
摘要: Compounds of the formula I ##STR1## in which n denotes 0-3,R.sup.1 and R.sup.1' are the same or different and denote hydrogen, alkyl or alkenyl, phenyl or benzyl, each substituted as desired;R.sup.2 denotes hydrogen, alkyl or alkenyl;R.sup.3 denotes hydrogen, alkyl, hydroxyalkyl, alkoxyalkyl or aminoalkyl, alkanoylaminoalkyl, guanidinoalkyl, imidazolylalkyl, indolylalkyl, mercaptoalkyl or alkylthioalkyl, phenylalkyl, hydroxyphenylalkyl, phenoxyalkyl or phenylthioalkyl, or R.sup.2 and R.sup.3, together with the C and N atoms carrying them, denote a saturated or unsaturated 4- to 8-membered monocyclic or 8- to 10-membered bicyclic isocycle or heterocycle, optionally monosubstituted or disubstituted by hydroxyl, alkoxy having 1 to 3 C atoms or alkyl,R.sup.4 denotes hydrogen, alkyl, alkenyl, alkadienyl, alkinyl, alkeninyl or alkadiinyl, cycloalkyl, phenyl, benzyl, phenethyl or phenylpropyl, each of which can be optionally monosubstituted or disubstituted;R.sup.5 denotes hydrogen or alkyl, hydroxyl or alkoxy andR.sup.6 denotes hydrogen, optionally substituted alkyl, cycloalkyl, alkenyl, optionally monosubstituted or disubstituted phenyl or naphthyl,their salts, a process for their preparation and their use as medicaments.
摘要翻译: 式I的化合物其中n表示0-3,R1和R1'相同或不同,表示氢,烷基或链烯基,苯基或苄基,各自根据需要取代; R2表示氢,烷基或烯基; R3表示氢,烷基,羟基烷基,烷氧基烷基或氨基烷基,烷酰基氨基烷基,胍基烷基,咪唑基烷基,吲哚基烷基,巯基烷基或烷硫基烷基,苯基烷基,羟基苯基烷基,苯氧基烷基或苯硫基烷基,或R2和R3与携带它们的C和N原子一起表示饱和 或不饱和的4至8元单环或8至10元双环的单环或杂环,任选被羟基,具有1至3个C原子的烷氧基或烷基单取代或二取代,R4表示氢,烷基,烯基,链烯基,炔基, 链烯基或烷撑基,环烷基,苯基,苄基,苯乙基或苯基丙基,它们各自可以任选被单取代或二取代; R5表示氢或烷基,羟基或烷氧基,R6表示氢,任选取代的烷基,环烷基,烯基,任选单取代或二取代的苯基或萘基,它们的盐,其制备方法及其作为药物的用途。
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