2- (2-pyridyl) -5-phenyl-6-aminopyrimidine, method and intermediate products for the production and use thereof for combating noxious fungi
    62.
    发明申请
    2- (2-pyridyl) -5-phenyl-6-aminopyrimidine, method and intermediate products for the production and use thereof for combating noxious fungi 失效
    2-(2-吡啶基)-5-苯基-6-氨基嘧啶,用于生产和用于对抗有害真菌的方法和中间产物

    公开(公告)号:US20050107401A1

    公开(公告)日:2005-05-19

    申请号:US10505146

    申请日:2003-02-06

    CPC分类号: C07D401/04

    摘要: The invention relates to 2-(2-pyridyl)-5-phenyl-6-amninopyrimidines of formula I, wherein the substitutes and the index have the following meaning: R1 represents halogen, hydroxy, hyano, hxo, nitro, amino, mercapto, alkyl, halogenalkyl, alkenyl, alkinyl, cycloalkyl, alkoxy, halogenalkoxy, carboxyl, alkoxycarbonyl, carbamoyl, alkylaminocarbonyl, dialkylamincarbonyl, morpholinocarbonyl, pyrrolidinocarbonyl, alkylcarbonylamino, alkylamino. dialkylamino, alkylthio, alkylsulfinyl, alkylsulfonyl, hydroxysulfonyl, aminosulfonyl, alkylaminosulfonyl, dialkylaminosulfonyl; m=0 or 1-4; R2 represents hydrogen, halogen, cyano, alkyl, halogenalkyl or alkoxy; R3, R4 represents hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl, R3 and R4 together with the nitrogen atom to which they are connected, form a five or six-membered ring which is interrupted by an atom from the group O, N or S and/or can be substituted according to the description; R5 represents halogen, alkyl or halogenalkyl; R6 represents hydrogen or one of the known groups in R5; R7, R8 represent hydrogen, halogen, alkyl or halogenalkyl; R9 represents hydrogen, halogen, hydroxy, cyano, alkyl, alkoxy, cycloalkoxy, halogenalkoxy, alkoxycarbonyl or alkylaminocarbonyl. The invention also relates to a method and intermediate product for the production of said compound in addition to the use thereof for combating undesirable plants.

    摘要翻译: 本发明涉及式I的2-(2-吡啶基)-5-苯基-6-脒嘧啶,其中取代基和指数具有以下含义:R 1表示卤素,羟基,杂环基, 烷氧基,烷氧基羰基,氨基甲酰基,烷基氨基羰基,二烷基氨基羰基,吗啉代羰基,吡咯烷基羰基,烷基羰基氨基,烷基氨基。 二烷基氨基,烷硫基,烷基亚磺酰基,烷基磺酰基,羟基磺酰基,氨基磺酰基,烷基氨基磺酰基,二烷基氨基磺酰基; m = 0或1-4; R 2表示氢,卤素,氰基,烷基,卤代烷基或烷氧基; R 3,R 4表示氢,烷基,卤代烷基,环烷基,卤代烷基,烯基,卤代烯基,环烯基,炔基,卤代炔基或环炔基,R 3 O 和R 4与它们连接的氮原子一起形成5或6元环,其被来自基团O,N或S的原子和/或可被取代 根据说明; R 5表示卤素,烷基或卤代烷基; R 6表示氢或R 5中的已知基团之一; R 7,R 8表示氢,卤素,烷基或卤代烷基; R 9表示氢,卤素,羟基,氰基,烷基,烷氧基,环烷氧基,卤代烷氧基,烷氧基羰基或烷基氨基羰基。 本发明还涉及用于生产所述化合物的方法和中间产物,除了其用于对抗不期望的植物之外。

    Benzyl amidoxime derivatives, intermediate products and method for their production and use as fungicides
    63.
    发明授权
    Benzyl amidoxime derivatives, intermediate products and method for their production and use as fungicides 失效
    苄基偕胺肟衍生物,中间产物及其生产和用作杀真菌剂的方法

    公开(公告)号:US06881742B1

    公开(公告)日:2005-04-19

    申请号:US10089148

    申请日:2000-10-05

    摘要: Novel benzamidoxime derivatives, processes and intermediates for their preparation and their use as fungicides are described.In the context of the present invention, benzamidoxime derivatives are compounds of the formula I where: A is an aryl or hetaryl radical; Y is a straight-chain or branched C1-C4-alkylene group, where one carbon can be replaced by oxygen, nitrogen or sulfur or by a cyclopropyl group; Rn1 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylthio, C1-C4-alkoxyalkoxy; R2 is unsubstituted or substituted phenyl-C1-C6-alkyl, thienyl-C1-C4-alkyl, or pyrazolyl-C1-C4-alkyl, Rp3 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylthio, C1-C4-alkoxyalkoxy, C1-C6-alkylcarbonyl; n is 0-5; p is, depending on the number of free valencies, 0-4.

    摘要翻译: 描述了新的苯甲酰胺肟衍生物,其制备方法和中间体及其作为杀真菌剂的用途。 在本发明的上下文中,苯甲酰胺肟衍生物是式I的化合物,其中:A是芳基或杂芳基; Y是直链或支链C 1 -C 4 - 亚烷基,其中一个碳可被氧,氮或硫取代或被环丙基取代; R 1是与以下组成的组中的一至五个相同或不同的基团:氢,卤素,C 1 -C 6 C 1 -C 6烷基,C 1 -C 6 - 烷氧基,C 1 -C 4 - 卤代烷基 ,C 1 -C 4 - 卤代烷氧基,C 1 -C 4 - 烷硫基,C 1 -C 4 - 烷氧基烷氧基; R 2是未取代或取代的苯基-C 1 -C 6 - 烷基,噻吩基-C 1 -C 或 - 吡唑基-C 1 -C 4 - C 1-4 - 烷基,R 3 - (CH 3)3 - / SUP>是与由以下组成的组中的一至五个相同或不同的基团:氢,卤素,C 1 -C 6 - 烷基,C 1 - C 1 -C 6 - 烷氧基,C 1 -C 4 - 卤代烷基,C 1 -C 3 > 4个 - 卤代烷氧基,C 1 -C 4 - 烷硫基,C 1 -C 4 - - 烷氧基烷氧基,C 1 -C 6 - 烷基羰基; n为0-5; p取决于自由价格的数量,0-4。

    Use of phenylacetamides as plant protectives having herbicidal and fungicidal effect
    64.
    发明授权
    Use of phenylacetamides as plant protectives having herbicidal and fungicidal effect 失效
    苯乙酰胺用作具有除草和杀真菌作用的植物保护剂

    公开(公告)号:US06613931B1

    公开(公告)日:2003-09-02

    申请号:US09913978

    申请日:2001-08-21

    IPC分类号: C07C25503

    CPC分类号: C07C255/41 A01N37/34

    摘要: The resent invention relates to the use of phenylacetamides as crop protection agents, to novel crop protection compositions comprising, as active compounds, phenylacetamides, and to novel phenylacetamides. The present invention provides the use of phenylacetamides of the formula I as crop protection agents having herbicidal and/or fungicidal action, where the radicals have the following meanings: A is an unsubstituted or substituted aryl radical; R1 is an unsubstituted or substituted aryl radical; R2, R3 are hydrogen, C1-C6-alkyl, C2-C6-alkenyl, C3-C7-cycloalkyl, C1-C6-alkylaryl, which may be unsubstituted or partially or fully halogenated or may carry one to three substituents selected from the group consisting of C1-C4-alkoxy, C1-C4-haloalkoxy, C1-C4-alkylthio, C3-C7-cycloalkyl, C5-C7-cycloalkenyl; R4 is hydrogen or C1-C6-alkyl; R5 is hydroxyl, C1-C4-alkoxy, aryl-C1-C4-alkoxy, aryloxy, and their agriculturally useful salts.

    摘要翻译: 本发明涉及苯基乙酰胺作为作物保护剂的用途,作为新的作物保护组合物,其包含作为活性化合物的苯乙酰胺和新的苯乙酰胺。本发明提供了下式的苯基乙酰胺的用途:具有除草和 /或杀真菌作用,其中基团具有以下含义:A是未取代或取代的芳基; R 1是未取代或取代的芳基; R 2,R 3是氢,C 1 -C 6 - 烷基,C 2 -C 6 - 烯基,C 3 C 1 -C 4 - 烷氧基,C 1 -C 4 - 烷氧基,C 1 -C 4 - 烷氧基,C 1 -C 4 - 烷氧基,C 1 -C 4 - 烷基芳基, C 3 -C 7 - 环烷基,C 5 -C 7 - 环烯基; R 4是氢或C 1 -C 6烷基; R 5是羟基,C 1 -C 4 - 烷氧基,芳基-C 1 -C 4 - 烷氧基,芳氧基和它们的农业上有用的盐。

    Fungicidal agents containing pyrrolidones as their active agents and use thereof for treating plants
    66.
    发明授权
    Fungicidal agents containing pyrrolidones as their active agents and use thereof for treating plants 失效
    含有吡咯烷酮作为其活性剂的杀真菌剂及其用于处理植物的用途

    公开(公告)号:US06586369B1

    公开(公告)日:2003-07-01

    申请号:US10204349

    申请日:2002-08-20

    IPC分类号: C07D20718

    摘要: Agrochemical compositions having fungicidal action and comprising as active compounds compounds of the formula I where R1 is hydrogen, C1-C6-alkyl, C1-C6-alkylcarbonyl, formyl or C1-C6-haloalkylcarbonyl; R2 is halogen, C1-C6-alkylthio, C1-C6-alkoxy, C3-C6-cycloalkyl-C1-C6-alkoxy, C1-C6-alkoxy-C1-C6-alkyl, halo-C1-C6-alkoxy, C1-C6-alkylsulfonyl, C1-C6-alkylsulfinyl, halo-C1-C6-alkylsulfonyl, cyano or a radical NR13R14; R3-R12 are hydrogen, halogen, C1-C8-cycloalkyl, C1-C6-alkyl, halo-C1-C6-alkyl, C1-C6-alkoxy, halo-C1-C6-alkoxy, C1-C6-alkylsulfonyl, halo-C1-C6-alkylsulfonyl, formyl, C1-C6-alkylcarbonyl, cyano, C1-C6-alkylthio or phenyl, which may be unsubstituted or substituted by halogen, C1-C6-alkyl or halo-C1-C6-alkyl, R13 is hydrogen, C1-C6-alkyl, R14 is C1-C6-alkyl, C1-C8-cycloalkyl or, together with R13 and the nitrogen atom to which they are attached, a saturated or unsaturated heterocyclic five- or six-membered ring which contains one or two heteroatoms selected from the group consisting of nitrogen and oxygen, and their agriculturally useful salts are described.

    摘要翻译: 具有杀真菌作用的农药组合物,包含作为活性化合物的式I化合物,其中R 1是氢,C 1 -C 6烷基,C 1 -C 6烷基羰基,甲酰基或C 1 -C 6卤代烷基羰基; R 2是卤素,C 1 -C 6烷硫基, C 1 -C 6烷氧基,C 1 -C 6烷氧基,C 1 -C 6烷氧基,C 1 -C 6 - 烷基亚磺酰基, C 1 -C 6 - 烷基磺酰基,氰基或NR 13 R 14基; R 3 -R 12是氢,卤素,C 1 -C 8 - 环烷基,C 1 -C 6烷基,卤代-C 1 -C 6 - 烷基,C 1 -C 6 - 烷氧基, C 1 -C 6 - 烷基磺酰基,卤代-C 1 -C 6 - 烷基磺酰基,甲酰基,C 1 -C 6 - 烷基羰基,氰基,C 1 -C 6 - 烷硫基或苯基,其可以是未取代的或被卤素取代, 或卤代-C 1 -C 6烷基,R 13是氢,C 1 -C 6烷基,R 14是C 1 -C 6 - 烷基,C 1 -C 8 - 环烷基,或者与R 13和它们所连接的氮原子一起是饱和或 不饱和杂环五元或六元环,其含有一个或两个选自组的杂原子 描述了氮和氧及其农业上有用的盐。