N-heteroaryl-N'-(pyrid-2-ylsulfonyl)ureas, processes for their
preparation, and their use as herbicides and plant growth regulators
    81.
    发明授权
    N-heteroaryl-N'-(pyrid-2-ylsulfonyl)ureas, processes for their preparation, and their use as herbicides and plant growth regulators 失效
    N-杂芳基-N' - (吡啶-2-基磺酰基)脲,其制备方法及其作为除草剂和植物生长调节剂的用途

    公开(公告)号:US5714436A

    公开(公告)日:1998-02-03

    申请号:US592393

    申请日:1996-03-22

    摘要: Compounds of the formula (I) or salts thereof ##STR1## in which R.sup.1 -R.sup.4, W, A, n and m are as defined in claim 1, for example R.sup.1 and R.sup.2 are H, (substituted) alkyl, (substituted) alkenyl or alkynyl, (substituted) cycloalkyl, (substituted) aryl or acyl and A is (substituted) pyrimidinyl or triazinyl are suitable as selective sulfonylurea herbicides and plant growth regulators. (I) is prepared analogously to known processes via intermediates, some of which are novel, for example via suitably substituted pyridylsulfonamides (II) and N-tert-butylsulfonamides (VIII) as claimed in claim 5.

    摘要翻译: PCT No.PCT / EP94 / 02628 Sec。 371日期:1996年3月22日 102(e)1996年3月22日PCT 1994年8月8日PCT公布。 第WO95 / 06049号公报 日期:1995年3月2日如权利要求1所定义的式(I)或其盐的化合物,例如R 1和R 2是H,(取代的)烷基,(取代的)烯基或炔基,(取代的)环烷基,(取代的) 或酰基,A是(取代的)嘧啶基或三嗪基作为选择性磺酰脲类除草剂和植物生长调节剂。 (I)类似于已知方法通过中间体制备,其中一些是新颖的,例如通过适当取代的如权利要求5所述的吡啶基磺酰胺(II)和N-叔丁基磺酰胺(VIII)。

    Plant protection agents based on pyrazolecarboxylic acid derivatives
    83.
    发明授权
    Plant protection agents based on pyrazolecarboxylic acid derivatives 失效
    基于吡唑羧酸衍生物的植物保护剂

    公开(公告)号:US5401700A

    公开(公告)日:1995-03-28

    申请号:US912659

    申请日:1992-07-13

    CPC分类号: A01N25/32 C07D231/14

    摘要: The present invention relates to agents for protecting crop plants from the phytotoxic side effects of herbicides, which agents contain a compound of the formula ##STR1## wherein Y denotes C--H or N,the symbols R.sub.1 independently of one another denote alkyl, halo-alkyl, alkoxy, haloalkoxy or halogen,R.sub.2 denotes alkyl or cycloalkyl,X denotes COOR.sub.3, CON(R.sub.4).sub.2, COSR.sub.3, CN or ##STR2## R.sub.3 denotes an alkali metal or alkaline earth metal, hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, or phenylalkyl, it being possible for phenyl to be substituted by halogen, or trisalkylsilylalkyl or alkoxyalkyl,the symbols R.sub.4 independently of one another denote H, alkyl or cycloalkyl, which can be substituted, or radicals R.sub.4 together with the N atom linking them form a 4- to 7-membered heterocyclic ring andn denotes 1 to 3,in combination with a herbicide.

    摘要翻译: 本发明涉及用于保护作物的植物免受除草剂的植物毒性副作用的药剂,该试剂含有式(I)的化合物,其中Y表示CH或N,符号R1彼此独立地表示烷基,卤代 - 烷基,卤代烷氧基或卤素,R 2表示烷基或环烷基,X表示COOR 3,CON(R 4)2,COSR 3,CN或R 3表示碱金属或碱土金属,氢,烷基,烯基,炔基, 环烷基或苯基烷基,苯基被卤素或三烷基甲硅烷基烷基或烷氧基烷基取代,符号R4彼此独立地表示可被取代的H,烷基或环烷基,或者与连接它们的N原子一起形成基团R4 形成4-至7-元杂环,n表示1至3,与除草剂组合。

    4,5,6,7-tetrahydro-3-aryl-indazoles and their use as herbicides
    85.
    发明授权
    4,5,6,7-tetrahydro-3-aryl-indazoles and their use as herbicides 失效
    4,5,6,7-四氢呋喃-3-磺酸钠及其作为除草剂的用途

    公开(公告)号:US5104442A

    公开(公告)日:1992-04-14

    申请号:US739687

    申请日:1991-08-02

    摘要: The invention relates to novel herbicidal compounds of the formula I or I' ##STR1## in which X is an oxygen or sulfur atom,R.sup.1 is H, C.sub.1 -C.sub.6 -alkyl, C.sub.2 -C.sub.6 -alkenyl, C.sub.2 -C.sub.6 -alkynyl, C.sub.1 -C.sub.6 -haloalkyl, (C.sub.1 -C.sub.4 -alkoxy-C.sub.1 -C.sub.4 -alkyl, (C.sub.1 -C.sub.6 -alkoxy)carbonyl, aryloxycarbonyl, (C.sub.1 -C.sub.6 -alkyl) aminocarbonyl, arylaminocarbonyl, phenyl, substituted phenyl or acyl,R.sup.2 is phenyl or substituted phenyl,R.sup.3 independently of other radicals R.sup.3 is H or C.sub.1 -C.sub.5 -alkyl andn is an integer from 0 to 6.The herbicides are suitable for selectively controlling harmful plants in cereal crops.

    摘要翻译: 本发明涉及式I或Ⅰ'其中X是氧或硫原子,R1是H,C1-C6-烷基,C2-C6的新颖除草化合物 - 烯基,C 2 -C 6 - 炔基,C 1 -C 6 - 卤代烷基,(C 1 -C 4 - 烷氧基-C 1 -C 4 - 烷基,(C 1 -C 6烷氧基)羰基,芳氧基羰基,(C 1 -C 6烷基)氨基羰基,芳基氨基羰基, 苯基,取代的苯基或酰基,R 2为苯基或取代的苯基,R 3独立地为其它基团,R 3为H或C 1 -C 5烷基,n为0至6的整数。除草剂适用于选择性地控制谷类作物中的有害植物 。

    Herbicidal imidazolinones
    86.
    发明授权
    Herbicidal imidazolinones 失效
    除草咪唑啉酮

    公开(公告)号:US4614535A

    公开(公告)日:1986-09-30

    申请号:US669620

    申请日:1984-11-08

    摘要: Imidazolinones of the formula ##STR1## in which A denotes N or C--R.sup.4 ; B denotes halogenoalkyl, alkoxymethyl, cyanomethyl or thiocyanatomethyl; X denotes alkyl; and Y denotes alkyl, cycloalkyl, alkenyl, phenyl or benzyl; or X and Y, together with C, denote a spiro-cycloalkyl group; Z denotes H, (substituted) alkyl, alkenyl, propargyl or an alkyl, carboxylic acid ester or sulfonic acid ester group; and R.sup.1 -R.sup.4 denote H, halogen, alkyl, alkoxy, alkoxycarbonyl, halogenoalkyl, NO.sub.2, CN, (substituted) phenoxy or (substituted) phenyl, or in each case two adjacent radicals together denote the radical --CH.dbd.CH--CH--CH--, are active herbicides and growth regulators.

    摘要翻译: 式(I)的咪唑啉酮,其中A表示N或C-R4; B表示卤代烷基,烷氧基甲基,氰基甲基或硫代氰基甲基; X表示烷基; Y表示烷基,环烷基,烯基,苯基或苄基; 或X和Y与C一起表示螺环烷基; Z表示H,(取代的)烷基,烯基,炔丙基或烷基,羧酸酯或磺酸酯基; 并且R 1 -R 4表示H,卤素,烷基,烷氧基,烷氧基羰基,卤代烷基,NO 2,CN,(取代的)苯氧基或(取代的)苯基,或者在每种情况下两个相邻的基团一起表示基团-CH = CH-CH-CH - 是活性除草剂和生长调节剂。

    Plant protection agents based on pyrazolecarboxylic acid derivatives
    88.
    发明授权
    Plant protection agents based on pyrazolecarboxylic acid derivatives 失效
    基于吡唑羧酸衍生物的植物保护剂

    公开(公告)号:US5945541A

    公开(公告)日:1999-08-31

    申请号:US356659

    申请日:1994-12-15

    CPC分类号: A01N25/32 C07D231/14

    摘要: The present invention relates to agents for protecting crop plants from the phytotoxic side effects of herbicides, which agents contain a compound of the formula I ##STR1## wherein Y denotes C--H or N,the symbols R.sub.1 independently of one another denote alkyl, halo-alkyl, alkoxy, haloalkoxy or halogen,R.sub.2 denotes alkyl or cycloalkyl,X denotes COOR.sub.3, CON(R.sub.4).sub.2, COSR.sub.3, CN or ##STR2## R.sub.3 denotes an alkali metal or alkaline earth metal, hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, or phenylalkyl, it being possible for phenyl to be substituted by halogen, or trialkylsilylalkyl or alkoxyalkyl,the symbols R.sub.4 independently of one another denote H, alkyl or cycloalkyl, which can be substituted, or 2 radicals R.sub.4 together with the N atom linking them form a 4- to 7-membered heterocyclic ring andn denotes 1 to 3, in combination with a herbicide.

    摘要翻译: 本发明涉及用于保护作物免受除草剂植物毒性副作用的试剂,该试剂含有式I化合物,其中Y表示CH或N,符号R 1彼此独立地表示烷基,卤代烷基,烷氧基, 卤代烷氧基或卤素,R2表示烷基或环烷基,X表示COOR3,CON(R4)2,COSR3,CN或R3表示碱金属或碱土金属,氢,烷基,烯基,炔基,环烷基或苯基烷基, 对于被卤素取代的苯基或三烷基甲硅烷基烷基或烷氧基烷基,符号R4彼此独立地表示可以被取代的H,烷基或环烷基,或2个基团R4与连接它们的N原子一起形成4-至7- 并且n表示1至3,与除草剂组合。

    Plant-protecting substituted isoxazolines, isoxazoles, isothiazolines
and isothiazoles, and also processes for their preparation and their use
    90.
    发明授权
    Plant-protecting substituted isoxazolines, isoxazoles, isothiazolines and isothiazoles, and also processes for their preparation and their use 失效
    植物保护取代的异恶唑啉,异恶唑,异噻唑啉和异噻唑,以及它们的制备和使用方法

    公开(公告)号:US5332715A

    公开(公告)日:1994-07-26

    申请号:US952895

    申请日:1992-11-18

    摘要: Plant-protecting substituted isoxazolines, isoxazoles, isothiazolines and isothiazoles, and also processes for their preparation and their useCompounds of the formula I(R.sup.1)(R.sup.2)(R.sup.3)Si--A--Het--B--CO--Z (I)whereHet is an isoxazole-, isoxazoline-, isothiazole- or isothiazoline-3,5-diyl radical,A and B are a bond or alkylene,R.sup.1, R.sup.2 and R.sup.3 are substituted or unsubstituted, saturated or unsaturated alkyl or, if desired, phenylalkyl or phenyl,Z is OH, OR where R is saturated or unsaturated, substituted or unsubstituted alkyl or substituted or unsubstituted phenyl or benzyl or trialkylsilylmethoxy, substituted or unsubstituted phenylamino or oxazolinyl or amino, mono- or dialkylamino or -hydrazino, cycloalkylamino, NH.sub.2 NH.sub.2, pyridino, morpholino, dimethylmorpholino, a radical --ON.dbd.CR.sup.4 R.sup.5 or O--CHR.sup.7 --CO--OR.sup.6 where R.sup.4, R.sup.5 =alkyl and/or R.sup.4 CR.sup.5 is cycloalkyl and R.sup.6, R.sup.7 are H or a saturated or unsaturated acyclic hydrocarbon radical,are suitable for protecting crop plants against phytotoxic side effects of herbicides.

    摘要翻译: 植物保护取代的异恶唑啉,异恶唑,异噻唑啉和异噻唑,以及其制备方法及用途式Ⅰ(R1)(R2)(R3)Si-A-Het-B-CO-Z(Ⅰ) Het是异恶唑,异恶唑啉,异噻唑或异噻唑啉-3,5-二基,A和B是键或亚烷基,R 1,R 2和R 3是取代或未取代的饱和或不饱和烷基,或者如果需要,苯基烷基 或苯基,Z是OH,OR,其中R是饱和或不饱和的,取代或未取代的烷基或取代或未取代的苯基或苄基或三烷基甲硅烷基甲氧基,取代或未取代的苯基氨基或恶唑啉基或氨基,单或二烷基氨基或肼基,环烷基氨基,NH 2 NH 2, 吡啶基,吗啉代,二甲基吗啉代,基团-ON = CR4R5或O-CHR7-CO-OR6,其中R4,R5 =烷基和/或R4CR5为环烷基,R6,R7为H或饱和或不饱和的无环烃基, 保护作物免受植物毒副作用 的除草剂。