摘要:
Novel benzoheterocyclic compounds of the formula: ##STR1## wherein R.sup.1 is H, halogen, OH, etc,; R.sup.2 is H, alkyl, halogen or alkoxy; R.sup.3 is phenyl-alkanoylamino, or ##STR2## R.sup.4 is H, --NR.sup.6 R.sup.7, alkenyloxy, HO-alkyl, --O--CO--A--NR.sup.8 R.sup.9, etc.; R.sup.5 is H, OH, etc., or a salt thereof, which have excellent vasopressin antagonistic activities and useful as vasodilator, hypotensive agent, water diuretics, platelet agglutination inhibitor, and a vasopressin antagonistic composition containing the compound as the active ingredient.
摘要:
Novel carbostyril derivatives of the formula: ##STR1## wherein R.sup.1 is H, NO.sub.2, alkoxy, alkoxycarbonyl, alkyl, halogen, optionally substituted amino, OH, CN, COOH, alkanoyloxy, hydrazinocarbonyl; q is 1 to 3, and R is a group of the formula ##STR2## [wherein R.sup.2 is H, alkoxycarbonyl, optionally substituted phenoxycarbonyl, phenylalkenyl-CO-, optionally substituted phenylalkanoyl, alkanoyl, alkenyl-CO-, optionally substituted phenyl--SO.sub.2 --, --CONR.sup.8 R.sup.9, optionally substituted heterocyclic group--CO--, naphthyl--CO--, thienylalkanoyl, tricyclo[3.3.1.1]alkanoyl, ##STR3## (R.sup.13 is OH, optionally substituted alkoxy, --NR.sup.32 R.sup.33, --O--A--(E).sub.l --NR.sup.4 R.sup.5, --(B).sub.l 'NR.sup.6 R.sup.7, etc.), n is 1 or 2, m is 0 or 1 to 3, R.sup.3 is alkyl, R.sup.10 is --(CO).sub.l --NR.sup.11 R.sup.12 ], and the bond between 3- and 4-position of carbostyril nucleus is single or double bond, which have excellent vasopressin antagonistic activities and are useful as vasodilator, hypotensive agent, water diuretics, platelet agglutination inhibitor, and a vasopressin antagonistic composition containing the compound as the active ingredient.
摘要翻译:其中R1是H,NO2,烷氧基,烷氧基羰基,烷基,卤素,任选取代的氨基,OH,CN,COOH,烷酰氧基,肼基羰基; q为1至3,并且R为下式的基团:其中R 2为H,烷氧基羰基,任选取代的苯氧基羰基,苯基烯基-CO-,任选取代的苯基烷酰基,烷酰基,烯基-CO-,任选取代的苯基-SO 2 - , - CONR 8 R 9,任选取代的杂环基-CO-,萘基-CO-,噻吩基烷酰基,三环[3.3.1.1]烷酰基,(R 13是OH,任选取代的烷氧基,-NR 32 R 33,-OA-(E) -NR 4 R 5, - (B)1 NR 6 R 7等),n为1或2,m为0或1〜3,R 3为烷基,R 10为 - (CO)1 -NR 11 R 12] 并且喹诺酮核的4-位是单或双键,其具有优异的加压素拮抗活性,并且可用作血管扩张剂,降血压剂,水利尿剂,血小板凝集抑制剂和含有该化合物作为活性成分的血管加压素拮抗剂组合物。
摘要:
Process for preparing NbN superconducting material, characterized in that a bulk Nb is placed in powder including at least one metal which can be nitriding-burned, and then the powder is heated to be nitriding-burned in pressurized N.sub.2 atmosphere so that the bulk Nb is nitrided by the nitriding-burning of the powder.
摘要:
A method of producing polymer particles having a particle size distribution of .+-.25% with respect to each average particle size in an amount of 95 wt. % or more, within the average particle sizes ranging from 1 .mu.m to 100 .mu.m, is disclosed, which comprises the steps of: (1) adding a polymer dispersion stabilizer in an amount of 0.1 to 10 wt. % to a hydrophilic organic liquid in which the polymer dispersion stabilizer is soluble; (2) adding thereto at least one vinyl monomer in an amount of not more than 50 times by weight the amount of the polymeric dispersion stabilizer, which monomer is soluble in the hydrophilic organic liquid, but a polymer synthesized from the monomer being swelled or substantially insoluble in the hydrophilic organic liquid; and (3) polymerizing the monomer under the condition that the amount of the vinyl monomer is 200 wt. % or less of the hydrophilic organic liquid.
摘要:
A position-detecting device comprising a scale, a first photo-interrupter, and a second photo-interrupter. The scale is attached to a movable member, and has a plurality of slits arranged at regular intervals. Each photo-interrupter includes a light source and a light detector, which are located at opposing sides of said scale, respectively. The first and second photo-interrupters are spaced apart such that when the scale moves, they generate, respectively, a first signal and a second signal which have a phase difference of .pi./2. These signals are processed, thereby to determine the position of the movable member with high accuracy.
摘要:
A surface treatment method for magnetic particles is disclosed, which comprises the steps of activating magnetic particles by application of heat thereto, treating the surface of the magnetic particles with a reactive silane coupling agent, bringing the treated magnetic particles into contact with at least one polymerizable vinyl-type monomer, polymerizing the monomer to form a polymer, and coating the surface of the magnetic particles with the polymer.
摘要:
Carbon material for de-sulfurization excellent in adsorptibility and mechanical strength can be produced from coal by controlling the physical properties of the raw material coal before its shaping to particular ranges, and subjecting the shaped coal to carbonization treatment.
摘要:
A recording and/or reproduction apparatus for an endless tape which includes a hollow fixed reel, the outer wall of which is wound with an endless tape which is conducted from the innermost portion and wound onto the outermost side a head mechanism for scanning the thus guided tape, a pinch roller and capstan which are driven with the tape held therebetween thereby causing the tape to be slackened downstream of the capstan, a swingable arm which releases the pinch roller from the capstan before its rotation is brought to an end, and a guide pin for releasing the tape from the head mechanism, capstan and pinch roller.
摘要:
A process for producing a developer for electrostatic latent images comprising adding a solution (A) of a high-molecular weight compound having electron-donating functional groups dissolved in an organic solvent (1) which is a good solvent for the high-molecular weight compound to an organic solvent (2) in which the high-molecular weight compound is substantially insoluble, thereby depositing the high-molecular weight compound in a finely divided particle form, wherein an organic resin which is soluble in both of organic solvent (1) and organic solvent (2) is dissolved in at least one of solution (A) and organic solvent (2).
摘要:
An image forming apparatus is provided that includes: first and second electrostatic latent image bearers; first and second electrostatic latent image forming devices; first and second developing devices configured to develop first and second electrostatic latent images with a colored toner and a special-color toner to form a colored toner image and a special-color toner image, respectively; a primary transfer device configured to transfer the colored toner image and the special-color toner image onto an intermediate image bearer in an overlapping manner to form a composite toner image; a secondary transfer device configured to transfer the composite toner image onto a recording medium; and a fixing device configured to fix the composite toner image thereon. The special-color toner comprises plate-like and/or film-like pigments. An absolute difference in volume resistivity between the special-color toner and the colored toner is 0.30 log Ω cm or less.