公开(公告)号：US4364958A

公开(公告)日：1982-12-21

申请号：US169439

申请日：1980-07-16

Applicant: Jeno Seres ,  Erika Varkonyi nee Schlavicsko ,  Sandor Virag ,  Gabor Kulcsar

Inventor： Jeno Seres ,  Erika Varkonyi nee Schlavicsko ,  Sandor Virag ,  Gabor Kulcsar

IPC: C07D207/40 ,  A61K31/40 ,  A61K31/4015 ,  A61P31/04 ,  A61P31/10 ,  C07D207/416 ,  C07D207/46 ,  A01N43/36

CPC classification number: C07D207/416 ,  C07D207/46

Abstract: A fungicidal compound of the formula: ##STR1## wherein A is C.sub.5-10 cycloalkyl, R is hydrogen, C.sub.1-6 alkyl, phenyl optionally substituted by one or more groups selected from C.sub.1-4 alkyl, nitro, hydroxy, carboxy, sulfo, sulfonylamino, halogen, C.sub.1-4 alkoxy, C.sub.1-4 acyloxy, C.sub.2-5 alkoxycarbonyl, C.sub.1-4 acyl, and N-(C.sub.2-5 alkoxycarbonyl)-sulfonylamino, or phenyl-(C.sub.1-4 alkyl) or a salt thereof.

Abstract translation: 一种下式的杀真菌化合物：其中A是C5-10环烷基，R是氢，C1-6烷基，任选被一个或多个选自C 1-4烷基，硝基，羟基，羧基的基团取代的苯基 ，磺基氨基，卤素，C 1-4烷氧基，C 1-4酰氧基，C 2-5烷氧基羰基，C 1-4酰基和N-（C 2-5烷氧基羰基） - 磺酰基氨基或苯基 - （C 1-4烷基）或 的盐。

公开(公告)号：US4065491A

公开(公告)日：1977-12-27

申请号：US758790

申请日：1977-01-12

Applicant: Todor Pfliegel ,  Jeno Seres ,  Antal Gajary ,  Klara Daroczy nee Csuka ,  Lajos T. Nagy

Inventor： Todor Pfliegel ,  Jeno Seres ,  Antal Gajary ,  Klara Daroczy nee Csuka ,  Lajos T. Nagy

IPC: C07F9/38

CPC classification number: C07F9/3813

Abstract: The invention relates to a new and improved method for the preparation of N-phosphonomethyl-glycine, a potent pre-emergence herbicide. According to the invention glycine, formaldehyde and a dialkyl phosphite are condensed in an aqueous alkaline medium to form a N-phosphonomethyl-glycine dialkyl ester, and the diester is hydrolyzed with a mineral acid.

Abstract translation: 本发明涉及一种新的和改进的N-膦酰基甲基 - 甘氨酸的制备方法，N-膦酰基甲基 - 甘氨酸是有效的出苗前除草剂。 根据本发明，甘氨酸，甲醛和亚磷酸二烷基酯在碱性水溶液中冷凝，形成N-膦酰基甲基 - 甘氨酸二烷基酯，二酯用无机酸水解。

公开(公告)号：US4353734A

公开(公告)日：1982-10-12

申请号：US927343

申请日：1978-07-24

Applicant: Jeno Seres ,  Istvanne Daroczi nee Csuka ,  Janosne Varkonyi nee Slovicsko ,  Gabor Horvath ,  Ildiko Szilagyi ,  Belane Radvanyi nee Hegedus

Inventor： Jeno Seres ,  Istvanne Daroczi nee Csuka ,  Janosne Varkonyi nee Slovicsko ,  Gabor Horvath ,  Ildiko Szilagyi ,  Belane Radvanyi nee Hegedus

IPC: A01N37/32 ,  A01N41/10 ,  A01N43/08 ,  A01N47/16 ,  C07D207/40 ,  C07D207/404 ,  C07D207/416 ,  C07D207/44 ,  C07D207/448 ,  C07D207/452 ,  C07D207/456 ,  A01N43/36

CPC classification number: C07D207/408 ,  A01N37/32 ,  A01N41/10 ,  A01N43/08 ,  A01N47/16 ,  C07D207/416 ,  C07D207/456

Abstract: Compounds of the formulae ##STR1## are disclosed wherein R is hydrogen, halogen, phenyl, phenyl-C.sub.1 to C.sub.4 alkylthio, C.sub.1 to C.sub.6 alkylthio, C.sub.5 to C.sub.7 cycloalkylthio, phenylthio or phenylsulfonyl;R.sub.1 is amino, C.sub.5 to C.sub.7 cycloalkylamino, C.sub.1 to C.sub.6 alkylamino, C.sub.1 to C.sub.4 -alkoxy-substituted-phenyl-(C.sub.1 to C.sub.4 -alkylamino), phenylamino, naphthylamino, furfurylamino, phenyl-(C.sub.1 to C.sub.4)-alkylamino, phenylamino-substituted by C.sub.1 to C.sub.4 alkoxy, halogen or C.sub.1 to C.sub.4 alkyl or phenylsulfonyl.R.sub.2 is hydrogen; andR.sub.3 is C.sub.1 to C.sub.6 alkyl, alkoxy or phenyl. The compounds have herbicidal properties.

Abstract translation: 公开了下式的化合物，其中R是氢，卤素，苯基，苯基-C 1至C 4烷硫基，C 1至C 6烷硫基，C 5至C 7环烷硫基，苯硫基或苯磺酰基; R1为氨基，C5至C7环烷基氨基，C1至C6烷基氨基，C1至C4烷氧基取代的苯基 - （C1至C4烷基氨基），苯基氨基，萘基氨基，糠基氨基，苯基 - （C1至C4） - 烷基氨基，苯基氨基 - 被C1至C4烷氧基，卤素或C1至C4烷基或苯基磺酰基取代。 R2是氢; 且R 3为C 1至C 6烷基，烷氧基或苯基。 该化合物具有除草性质。

公开(公告)号：US4051156A

公开(公告)日：1977-09-27

申请号：US376445

申请日：1973-07-05

Applicant: Lajos Guczoghy ,  Todor Pfliegel ,  Maria Puklics ,  Laszlo Institoris ,  Jeno Seres

Inventor： Lajos Guczoghy ,  Todor Pfliegel ,  Maria Puklics ,  Laszlo Institoris ,  Jeno Seres

IPC: A01N37/52 ,  A61K31/155 ,  C07C67/00 ,  C07C239/00 ,  C07C257/10 ,  C09B11/10

CPC classification number: A61K31/155

Abstract: A compound selected from the group which consists of the amidine of formula ##STR1## and the phytotoxically acceptable addition salts, hemihydrates and hydrates thereof,R.sup.1, r.sup.2 and R.sup.3 being phenyl or a phenyl group substituted with chlorine, bromine, iodine or fluorine, alkoxy having 1-4 carbon atoms or alkyl having 1 to 4 carbon atoms,R.sup.4 being methyl.

Abstract translation: 选自由式的脒组成的化合物及其植物学上可接受的加成盐，半水合物和水合物，R1，R2和R3是苯基或被氯，溴，碘或氟取代的苯基，烷氧基 具有1-4个碳原子或具有1至4个碳原子的烷基，R 4是甲基。