Piperazinylacylpiperidine derivatives, their preparation and therapeutic use thereof
    5.
    发明授权
    Piperazinylacylpiperidine derivatives, their preparation and therapeutic use thereof 有权
    哌嗪酰基哌啶衍生物,其制备和治疗用途

    公开(公告)号:US07294628B2

    公开(公告)日:2007-11-13

    申请号:US10516808

    申请日:2003-06-05

    CPC分类号: C07D417/14 C07D401/14

    摘要: The invention relates to substituted 1-piperazinylacylpiperidine derivatives of general formula (I) in which: n is 1 or 2; R1 represents a halogen atom; a trifluoromethyl radical; a (C1-C4) alkyl; a (C1-C4)alkoxy; a trifluoromethoxy radical; R2 represents a hydrogen atom or a halogen atom; R3 represents a hydrogen atom; a group —OR5; a group —CH2OR5; a group —NR6R7; a group —NR8COR9; a group —NR8CONR10R11; a group —CH2NR12R13; a group —CH2NR8CONR14R15; a (C1-C4)alkoxycarbonyl; a group —CONR16R17; or else R3 constitutes a double bond between the carbon atom to which it is attached and the adjacent carbon atom of the piperidine ring; R4 represents the aromatic group 1,3-thiazol-2-yl of formula: Preparation process and therapeutic application.

    摘要翻译: 本发明涉及通式(I)的取代的1-哌嗪基酰基哌啶衍生物,其中n为1或2; R 1表示卤素原子; 三氟甲基; (C 1 -C 4 -C 4)烷基; (C 1 -C 4 -C 4)烷氧基; 三氟甲氧基; R 2表示氢原子或卤素原子; R 3代表氢原子; 一个基团-OR 5; 基团-CH 2或OR 5; 基团-NR 6 R 7; 基团-NR 8 COR 9; 基团-NR 8 CONR 10 R 11; 基团-CH 2 NR 12 R 13; 基团-CH 2 NR 8 CONR 14 R 15 15; (C 1 -C 4 -C 4)烷氧基羰基; 基团-CONR 16 R 17 R 17; 或者R 3 3在其所连接的碳原子和哌啶环的相邻碳原子之间构成双键; R 4代表下式的芳族基团1,3-噻唑-2-基:制备方法和治疗应用。

    VEHICLE ALTERNATOR HAVING SYNCHRONOUS RECTIFICATION AND ELECTRONIC FAULT MANAGEMENT
    6.
    发明申请
    VEHICLE ALTERNATOR HAVING SYNCHRONOUS RECTIFICATION AND ELECTRONIC FAULT MANAGEMENT 有权
    具有同步修复和电子故障管理的车辆交换机

    公开(公告)号:US20120286744A1

    公开(公告)日:2012-11-15

    申请号:US13393586

    申请日:2010-07-22

    IPC分类号: H02P9/30 H02P9/02

    摘要: A synchronous rectification alternator for a motor vehicle is disclosed. The alternator includes a stator, a rotor, and a synchronous rectification system for rectifying into a DC voltage the alternating voltages supplied by the stator, and a voltage regulator for regulating the DC voltage. The alternator also includes fault detection for detecting faults in the synchronous rectification and supplying fault detection information to the voltage regulator. In one version, the fault information is supplied to the voltage regulator at fault inputs also receiving phase signals representing the alternating voltages supplied by the stator. At least one of the items of fault information is used to cause, in the voltage regulator, opening of an excitation circuit supplying current to an excitation coil of the rotor so as to produce, in the voltage regulator, a fault indication. The opening of the excitation circuit is preferably caused through a suitable command of a fast demagnetisation transistor included in the excitation circuit.

    摘要翻译: 公开了一种用于机动车辆的同步整流交流发电机。 交流发电机包括定子,转子和用于将由定子提供的交流电压整流为直流电压的同步整流系统和用于调节直流电压的电压调节器。 交流发电机还包括故障检测,用于检测同步整流中的故障,并向电压调节器提供故障检测信息。 在一个版本中,故障信息被提供给电压调节器,故障输入端还接收表示由定子提供的交流电压的相位信号。 使用故障信息中的至少一个,在电压调节器中,使得向转子的励磁线圈提供电流的励磁电路打开,以便在电压调节器中产生故障指示。 激励电路的打开优选地通过包括在激励电路中的快速去磁晶体管的合适命令来引起。

    Piperazinylacylpiperidine derivatives, their preparation and therapeutic use thereof
    8.
    发明申请
    Piperazinylacylpiperidine derivatives, their preparation and therapeutic use thereof 有权
    哌嗪酰基哌啶衍生物,其制备和治疗用途

    公开(公告)号:US20060167007A1

    公开(公告)日:2006-07-27

    申请号:US10516808

    申请日:2003-06-05

    CPC分类号: C07D417/14 C07D401/14

    摘要: The invention relates to substituted 1-piperazinylacylpiperidine derivatives of general formula (I) in which: n is 1 or 2; R1 represents a halogen atom; a trifluoromethyl radical; a (C1-C4) alkyl; a (C1-C4)alkoxy; a trifluoromethoxy radical; R2 represents a hydrogen atom or a halogen atom; R3 represents a hydrogen atom; a group —OR5; a group —CH2OR5; a group —NR6R7; a group —NR8COR9; a group —NR8CONR10R11; a group —CH2NR12R13; a group —CH2NR8CONR14R15; a (C1-C4)alkoxycarbonyl; a group —CONR16R17; or else R3 constitutes a double bond between the carbon atom to which it is attached and the adjacent carbon atom of the piperidine ring; R4 represents the aromatic group 1,3-thiazol-2-yl of formula: Preparation process and therapeutic application.

    摘要翻译: 本发明涉及通式(I)的取代的1-哌嗪基酰基哌啶衍生物,其中n为1或2; R 1表示卤素原子; 三氟甲基; (C 1 -C 4 -C 4)烷基; (C 1 -C 4 -C 4)烷氧基; 三氟甲氧基; R 2表示氢原子或卤素原子; R 3表示氢原子; 一个基团-OR 5; 基团-CH 2或OR 5; 基团-NR 6 R 7; 基团-NR 8 COR 9; 基团-NR 8 CONR 10 R 11; 基团-CH 2 NR 12 R 13; 基团-CH 2 NR 8 CONR 14 R 15 15; (C 1 -C 4 -C 4)烷氧基羰基; 基团-CONR 16 R 17 R 17; 或者R 3 3在其所连接的碳原子和哌啶环的相邻碳原子之间构成双键; R 4代表下式的芳族基团1,3-噻唑-2-基:制备方法和治疗应用。