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1.Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivates and intermediates therein 有权
标题翻译: 制备吡喃葡萄糖基取代的苄基苯衍生物及其中间体的方法公开(公告)号:US09127034B2
公开(公告)日:2015-09-08
申请号:US12789859
申请日:2010-05-28
申请人: Matthias Eckhardt , Frank Himmelsbach , Xiao-jun Wang , Wenjun Tang , Xiufeng Sun , Li Zhang , Dhileepkumar Krishnamurthy , Christopher Hugh Senanayake , Zhengxu Han
发明人: Matthias Eckhardt , Frank Himmelsbach , Xiao-jun Wang , Wenjun Tang , Xiufeng Sun , Li Zhang , Dhileepkumar Krishnamurthy , Christopher Hugh Senanayake , Zhengxu Han
IPC分类号: C07D307/32 , C07C49/786 , C07C41/05 , C07C43/184 , C07C43/205 , C07C25/06 , C07H15/203
CPC分类号: C07D407/12 , C07D309/10 , C07F1/02 , C07F3/02 , C07H15/04 , C07H15/203 , C07H19/01
摘要: The present invention relates to processes for preparing the compounds of general formula I, wherein the groups R1 and R3 are defined according to claim 1. Furthermore this inventions relates to intermediates obtained in these processes.
摘要翻译: 本发明涉及制备通式I化合物的方法,其中基团R1和R3根据权利要求1定义。此外,本发明涉及在这些方法中获得的中间体。
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2.Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives and intermediates therein 有权
标题翻译: 制备吡喃葡萄糖基取代的苄基苯衍生物及其中间体的方法公开(公告)号:US20060258749A1
公开(公告)日:2006-11-16
申请号:US11416683
申请日:2006-05-03
申请人: Matthias Eckhardt , Frank Himmelsbach , Xiao-jun Wang , Wenjun Tang , Xiufeng Sun , Li Zhang , Dhileepkumar Krishnamurthy , Christopher Senanayake , Zhengxu Han
发明人: Matthias Eckhardt , Frank Himmelsbach , Xiao-jun Wang , Wenjun Tang , Xiufeng Sun , Li Zhang , Dhileepkumar Krishnamurthy , Christopher Senanayake , Zhengxu Han
IPC分类号: A61K31/135
CPC分类号: C07D407/12 , C07D309/10 , C07F1/02 , C07F3/02 , C07H15/04 , C07H15/203 , C07H19/01
摘要: The present invention relates to processes for preparing the compounds of general formula I, wherein the groups R1 and R3 are defined according to claim 1. Furthermore this inventions relates to intermediates obtained in these processes.
摘要翻译: 本发明涉及制备通式I化合物的方法,其中R 1和R 3基团根据权利要求1定义。此外,本发明涉及中间体 在这些过程中获得。
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3.PROCESSES FOR PREPARING OF GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZENE DERIVATES AND INTERMEDIATES THEREIN 有权
标题翻译: 制备葡萄糖苷取代的苄基苯甲酸衍生物及其中间体的方法公开(公告)号:US20100240879A1
公开(公告)日:2010-09-23
申请号:US12789859
申请日:2010-05-28
申请人: Matthias ECKHARDT , Frank HIMMELSBACH , Xiao-jun WANG , Wenjun TANG , Xiufeng SUN , Li ZHANG , Dhileepkumar KRISHNAMURTHY , Chris Hugh SENANAYAKE , Zhengxu HAN
发明人: Matthias ECKHARDT , Frank HIMMELSBACH , Xiao-jun WANG , Wenjun TANG , Xiufeng SUN , Li ZHANG , Dhileepkumar KRISHNAMURTHY , Chris Hugh SENANAYAKE , Zhengxu HAN
IPC分类号: C07G3/00 , C07H1/00 , C07D307/04
CPC分类号: C07D407/12 , C07D309/10 , C07F1/02 , C07F3/02 , C07H15/04 , C07H15/203 , C07H19/01
摘要: The present invention relates to processes for preparing the compounds of general formula I, wherein the groups R1 and R3 are defined according to claim 1. Furthermore this inventions relates to intermediates obtained in these processes.
摘要翻译: 本发明涉及制备通式I化合物的方法,其中基团R1和R3根据权利要求1定义。此外,本发明涉及在这些方法中获得的中间体。
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4.Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives and intermediates therein 有权
标题翻译: 制备吡喃葡萄糖基取代的苄基苯衍生物及其中间体的方法公开(公告)号:US07772191B2
公开(公告)日:2010-08-10
申请号:US11416683
申请日:2006-05-03
申请人: Matthias Eckhardt , Frank Himmelsbach , Xiao-jun Wang , Wenjun Tang , Xiufeng Sun , Li Zhang , Dhileepkumar Krishnamurthy , Chris Hugh Senanayake , Zhengxu Han
发明人: Matthias Eckhardt , Frank Himmelsbach , Xiao-jun Wang , Wenjun Tang , Xiufeng Sun , Li Zhang , Dhileepkumar Krishnamurthy , Chris Hugh Senanayake , Zhengxu Han
IPC分类号: A61K31/341 , A61K31/351 , A61K31/7034 , A61K31/7048 , C07H7/04 , C07D309/12 , C07D307/20
CPC分类号: C07D407/12 , C07D309/10 , C07F1/02 , C07F3/02 , C07H15/04 , C07H15/203 , C07H19/01
摘要: The present invention relates to processes for preparing the compounds of general formula I, wherein the groups R1 and R3 are defined according to claim 1. Furthermore this inventions relates to intermediates obtained in these processes.
摘要翻译: 本发明涉及制备通式I化合物的方法,其中基团R1和R3根据权利要求1定义。此外,本发明涉及在这些方法中获得的中间体。
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公开(公告)号:US20060258888A1
公开(公告)日:2006-11-16
申请号:US11380956
申请日:2006-05-01
IPC分类号: C07C209/10
CPC分类号: C07C209/10 , C07C213/02 , C07C2601/02 , C07C211/51 , C07C211/52 , C07C211/58 , C07C217/84 , C07C211/56
摘要: Disclosed are methods for making 1,3- and 1,4-diamino-phenyl intermediates by utilizing bis-amination of ortho-substituted aryl halides.
摘要翻译: 公开了通过利用邻位取代的芳基卤化物的双 - 胺化制备1,3-和1,4-二氨基 - 苯基中间体的方法。
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