公开(公告)号：US20050101783A1

公开(公告)日：2005-05-12

申请号：US10477338

申请日：2001-05-09

申请人： Atsushi Ito ,  Keiichi Sudo ,  Tsumoru Watanabe ,  Nobuyuki Kusano ,  Nobuyuki Araki ,  Takayoshi Eizuka ,  Yoshitaka Niizeki

发明人： Atsushi Ito ,  Keiichi Sudo ,  Tsumoru Watanabe ,  Nobuyuki Kusano ,  Nobuyuki Araki ,  Takayoshi Eizuka ,  Yoshitaka Niizeki

IPC分类号： C07D249/08 ,  A01N43/36 ,  A01N43/40 ,  A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/60 ,  A01N43/653 ,  A01N43/78 ,  A61K31/40 ,  A61K31/415 ,  A61K31/417 ,  A61K31/4196 ,  A61K31/425 ,  A61K31/426 ,  A61K31/44 ,  A61K31/4965 ,  A61K31/505 ,  A61P31/10 ,  C07D207/323 ,  C07D213/38 ,  C07D213/61 ,  C07D231/12 ,  C07D233/64 ,  C07D239/26 ,  C07D241/16 ,  C07D277/20 ,  C07D277/32 ,  C07D213/26

CPC分类号： A01N43/60 ,  A01N43/36 ,  A01N43/40 ,  A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/653 ,  A01N43/78

摘要： A N-heterocyclicmethyl-alkylamine derivative according to the present invention is a N-heterocyclicmethyl-alkylamine derivative represented by the following general formula (I): or an acid addition salt thereof. [in the formula, R1 represents a heterocycle which has at least one nitrogen atom as a hetero atom and may have a substituent on a ring; R2 represents a hydrogen or the like; R3 represents an alkyl group having a carbon number of 1 to 5 or the like; R4 represents an alkyl group having a carbon number of 1 to 5 or the like; when R4 is an alkyl group having a carbon number of 1 to 5 or a halogenated alkyl group having a carbon number of 1 to 5, carbon atoms in R3 and R4 may be bonded to form a ring structure; m represents an integer of 1 to 3; R5 represents a cycloalkyl group or the like described by the following formula (III): (in the formula, Y and Z each represents a hydrogen atom or the like, the letter p represents an integer of 2 to 5, and the groups described by CYZ may be each the same or different), when m is 1 and R4 is a hydrogen atom, R5 is a cycloalkyl group described by the foregoing formula (III).]

摘要翻译： 根据本发明的N-杂环甲基 - 烷基胺衍生物是由以下通式（I）表示的N-杂环甲基 - 烷基胺衍生物或其酸加成盐。 [式中，R 1表示具有至少一个氮原子作为杂原子并且可以在环上具有取代基的杂环; R 2表示氢等; R 3表示碳数为1〜5的烷基等; R 4表示碳数为1〜5的烷基等; 当R 4是碳数为1至5的烷基或碳数为1至5的卤代烷基时，R 3和R 3中的碳原子 可以键合4个以​​形成环结构; m表示1〜3的整数， R 5表示下述式（III）所示的环烷基等：（式中，Y和Z各自表示氢原子等，字母p表示2以上的整数） 至5，并且由CYZ描述的基团可各自相同或不同），当m为1且R 4为氢原子时，R 5为环烷基 由上述式（III）表示。]

公开(公告)号：US06271385B1

公开(公告)日：2001-08-07

申请号：US09508347

申请日：2000-03-10

申请人： Atsushi Ito ,  Satoru Kumazawa ,  Keiichi Sudo ,  Tsumoru Watanabe ,  Takayoshi Eizuka ,  Yoshitaka Niizeki

发明人： Atsushi Ito ,  Satoru Kumazawa ,  Keiichi Sudo ,  Tsumoru Watanabe ,  Takayoshi Eizuka ,  Yoshitaka Niizeki

IPC分类号： A01N5718

CPC分类号： A01N43/78 ,  A01N43/36 ,  A01N43/40 ,  A01N43/54 ,  A01N43/56 ,  A01N43/80

摘要： N-heterocyclicmethylpropylamine derivatives of formula (I): and acid addition salts thereof; wherein R1 represents hydrogen, halogen, alkyl, alkenyl, halogenated alkyl, alkoxy, halogenated alkoxy, hydroxyl, cyano, nitro, phenyl optionally having a substituent on a ring thereof or phenoxy; n represents an integer of 0-5; R2 represents a heterocycle containing at least one nitrogen atom as the hetero atom and optionally having a substituent on a ring thereof; and R3 represents hydrogen or C1-C5 alkyl.

摘要翻译： 式（I）的N-杂环甲基丙胺衍生物及其酸加成盐;其中R1表示氢，卤素，烷基，烯基，卤代烷基，烷氧基，卤代烷氧基，羟基，氰基，硝基，任选在其环上具有取代基的苯基 或苯氧基; n表示0〜5的整数。 R2表示含有至少一个氮原子作为杂原子并且在其环上任选具有取代基的杂环; 并且R 3表示氢或C 1 -C 5烷基。

公开(公告)号：US20120277440A1

公开(公告)日：2012-11-01

申请号：US13520668

申请日：2011-01-06

申请人： Shinzo Kagabu ,  Satoru Kumazawa ,  Tsumoru Watanabe ,  Taiji Miyake ,  Masahiro Nomura ,  Satoshi Nakamura ,  Masaaki Mitomi

发明人： Shinzo Kagabu ,  Satoru Kumazawa ,  Tsumoru Watanabe ,  Taiji Miyake ,  Masahiro Nomura ,  Satoshi Nakamura ,  Masaaki Mitomi

IPC分类号： C07D417/06

CPC分类号： C07D417/06 ,  A01N43/78 ,  C07D417/14

摘要： To provide a novel imino derivative capable of being an insecticide compound which is excellent in characteristics such as sustained effects and a broad spectrum.An imino derivative represented by Formula (A) shown below: wherein “Ar” represents a heterocyclic group which may have a substituent on the ring, “X” represents a sulfur atom or CH2, NR; “R” represents a hydrogen atom or an alkyl group; “Ya” is selected from “C(═S)NR1R2”, “C(═S)SR3”, “C(═O)SR4”, “C(═S)OR4”, “SO2Zα”, and “OZβ”; and, each of “R1” to “R4”, “Zα”, and “Zβ” represents a hydrogen atom or a certain substituent; is provided.

摘要翻译： 提供能够成为持续效果和广谱特性优异的杀虫剂化合物的新型亚氨基衍生物。 由下式（A）表示的亚氨基衍生物：其中Ar表示可在环上具有取代基的杂环基，X表示硫原子或CH2，NR; R表示氢原子或烷基; Ya选自C（= S）NR1R2，C（= S）SR3，C（= O）SR4，C（= ORS）OR4，SO2Zα和OZ。 并且R 1至R 4，Z a和Z bb中的每一个; 表示氢原子或某一取代基; 被提供。

公开(公告)号：US5279719A

公开(公告)日：1994-01-18

申请号：US970305

申请日：1992-11-02

申请人： Kazuhiko Sunagawa ,  Hajime Hoshi ,  Tsumoru Watanabe

发明人： Kazuhiko Sunagawa ,  Hajime Hoshi ,  Tsumoru Watanabe

IPC分类号： C07C17/12 ,  C07C17/14 ,  C07C25/02 ,  C07C25/125 ,  C07C25/22 ,  C07C17/00

CPC分类号： C07C17/12 ,  C07C17/14 ,  C07C25/125

摘要： A process for chlorination of methylated aromatic compounds in a titanium tetrachloride is disclosed. The ring chlorination is first carried out by reacting said methylated aromatic compounds with chlorine gas under reduced light conditions, and then the side chain chlorination is carried out by reacting the resulting mixture with chlorine gas under light irradiation conditions. The process ensures continuous chlorination of aromatic rings and side chains of methylated aromatic compounds at a high yield without using any catalysts or perilous solvents such as carbon tetrachloride.

摘要翻译： 公开了一种在四氯化钛中氯化甲基化芳族化合物的方法。 环氯化首先通过使所述甲基化芳香族化合物与降低光照条件下的氯气反应进行，然后通过在光照射条件下使所得混合物与氯气反应来进行侧链氯化。 该方法确保甲基化芳族化合物的芳香环和侧链在不使用任何催化剂或危险溶剂如四氯化碳的情况下以高产率连续氯化。