公开(公告)号：US20050101783A1

公开(公告)日：2005-05-12

申请号：US10477338

申请日：2001-05-09

申请人： Atsushi Ito ,  Keiichi Sudo ,  Tsumoru Watanabe ,  Nobuyuki Kusano ,  Nobuyuki Araki ,  Takayoshi Eizuka ,  Yoshitaka Niizeki

发明人： Atsushi Ito ,  Keiichi Sudo ,  Tsumoru Watanabe ,  Nobuyuki Kusano ,  Nobuyuki Araki ,  Takayoshi Eizuka ,  Yoshitaka Niizeki

IPC分类号： C07D249/08 ,  A01N43/36 ,  A01N43/40 ,  A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/60 ,  A01N43/653 ,  A01N43/78 ,  A61K31/40 ,  A61K31/415 ,  A61K31/417 ,  A61K31/4196 ,  A61K31/425 ,  A61K31/426 ,  A61K31/44 ,  A61K31/4965 ,  A61K31/505 ,  A61P31/10 ,  C07D207/323 ,  C07D213/38 ,  C07D213/61 ,  C07D231/12 ,  C07D233/64 ,  C07D239/26 ,  C07D241/16 ,  C07D277/20 ,  C07D277/32 ,  C07D213/26

CPC分类号： A01N43/60 ,  A01N43/36 ,  A01N43/40 ,  A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/653 ,  A01N43/78

摘要： A N-heterocyclicmethyl-alkylamine derivative according to the present invention is a N-heterocyclicmethyl-alkylamine derivative represented by the following general formula (I): or an acid addition salt thereof. [in the formula, R1 represents a heterocycle which has at least one nitrogen atom as a hetero atom and may have a substituent on a ring; R2 represents a hydrogen or the like; R3 represents an alkyl group having a carbon number of 1 to 5 or the like; R4 represents an alkyl group having a carbon number of 1 to 5 or the like; when R4 is an alkyl group having a carbon number of 1 to 5 or a halogenated alkyl group having a carbon number of 1 to 5, carbon atoms in R3 and R4 may be bonded to form a ring structure; m represents an integer of 1 to 3; R5 represents a cycloalkyl group or the like described by the following formula (III): (in the formula, Y and Z each represents a hydrogen atom or the like, the letter p represents an integer of 2 to 5, and the groups described by CYZ may be each the same or different), when m is 1 and R4 is a hydrogen atom, R5 is a cycloalkyl group described by the foregoing formula (III).]

摘要翻译： 根据本发明的N-杂环甲基 - 烷基胺衍生物是由以下通式（I）表示的N-杂环甲基 - 烷基胺衍生物或其酸加成盐。 [式中，R 1表示具有至少一个氮原子作为杂原子并且可以在环上具有取代基的杂环; R 2表示氢等; R 3表示碳数为1〜5的烷基等; R 4表示碳数为1〜5的烷基等; 当R 4是碳数为1至5的烷基或碳数为1至5的卤代烷基时，R 3和R 3中的碳原子 可以键合4个以​​形成环结构; m表示1〜3的整数， R 5表示下述式（III）所示的环烷基等：（式中，Y和Z各自表示氢原子等，字母p表示2以上的整数） 至5，并且由CYZ描述的基团可各自相同或不同），当m为1且R 4为氢原子时，R 5为环烷基 由上述式（III）表示。]

公开(公告)号：US08710090B2

公开(公告)日：2014-04-29

申请号：US13508269

申请日：2010-12-07

申请人： Nobuyuki Araki ,  Toru Yamazaki ,  Nobuyuki Kusano ,  Eiyu Imai ,  Hisashi Kanno ,  Masaru Mori ,  Taiji Miyake

发明人： Nobuyuki Araki ,  Toru Yamazaki ,  Nobuyuki Kusano ,  Eiyu Imai ,  Hisashi Kanno ,  Masaru Mori ,  Taiji Miyake

IPC分类号： A01N43/50 ,  A61K31/4164 ,  C07D233/60 ,  C07D249/08

CPC分类号： C07C67/31 ,  A01N37/10 ,  A01N43/50 ,  A01N43/653 ,  C07C201/12 ,  C07C2601/08 ,  C07D405/06

摘要： An azole derivative according to the invention is represented by Formula (I), wherein each of Ra and Rb denotes a hydrogen atom, or a C1-C6 alkyl group, a C2-C6 alkenyl group or a C2-C6 alkynyl group; Ra and Rb may be substituted with Xa or Xb which is a halogen atom; each of na and nb denotes 0 or the number of Xa- or Xb-substituted hydrogen atoms among the hydrogen atoms in Ra or Rb; each Y denotes a halogen atom, a C1-C4 alkyl group, a C1-C4 haloalkyl group, a C1-C4 alkoxy group, a C1-C4 haloalkoxy group, a phenyl group, a cyano group or a nitro group; m denotes 0 to 5; and A denotes a nitrogen atom or a methyne group. As a result, an azole derivative contained as an active ingredient in an agro-horticultural agent having an excellent controlling effect on diseases can be provided.

摘要翻译： 根据本发明的唑衍​​生物由式（I）表示，其中R a和R b各自表示氢原子或C 1 -C 6烷基，C 2 -C 6烯基或C 2 -C 6炔基; Ra和Rb可以被Xa或Xb取代，Xb或Xb是卤素原子; na和nb中的每一个表示0或Ra或Rb中的氢原子中的X a或X b取代的氢原子的数目; 每个Y表示卤素原子，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，苯基，氰基或硝基; m表示0〜5; A表示氮原子或甲炔基。 结果，可以提供在对疾病具有优异控制作用的农业园艺剂中作为活性成分含有的唑衍生物。

公开(公告)号：US20120232286A1

公开(公告)日：2012-09-13

申请号：US13508269

申请日：2010-12-07

申请人： Nobuyuki Araki ,  Toru Yamazaki ,  Nobuyuki Kusano ,  Eiyu Imai ,  Hisashi Kanno ,  Masaru Mori ,  Taiji Miyake

发明人： Nobuyuki Araki ,  Toru Yamazaki ,  Nobuyuki Kusano ,  Eiyu Imai ,  Hisashi Kanno ,  Masaru Mori ,  Taiji Miyake

IPC分类号： C07D249/08 ,  C07D233/64 ,  C07C69/757

CPC分类号： C07C67/31 ,  A01N37/10 ,  A01N43/50 ,  A01N43/653 ,  C07C201/12 ,  C07C2601/08 ,  C07D405/06

摘要： An azole derivative according to the invention is represented by Formula (I), wherein each of Ra and Rb denotes a hydrogen atom, or a C1-C6 alkyl group, a C2-C6 alkenyl group or a C2-C6 alkynyl group; Ra and Rb may be substituted with Xa or Xb which is a halogen atom; each of na and nb denotes 0 or the number of Xa- or Xb-substituted hydrogen atoms among the hydrogen atoms in Ra or Rb; each Y denotes a halogen atom, a C1-C4 alkyl group, a C1-C4 haloalkyl group, a C1-C4 alkoxy group, a C1-C4 haloalkoxy group, a phenyl group, a cyano group or a nitro group; m denotes 0 to 5; and A denotes a nitrogen atom or a methyne group. As a result, an azole derivative contained as an active ingredient in an agro-horticultural agent having an excellent controlling effect on diseases can be provided.

摘要翻译： 根据本发明的唑衍​​生物由式（I）表示，其中R a和R b各自表示氢原子或C 1 -C 6烷基，C 2 -C 6烯基或C 2 -C 6炔基; Ra和Rb可以被Xa或Xb取代，Xb或Xb是卤素原子; na和nb中的每一个表示0或Ra或Rb中的氢原子中的X a或X b取代的氢原子的数目; 每个Y表示卤素原子，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，苯基，氰基或硝基; m表示0〜5; A表示氮原子或甲炔基。 结果，可以提供在对疾病具有优异控制作用的农业园艺剂中作为活性成分含有的唑衍生物。

公开(公告)号：US20140113899A1

公开(公告)日：2014-04-24

申请号：US14124168

申请日：2012-06-06

申请人： Hideaki Tateishi ,  Nobuyuki Araki ,  Toru Yamazaki ,  Taiji Miyake ,  Keiichi Sudo ,  Hisashi Kanno

发明人： Hideaki Tateishi ,  Nobuyuki Araki ,  Toru Yamazaki ,  Taiji Miyake ,  Keiichi Sudo ,  Hisashi Kanno

IPC分类号： A01N43/653 ,  A01N43/40 ,  A01N37/22 ,  A01N37/34 ,  A01N43/84 ,  A01N47/34 ,  A01N47/38 ,  A01N43/56 ,  A01N43/54

CPC分类号： A01N43/653 ,  A01N37/22 ,  A01N37/34 ,  A01N43/40 ,  A01N43/54 ,  A01N43/56 ,  A01N43/84 ,  A01N47/34 ,  A01N47/38 ,  A01N45/02 ,  A01N2300/00

摘要： An agro-horticultural agent of the present invention is intended to provide an agro-horticultural agent capable of providing, with a smaller spray amount, the same effect as compared to a conventional agro-horticultural agent. The agro-horticultural agent of the present invention includes a plurality of active ingredients and one of the plurality of active ingredients is an azole derivative represented by the following general formula (I); where: Ra and Rb each represent a predetermined hydrocarbon group and at least one of Ra and Rb has a chlorine atom or a bromine atom substituted for a hydrogen atom; Y represents a chlorine atom or a fluorine atom; and m represents 0 or 1.

摘要翻译： 本发明的农业园艺剂旨在提供能够以较小喷雾量提供与常规农业园艺剂相比相同效果的农业园艺剂。 本发明的农业园艺剂包括多种活性成分，多种活性成分之一是由以下通式（I）表示的唑衍生物。 其中：Ra和Rb各自表示预定的烃基，Ra和Rb中的至少一个具有取代氢原子的氯原子或溴原子; Y表示氯原子或氟原子; m表示0或1。

公开(公告)号：US20140094362A1

公开(公告)日：2014-04-03

申请号：US14122944

申请日：2012-05-30

申请人： Taiji Miyake ,  Nobuyuki Araki ,  Toru Yamazaki

发明人： Taiji Miyake ,  Nobuyuki Araki ,  Toru Yamazaki

IPC分类号： A01N43/653

CPC分类号： A01N43/653 ,  C07B57/00 ,  C07D249/08 ,  A01N25/00

摘要： In order to provide a compound that shows a strong effect on controlling a plant disease, a triazole compound of the present invention (i) is a compound in which —OH group, —R2 group, and CH2—Ar group are bonded in cis configuration with a cyclopentane, (ii) is (−)-enantiomer or (+) enantiomer, and (iii) is represented by Formula (I): (wherein R1 represents an alkyl group; R2 represents a haloalkyl group; and Ar represents a substituted/unsubstituted aromatic hydrocarbon group or a substituted/unsubstituted aromatic heterocyclic group.

摘要翻译： 为了提供对控制植物病害具有强效果的化合物，本发明的三唑化合物（i）是其中-OH基，-R2基和CH2-Ar基以顺式结构键合的化合物 （ii）为（ - ） - 对映体或（+）对映异构体，（iii）由式（I）表示：（其中R 1表示烷基; R 2表示卤代烷基; Ar表示取代基 /未取代的芳香族烃基或取代/未取代的芳香族杂环基。

公开(公告)号：US4381178A

公开(公告)日：1983-04-26

申请号：US171045

申请日：1980-07-22

申请人： Shozo Nakayama ,  Kimio Kato ,  Nobuyuki Araki ,  Kenji Takenaka

发明人： Shozo Nakayama ,  Kimio Kato ,  Nobuyuki Araki ,  Kenji Takenaka

IPC分类号： F04B27/08 ,  F04B25/04 ,  F04B27/12 ,  F04B1/16 ,  F04B1/18

CPC分类号： F04B27/12

摘要： A swash-plate type compressor wherein a plurality of pistons fitted into a plurality of cylinder bores having their center on a circle are reciprocated by a swash-plate secured to a rotary shaft at a tilt angle. A swash-plate chamber rotatably accommodating the swash-plate concurrently functions as a passage for the refrigerant gas sucked, and an annular refrigerant gas passage, whose external diameter is larger than that of a circumcircle of the aforementioned cylinder bores and whose inner side is open to the swash-plate chamber, is formed on the external side of the swash-plate chamber. This annular passage for the refrigerant gas sucked functions as a by-pass therefor, diminishes the flow resistance of the refrigerant gas, and facilitates the cooling of the pistons with a result of reducing the operation noise produced from the engaging portion of the pistons and the swash-plate.

摘要翻译： 旋转斜盘式压缩机，其中装配在其圆周中心的多个气缸孔中的多个活塞通过以倾斜角固定到旋转轴的斜盘往复运动。 可旋转地容纳旋转斜盘的旋转斜盘室同时用作吸入的制冷剂气体的通道，并且其外径大于上述气缸孔的外接圆的内周侧敞开的环状制冷剂气体通道 到斜盘室，形成在旋转斜盘室的外侧。 用于被吸入的制冷剂气体的该环形通道用作旁路，从而减小制冷剂气体的流动阻力，并且有助于活塞的冷却，从而减少由活塞的接合部分产生的操作噪声和 斜盘

公开(公告)号：US4101250A

公开(公告)日：1978-07-18

申请号：US755480

申请日：1976-12-29

申请人： Shozo Nakayama ,  Masayuki Kurahashi ,  Nobuyuki Araki

发明人： Shozo Nakayama ,  Masayuki Kurahashi ,  Nobuyuki Araki

IPC分类号： F04B27/10 ,  F04B27/12 ,  F04B1/12 ,  F04B27/08

CPC分类号： F04B27/12 ,  F04B27/1045

摘要： A swash plate type compressor adapted for use in an automotive cooling system is disclosed. A cylinder block, which forms a principal part of the compressor and is axially divided into two portions, has at least four bores arranged at equal distances along the circumference thereof. A clamping bolt for uniting all principal members of the compressor extends through a hole provided through a narrow interzone lying between each two adjacent bores. The through hole has a diameter considerably greater than that of the clamping bolt. The space between the inner surface of the hole and the outer surface of the bolt serves as a passage through which a low pressure refrigerant gas flows, and this helps simplification in construction and improvement in capacity of the swash plate type compressor.

摘要翻译： 公开了一种适用于汽车冷却系统的旋转斜盘式压缩机。 形成压缩机的主要部分并被轴向分成两部分的气缸体具有至少四个沿其圆周等距离布置的孔。 用于将压缩机的所有主要构件联合的夹紧螺栓延伸通过位于每两个相邻孔之间的狭窄区域提供的孔。 通孔的直径大大大于夹紧螺栓的直径。 孔的内表面和螺栓的外表面之间的空间用作低压制冷剂气体流过的通道，这有助于简化结构并提高斜盘式压缩机的容量。

公开(公告)号：US20140179517A1

公开(公告)日：2014-06-26

申请号：US14124546

申请日：2012-06-06

申请人： Nobuyuki Araki ,  Taiji Miyake ,  Eiyu Imai ,  Emiko Obata

发明人： Nobuyuki Araki ,  Taiji Miyake ,  Eiyu Imai ,  Emiko Obata

IPC分类号： A01N43/653

CPC分类号： C07D249/12 ,  A01N43/50 ,  A01N43/653 ,  A01N43/80 ,  C07D233/56 ,  C07D233/60 ,  C07D249/08 ,  C07D405/04 ,  C07D405/06 ,  A01N25/04 ,  A01N25/28

摘要： Provided is an azole derivative superior in disease-controlling activity contained as an active ingredient in agricultural or horticultural chemical agents.The azole derivative according to the present invention is represented by the following General Formula (I): (in Formula (I), R1 represents an unsubstituted or substituted C1-C6-alkyl group; R2 represents a carbonyl group-containing functional group, wherein the carbon atom in the carbonyl group is bound to the carbon atom in the cyclopentane ring substituted with R1 and to a hydrogen atom, a hydroxyl group, R3, OR3, or NR3R4; R3 and R4 each represent a C1-C6-alkyl group, a C2-C6-alkenyl group, or a C2-C6-alkynyl group; Y represents a halogen atom, a C1-C4-alkyl group, a C1-C4-haloalkyl group, a C1-C4-alkoxy group, a C1-C4-haloalkoxy group, a phenyl group, a cyano group, or a nitro group; m is 0 to 5; and A represents a nitrogen atom or a methine group).

摘要翻译： 提供在农业或园艺化学试剂中作为活性成分含有的疾病控制活性优异的唑衍生物。 根据本发明的唑衍​​生物由以下通式（I）表示：（在式（I）中，R 1表示未取代或取代的C 1 -C 6 - 烷基; R 2表示含羰基的官能团，其中 羰基中的碳原子与被R 1取代的环戊烷环中的碳原子结合，并与氢原子，羟基，R3，OR3或NR3R4结合; R3和R4各自表示C1-C6-烷基， C2-C6-烯基或C2-C6-炔基; Y表示卤素原子，C1-C4-烷基，C1-C4-卤代烷基，C1-C4-烷氧基，C1- C4卤代烷氧基，苯基，氰基或硝基; m为0-5; A表示氮原子或次甲基）。

公开(公告)号：US09253983B2

公开(公告)日：2016-02-09

申请号：US14122944

申请日：2012-05-30

申请人： Taiji Miyake ,  Nobuyuki Araki ,  Toru Yamazaki

发明人： Taiji Miyake ,  Nobuyuki Araki ,  Toru Yamazaki

IPC分类号： A01N43/653 ,  C07B57/00 ,  C07D249/08

CPC分类号： A01N43/653 ,  C07B57/00 ,  C07D249/08 ,  A01N25/00

摘要： In order to provide a compound that shows a strong effect on controlling a plant disease, a triazole compound of the present invention (i) is a compound in which —OH group, —R2 group, and CH2—Ar group are bonded in cis configuration with a cyclopentane, (ii) is (−)-enantiomer or (+) enantiomer, and (iii) is represented by Formula (I): (wherein R1 represents an alkyl group; R2 represents a haloalkyl group; and Ar represents a substituted/unsubstituted aromatic hydrocarbon group or a substituted/unsubstituted aromatic heterocyclic group.

摘要翻译： 为了提供对控制植物病害具有强效果的化合物，本发明的三唑化合物（i）是其中-OH基，-R2基和CH2-Ar基以顺式结构键合的化合物 （ii）为（ - ） - 对映体或（+）对映异构体，（iii）由式（I）表示：（其中R 1表示烷基; R 2表示卤代烷基; Ar表示取代基 /未取代的芳香族烃基或取代/未取代的芳香族杂环基。

公开(公告)号：US09035069B2

公开(公告)日：2015-05-19

申请号：US14124546

申请日：2012-06-06

申请人： Nobuyuki Araki ,  Taiji Miyake ,  Eiyu Imai ,  Emiko Obata

发明人： Nobuyuki Araki ,  Taiji Miyake ,  Eiyu Imai ,  Emiko Obata

IPC分类号： C07D233/56 ,  C07D249/08 ,  A01N43/653 ,  A01N43/50 ,  C07D233/60 ,  C07D405/06 ,  A01N43/80

CPC分类号： C07D249/12 ,  A01N43/50 ,  A01N43/653 ,  A01N43/80 ,  C07D233/56 ,  C07D233/60 ,  C07D249/08 ,  C07D405/04 ,  C07D405/06 ,  A01N25/04 ,  A01N25/28

摘要： Provided is an azole derivative superior in disease-controlling activity contained as an active ingredient in agricultural or horticultural chemical agents.The azole derivative according to the present invention is represented by the following General Formula (I): (in Formula (I), R1 represents an unsubstituted or substituted C1-C6-alkyl group; R2 represents a carbonyl group-containing functional group, wherein the carbon atom in the carbonyl group is bound to the carbon atom in the cyclopentane ring substituted with R1 and to a hydrogen atom, a hydroxyl group, R3, OR3, or NR3R4; R3 and R4 each represent a C1-C6-alkyl group, a C2-C6-alkenyl group, or a C2-C6-alkynyl group; Y represents a halogen atom, a C1-C4-alkyl group, a C1-C4-haloalkyl group, a C1-C4-alkoxy group, a C1-C4-haloalkoxy group, a phenyl group, a cyano group, or a nitro group; m is 0 to 5; and A represents a nitrogen atom or a methine group).

摘要翻译： 提供在农业或园艺化学试剂中作为活性成分含有的疾病控制活性优异的唑衍生物。 根据本发明的唑衍​​生物由以下通式（I）表示：（在式（I）中，R 1表示未取代或取代的C 1 -C 6 - 烷基; R 2表示含羰基的官能团，其中 羰基中的碳原子与被R 1取代的环戊烷环中的碳原子结合，并与氢原子，羟基，R3，OR3或NR3R4结合; R3和R4各自表示C1-C6-烷基， C2-C6-烯基或C2-C6-炔基; Y表示卤素原子，C1-C4-烷基，C1-C4-卤代烷基，C1-C4-烷氧基，C1- C4卤代烷氧基，苯基，氰基或硝基; m为0-5; A表示氮原子或次甲基）。