公开(公告)号：US4957535A

公开(公告)日：1990-09-18

申请号：US250888

申请日：1988-09-29

申请人： Beat Bohner ,  Georg Pissiotasa ,  Hans Moser

发明人： Beat Bohner ,  Georg Pissiotasa ,  Hans Moser

IPC分类号： A01N37/32 ,  A01N43/90 ,  A01N47/02 ,  C07D209/48 ,  C07D471/04 ,  C07D487/04 ,  C07D513/04

CPC分类号： C07D209/48 ,  A01N37/32 ,  A01N43/90 ,  A01N47/02 ,  C07D471/04 ,  C07D487/04 ,  C07D513/04

摘要： Novel bicyclic triazole compounds of the formula I have an excellent herbicidal and plant-growth regulating action.The compounds correspond to the formula I ##STR1## wherein Q is hydrogen or halogen,T is halogen, andZ is a radical --XR or --COXR, in whichX is oxygen, sulfur or a radical --NR.sub.2 --,R is hydrogen, a C.sub.1 -C.sub.6 -alkyl, C hd 3-C.sub.6 -cycloalkyl, C hd 2-C.sub.6 -alkenyl or C.sub.3 -C.sub.6 -alkynyl radical, which is unsubstituted or substituted by halogen, or is a radical --A--COXR.sub.1, in whichA is a C.sub.1 -C.sub.4 -alkylene bridge andR.sub.1 is hydrogen or C.sub.1 -C.sub.4 -alkyl, C.sub.3 -C.sub.6 -cycloalkyl, C.sub.3 -C.sub.4 -alkenyl or C.sub.3 -C.sub.4 -alkynyl.

摘要翻译： 式I的新型双环三唑化合物具有优异的除草和植物生长调节作用。 化合物对应于其中Q为氢或卤素，T为卤素且Z为基团-XR或-COXR的式I（I）其中X为氧，硫或基团-NR 2 - ，R 是未取代或被卤素取代的氢，C 1 -C 6 - 烷基，C 5d 3 -C 6环烷基，C 2d-C 2 -C 6链烯基或C 3 -C 6炔基，或者是-A-COXR1基团， 其中A是C1-C4-亚烷基桥，R1是氢或C1-C4-烷基，C3-C6-环烷基，C3-C4-烯基或C3-C4-炔基。

公开(公告)号：US5078780A

公开(公告)日：1992-01-07

申请号：US109667

申请日：1987-10-16

申请人： Hans Moser ,  Beat Bohner ,  Werner Fory

发明人： Hans Moser ,  Beat Bohner ,  Werner Fory

IPC分类号： C07F7/18 ,  A01N25/04 ,  A01N25/32 ,  A01N43/40 ,  A01N43/56 ,  A01P13/00 ,  C07D231/14 ,  C07D401/12 ,  C07D405/12 ,  C07D409/12 ,  C07D417/12 ,  C07D487/04 ,  C07D521/00

CPC分类号： C07D231/12 ,  A01N25/32 ,  C07D231/14 ,  C07D233/56 ,  C07D249/08 ,  C07D401/12 ,  C07D405/12 ,  C07D409/12 ,  C07D417/12 ,  C07D487/04

摘要： 1,5-diphenylpyrazole-3-carboxylic acid derivatives of the formula ##STR1## are capable of antagonising specifically the phytotoxic action of phenoxypropionic acid ester herbicides of the formula II ##STR2## in which G represents ##STR3## Compositions, containing those compositions, as selective herbicides and the use of those two active ingredients for controlling weeds in crops of useful plants are described, as are also novel 1,5-diphenylpyrazole-3-carboxylic acid derivatives corresponding to the formula I and the preparation thereof.

公开(公告)号：US4944790A

公开(公告)日：1990-07-31

申请号：US325833

申请日：1989-03-20

申请人： Hans Moser ,  Beat Bohner ,  Werner Fory

发明人： Hans Moser ,  Beat Bohner ,  Werner Fory

IPC分类号： C07F7/18 ,  A01N25/04 ,  A01N25/32 ,  A01N43/40 ,  A01N43/56 ,  A01P13/00 ,  C07D231/14 ,  C07D401/12 ,  C07D405/12 ,  C07D409/12 ,  C07D417/12 ,  C07D487/04 ,  C07D521/00

CPC分类号： C07D231/12 ,  A01N25/32 ,  C07D231/14 ,  C07D233/56 ,  C07D249/08 ,  C07D401/12 ,  C07D405/12 ,  C07D409/12 ,  C07D417/12 ,  C07D487/04

摘要： 1,5-diphenylpyrazole-3-carboxylic acid derivatives of the formula ##STR1## in which each of R.sub.a and R.sub.b, independently of the other represents halogen, C.sub.1 -C.sub.5 -alkyl, C.sub.1 -C.sub.5 -haloalkyl, C.sub.2 -C.sub.5 -alkenyl, C.sub.2 -C.sub.5 -alkynyl or cyano, n represents zero or an integer from 1 to 3, and OR.sub.1 represents hydroxy, a plant-physiologically tolerable salt radical or any desired ester radical, are capable of antagonizing specifically the phytotoxic action of phenoxypropionic acid ester herbicides of the formula II ##STR2## in which G represents ##STR3## in which Hal.sub.1 represents fluorine, chlorine, bromine, iodine or trifluoromethyl, Hal.sub.2 represents hydrogen, fluorine, chlorine, bromine or trifluoromethyl, Z represents nitrogen or methine (--CH.dbd.), X represents an oxygen or sulphur atom, R.sub.1 ' represents halogen, trifluoromethyl, nitro, cyano, C.sub.1 -C.sub.4 -alkyl or C.sub.1 -C.sub.4 -alkoxy and n represents 0, 1, 2 or 3 and T represents an ester, amide, cyanamide or oxime radical.Compositions, containing those components, as selective herbicides and the use of those two active ingredients for controlling weeds in crops of useful plants are described, as are also novel 1,5-diphenylpyrazole-3-carboxylic acid derivatives corresponding to the formula I and the preparation thereof.

摘要翻译： 其中R a和R b各自独立地表示卤素，C 1 -C 5 - 烷基，C 1 -C 5 - 卤代烷基，C 2 -C 5 - 烯基的1,5-二苯基吡唑-3-羧酸衍生物 ，C 2 -C 5炔基或氰基，n表示0或1至3的整数，OR 1表示羟基，植物 - 生理上可耐受的盐基或任何所需的酯基，能够特异性地拮抗苯氧基丙酸酯的植物毒性作用 其中G代表其中Hal1代表氟，氯，溴，碘或三氟甲基的式Ⅱ的除草剂，其中G代表氢，氯，溴，碘或三氟甲基，Hal2代表氢，氟，氯，溴或三氟甲基，Z 表示氮或次甲基（-CH =），X表示氧或硫原子，R1'表示卤素，三氟甲基，硝基，氰基，C1-C4-烷基或C1-C4-烷氧基，n表示0,1,2或3 T代表酯，酰胺，氰胺或肟基。 描述了含有这些成分的作为选择性除草剂的组合物以及这两种活性成分用于控制有用植物作物中的杂草的用途，以及对应于式I的新的1,5-二苯基吡唑-3-羧酸衍生物和 的制备。

公开(公告)号：US5114462A

公开(公告)日：1992-05-19

申请号：US325834

申请日：1989-03-20

申请人： Hans Moser ,  Beat Bohner ,  Werner Fory

发明人： Hans Moser ,  Beat Bohner ,  Werner Fory

IPC分类号： C07F7/18 ,  A01N25/04 ,  A01N25/32 ,  A01N43/40 ,  A01N43/56 ,  A01P13/00 ,  C07D231/14 ,  C07D401/12 ,  C07D405/12 ,  C07D409/12 ,  C07D417/12 ,  C07D487/04 ,  C07D521/00

CPC分类号： C07D231/12 ,  A01N25/32 ,  C07D231/14 ,  C07D233/56 ,  C07D249/08 ,  C07D401/12 ,  C07D405/12 ,  C07D409/12 ,  C07D417/12 ,  C07D487/04

摘要： 1,5-diphenylpyrazole-3-carboxylic acid derivatives of the formula ##STR1## in which each of R.sub.a and R.sub.b, independently of the other, represents halogen, C.sub.1 -C.sub.5 -alkyl, C.sub.1 -C.sub.5 -haloalkyl, C.sub.2 -C.sub.5 -alkenyl, C.sub.2 -C.sub.5 -alkynyl or cyano, n represents zero or an integer from 1 to 3, and OR.sub.1 represents hydroxy, a plant-physiologically tolerable salt radical or any desired ester radical, are capable of antagonizing specifically the phytotoxic action of phenoxypropionic acid ester herbicides of the formula II ##STR2## in which G represents ##STR3## in which Hal.sub.1 represents fluorine, chlorine, bromine, iodine or trifluoromethyl, Hal.sub.2 represents hydrogen, fluorine, chlorine, bromine or trifluoromethyl, Z represents nitrogen or methine (--CH.dbd.), X represents an oxygen or sulphur atom, R.sub.1 ' represents halogen, trifluoromethyl, nitro, cyano, C.sub.1 -C.sub.4 -alkyl or C.sub.1 -C.sub.4 -alkoxy and n represents, 0, 1, 2 or 3 and T represents an ester, amide, cyanamide or oxime radical.Compositions, containing those components, as selective herbicides and the use of those two active ingredients for controlling weeds in crops of useful plants are described, as are also novel 1,5-diphenyl-pyrazole-3-carboxylic acid derivatives corresponding to the formula I and the preparation thereof.

公开(公告)号：US4940485A

公开(公告)日：1990-07-10

申请号：US277090

申请日：1988-11-28

申请人： Beat Bohner ,  Hans Moser ,  Georg Pissiotas

发明人： Beat Bohner ,  Hans Moser ,  Georg Pissiotas

IPC分类号： A01N37/22 ,  A01N37/32 ,  A01N37/34 ,  A01N37/36 ,  A01N39/04 ,  C07C67/00 ,  C07C213/00 ,  C07C217/82 ,  C07C253/00 ,  C07C255/13 ,  C07C313/00 ,  C07C323/35 ,  C07C323/36 ,  C07C325/00 ,  C07C327/22 ,  C07D209/48

CPC分类号： C07D209/48 ,  A01N37/32 ,  A01N39/04

摘要： The invention relates to novel 3-methyltetrahydrophthalimides of the formula I in which the substituents R.sub.1 is hydrogen or fluorine, R.sub.2 is halogen, X is O or S and R.sub.3 is C.sub.3 -C.sub.10 -alkenyl, C.sub.5 -C.sub.6 -cycloakly, C.sub.5 -C.sub.6 -cycloalkenyl, C.sub.3 -C.sub.10 -alkynyl, or C.sub.1 -C.sub.10 -alkyl which if desired, is mono- or poly-substituted by halogen, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -alkoxycarbonyl, cyano, C.sub.1 -C.sub.4 -alkylthio or by C.sub.1 -C.sub.4 -alkylthiocarbonyl, to processes for their preparation, and to novel selective herbicidal compositions containing compounds of the formula I.

摘要翻译： 本发明涉及式Ⅰ（I）的新型3-甲基四氢邻苯二酰亚胺，其中取代基R 1为氢或氟，R 2为卤素，X为O或S，R 3为C 3 -C 10 - 链烯基，C 5 -C 6 - C 1 -C 4 - 烷氧基，C 1 -C 4 - 烷氧基羰基，氰基，C 1 -C 4 - 烷氧基，C 1 -C 4 - 烷氧基，C 1 -C 4 - C4烷硫基或C1-C4烷硫基羰基，其制备方法，以及含有式I化合物的新型选择性除草组合物。

公开(公告)号：US4789394A

公开(公告)日：1988-12-06

申请号：US886501

申请日：1986-07-17

申请人： Beat Bohner ,  Georg Pissiotas ,  Hans Moser

发明人： Beat Bohner ,  Georg Pissiotas ,  Hans Moser

IPC分类号： A01N43/90 ,  C07D513/04

CPC分类号： C07D513/04 ,  A01N43/90

摘要： Novel bicyclic triazole compounds of the formula I have an excellent herbicidal and plant-growth regulating action.The compounds correspond to the formula I ##STR1## wherein Q is hydrogen or halogen,T is halogen, andZ is a radical --XR or --COXR, in whichX is oxygen, sulfur or a radical --NR.sub.1 --,R is hydrogen, a C.sub.1 -C.sub.6 -alkyl, C.sub.3 -C.sub.6 -cycloalkyl, C.sub.3 -C.sub.6 -alkenyl or C.sub.3 -C.sub.6 -alkynyl radical, which is unsubstituted or substituted by halogen, or is a radical --A--COXR.sub.1, in whichA is a C.sub.1 -C.sub.4 -alkylene bridge andR.sub.1 is hydrogen or C.sub.1 -C.sub.4 -alkyl, C.sub.3 -C.sub.6 -cycloalkyl, C.sub.3 -C.sub.4 -alkenyl or C.sub.3 -C.sub.4 -alkynyl.

摘要翻译： 式I的新型双环三唑化合物具有优异的除草和植物生长调节作用。 该化合物对应于其中Q为氢或卤素，T为卤素且Z为基团-XR或-COXR的式I（I）其中X为氧，硫或基团-NR 1 - ，R 是未取代的或被卤素取代的C 1 -C 6 - 烷基，C 3 -C 6 - 环烷基，C 3 -C 6 - 烯基或C 3 -C 6 - 炔基，或者是A-COXR1基团，其中A是 C1-C4-亚烷基桥，R1是氢或C1-C4-烷基，C3-C6-环烷基，C3-C4-烯基或C3-C4-炔基。

公开(公告)号：US5217524A

公开(公告)日：1993-06-08

申请号：US764756

申请日：1991-09-24

申请人： Beat Bohner ,  Hans Moser

发明人： Beat Bohner ,  Hans Moser

IPC分类号： A01N25/32 ,  A01N43/653 ,  C07D249/10

CPC分类号： A01N25/32 ,  A01N43/653 ,  C07D249/10

摘要： 1,5-Diphenyl-1,2,4-triazole-3-carboxylic acid derivatives of formula ##STR1## wherein each of R.sub.a and R.sub.b, independently of the other, is halogen, C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.5 haloalkyl, C.sub.2 -C.sub.5 alkenyl, C.sub.2 -C.sub.5 alkynyl or cyano, n is zero or a number from 1 to 3 and OR is hydroxy, a phytophysiologically tolerable metal or ammonium salt radical, or an ester radical defined in the description, are capable of specifically antagonising the phytotoxic action of herbicides.1,5-Diphenyl-1,2,4-triazole-3-carboxylic acid derivatives of formula I and the preparation thereof, compositions containing these components as selective herbicides and the use of these two active ingredient components for controlling weeds in crops of useful plants are described.

摘要翻译： 式（I）的1,5-二苯基-1,2,4-三唑-3-羧酸衍生物，其中R a和R b各自独立地为卤素，C 1 -C 5烷基，C 1 -C 5卤代烷基， C 2 -C 5烯基，C 2 -C 5炔基或氰基，n为0或1至3的数，OR为羟基，植物生理学上可耐受的金属或铵盐基团或描述中定义的酯基能够特异性拮抗植物毒素 除草剂的作用 式I的1,5-二苯基-1,2,4-三唑-3-羧酸衍生物及其制备方法，含有这些组分作为选择性除草剂的组合物以及这两种活性成分组分用于控制作物中杂草的用途 描述植物。

公开(公告)号：US5034048A

公开(公告)日：1991-07-23

申请号：US465719

申请日：1990-01-16

申请人： Georg Pissiotas ,  Hans Moser ,  Beat Bohner

发明人： Georg Pissiotas ,  Hans Moser ,  Beat Bohner

IPC分类号： A01N43/00 ,  C07D209/48 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12 ,  C07D521/00

CPC分类号： C07D209/48 ,  C07D231/12 ,  C07D233/56 ,  C07D249/08 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D417/12

摘要： 5-(N-3,4,5,6-tetrahydrophthalimido)benzoic acid esters of formula I below have good selective herbicidal properties pre- and postemergence and also influence or inhibit plant growth.The novel compounds are of formula I ##STR1## wherein n is 0, 1, or 2,R is C.sub.1 -C.sub.3 alkyl,R.sub.1 is hydrogen or halogen,R.sub.2 is halogen,X is oxygen or sulfur,A is a straight chain or branched C.sub.1 -C.sub.4 alkylene bridge,Q is a 5- or 6-membered heterocycle which is bound through carbon or nitrogen and contains 1 to 3 hetero atoms and may further contain one or two carbonyl groups, which heterocycle may be fused to benzene rings and substituted by halogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.3 haloalkyl, C.sub.1 -C.sub.3 alkoxy, C.sub.1 -C.sub.3 haloalkoxy, nitro, cyano, C.sub.1 -C.sub.3 alkylamino or di(C.sub.1 -C.sub.3)alkylamino, or Q is C.sub.1 -C.sub.4 alkylthio, C.sub.1 -C.sub.4 alkylsulfonyl, C.sub.2 -C.sub.8 alkoxyalkyl, nitro or di(C.sub.1 -C.sub.4)alkylamino, or is a benzyloxy, phenoxy or phenylthio radical, each of which may be substituted in the phenyl nucleus by halogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.3 haloalkyl, C.sub.1 -C.sub.3 alkoxy, C.sub.1 -C.sub.3 haloalkoxy, nitro, cyano, C.sub.1 -C.sub.3 alkylamino or di(C.sub.1 -C.sub.3)alkylamino, or, if X is sulfur, Q may also be a COOR.sub.3 radical, in whichR.sub.3 is C.sub.1 -C.sub.20 alkyl, C.sub.3 -C.sub.6 alkenyl, C.sub.3 -C.sub.6 alkynyl or C.sub.3 -C.sub.7 cycloalkyl, each of which is unsubstituted or substituted by halogen or C.sub.1 -C.sub.4 alkoxy.

公开(公告)号：US4929272A

公开(公告)日：1990-05-29

申请号：US281562

申请日：1988-12-08

申请人： Hans Moser ,  Georg Pissiotas ,  Hans-Georg Brunner ,  Beat Bohner ,  Marcus Baumann

发明人： Hans Moser ,  Georg Pissiotas ,  Hans-Georg Brunner ,  Beat Bohner ,  Marcus Baumann

IPC分类号： C07D207/40 ,  C07D207/404 ,  C07D207/44 ,  C07D207/448 ,  C07D405/10

CPC分类号： C07D207/404 ,  C07D207/448 ,  C07D405/10

摘要： Novel derivatives of N-phenylmaleic acid imide and N-phenylsuccinimide have good pre- and post-emergence selective herbicidal properties and they influence plant growth. The compounds correspond to the formula I in which.vertline.: represents a single or double bond,R.sup.1 represents hydrogen or fluorine,R.sup.2 represents halogen,Y represents C.sub.1 -C.sub.8 -alkyl,Z represents hydrogen or C.sub.1 -C.sub.8 -alkyl, andA represents hydrogen or a group ##STR1## wherein R.sup.3, R.sup.4, R.sup.5, R.sup.6, R.sup.7 and R.sup.8 represent customary organic radicals and X represents oxygen, sulphur, SO, SO.sub.2, NH, alkylimino or alkenylimino.

公开(公告)号：US5077413A

公开(公告)日：1991-12-31

申请号：US248077

申请日：1988-09-23

申请人： Beat Bohner ,  Hans Moser

发明人： Beat Bohner ,  Hans Moser

IPC分类号： C07D261/14 ,  A01N25/04 ,  A01N25/32 ,  A01N43/40 ,  A01N43/653 ,  A01P13/00 ,  C07D249/08 ,  C07D249/10

CPC分类号： A01N43/653 ,  A01N25/32 ,  C07D249/10

摘要： 1,5-Diphenyl-1,2,4-triazole-3-carboxylic acid derivatives of formula ##STR1## wherein each of R.sub.a and R.sub.b, independently of the other, is halogen, C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.5 haloalkyl, C.sub.2 -C.sub.5 alkenyl, C.sub.2 -C.sub.5 alkynyl or cyano, n is zero or a number from 1 to 3 and OR is hydroxy, a phytophysiologically tolerable metal or ammonium salt radical, or an ester radical defined in the description, are capable of specifically antagonizing the phytotoxic action of herbicides.1,5-Diphenyl-1,2,4-triazole-3-carboxylic acid derivatives of formula I and the preparation thereof, compositions containing these components as selective herbicides and the use of these two active ingredient components for controlling weeds in crops of useful plants are described.

摘要翻译： 式（I）的1,5-二苯基-1,2,4-三唑-3-羧酸衍生物，其中R a和R b各自独立地为卤素，C 1 -C 5烷基，C 1 -C 5卤代烷基， C 2 -C 5烯基，C 2 -C 5炔基或氰基，n为0或1至3的数，OR为羟基，植物生理学上可耐受的金属或铵盐基团或描述中定义的酯基能够特异性拮抗植物毒素 除草剂的作用 式I的1,5-二苯基-1,2,4-三唑-3-羧酸衍生物及其制备方法，含有这些组分作为选择性除草剂的组合物以及这两种活性成分组分用于控制作物中杂草的用途 描述植物。