NOVEL PYRIDAZINE DERIVATIVES
    9.
    发明申请
    NOVEL PYRIDAZINE DERIVATIVES 审中-公开
    新的吡咯烷酮衍生物

    公开(公告)号:US20100029668A1

    公开(公告)日:2010-02-04

    申请号:US12374052

    申请日:2007-07-16

    IPC分类号: A01N43/58 C07D405/04 A01P3/00

    摘要: The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is hydrogen, C1-C6alkyl, C1-C6haloalkyl or C3-C6cycloalkyl; R2 is an optionally substituted heteroaryl; R3 is an optionally substituted heteroaryl; and R4 is hydrogen, halogen, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy, C1-C6haloalkoxy, hydroxy or cyano; or an agrochemically usable salt form thereof.

    摘要翻译: 本发明涉及具有杀微生物活性,特别是杀真菌活性的活性成分的式(I)的新哒嗪衍生物,其中R1是氢,C1-C6烷基,C1-C6卤代烷基或C3-C6环烷基; R2是任选取代的杂芳基; R3是任选取代的杂芳基; R4是氢,卤素,C1-C6烷基,C1-C6卤代烷基,C1-C6烷氧基,C1-C6卤代烷氧基,羟基或氰基; 或其农业化学上可用的盐形式。

    PYRIDAZINE DERIVATIVES USEFUL AS FUNGICIDES AND FOR THE TREATMENT OF CANCER
    10.
    发明申请
    PYRIDAZINE DERIVATIVES USEFUL AS FUNGICIDES AND FOR THE TREATMENT OF CANCER 审中-公开
    用作杀真菌剂和治疗癌症的吡咯烷酮衍生物

    公开(公告)号:US20100273804A1

    公开(公告)日:2010-10-28

    申请号:US12809604

    申请日:2008-12-19

    摘要: The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: formula (I) wherein R1 is C1-C6alkyl, C1-C6haloalkyl or C3-C6cycloalkyl; R2 is hydrogen or an optionally substituted alkyl, aryl or heteroaryl; R3 is hydrogen, C1-C6alkyl or C1-C6haloalkyl; R4 is hydrogen, C1-C6alkyl or C1-C6haloalkyl; or R3 and R4 together can be part of a carbocyclic or heterocyclic 3- to 8-membered ring; R5 is optionally substituted aryl or heteroaryl; and R6 is hydroxy, halogen, C1-C6alkoxy, C1-C6haloalkoxy, C1-C6alkylthio or C1-C6haloalkylthio; or an agrochemically usable salt form thereof.

    摘要翻译: 本发明涉及具有杀微生物活性,特别是杀真菌活性的作为活性成分的式(I)的新哒嗪衍生物:式(I)其中R 1是C 1 -C 6烷基,C 1 -C 6卤代烷基或C 3 -C 6环烷基; R 2是氢或任选取代的烷基,芳基或杂芳基; R3是氢,C1-C6烷基或C1-C6卤代烷基; R4是氢,C1-C6烷基或C1-C6卤代烷基; 或者R 3和R 4一起可以是碳环或杂环的3至8元环的一部分; R5是任选取代的芳基或杂芳基; R 6为羟基,卤素,C 1 -C 6烷氧基,C 1 -C 6卤代烷氧基,C 1 -C 6烷硫基或C 1 -C 6卤代烷硫基; 或其农业化学上可用的盐形式。