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    NOVEL MICROBICIDES
    1.
    发明申请
    NOVEL MICROBICIDES 审中-公开
    新型微生物

    公开(公告)号：US20130281467A1

    公开(公告)日：2013-10-24

    申请号：US13881648

    申请日：2011-10-28

    Applicant: Stephan Trah ,  Laura Quaranta ,  Clemens Lamberth ,  Martin Pouliot

    Inventor： Stephan Trah ,  Laura Quaranta ,  Clemens Lamberth ,  Martin Pouliot

    IPC: A01N43/54 ,  A01N43/90

    CPC classification number: A01N43/54 ,  A01N43/90 ,  C07D401/04 ,  C07D491/04 ,  C07D491/10

    Abstract: Compounds of formula (I), wherein G represents together with the two carbon atoms of the pyrimidine ring to which it is attached, a 5- to 7-membered aliphatic carbocyclic or heterocyclic ring system which contain 0 to 2 heteroatoms selected from the group consisting of nitrogen, oxygen and sulfur; and wherein said 5- to 7-membered aliphatic carbocyclic or heterocyclic ring system can be mono-, di- or trisubstituted by substituents selected from the group consisting of halogen, keto, C1-C6alkyl, C1-C6alkoxy, C1-C6alkyloximino and C1-C6alkylendioxy; and wherein the other substituents R1, R2, R3, R4, R5 and R6 are as defined in claim 1, and their use as microbicides.

    Abstract translation: 式（I）化合物，其中G代表与其连接的嘧啶环的两个碳原子一起，含有0至2个选自以下的杂原子的5-至7-元脂族碳环或杂环系： 的氮，氧和硫; 并且其中所述5-至7-元脂族碳环或杂环系统可以被选自卤素，酮，C 1 -C 6烷基，C 1 -C 6烷氧基，C 1 -C 6烷氧基肟基和C 1 -C 6烷氧基的取代基单，二或三取代， C6烷基二氧基; 并且其中其它取代基R 1，R 2，R 3，R 4，R 5和R 6如权利要求1中所定义，及其作为杀微生物剂的用途。

    PYRIDAZINE DERIVATIVES
    3.
    发明申请
    PYRIDAZINE DERIVATIVES 审中-公开
    吡啶衍生物

    公开(公告)号：US20100144674A1

    公开(公告)日：2010-06-10

    申请号：US12447028

    申请日：2007-10-23

    Applicant: Stephan Trah ,  Clemens Lamberth ,  Sebastian Wendeborn

    Inventor： Stephan Trah ,  Clemens Lamberth ,  Sebastian Wendeborn

    IPC: A01N57/00 ,  C07D237/02 ,  A01N43/58 ,  A01N43/54 ,  A01N43/84 ,  A01P3/00 ,  A01P15/00

    CPC classification number: C07D237/14 ,  A01N43/58 ,  C07D237/08 ,  C07D237/12 ,  C07D307/60 ,  C07D307/79 ,  C07D401/04 ,  C07D401/12 ,  C07D403/04 ,  C07D405/04 ,  C07D405/12 ,  C07D407/04 ,  C07D409/04 ,  C07D409/12 ,  C07D413/04 ,  C07D417/04

    Abstract: The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is hydrogen, C1-C6alkyl, C1-C8haloalkyl or C3-C6cycloalkyl; R2 is cycloalkyl, cycloalkylalkyl, halocycloalkyl, cycloalkoxy, halocycloalkoxy, cycloalkylalkoxy, halocycloalkylalkoxy, alkoxyalkyl, cycloalkoxyalkoxyalkyl, haloalkoxyalkyl, trialkylsilyl, alkylthioalkyl, haloalkylthioalkyl, cycloalkylthio, halocycloalkylthio, cycloalkylalkylthio, halocycloalkylalkylthio, alkylsulfinylalkyl, alkylsulfonylalkyl, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl, C2-C6alkenyl, C2-C6alkynyl, optionally substituted arylsulfonyl, optionally substituted aryloxy, optionally optionally substituted heteroaryloxy, optionally substituted arylthio, optionally substituted heteroarylthio; or R2 together with an adjacent carbon atom forms an optionally substituted fused ring; R3 is an optionally substituted aryl; R4 is hydrogen, halogen, C1-C6alkyl, C1-C6haloalkyl, C1-C8alkoxy, C1-C6haloalkoxy, hydroxy or cyano; and n is a whole number from 1 to 4; or an agrochemically usable salt form thereof.

    Abstract translation: 本发明涉及具有杀微生物活性，特别是杀真菌活性的活性成分的式（I）的新哒嗪衍生物，其中R1是氢，C1-C6烷基，C1-C8卤代烷基或C3-C6环烷基; R 2是环烷基，环烷基烷基，卤代环烷基，环烷氧基，卤代环烷氧基，环烷基烷氧基，卤代环烷基烷氧基，烷氧基烷基，环烷氧基烷氧基烷基，卤代烷氧基烷基，三烷基甲硅烷基，烷硫基烷基，卤代烷硫基烷基，环烷硫基，卤代环烷硫基，环烷基烷硫基，卤代环烷基烷硫基，烷基亚磺酰基烷基，烷基磺酰基烷基，烷基亚磺酰基，卤代烷基亚磺酰基，烷基磺酰基，卤代烷基磺酰基， C 6链烯基，C 2 -C 6炔基，任选取代的芳基磺酰基，任选取代的芳氧基，任选任选取代的杂芳氧基，任选取代的芳硫基，任选取代的杂芳硫基; 或R 2与相邻的碳原子一起形成任选取代的稠环; R3是任选取代的芳基; R4是氢，卤素，C1-C6烷基，C1-C6卤代烷基，C1-C8烷氧基，C1-C6卤代烷氧基，羟基或氰基; n为1〜4的整数; 或其农业化学上可用的盐形式。

    PESTICIDALLY ACTIVE KETONE AND OXIME DERIVATIVES
    4.
    发明申请
    PESTICIDALLY ACTIVE KETONE AND OXIME DERIVATIVES 审中-公开
    杀虫活性酮和氧化衍生物

    公开(公告)号：US20090298898A1

    公开(公告)日：2009-12-03

    申请号：US12533302

    申请日：2009-07-31

    Applicant: Werner Zambach ,  Roger Graham Hall ,  Peter Renold ,  Stephan Trah

    Inventor： Werner Zambach ,  Roger Graham Hall ,  Peter Renold ,  Stephan Trah

    IPC: A01N43/80 ,  C07C233/02 ,  C07C249/02 ,  C07D261/06 ,  A01N37/18 ,  A01N33/02 ,  A01P7/00

    CPC classification number: C07D333/58 ,  A01N33/24 ,  A01N35/10 ,  A01N37/52 ,  A01N41/06 ,  A01N43/10 ,  A01N43/40 ,  A01N43/78 ,  A01N43/80 ,  C07C49/753 ,  C07C49/755 ,  C07C49/84 ,  C07C235/84 ,  C07C251/44 ,  C07C251/48 ,  C07C251/54 ,  C07C251/58 ,  C07C311/04 ,  C07C311/05 ,  C07C311/09 ,  C07C323/47 ,  C07D213/50 ,  C07D213/53 ,  C07D213/61 ,  C07D213/64 ,  C07D261/08 ,  C07D277/24 ,  C07D277/28 ,  C07D307/52 ,  C07D307/81 ,  C07D333/22

    Abstract: Compounds of formula wherein A0, A1 and A2 are each independently of the others a bond or a C1-C6alkylene bridge; A3 is a C1-C6alkylene bridge which is unsubstituted or substituted by from one to six identical or different substituents selected from halogen and C3-C8cycloalkyl; Y is, for example, O, S, SO or SO2; M is O or NOR6, X1 and X2 are each independently of the other fluorine, chlorine or bromine; R1, R2 and R3 are, for example, H, halogen, OH, SH, CN, nitro, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkylcarbonyl, C2-C6alkenyl, C2-C6haloalkenyl or C2-C6alkynyl; Q is, for example, O, S, SO or SO2; W is, for example, O, S, SO, SO2, —C(═O)—O— or —O—C(═O)—; T is, for example, a bond, O, S, SO, SO2, —C(═O)—O— or —O—C(═O)—; D is CH or N; R4 is, for example, H, halogen, OH, SH, CN, nitro, C1-C6alkyl or C1-C6haloalkyl; R5 is, for example, C1-C12alkyl, C3-C8cycloalkyl or —N(R7)2; R7 is H, C1-C6alkyl, C1-C3haloalkyl, C1-C6alkylcarbonyl, C1-C3haloalkylcarbonyl, C1-C6alkoxycarbonyl, C3-C8cycloalkyl, C3-C8 cycloalkylcarbonyl or formyl; k is 0, 1, 2, 3 or 4; m is 1 or 2; and q is 0, 1 or 2; and, where applicable, their possible E/Z isomers, E/Z isomeric mixtures and/or tautomers, in each case in free form or in salt form, a process for the preparation of those compounds and their use, pesticidal compositions in which the active ingredient has been selected from those compounds and agrochemically acceptable salts thereof, and a process for the preparation of those compositions and their use, to plant propagation material treated with those compositions, and a method of controlling pests.

    Abstract translation: 下式化合物其中A0，A1和A2各自独立地为键或C1-C6亚烷基桥; A3是C1-C6亚烷基桥，其未被取代或被1-6个相同或不同的选自卤素和C 3 -C 8环烷基的取代基取代; Y是例如O，S，SO或SO 2; M为O或NOR6，X1和X2各自独立地为氟，氯或溴; R1，R2和R3是例如H，卤素，OH，SH，CN，硝基，C1-C6烷基，C1-C6卤代烷基，C1-C6烷基羰基，C2-C6链烯基，C2-C6卤代烯基或C2-C6炔基; Q是例如O，S，SO或SO 2; W是例如O，S，SO，SO 2，-C（-O）-O-或-O-C（-O） - ; T是例如键O，S，SO，SO 2，-C（-O）-O-或-O-C（-O） - ; D是CH或N; R4是例如H，卤素，OH，SH，CN，硝基，C1-C6烷基或C1-C6卤代烷基; R5是例如C1-C12烷基，C3-C8环烷基或-N（R7）2; R 7是H，C 1 -C 6烷基，C 1 -C 3卤代烷基，C 1 -C 6烷基羰基，C 1 -C 3卤代烷基羰基，C 1 -C 6烷氧基羰基，C 3 -C 8环烷基，C 3 -C 8环烷基羰基或甲酰基; k为0，1，2，3或4; m为1或2; q为0,1或2; 在适用情况下，它们可能的E / Z异构体，E / Z异构体混合物和/或互变异构体，在每种情况下为游离形式或盐形式，制备这些化合物及其用途的方法，其中 已经从这些化合物和农业化学上可接受的盐中选择活性成分，以及这些组合物的制备方法及其用途，用这些组合物处理的繁殖材料以及控制害虫的方法。

    4-(3,3-dihalo-allyloxy) phenol derivatives having pesticidal properties
    5.
    发明授权
    4-(3,3-dihalo-allyloxy) phenol derivatives having pesticidal properties 失效
    具有杀虫特性的4-（3,3-二卤代烯丙氧基）苯酚衍生物

    公开(公告)号：US07608631B2

    公开(公告)日：2009-10-27

    申请号：US10525891

    申请日：2003-08-29

    Applicant: Wemer Zambach ,  Arthur Steiger ,  Peter Renold ,  Stephan Trah ,  Roger Graham Hall

    Inventor： Wemer Zambach ,  Arthur Steiger ,  Peter Renold ,  Stephan Trah ,  Roger Graham Hall

    IPC: A01N43/40

    CPC classification number: C07D207/325 ,  A01N43/36 ,  A01N43/56 ,  A01N43/653 ,  A01N43/713 ,  A01N43/76 ,  A01N43/78 ,  A01N43/80 ,  A01N43/82 ,  A01N43/90 ,  A01N47/18 ,  A01N47/20 ,  C07D207/333 ,  C07D207/34 ,  C07D231/12 ,  C07D231/22 ,  C07D231/38 ,  C07D249/08 ,  C07D249/10 ,  C07D257/04 ,  C07D261/08 ,  C07D261/10 ,  C07D261/18 ,  C07D263/32 ,  C07D263/34 ,  C07D271/06 ,  C07D271/07 ,  C07D277/24 ,  C07D277/30 ,  C07D277/40 ,  C07D277/48 ,  C07D277/56 ,  C07D285/08 ,  C07D285/12 ,  C07D333/16 ,  C07D333/38 ,  C07D471/04

    Abstract: Compounds of formula (I) wherein Ao is a bond or a C1-C6alkylene bridge; A1, A2 and A3 are a C1-C6alkylene bridge; D is CH or N; W is, for example, O, S, SO, S02, —C(═O)—O— or —O—C(═O)—; T is a bond or, for example, O, NH, S, SO or SR2; Q is, for example, O, S, SO or SO2; Y is, for example, O, S, SO or SO2; X1 and X2 are each independently of the other fluorine, chlorine or bromine; R1, R2 and R3 are, for example, H, halogen, OH, SH, CN or nitro; R4 is, for example, H, halogen, OH, SH, CN, nitro or C1-C6alkyl; R5 is, for example, H, CN, OH, C1-C6alkyl or C3-C8cycloalkyl; k is 1, 2 or 3 when D is nitrogen; or is 1, 2, 3 or 4 when D is CH; m is 1 or 2; E is heteroaryl which is unsubstituted or substituted—depending upon the substitutions possible on the ring—by from one to four identical or different substituents selected from R10; and R10 is, for example, halogen, CN, NO2, OH, SH or C1-C6alkyl; and, where applicable, their possible E/Z isomers, E/Z isomeric mixtures and/or tautomers, in each case in free form or in salt form, a process for the preparation of those compounds and their use, pesticidal compositions in which the active ingredient has been selected from those compounds or an agrochemically acceptable salt thereof, a process for the preparation of those compositions and their use, plant propagation material treated with those compositions, and a method of controlling pests.

    Abstract translation: 式（I）的化合物，其中Ao是一个键或C1-C6亚烷基桥; A1，A2和A3是C1-C6亚烷基桥; D是CH或N; W是例如O，S，SO，SO 2，-C（-O）-O-或-O-C（-O） - ; T是键或例如O，NH，S，SO或SR2; Q是例如O，S，SO或SO 2; Y是例如O，S，SO或SO 2; X1和X2各自独立地为氟，氯或溴; R1，R2和R3是例如H，卤素，OH，SH，CN或硝基; R4是例如H，卤素，OH，SH，CN，硝基或C1-C6烷基; R5是例如H，CN，OH，C1-C6烷基或C3-C8环烷基; 当D为氮时，k为1,2或3; 或D为CH时为1,2,3或4; m为1或2; E是未被取代或被取代的杂芳基，这取决于环上通过1-4个相同或不同的选自R 10的取代基取代的取代基; R 10为例如卤素，CN，NO 2，OH，SH或C 1 -C 6烷基; 在适用情况下，它们可能的E / Z异构体，E / Z异构体混合物和/或互变异构体，在每种情况下为游离形式或盐形式，制备这些化合物及其用途的方法，其中 从这些化合物或其农业化学上可接受的盐中选择活性成分，制备这些组合物的方法及其用途，用这些组合物处理的植物繁殖材料以及控制害虫的方法。

    Process for the preparation of pesticides
    10.
    发明授权
    Process for the preparation of pesticides 失效
    农药制备工艺

    公开(公告)号：US6156923A

    公开(公告)日：2000-12-05

    申请号：US762217

    申请日：1996-12-06

    Applicant: Saleem Farooq ,  Stephan Trah ,  Hugo Ziegler ,  Rene Zurfluh

    Inventor： Saleem Farooq ,  Stephan Trah ,  Hugo Ziegler ,  Rene Zurfluh

    IPC: C07C249/04 ,  C07C249/12 ,  C07C251/48 ,  C07C251/60

    CPC classification number: C07C249/12 ,  C07C251/48 ,  C07C251/60

    Abstract: The invention relates to a process for the preparation of compounds of the formula ##STR1## or, if appropriate, a tautomer thereof, in each case in the free form or in salt form, in whichA, X, Y, Z, R.sub.2, R.sub.3, R.sub.4, R.sub.5, R.sub.7, R.sub.9 and n are as defined in claim 1 and the C.dbd.N double bond marked with E has the E configuration, which comprisesa1) reacting either a compound of the formula (II) mentioned above with a compound of the formula (III) mentioned above, in which X.sub.1 is a leaving group, ora2) a compound of the formula (IV) mentioned above, if appropriate in the presence of a base, with a compound of the formula (V) mentioned above, orb1) reacting a compound of the formula (VI) mentioned above with a compound of the formula R.sub.7 --A--X.sub.2 (VII), in which X.sub.2 is a leaving group, and either further reacting the compound thus obtainable, of the formula (IV), for example according to method a2), orb2) reacting it with hydroxylamine or a salt thereof, if appropriate in the presence of a basic or acid catalyst, and further reacting the compound thus obtainable, of the formula (II), for example according to method a1), orc) reacting a compound of the formula (VII), mentioned above with a C.sub.1 -C.sub.6 alkyl nitrite and further reacting the compound thus obtainable, of the formula (VI), for example according to method b), the E isomers of the compounds of the formulae (II), (IV) and (VI), a process for their preparation and their use for the preparation of compounds of the formula (I).

    Abstract translation: 本发明涉及一种制备下式的化合物或其合适的互变异构体的方法，其各自为游离形式或盐形式，其中A，X，Y，Z，R 2，R 3，R 4 ，R 5，R 7，R 9和n如权利要求1中所定义，并且用E标记的C = N双键具有E构型，其包括a1）使上述式（II）的化合物与 上述式（III），其中X1是离去基团，或a2）上述式（Ⅳ）化合物，如果合适，在碱的存在下，与上述式（Ⅴ）化合物， 或b1）使上述式（Ⅵ）化合物与式R7-A-X2（Ⅶ）化合物反应，其中X 2为离去基团，并进一步使由此得到的化合物（式（Ⅴ） IV），例如根据方法a2），或b2）如果合适，在碱性或酸性催化剂存在下，使其与羟胺或其盐反应， 进一步使由式（II）得到的化合物，例如按照方法a1）进行反应，或c）使上述式（Ⅶ）化合物与亚硝酸C 1 -C 6烷基酯反应，然后进一步使化合物 式（Ⅵ）化合物的E异构体，其制备方法及其制备方法（Ⅵ）的制备方法及其制备方法 式（I）的化合物。

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