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    PYRIDAZINE DERIVATIVES USEFUL AS FUNGICIDES AND FOR THE TREATMENT OF CANCER
    1.
    发明申请
    PYRIDAZINE DERIVATIVES USEFUL AS FUNGICIDES AND FOR THE TREATMENT OF CANCER 审中-公开
    用作杀真菌剂和治疗癌症的吡咯烷酮衍生物

    公开(公告)号：US20100273804A1

    公开(公告)日：2010-10-28

    申请号：US12809604

    申请日：2008-12-19

    申请人： Clemens Lamberth ,  Stephan Trah ,  Raphael Dumeunier ,  Sebastian Volker Wendeborn

    发明人： Clemens Lamberth ,  Stephan Trah ,  Raphael Dumeunier ,  Sebastian Volker Wendeborn

    IPC分类号： A61K31/501 ,  A01N43/58 ,  C07D403/04 ,  C07D237/08 ,  A01P3/00 ,  A61K31/50 ,  A61P35/00

    CPC分类号： C07D237/12 ,  A01N43/58 ,  C07D237/14

    摘要： The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: formula (I) wherein R1 is C1-C6alkyl, C1-C6haloalkyl or C3-C6cycloalkyl; R2 is hydrogen or an optionally substituted alkyl, aryl or heteroaryl; R3 is hydrogen, C1-C6alkyl or C1-C6haloalkyl; R4 is hydrogen, C1-C6alkyl or C1-C6haloalkyl; or R3 and R4 together can be part of a carbocyclic or heterocyclic 3- to 8-membered ring; R5 is optionally substituted aryl or heteroaryl; and R6 is hydroxy, halogen, C1-C6alkoxy, C1-C6haloalkoxy, C1-C6alkylthio or C1-C6haloalkylthio; or an agrochemically usable salt form thereof.

    摘要翻译： 本发明涉及具有杀微生物活性，特别是杀真菌活性的作为活性成分的式（I）的新哒嗪衍生物：式（I）其中R 1是C 1 -C 6烷基，C 1 -C 6卤代烷基或C 3 -C 6环烷基; R 2是氢或任选取代的烷基，芳基或杂芳基; R3是氢，C1-C6烷基或C1-C6卤代烷基; R4是氢，C1-C6烷基或C1-C6卤代烷基; 或者R 3和R 4一起可以是碳环或杂环的3至8元环的一部分; R5是任选取代的芳基或杂芳基; R 6为羟基，卤素，C 1 -C 6烷氧基，C 1 -C 6卤代烷氧基，C 1 -C 6烷硫基或C 1 -C 6卤代烷硫基; 或其农业化学上可用的盐形式。

    NOVEL IMIDAZOLE DERIVATIVES
    3.
    发明申请
    NOVEL IMIDAZOLE DERIVATIVES 审中-公开
    新咪唑衍生物

    公开(公告)号：US20110311649A1

    公开(公告)日：2011-12-22

    申请号：US12739852

    申请日：2008-10-24

    申请人： Raphael Dumeunier ,  Clemens Lamberth ,  Stephan Trah ,  Sebastian Volker Wendeborn

    发明人： Raphael Dumeunier ,  Clemens Lamberth ,  Stephan Trah ,  Sebastian Volker Wendeborn

    IPC分类号： A01N43/40 ,  C07D401/14 ,  A01N43/42 ,  A01N57/00 ,  A01N43/54 ,  A01N43/84 ,  A01N59/20 ,  C07D401/04 ,  A01P3/00

    CPC分类号： C07D233/61 ,  C07D233/68 ,  C07D401/04 ,  C07D401/14 ,  C07D409/04 ,  C07D409/14

    摘要： The present invention relates to novel imidazole derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is halogen, C1-C4alkyl or C1-C4haloalkyl; R2 is an optionally substituted aryl or heteroaryl; R3 is halogen; R4 is hydrogen, halogen, C1-C4alkyl, C1-C4haloalkyl, hydroxyl, C1-C4alkoxy, OR6, C1-C4haloalkoxy or cyano; R5 is halogen; R6 is hydrogen, C3-C7 cycloalkyl, C3-C10 alkylcycloalkyl, C1-C6 haloalkyl, C2-C6 alkenyl, C2-C6 haloalkenyl, C3-C7 cycloalkenyl, C2-C6 alkynyl, C2-C6 haloalkynyl or C2-C6 alkyloxyalkyl; X is N or C(R); and R is hydrogen, halogen, C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy or cyano; or an agrochemically usable salt form thereof; provided that when X is C(R), R2 cannot be an optionally substituted aryl.

    摘要翻译： 本发明涉及式（I）的新咪唑衍生物作为具有杀微生物活性，特别是杀真菌活性的活性成分：其中R1是卤素，C1-C4烷基或C1-C4卤代烷基; R2是任选取代的芳基或杂芳基; R3是卤素; R4是氢，卤素，C1-C4烷基，C1-C4卤代烷基，羟基，C1-C4烷氧基，OR6，C1-C4卤代烷氧基或氰基; R5是卤素; R6是氢，C3-C7环烷基，C3-C10烷基环烷基，C1-C6卤代烷基，C2-C6烯基，C2-C6卤代烯基，C3-C7环烯基，C2-C6炔基，C2-C6卤代炔基或C2-C6烷氧基烷基; X是N或C（R）; 且R为氢，卤素，C 1 -C 4烷基，C 1 -C 4卤代烷基，C 1 -C 4烷氧基，C 1 -C 4卤代烷氧基或氰基; 或其农业化学可用的盐形式; 条件是当X是C（R）时，R 2不能是任选取代的芳基。

    Pyridazine fungicides
    4.
    发明授权
    Pyridazine fungicides 失效
    哒嗪类杀菌剂

    公开(公告)号：US08410026B2

    公开(公告)日：2013-04-02

    申请号：US12863377

    申请日：2009-01-14

    申请人： Stephan Trah ,  Clemens Lamberth ,  Raphael Dumeunier ,  Sebastian Volker Wendeborn

    发明人： Stephan Trah ,  Clemens Lamberth ,  Raphael Dumeunier ,  Sebastian Volker Wendeborn

    IPC分类号： A01N43/58 ,  A61K31/50 ,  C07D237/00

    CPC分类号： C07D401/04

    摘要： The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is methyl, ethyl or isopropyl; R2 is chloro, fluoro, hydroxy or C1-C2alkoxy; R3 is H, chloro, fluoro, methoxy or C1-C3alkyl; R4 is chloro, fluoro or bromo; and R5 is H, fluoro or methoxy; or an agrochemically usable salt form thereof; with the proviso that when R1 is methyl, R2 is chloro and R3 is H, then R4 or R5 is different from fluoro.

    摘要翻译： 本发明涉及式（I）的新的哒嗪衍生物作为具有杀微生物活性的活性成分，特别是杀真菌活性：其中R1是甲基，乙基或异丙基; R 2是氯，氟，羟基或C 1 -C 2烷氧基; R3是H，氯，氟，甲氧基或C1-C3烷基; R4是氯，氟或溴; R5为H，氟或甲氧基; 或其农业化学可用的盐形式; 条件是当R 1为甲基时，R 2为氯且R 3为H，则R 4或R 5不同于氟。

    NOVEL PYRIDAZINE DERIVATIVES
    6.
    发明申请
    NOVEL PYRIDAZINE DERIVATIVES 审中-公开
    新的吡咯烷酮衍生物

    公开(公告)号：US20100029668A1

    公开(公告)日：2010-02-04

    申请号：US12374052

    申请日：2007-07-16

    申请人： Stephan Trah ,  Clemens Lamberth ,  Sebastian Volker Wendeborn

    发明人： Stephan Trah ,  Clemens Lamberth ,  Sebastian Volker Wendeborn

    IPC分类号： A01N43/58 ,  C07D405/04 ,  A01P3/00

    CPC分类号： C07D401/14 ,  A01N43/58 ,  C07D403/14 ,  C07D405/14 ,  C07D407/14 ,  C07D409/14 ,  C07D417/14

    摘要： The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is hydrogen, C1-C6alkyl, C1-C6haloalkyl or C3-C6cycloalkyl; R2 is an optionally substituted heteroaryl; R3 is an optionally substituted heteroaryl; and R4 is hydrogen, halogen, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy, C1-C6haloalkoxy, hydroxy or cyano; or an agrochemically usable salt form thereof.

    摘要翻译： 本发明涉及具有杀微生物活性，特别是杀真菌活性的活性成分的式（I）的新哒嗪衍生物，其中R1是氢，C1-C6烷基，C1-C6卤代烷基或C3-C6环烷基; R2是任选取代的杂芳基; R3是任选取代的杂芳基; R4是氢，卤素，C1-C6烷基，C1-C6卤代烷基，C1-C6烷氧基，C1-C6卤代烷氧基，羟基或氰基; 或其农业化学上可用的盐形式。

    FUNGICIDAL COMPOUNDS AND COMPOSITIONS
    8.
    发明申请
    FUNGICIDAL COMPOUNDS AND COMPOSITIONS 审中-公开
    杀真菌化合物和组合物

    公开(公告)号：US20100016339A1

    公开(公告)日：2010-01-21

    申请号：US12375839

    申请日：2007-07-30

    申请人： Jeremy Godwin ,  Stephan Trah ,  Clemens Lamberth ,  Sebastian Volker Wendeborn

    发明人： Jeremy Godwin ,  Stephan Trah ,  Clemens Lamberth ,  Sebastian Volker Wendeborn

    IPC分类号： A01N43/90 ,  C07D237/02 ,  A01N43/58 ,  A01P3/00

    CPC分类号： C07D237/12 ,  A01N43/58

    摘要： The present invention relates, inter alia, to a compound having the formula (I):—wherein (R)n is selected from the group consisting of 4-Br, 4-OCH2CH3, 4-OCH2CF3, 2-CH3-4-Cl, 2-CH3-4-OCH3, 2-CH3-4-OCF3, 2-F-4-Br, 2-F-4-CF3, 3-CH3-4-Br, 3-F-4-Cl, 3-F-4-CH3, 3-F-4-Br, 3-F-4-OCH3 and 3-F-4-F. The present invention further relates to a fungicidal composition comprising a compound having the formula (I)—and also to fungicidal compositions comprising compounds having the formula (II) and/or (III): Furthermore, the present invention relates to methods for controlling pathogenic organisms using the compositions.

    摘要翻译： 本发明特别涉及具有式（I）的化合物：其中（R）n选自4-Br，4-OCH2CH3,4-OCH2CF3,2-CH3-4-Cl ，2-CH3-4-OCH3,2-CH3-4-OCF3,2-F-4-Br，2-F-4-CF3,3-CH3-4-Br，3-F-4-Cl，3 -F-4-CH 3，3-F-4-Br，3-F-4-OCH 3和3-F-4-F。 本发明还涉及包含具有式（I）的化合物的杀真菌组合物，还涉及包含具有式（II）和/或（III）的化合物的杀真菌组合物：此外，本发明涉及控制致病性的方法 使用组合物的生物体。

    PYRIDAZINE FUNGICIDES
    9.
    发明申请
    PYRIDAZINE FUNGICIDES 失效
    吡咯烷类杀真菌剂

    公开(公告)号：US20110112108A1

    公开(公告)日：2011-05-12

    申请号：US12863377

    申请日：2009-01-14

    申请人： Stephan Trah ,  Clemens Lamberth ,  Raphael Dumeunier ,  Sebastian Volker Wenderborn

    发明人： Stephan Trah ,  Clemens Lamberth ,  Raphael Dumeunier ,  Sebastian Volker Wenderborn

    IPC分类号： A61K31/501 ,  C07D401/04 ,  A01N43/48 ,  A61P35/00 ,  A01P3/00

    CPC分类号： C07D401/04

    摘要： The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is methyl, ethyl or isopropyl; R2 is chloro, fluoro, hydroxy or C1-C2alkoxy; R3 is H, chloro, fluoro, methoxy or C1-C3alkyl; R4 is chloro, fluoro or bromo; and R3 is H, fluoro or methoxy; or an agrochemically usable salt form thereof; with the proviso that when R1 is methyl, R2 is chloro and R3 is H, then R4 or R5 is different from fluoro.

    摘要翻译： 本发明涉及式（I）的新的哒嗪衍生物作为具有杀微生物活性的活性成分，特别是杀真菌活性：其中R1是甲基，乙基或异丙基; R2是氯，氟，羟基或C1-C2烷氧基; R3是H，氯，氟，甲氧基或C1-C3烷基; R4是氯，氟或溴; 且R 3为H，氟或甲氧基; 或其农业化学可用的盐形式; 条件是当R 1为甲基时，R 2为氯且R 3为H，则R 4或R 5不同于氟。

    IMIDAZOLE DERIVATIVES
    10.
    发明申请
    IMIDAZOLE DERIVATIVES 审中-公开
    咪唑衍生物

    公开(公告)号：US20120010195A1

    公开(公告)日：2012-01-12

    申请号：US13256074

    申请日：2010-02-08

    申请人： Raphael Dumeunier ,  Clemens Lamberth ,  Stephan Trah

    发明人： Raphael Dumeunier ,  Clemens Lamberth ,  Stephan Trah

    IPC分类号： A01N43/46 ,  A01P3/00 ,  C07D403/04

    CPC分类号： C07D233/88

    摘要： The present invention relates to novel imidazole derivatives of formula (I) having microbiocidal, in particular fungicidal, activity, to processes for their preparation and intermediates used in their preparation, to agrochemical compositions comprising them and to the use in agriculture or horticulture for controlling or preventing infestation of plants, harvested food crops, seeds or non-living materials by phytopathogenic microorganisms, preferably fungi.

    摘要翻译： 本发明涉及式（I）的新型咪唑衍生物，其具有杀微生物，特别是杀真菌活性，其制备方法和用于其制备的中间体，包含它们的农用化学组合物以及在农业或园艺中用于控制或 通过植物病原微生物，优选真菌预防植物，收获的食物作物，种子或非生物材料的侵染。