FUNGICIDAL COMPOUNDS AND COMPOSITIONS
    1.
    发明申请
    FUNGICIDAL COMPOUNDS AND COMPOSITIONS 审中-公开
    杀真菌化合物和组合物

    公开(公告)号:US20100016339A1

    公开(公告)日:2010-01-21

    申请号:US12375839

    申请日:2007-07-30

    CPC分类号: C07D237/12 A01N43/58

    摘要: The present invention relates, inter alia, to a compound having the formula (I):—wherein (R)n is selected from the group consisting of 4-Br, 4-OCH2CH3, 4-OCH2CF3, 2-CH3-4-Cl, 2-CH3-4-OCH3, 2-CH3-4-OCF3, 2-F-4-Br, 2-F-4-CF3, 3-CH3-4-Br, 3-F-4-Cl, 3-F-4-CH3, 3-F-4-Br, 3-F-4-OCH3 and 3-F-4-F. The present invention further relates to a fungicidal composition comprising a compound having the formula (I)—and also to fungicidal compositions comprising compounds having the formula (II) and/or (III): Furthermore, the present invention relates to methods for controlling pathogenic organisms using the compositions.

    摘要翻译: 本发明特别涉及具有式(I)的化合物:其中(R)n选自4-Br,4-OCH2CH3,4-OCH2CF3,2-CH3-4-Cl ,2-CH3-4-OCH3,2-CH3-4-OCF3,2-F-4-Br,2-F-4-CF3,3-CH3-4-Br,3-F-4-Cl,3 -F-4-CH 3,3-F-4-Br,3-F-4-OCH 3和3-F-4-F。 本发明还涉及包含具有式(I)的化合物的杀真菌组合物,还涉及包含具有式(II)和/或(III)的化合物的杀真菌组合物:此外,本发明涉及控制致病性的方法 使用组合物的生物体。

    NOVEL PYRIDAZINE DERIVATIVES
    2.
    发明申请
    NOVEL PYRIDAZINE DERIVATIVES 审中-公开
    新的吡咯烷酮衍生物

    公开(公告)号:US20100029668A1

    公开(公告)日:2010-02-04

    申请号:US12374052

    申请日:2007-07-16

    IPC分类号: A01N43/58 C07D405/04 A01P3/00

    摘要: The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is hydrogen, C1-C6alkyl, C1-C6haloalkyl or C3-C6cycloalkyl; R2 is an optionally substituted heteroaryl; R3 is an optionally substituted heteroaryl; and R4 is hydrogen, halogen, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy, C1-C6haloalkoxy, hydroxy or cyano; or an agrochemically usable salt form thereof.

    摘要翻译: 本发明涉及具有杀微生物活性,特别是杀真菌活性的活性成分的式(I)的新哒嗪衍生物,其中R1是氢,C1-C6烷基,C1-C6卤代烷基或C3-C6环烷基; R2是任选取代的杂芳基; R3是任选取代的杂芳基; R4是氢,卤素,C1-C6烷基,C1-C6卤代烷基,C1-C6烷氧基,C1-C6卤代烷氧基,羟基或氰基; 或其农业化学上可用的盐形式。

    PYRIDAZINE DERIVATIVES USEFUL AS FUNGICIDES AND FOR THE TREATMENT OF CANCER
    3.
    发明申请
    PYRIDAZINE DERIVATIVES USEFUL AS FUNGICIDES AND FOR THE TREATMENT OF CANCER 审中-公开
    用作杀真菌剂和治疗癌症的吡咯烷酮衍生物

    公开(公告)号:US20100273804A1

    公开(公告)日:2010-10-28

    申请号:US12809604

    申请日:2008-12-19

    摘要: The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: formula (I) wherein R1 is C1-C6alkyl, C1-C6haloalkyl or C3-C6cycloalkyl; R2 is hydrogen or an optionally substituted alkyl, aryl or heteroaryl; R3 is hydrogen, C1-C6alkyl or C1-C6haloalkyl; R4 is hydrogen, C1-C6alkyl or C1-C6haloalkyl; or R3 and R4 together can be part of a carbocyclic or heterocyclic 3- to 8-membered ring; R5 is optionally substituted aryl or heteroaryl; and R6 is hydroxy, halogen, C1-C6alkoxy, C1-C6haloalkoxy, C1-C6alkylthio or C1-C6haloalkylthio; or an agrochemically usable salt form thereof.

    摘要翻译: 本发明涉及具有杀微生物活性,特别是杀真菌活性的作为活性成分的式(I)的新哒嗪衍生物:式(I)其中R 1是C 1 -C 6烷基,C 1 -C 6卤代烷基或C 3 -C 6环烷基; R 2是氢或任选取代的烷基,芳基或杂芳基; R3是氢,C1-C6烷基或C1-C6卤代烷基; R4是氢,C1-C6烷基或C1-C6卤代烷基; 或者R 3和R 4一起可以是碳环或杂环的3至8元环的一部分; R5是任选取代的芳基或杂芳基; R 6为羟基,卤素,C 1 -C 6烷氧基,C 1 -C 6卤代烷氧基,C 1 -C 6烷硫基或C 1 -C 6卤代烷硫基; 或其农业化学上可用的盐形式。

    NOVEL IMIDAZOLE DERIVATIVES
    5.
    发明申请
    NOVEL IMIDAZOLE DERIVATIVES 审中-公开
    新咪唑衍生物

    公开(公告)号:US20110311649A1

    公开(公告)日:2011-12-22

    申请号:US12739852

    申请日:2008-10-24

    摘要: The present invention relates to novel imidazole derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is halogen, C1-C4alkyl or C1-C4haloalkyl; R2 is an optionally substituted aryl or heteroaryl; R3 is halogen; R4 is hydrogen, halogen, C1-C4alkyl, C1-C4haloalkyl, hydroxyl, C1-C4alkoxy, OR6, C1-C4haloalkoxy or cyano; R5 is halogen; R6 is hydrogen, C3-C7 cycloalkyl, C3-C10 alkylcycloalkyl, C1-C6 haloalkyl, C2-C6 alkenyl, C2-C6 haloalkenyl, C3-C7 cycloalkenyl, C2-C6 alkynyl, C2-C6 haloalkynyl or C2-C6 alkyloxyalkyl; X is N or C(R); and R is hydrogen, halogen, C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy or cyano; or an agrochemically usable salt form thereof; provided that when X is C(R), R2 cannot be an optionally substituted aryl.

    摘要翻译: 本发明涉及式(I)的新咪唑衍生物作为具有杀微生物活性,特别是杀真菌活性的活性成分:其中R1是卤素,C1-C4烷基或C1-C4卤代烷基; R2是任选取代的芳基或杂芳基; R3是卤素; R4是氢,卤素,C1-C4烷基,C1-C4卤代烷基,羟基,C1-C4烷氧基,OR6,C1-C4卤代烷氧基或氰基; R5是卤素; R6是氢,C3-C7环烷基,C3-C10烷基环烷基,C1-C6卤代烷基,C2-C6烯基,C2-C6卤代烯基,C3-C7环烯基,C2-C6炔基,C2-C6卤代炔基或C2-C6烷氧基烷基; X是N或C(R); 且R为氢,卤素,C 1 -C 4烷基,C 1 -C 4卤代烷基,C 1 -C 4烷氧基,C 1 -C 4卤代烷氧基或氰基; 或其农业化学可用的盐形式; 条件是当X是C(R)时,R 2不能是任选取代的芳基。

    Pyridazine fungicides
    6.
    发明授权
    Pyridazine fungicides 失效
    哒嗪类杀菌剂

    公开(公告)号:US08410026B2

    公开(公告)日:2013-04-02

    申请号:US12863377

    申请日:2009-01-14

    CPC分类号: C07D401/04

    摘要: The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is methyl, ethyl or isopropyl; R2 is chloro, fluoro, hydroxy or C1-C2alkoxy; R3 is H, chloro, fluoro, methoxy or C1-C3alkyl; R4 is chloro, fluoro or bromo; and R5 is H, fluoro or methoxy; or an agrochemically usable salt form thereof; with the proviso that when R1 is methyl, R2 is chloro and R3 is H, then R4 or R5 is different from fluoro.

    摘要翻译: 本发明涉及式(I)的新的哒嗪衍生物作为具有杀微生物活性的活性成分,特别是杀真菌活性:其中R1是甲基,乙基或异丙基; R 2是氯,氟,羟基或C 1 -C 2烷氧基; R3是H,氯,氟,甲氧基或C1-C3烷基; R4是氯,氟或溴; R5为H,氟或甲氧基; 或其农业化学可用的盐形式; 条件是当R 1为甲基时,R 2为氯且R 3为H,则R 4或R 5不同于氟。