公开(公告)号：US20060270726A1

公开(公告)日：2006-11-30

申请号：US10554328

申请日：2004-04-27

申请人： George Theodoridis ,  Edward Barron ,  John Lyga ,  Y. Zhang ,  Ping Ding ,  Frank Zawacki ,  Daniel Cohen ,  Matthew Whiteside

发明人： George Theodoridis ,  Edward Barron ,  John Lyga ,  Y. Zhang ,  Ping Ding ,  Frank Zawacki ,  Daniel Cohen ,  Matthew Whiteside

IPC分类号： A01N43/56 ,  A01N43/50 ,  C07D233/54 ,  C07D231/44

CPC分类号： A01N43/30 ,  A01N43/32 ,  A01N43/40 ,  A01N43/60 ,  A01N47/16 ,  C07D211/22 ,  C07D307/79 ,  C07D307/83 ,  C07D311/04 ,  C07D401/04 ,  C07D495/10

摘要： Certain novel phenyl substituted cyclic derivatives have unexpected insecticidal activity. These compounds are represented by formula I: where B is a cyclic bridging group containing at least one N or N oxide link and a, A, b, B, c, d, D, L, M, R1 through R9, inclusively, and R13, R14 and R15 are fully described herein. In addition, novel intermediates useful in preparing compounds of Formula I, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 某些新的苯基取代的环状衍生物具有出人意料的杀虫活性。 这些化合物由式I表示：其中B是含有至少一个N或N氧化物键的环状桥连基团，A，b，B，c，d，D，L，M，R 1， 包括R 9，R 14，R 14和R 15在本文中被完整描述。 此外，可用于制备式I化合物的新型中间体，包含杀虫有效量的至少一种式I化合物的组合物，以及任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体 也披露; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US20060094776A1

公开(公告)日：2006-05-04

申请号：US11292023

申请日：2005-12-01

申请人： George Theodoridis ,  Edward Barron ,  Dominic Suarez ,  Y. Zhang ,  Ping Ding ,  David Roush ,  Stephen Donovan ,  Frank Zawacki ,  Walter Yeager ,  John Lyga ,  Daniel Cohen

发明人： George Theodoridis ,  Edward Barron ,  Dominic Suarez ,  Y. Zhang ,  Ping Ding ,  David Roush ,  Stephen Donovan ,  Frank Zawacki ,  Walter Yeager ,  John Lyga ,  Daniel Cohen

IPC分类号： A01N43/16 ,  A01N43/08 ,  C07D311/04 ,  C07D307/87

CPC分类号： A01N43/30 ,  A01N43/32 ,  A01N43/40 ,  A01N43/60 ,  A01N47/16 ,  C07D211/22 ,  C07D307/79 ,  C07D307/83 ,  C07D311/04 ,  C07D401/04 ,  C07D495/10

摘要： Insecticidal (dihalopropenyl) phenylalkyl substituted dihydrobenzofuran and dihydrobenzopyran derivatives of Formula I are disclosed. These compounds provide unexpected insecticidal activity across a spectrum of insect pests combined with desirable physical properties including improved photostability. wherein x and y are integers independently selected from 0 or 1; and B is a bridging group *—(CR16R17)q—(CR18R19)r—(CR20R21)s-Lt-(CR22R23)u—(CR24R25)v—(CR26R27)w—, where the asterisk denotes attachment at A; and q, r, s, u, v and w are integers independently selected from 0, 1 and 2; and t is an integer selected from 0 and 1. A, D, E, G, M, R through R11, and R16 through R27, inclusively, are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I and methods of controlling insects by applying said compositions to a locus where insects are present or are expected to be present are also disclosed.

摘要翻译： 公开了杀虫（二卤代丙烯基）苯基烷基取代的二氢苯并呋喃和式I的二氢苯并吡喃衍生物。 这些化合物在一系列昆虫害虫中提供了意想不到的杀虫活性，并结合所需的物理性质，包括改善的光稳定性。 其中x和y是独立地选自0或1的整数; 并且B是桥接基团<？in-line-formula description =“In-line Formulas”end =“lead”？> * - （CR ^{16 17 ） - （CR 20） - （CR 20） - （CR 20） - （CR 20） - （CR 22）23 - - - （CR 22）23 （CR 26）25（ - ） - （CR 26）25 ） q，r，s，u，v和w是独立地选自0,1和2的整数; A，D，E，G，M，R至R 11和R 16至R 27中的一个整数。 / SUP>，包括这里完全描述。 此外，还公开了包含杀虫有效量的至少一种式I化合物的组合物和通过将所述组合物施用于存在昆虫或预期存在的场所来控制昆虫的方法。}

公开(公告)号：US20060247283A1

公开(公告)日：2006-11-02

申请号：US10554347

申请日：2004-04-28

申请人： George Theodoridis ,  Edward Barron ,  Dominic Suarer ,  Y. Zhang ,  Ping Ding ,  John Lyga ,  Mathew Whiteside ,  Frank Zawacki

发明人： George Theodoridis ,  Edward Barron ,  Dominic Suarer ,  Y. Zhang ,  Ping Ding ,  John Lyga ,  Mathew Whiteside ,  Frank Zawacki

IPC分类号： A01N43/82 ,  A01N43/76 ,  A01N43/56 ,  A01N43/78 ,  A01N43/50 ,  C07D417/02 ,  C07D405/02 ,  C07D413/02

CPC分类号： A01N43/30 ,  A01N43/32 ,  A01N43/40 ,  A01N43/60 ,  A01N47/16 ,  C07D211/22 ,  C07D307/79 ,  C07D307/83 ,  C07D311/04 ,  C07D401/04 ,  C07D495/10

摘要： Certain novel (dihalopropenyl)phenylalkyl substituted benzodioxolane and benzodioxane derivatives have provided unexpected insecticidal activity. These compounds are represented by formula I: where R through R10, inclusively, x, A, B, y, D, E, G and M are fully described herein. Preferred compounds of the present invention are those wherein the benzofused ring moiety is attached to the remainder of the molecule at the positions designated as 1- or 2-. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 某些新的（二卤代丙烯基）苯基烷基取代的苯并二氧杂环戊烷和苯并二恶烷衍生物提供了意想不到的杀虫活性。 这些化合物由式I表示：其中R至R 10，包括x，A，B，y，D，E，G和M在本文中被完整描述。 本发明优选的化合物是其中苯并稠环部分在指定为1-或2-的位置连接到分子的其余部分的化合物。 此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US20050171356A1

公开(公告)日：2005-08-04

申请号：US10510331

申请日：2004-04-28

申请人： George Theodoridis ,  Edward Barron ,  Dominic Suarez ,  Y. Larry Zhang ,  Ping Ding ,  John Lyga ,  Matthew Whiteside

发明人： George Theodoridis ,  Edward Barron ,  Dominic Suarez ,  Y. Larry Zhang ,  Ping Ding ,  John Lyga ,  Matthew Whiteside

IPC分类号： A01N43/30 ,  A01N43/32 ,  C07D307/79 ,  C07D307/83 ,  C07D311/04 ,  C07D495/10 ,  C07D277/82

CPC分类号： A01N43/30 ,  A01N43/32 ,  A01N43/40 ,  A01N43/60 ,  A01N47/16 ,  C07D211/22 ,  C07D307/79 ,  C07D307/83 ,  C07D311/04 ,  C07D401/04 ,  C07D495/10

摘要： Certain novel (dihalopropenyl)phenylalkyl substituted benzoxazole and benzothiazole derivatives have unexpected insecticidal activity. These compounds are represented by formula (I): where R through R11, inclusively. x, A, B, y, D, E and G are fully described herein. Preferred compounds of the present invention are those wherein the benzo-fused ring moiety is attached to the remainder of the molecule at the positions designated as (5) or (6) and where R11 is either C1-C3 alkyl or halo C1-C3 alkyl. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula (I), and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 某些新的（二卤代丙烯基）苯基烷基取代的苯并恶唑和苯并噻唑衍生物具有出人意料的杀虫活性。 这些化合物由式（I）表示：其中R 1至R 11包括。 这里完整地描述了x，A，B，y，D，E和G。 本发明优选的化合物是其中苯并稠环部分在（5）或（6）表示的位置连接到分子的其余部分，其中R 11是C < C 1 -C 3烷基或卤素C 1 -C 3烷基。 此外，还公开了包含杀虫有效量的至少一种式（I）化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US20080090828A1

公开(公告)日：2008-04-17

申请号：US11874015

申请日：2007-10-17

申请人： Ping Ding ,  Robert Henrie ,  Daniel Cohen ,  John Lyga ,  David Rosen ,  George Theodoridis ,  Qun Zhang ,  Walter Yeager ,  Stephen Donovan ,  Stephen Zhang ,  Inna Shulman ,  Seong Yu ,  Guozhi Wang ,  Y. Zhang ,  Ariamala Gopalsamy ,  Dennis Warkentin ,  Paul Rensner ,  Ian Silverman ,  Thomas Cullen

发明人： Ping Ding ,  Robert Henrie ,  Daniel Cohen ,  John Lyga ,  David Rosen ,  George Theodoridis ,  Qun Zhang ,  Walter Yeager ,  Stephen Donovan ,  Stephen Zhang ,  Inna Shulman ,  Seong Yu ,  Guozhi Wang ,  Y. Zhang ,  Ariamala Gopalsamy ,  Dennis Warkentin ,  Paul Rensner ,  Ian Silverman ,  Thomas Cullen

IPC分类号： C07D453/02 ,  A61K31/4745 ,  A61K31/50

CPC分类号： C07D405/14 ,  A01N43/40 ,  A01N43/54 ,  A01N43/713 ,  C07D211/14 ,  C07D211/18 ,  C07D211/22 ,  C07D211/24 ,  C07D211/26 ,  C07D211/28 ,  C07D211/32 ,  C07D211/94 ,  C07D401/06 ,  C07D401/10 ,  C07D401/12 ,  C07D401/14 ,  C07D413/12 ,  C07D417/12 ,  C07D451/14 ,  C07D513/04

摘要： It has now been found that certain novel N-(substituted aryl)-4-(disubstituted methyl)piperidine and pyridine derivatives have provided unexpected insecticidal activity. These compounds are represented by formula (I): wherein m, n, q, r, and s are independently selected from 0 or 1; and p is 0, 1, 2, or 3; A is C or CH; and B, D, E, R, R1, R2, R3, R4, R5, R6, R7 and R8 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 现在已经发现某些新的N-（取代的芳基）-4-（二取代的甲基）哌啶和吡啶衍生物提供了意想不到的杀虫活性。 这些化合物由式（I）表示：其中m，n，q，r和s独立地选自0或1; 且p为0,1,2或3; A是C或CH; 和B，D，E，R，R 1，R 2，R 3，R 4，R 本文中充分描述了本发明的第5，第6，第七和第八和第八。 此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US20060135504A1

公开(公告)日：2006-06-22

申请号：US10538998

申请日：2003-12-08

申请人： Ping Ding ,  Robert Henrie II ,  Daniel Cohen ,  John Lyga ,  David Rosen ,  George Theodoridis ,  Qun Zhang ,  Walter Yeager ,  Stephen Donovan ,  Steven Zhang ,  Inna Shulman ,  Seong Yu ,  Guozhi Wang ,  Y. Larry Zhang ,  Araimala Gopalsamy ,  Dennis Warkentin ,  Paul Rensner ,  Ian Silverman ,  Thomas Cullen

发明人： Ping Ding ,  Robert Henrie II ,  Daniel Cohen ,  John Lyga ,  David Rosen ,  George Theodoridis ,  Qun Zhang ,  Walter Yeager ,  Stephen Donovan ,  Steven Zhang ,  Inna Shulman ,  Seong Yu ,  Guozhi Wang ,  Y. Larry Zhang ,  Araimala Gopalsamy ,  Dennis Warkentin ,  Paul Rensner ,  Ian Silverman ,  Thomas Cullen

IPC分类号： A61K31/397 ,  C07D213/63 ,  C07D205/10

CPC分类号： C07D405/14 ,  A01N43/40 ,  A01N43/54 ,  A01N43/713 ,  C07D211/14 ,  C07D211/18 ,  C07D211/22 ,  C07D211/24 ,  C07D211/26 ,  C07D211/28 ,  C07D211/32 ,  C07D211/94 ,  C07D401/06 ,  C07D401/10 ,  C07D401/12 ,  C07D401/14 ,  C07D413/12 ,  C07D417/12 ,  C07D451/14 ,  C07D513/04

摘要： It has now been found that certain novel N-(substituted aryl)-4(disubstituted methyl)piperidine and pyridine derivatives have provided unexpected insecticidal activity. These compounds are represented by formula (I): wherein m, n, q, r, and s are independently selected from 0 or 1; and p is 0, 1, 2, or 3; A is C or CH; and B, D, E, R, R1, R2, R3, R4, R5, R6, R7 and R8 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 现在已经发现，某些新的N-（取代的芳基）-4（二取代的甲基）哌啶和吡啶衍生物已经提供了意想不到的杀虫活性。 这些化合物由式（I）表示：其中m，n，q，r和s独立地选自0或1; 且p为0,1,2或3; A是C或CH; 和B，D，E，R，R 1，R 2，R 3，R 4，R 本文中充分描述了本发明的第5，第6，第七和第八和第八。 此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US07671201B2

公开(公告)日：2010-03-02

申请号：US10554328

申请日：2004-04-27

申请人： George Theodoridis ,  Edward J. Barron ,  John W. Lyga ,  Y. Larry Zhang ,  Ping Ding ,  Frank J. Zawacki ,  Daniel H. Cohen ,  Matthew P. Whiteside

发明人： George Theodoridis ,  Edward J. Barron ,  John W. Lyga ,  Y. Larry Zhang ,  Ping Ding ,  Frank J. Zawacki ,  Daniel H. Cohen ,  Matthew P. Whiteside

IPC分类号： C07D241/00 ,  C07D211/68 ,  C07D401/00 ,  A01N25/00

CPC分类号： A01N43/30 ,  A01N43/32 ,  A01N43/40 ,  A01N43/60 ,  A01N47/16 ,  C07D211/22 ,  C07D307/79 ,  C07D307/83 ,  C07D311/04 ,  C07D401/04 ,  C07D495/10

摘要： Certain novel phenyl substituted cyclic derivatives have unexpected insecticidal activity. These compounds are represented by formula I: where B is a cyclic bridging group containing at least one N or N oxide link and a, A, b, B, c, d, D, L, M, R1 through R9, inclusively, and R13, R14 and R15 are fully described herein. In addition, novel intermediates useful in preparing compounds of Formula I, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 某些新的苯基取代的环状衍生物具有出人意料的杀虫活性。 这些化合物由式I表示：其中B是含有至少一个N或N氧化物连接的环状桥连基团和a，A，b，B，c，d，D，L，M，R 1至R 9，包括和 R13，R14和R15在此完全描述。 此外，可用于制备式I化合物的新型中间体，包含杀虫有效量的至少一种式I化合物的组合物，以及任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体 也披露; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US06987194B2

公开(公告)日：2006-01-17

申请号：US10832624

申请日：2004-04-27

申请人： George Theodoridis ,  Edward J. Barron ,  Dominic P. Suarez ,  Y. Larry Zhang ,  Ping Ding ,  David M. Roush ,  Stephen F. Donovan ,  Frank J. Zawacki ,  Walter H. Yeager ,  John W. Lyga ,  Daniel H. Cohen

发明人： George Theodoridis ,  Edward J. Barron ,  Dominic P. Suarez ,  Y. Larry Zhang ,  Ping Ding ,  David M. Roush ,  Stephen F. Donovan ,  Frank J. Zawacki ,  Walter H. Yeager ,  John W. Lyga ,  Daniel H. Cohen

IPC分类号： C07D307/83 ,  C07D311/04 ,  A61K31/343 ,  A61K31/353

CPC分类号： A01N43/30 ,  A01N43/32 ,  A01N43/40 ,  A01N43/60 ,  A01N47/16 ,  C07D211/22 ,  C07D307/79 ,  C07D307/83 ,  C07D311/04 ,  C07D401/04 ,  C07D495/10

摘要： Insecticidal (dihalopropenyl) phenylalkyl substituted dihydrobenzofuran and dihydrobenzopyran derivatives of Formula I are disclosed. These compounds provide unexpected insecticidal activity across a spectrum of insect pests combined with desirable physical properties including improved photostability. wherein x and y are integers independently selected from 0 or 1; and B is a bridging group *—(CR16R17)q—(CR18R19)r—(CR20R21)s—Lt—(CR22R23)u—(CR24R25)v—(CR26R27)w—, where the asterisk denotes attachment at A; and q, r, s, u, v and w are integers independently selected from 0, 1 and 2; and t is an integer selected from 0 and 1. A, D, E, G, M, R through R11, and R16 through R27, inclusively, are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I and methods of controlling insects by applying said compositions to a locus where insects are present or are expected to be present are also disclosed.

摘要翻译： 公开了杀虫（二卤代丙烯基）苯基烷基取代的二氢苯并呋喃和式I的二氢苯并吡喃衍生物。 这些化合物在一系列昆虫害虫中提供了意想不到的杀虫活性，并结合所需的物理性质，包括改善的光稳定性。 其中x和y是独立地选自0或1的整数; 并且B是桥接基团<？in-line-formula description =“In-line Formulas”end =“lead”？> * - （CR ^{16 17 ） - （CR 20） - （CR 20） - （CR 20） - （CR 20） - （CR 22）23 - - - （CR 22）23 （CR 26）25（ - ） - （CR 26）25 ） q，r，s，u，v和w是独立地选自0,1和2的整数; A，D，E，G，M，R至R 11和R 16至R 27中的一个整数。 / SUP>，包括这里完全描述。 此外，还公开了包含杀虫有效量的至少一种式I化合物的组合物和通过将所述组合物施用于存在昆虫或预期存在的场所来控制昆虫的方法。}

公开(公告)号：US07683070B2

公开(公告)日：2010-03-23

申请号：US11874015

申请日：2007-10-17

申请人： Ping Ding ,  Robert N. Henrie, II ,  Daniel H. Cohen ,  John W. Lyga ,  David S. Rosen ,  George Theodoridis ,  Qun Zhang ,  Walter H. Yeager ,  Stephen F. Donovan ,  Stephen Shunxiang Zhang ,  Inna Shulman ,  Seong Jae Yu ,  Guozhi Wang ,  Y. Larry Zhang ,  Ariamala Gopalsamy ,  Dennis L. Warkentin ,  Paul E. Rensner ,  Ian R. Silverman ,  Thomas G. Cullen

发明人： Ping Ding ,  Robert N. Henrie, II ,  Daniel H. Cohen ,  John W. Lyga ,  David S. Rosen ,  George Theodoridis ,  Qun Zhang ,  Walter H. Yeager ,  Stephen F. Donovan ,  Stephen Shunxiang Zhang ,  Inna Shulman ,  Seong Jae Yu ,  Guozhi Wang ,  Y. Larry Zhang ,  Ariamala Gopalsamy ,  Dennis L. Warkentin ,  Paul E. Rensner ,  Ian R. Silverman ,  Thomas G. Cullen

IPC分类号： A61K31/4523 ,  A61K31/4545 ,  C07D211/06 ,  C07D239/02

CPC分类号： C07D405/14 ,  A01N43/40 ,  A01N43/54 ,  A01N43/713 ,  C07D211/14 ,  C07D211/18 ,  C07D211/22 ,  C07D211/24 ,  C07D211/26 ,  C07D211/28 ,  C07D211/32 ,  C07D211/94 ,  C07D401/06 ,  C07D401/10 ,  C07D401/12 ,  C07D401/14 ,  C07D413/12 ,  C07D417/12 ,  C07D451/14 ,  C07D513/04

摘要： It has now been found that certain novel N-(substituted aryl)-4-(disubstituted methyl)piperidine and pyridine derivatives have provided unexpected insecticidal activity. These compounds are represented by formula (I): wherein m, n, q, r, and s are independently selected from 0 or 1; and p is 0, 1, 2, or 3; A is C or CH; and B, D, E, R, R1, R2, R3, R4, R5, R6, R7 and R8 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 现在已经发现某些新的N-（取代的芳基）-4-（二取代的甲基）哌啶和吡啶衍生物提供了意想不到的杀虫活性。 这些化合物由式（I）表示：其中m，n，q，r和s独立地选自0或1; 且p为0,1,2或3; A是C或CH; 本文完整地描述了B，D，E，R，R 1，R 2，R 3，R 4，R 5，R 6，R 7和R 8。 此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

公开(公告)号：US07576224B2

公开(公告)日：2009-08-18

申请号：US11292023

申请日：2005-12-01

申请人： George Theodoridis ,  Edward J. Barron ,  Dominic P. Suarez ,  Y. Larry Zhang ,  Ping Ding ,  David M. Roush ,  Stephen F. Donovan ,  Frank J. Zawacki ,  Walter H. Yeager ,  John W. Lyga ,  Daniel H. Cohen

发明人： George Theodoridis ,  Edward J. Barron ,  Dominic P. Suarez ,  Y. Larry Zhang ,  Ping Ding ,  David M. Roush ,  Stephen F. Donovan ,  Frank J. Zawacki ,  Walter H. Yeager ,  John W. Lyga ,  Daniel H. Cohen

IPC分类号： C07D307/80 ,  C07D495/10

CPC分类号： A01N43/30 ,  A01N43/32 ,  A01N43/40 ,  A01N43/60 ,  A01N47/16 ,  C07D211/22 ,  C07D307/79 ,  C07D307/83 ,  C07D311/04 ,  C07D401/04 ,  C07D495/10

摘要： Insecticidal (dihalopropenyl) phenylalkyl substituted dihydrobenzofuran and dihydrobenzopyran derivatives of Formula I are disclosed. These compounds provide unexpected insecticidal activity across a spectrum of insect pests combined with desirable physical properties including improved photostability. wherein x and y are integers independently selected from 0 or 1; and B is a bridging group *—(CR16R17)q—(CR18R19)r—(CR20R21)s-Lt-(CR22R23)u—(CR24R25)v—(CR26R27)w—, where the asterisk denotes attachment at A; and q, r, s, u, v and w are integers independently selected from 0, 1 and 2; and t is an integer selected from 0 and 1. A, D, E, G, M, R through R11, and R16 through R27, inclusively, are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I and methods of controlling insects by applying said compositions to a locus where insects are present or are expected to be present are also disclosed.

摘要翻译： 公开了杀虫（二卤代丙烯基）苯基烷基取代的二氢苯并呋喃和式I的二氢苯并吡喃衍生物。 这些化合物在一系列昆虫害虫中提供了意想不到的杀虫活性，并结合所需的物理性质，包括改善的光稳定性。 其中x和y是独立地选自0或1的整数; * - （CR16R17）q-（CR18R19）r-（CR20R21）s-Lt-（CR22R23），而B是桥接基团<？in-line-formula description =“In-line Formulas”end =“lead” u-（CR24R25）v-（CR26R27）w - ，<？在线公式描述=“在线公式”end =“tail”？>其中星号表示在A附近; q，r，s，u，v和w是独立地选自0,1和2的整数; 并且t是选自0和1的整数。本文充分描述了A，D，E，G，M，R至R 11和R 16至R 27。 此外，还公开了包含杀虫有效量的至少一种式I化合物的组合物和通过将所述组合物施用于存在昆虫或预期存在的场所来控制昆虫的方法。