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    Heterocyclic amide derivatives useful as microbiocides
    3.
    发明授权
    Heterocyclic amide derivatives useful as microbiocides 有权
    用作杀微生物剂的杂环酰胺衍生物

    公开(公告)号：US08183416B2

    公开(公告)日：2012-05-22

    申请号：US12765929

    申请日：2010-04-23

    申请人： Hans Tobler ,  Harald Walter ,  Josef Ehrenfreund ,  Camilla Corsi

    发明人： Hans Tobler ,  Harald Walter ,  Josef Ehrenfreund ,  Camilla Corsi

    IPC分类号： C07C205/06

    CPC分类号： C07C205/06 ,  A01N43/32 ,  A01N43/36 ,  A01N43/40 ,  A01N43/56 ,  A01N43/647 ,  A01N43/76 ,  A01N43/78 ,  C07C205/11 ,  C07C205/12 ,  C07C205/37 ,  C07C205/45 ,  C07C211/61 ,  C07C2603/66 ,  C07D207/34 ,  C07D207/46 ,  C07D213/89 ,  C07D231/14 ,  C07D249/04 ,  C07D263/34 ,  C07D277/56 ,  C07D327/06

    摘要： The invention relates to a fungicidally active compound of formula (I): where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by the groups R6, R7 and R8; R1 is hydrogen, C1-4 alkyl, C1-4 haloalkyl, C1-4alkoxy, C1-4haloalkoxy, CH2C≡CR9, CH2CR10═CHR11, CH═C═CH2 or COR12; R2 and R3 are each, independently, hydrogen, halo, C1-4 alkyl, C1-4 alkoxy, C1-4 haloalkyl or C1-4 haloalkoxy; R4 and R5 are each independently selected from halo, cyano and nitro; or one of R4 and R5 is hydrogen and the other is selected from halo, cyano and nitro; R6, R7 and R8 are each, independently, hydrogen, halo, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy(C1-4)alkyl, C1-4haloalkoxy(C1-4)alkyl or C1-4haloalkoxy, provided that at least one of R6, R7 and R8 is not hydrogen; R9, R10 and R11 are each, independently, hydrogen, halo, C1-4 alkyl, C1-4 haloalkyl or C1-4 alkoxy(C1-4)alkyl; and R12 is hydrogen, C1-6 alkyl, C1-6haloalkyl, C1-4 alkoxy(C1-4)alkyl, C1-4 alkylthio(C1-4)-alkyl, C1-4 alkoxy or aryl; to the preparation of these compounds, to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient, to the preparation of the compositions mentioned and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.

    摘要翻译： 本发明涉及式（I）的杀真菌活性化合物：其中Het是含有一至三个杂原子的5-或6-元杂环，各自独立地选自氧，氮和硫，该环被R6基团取代 ，R7和R8; R 1是氢，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基，C 1-4卤代烷氧基，CH 2C≡CR9，CH 2 CR 10 = CHR 11，CH = C = CH 2或COR 12; R 2和R 3各自独立地为氢，卤素，C 1-4烷基，C 1-4烷氧基，C 1-4卤代烷基或C 1-4卤代烷氧基; R4和R5各自独立地选自卤素，氰基和硝基; 或者R 4和R 5中的一个是氢，另一个选自卤素，氰基和硝基; R 6，R 7和R 8各自独立地为氢，卤素，氰基，硝基，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基（C 1-4）烷基，C 1-4卤代烷氧基（C 1-4）烷基或C 1 -4卤代烷氧基，条件是R 6，R 7和R 8中的至少一个不是氢; R 9，R 10和R 11各自独立地为氢，卤素，C 1-4烷基，C 1-4卤代烷基或C 1-4烷氧基（C 1-4）烷基; 并且R 12是氢，C 1-6烷基，C 1-6卤代烷基，C 1-4烷氧基（C 1-4）烷基，C 1-4烷硫基（C 1-4） - 烷基，C 1-4烷氧基或芳基; 涉及这些化合物的制备，用于制备这些化合物的新型中间体，包括至少一种新化合物作为活性成分的农用化学组合物，所述组合物的制备以及使用活性成分或 用于通过植物病原微生物，优选真菌控制或预防植物感染的农业或园艺成分。

    Process for the production of carboxanilides
    5.
    发明授权
    Process for the production of carboxanilides 有权
    生产甲酰苯胺的方法

    公开(公告)号：US07820830B2

    公开(公告)日：2010-10-26

    申请号：US12093619

    申请日：2006-11-13

    申请人： Harald Walter ,  Camilla Corsi ,  Josef Ehrenfreund ,  Hans Tobler

    发明人： Harald Walter ,  Camilla Corsi ,  Josef Ehrenfreund ,  Hans Tobler

    IPC分类号： C07D231/14

    CPC分类号： C07D231/14

    摘要： The present invention relates to a novel process for the preparation of a compound of general formula (I): wherein R1 is H or C1-4 alkyl and R2 is difluoromethyl or trifluoromethyl, which comprises reacting a compound of general formula (II): wherein R1 has the meaning given above and X is chloro or bromo, with a compound of general formula (III): wherein R2 has the meaning given above, in the presence of a base, a palladium catalyst and a ferrocenyl biphoshine ligand of the Josiphos type, the reaction being carried out in an ether solvent at a reflux temperature of at least 100° C.

    摘要翻译： 本发明涉及一种制备通式（I）化合物的新方法：其中R1是H或C1-4烷基，R2是二氟甲基或三氟甲基，其包括使通式（II）的化合物：其中 R1具有上面给出的含义，X是氯或溴，与通式（III）的化合物：其中R 2具有上面给出的含义，在碱存在下，钯催化剂和Josiphos型的二茂铁基二膦配体 ，反应在乙醚溶剂中在至少100℃的回流温度下进行。

    HETEROCYCLIC AMIDE DERIVATIVES USEFUL AS MICROBIOCIDES
    6.
    发明申请
    HETEROCYCLIC AMIDE DERIVATIVES USEFUL AS MICROBIOCIDES 有权
    杂环酰胺衍生物作为微生物有用

    公开(公告)号：US20100204482A1

    公开(公告)日：2010-08-12

    申请号：US12765929

    申请日：2010-04-23

    申请人： Hans Tobler ,  Harald Walter ,  Josef Ehrenfreund ,  Camilla Corsi

    发明人： Hans Tobler ,  Harald Walter ,  Josef Ehrenfreund ,  Camilla Corsi

    IPC分类号： C07C205/06 ,  C07D277/56

    CPC分类号： C07C205/06 ,  A01N43/32 ,  A01N43/36 ,  A01N43/40 ,  A01N43/56 ,  A01N43/647 ,  A01N43/76 ,  A01N43/78 ,  C07C205/11 ,  C07C205/12 ,  C07C205/37 ,  C07C205/45 ,  C07C211/61 ,  C07C2603/66 ,  C07D207/34 ,  C07D207/46 ,  C07D213/89 ,  C07D231/14 ,  C07D249/04 ,  C07D263/34 ,  C07D277/56 ,  C07D327/06

    摘要： The invention relates to a fungicidally active compound of formula (I): where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by the groups R6, R7 and R8; R1 is hydrogen, C1-4 alkyl, C1-4 haloalkyl, C1-4alkoxy, C1-4haloalkoxy, CH2C≡CR9, CH2CR10═CHR11, CH═C═CH2 or COR12; R2 and R3 are each, independently, hydrogen, halo, C1-4 alkyl, C1-4 alkoxy, C1-4 haloalkyl or C1-4 haloalkoxy; R4 and R5 are each independently selected from halo, cyano and nitro; or one of R4 and R5 is hydrogen and the other is selected from halo, cyano and nitro; R6, R7 and R8 are each, independently, hydrogen, halo, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy(C1-4)alkyl, C1-4haloalkoxy(C1-4)alkyl or C1-4haloalkoxy, provided that at least one of R6, R7 and R8 is not hydrogen; R9, R10 and R11 are each, independently, hydrogen, halo, C1-4 alkyl, C1-4 haloalkyl or C1-4 alkoxy(C1-4)alkyl; and R12 is hydrogen, C1-6 alkyl, C1-6haloalkyl, C1-4 alkoxy(C1-4)alkyl, C1-4 alkylthio(C1-4)-alkyl, C1-4 alkoxy or aryl; to the preparation of these compounds, to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient, to the preparation of the compositions mentioned and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.

    摘要翻译： 本发明涉及式（I）的杀真菌活性化合物：其中Het是含有一至三个杂原子的5-或6-元杂环，各自独立地选自氧，氮和硫，该环被R6基团取代 ，R7和R8; R 1是氢，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基，C 1-4卤代烷氧基，CH 2C≡CR9，CH 2 CR 10 = CHR 11，CH = C = CH 2或COR 12; R 2和R 3各自独立地是氢，卤素，C 1-4烷基，C 1-4烷氧基，C 1-4卤代烷基或C 1-4卤代烷氧基; R4和R5各自独立地选自卤素，氰基和硝基; 或者R4和R5之一是氢，另一个选自卤素，氰基和硝基; R 6，R 7和R 8各自独立地为氢，卤素，氰基，硝基，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基（C 1-4）烷基，C 1-4卤代烷氧基（C 1-4）烷基或C 1 -4卤代烷氧基，条件是R 6，R 7和R 8中的至少一个不是氢; R 9，R 10和R 11各自独立地为氢，卤素，C 1-4烷基，C 1-4卤代烷基或C 1-4烷氧基（C 1-4）烷基; 并且R 12是氢，C 1-6烷基，C 1-6卤代烷基，C 1-4烷氧基（C 1-4）烷基，C 1-4烷硫基（C 1-4） - 烷基，C 1-4烷氧基或芳基; 涉及这些化合物的制备，用于制备这些化合物的新型中间体，包括至少一种新化合物作为活性成分的农用化学组合物，所述组合物的制备以及使用活性成分或 用于通过植物病原微生物，优选真菌控制或预防植物感染的农业或园艺成分。

    Microbiocides
    7.
    发明授权
    Microbiocides 失效
    杀微生物剂

    公开(公告)号：US07723371B2

    公开(公告)日：2010-05-25

    申请号：US12092338

    申请日：2006-11-13

    申请人： Harald Walter ,  Camilla Corsi ,  Josef Ehrenfreund ,  Hans Tobler

    发明人： Harald Walter ,  Camilla Corsi ,  Josef Ehrenfreund ,  Hans Tobler

    IPC分类号： A01N43/56

    CPC分类号： A01N43/36 ,  A01N43/40 ,  A01N43/56 ,  A01N43/78 ,  A01N43/84 ,  C07C211/45 ,  C07C211/52 ,  C07C2601/02 ,  C07C2601/04 ,  C07D207/34 ,  C07D213/82 ,  C07D231/14 ,  C07D249/04 ,  C07D277/56 ,  C07D327/06

    摘要： The invention relates to a fungicidally active compound of the general Formula (I): where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by the groups R3, R4 and R5; R1 and R2 are independently H, halo, C1-4 alkyl or C1-4 haloalkyl; and R3, R4 and R5 are each, independently, H, halo, C1-4 alkyl, C1-4 haloalkyl or C1-4 haloalkoxy, provided that at least one of R3, R4 and R5 is not H; to the preparation of these compounds, to novel intermediates used in their preparation, to agrochemical compositions which comprise at least one of the novel compounds as an active ingredient, to the preparation of the compositions and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestations of plants by phytopathogenic microorganisms, especially fungi.

    摘要翻译： 本发明涉及通式（I）的杀真菌活性化合物：其中Het是含有一至三个杂原子的5-或6-元杂环，各自独立地选自氧，氮和硫，所述环被 基团R3，R4和R5; R 1和R 2独立地为H，卤素，C 1-4烷基或C 1-4卤代烷基; 并且R 3，R 4和R 5各自独立地为H，卤素，C 1-4烷基，C 1-4卤代烷基或C 1-4卤代烷氧基，条件是R 3，R 4和R 5中的至少一个不为H; 涉及这些化合物的制备，其制备中使用的新型中间体，包含至少一种新化合物作为活性成分的农用化学组合物，用于制备组合物以及在农业中使用活性成分或组合物 或园艺用于通过植物病原微生物，特别是真菌控制或预防植物侵染。

    Process for the Preparation of 4,4-Difluoro-3-Oxobutanoic Acid Esters
    9.
    发明申请
    Process for the Preparation of 4,4-Difluoro-3-Oxobutanoic Acid Esters 有权
    制备4,4-二氟-3-氧代丁酸酯的方法

    公开(公告)号：US20080004465A1

    公开(公告)日：2008-01-03

    申请号：US11572053

    申请日：2005-07-13

    申请人： Harald Walter ,  Camilla Corsi ,  Josef Ehrenfreund ,  Clemens Lamberth ,  Hans Tobler

    发明人： Harald Walter ,  Camilla Corsi ,  Josef Ehrenfreund ,  Clemens Lamberth ,  Hans Tobler

    IPC分类号： C07C69/66

    CPC分类号： C07C67/343 ,  C07C69/716

    摘要： The present invention relates to a process for the preparation of a compound of the formula (I), wherein R is C1-12 alkyl, by the contact of a compound of the general formula (II), wherein R1 and R2 are each, independently, C1-12 alkyl; or R1 and R2 join together with the nitrogen atom to which they are attached to form an alicyclic amine ring containing 4 to 7 carbon atoms or a morpholine ring, with an acetic acid ester of the general formula (III) CH3COOR, wherein R is as defined under formula (I), in the presence of a base.

    摘要翻译： 本发明涉及制备式（I）化合物的方法，其中R是C 1-12烷基，通过通式（II）的化合物与 其中R 1和R 2各自独立地为C 1-12烷基; 或R 1和R 2 2与它们所连接的氮原子一起形成含有4至7个碳原子的脂环族胺环或吗啉环，其中 （III）CH 3 COOR的乙酸酯，其中R如式（I）所定义，在碱的存在下。