NOVEL CRYSTALS OF PYRIMIDINE COMPOUND AND PROCESS FOR PRODUCING THE SAME
    2.
    发明申请
    NOVEL CRYSTALS OF PYRIMIDINE COMPOUND AND PROCESS FOR PRODUCING THE SAME 失效
    吡啶化合物的新型结晶及其制造方法

    公开(公告)号:US20090111986A1

    公开(公告)日:2009-04-30

    申请号:US12346544

    申请日:2008-12-30

    IPC分类号: C07D405/14 C07D405/02

    CPC分类号: C07D405/14 C07D405/06

    摘要: Crystals of 5-[2-amino-4-(2-furyl)pyrimidin-5-yl]-1-methylpyridin-2(1H)-one having a diffraction peak at a diffraction angle (2θ±0.2°) of 9.7° and/or 21.9° in a powder X-ray diffraction are suitable for an active ingredient of a preventing and therapeutic agent for diseases such as constipation. Crystals of 5-[2-amino-4-(2-furyl)pyrimidin-5-yl]-1-methylpyridin-2(1H)-one hydrate and amorphous 5-[2-amino-4-(2-furyl)pyrimidin-5-yl]-1-methylpyridin-2(1H)-one hydrate are also suitable for an active ingredient of a preventing and therapeutic agent for diseases such as constipation.

    摘要翻译: 在衍射角(2θ±0.2°)为9.7°的衍射峰的5- [2-氨基-4-(2-呋喃基)嘧啶-5-基] -1-甲基吡啶-2(1H) - 酮的晶体 和/或21.9°在粉末X射线衍射中适用于诸如便秘的疾病的预防和治疗剂的活性成分。 5- [2-氨基-4-(2-呋喃基)嘧啶-5-基] -1-甲基吡啶-2(1H) - 酮水合物和无定形的5- [2-氨基-4-(2-呋喃基) 嘧啶-5-基] -1-甲基吡啶-2(1H) - 酮水合物也适用于诸如便秘等疾病的预防和治疗剂的活性成分。

    Crystalline and amorphous pyrimidine compounds and processes for preparing pyrimidine compounds
    4.
    发明申请
    Crystalline and amorphous pyrimidine compounds and processes for preparing pyrimidine compounds 失效
    结晶和无定形嘧啶化合物及制备嘧啶化合物的方法

    公开(公告)号:US20070078151A1

    公开(公告)日:2007-04-05

    申请号:US11378307

    申请日:2006-03-20

    IPC分类号: A61K31/506 C07D405/14

    CPC分类号: C07D405/14 C07D405/06

    摘要: Crystals of 5-[2-amino-4-(2-furyl)pyrimidin-5-yl]-1-methylpyridin-2(1H)-one having a diffraction peak at a diffraction angle (2θ±0.2°) of 9.7° and/or 21.9° in a powder X-ray diffraction are suitable for an active ingredient of a preventing and therapeutic agent for diseases such as constipation. Crystals of 5-[2-amino-4-(2-furyl)pyrimidin-5-yl]-1-methylpyridin-2(1H)-one hydrate and amorphous 5-[2-amino-4-(2-furyl)pyrimidin-5-yl]-1-methylpyridin-2(1H)-one hydrate are also suitable for an active ingredient of a preventing and therapeutic agent for diseases such as constipation.

    摘要翻译: 在衍射角(2θ±0.2°)为9.7°的衍射峰的5- [2-氨基-4-(2-呋喃基)嘧啶-5-基] -1-甲基吡啶-2(1H) - 酮的晶体 和/或21.9°在粉末X射线衍射中适用于诸如便秘的疾病的预防和治疗剂的活性成分。 5- [2-氨基-4-(2-呋喃基)嘧啶-5-基] -1-甲基吡啶-2(1H) - 酮水合物和无定形的5- [2-氨基-4-(2-呋喃基) 嘧啶-5-基] -1-甲基吡啶-2(1H) - 酮水合物也适用于诸如便秘等疾病的预防和治疗剂的活性成分。

    Muscle training apparatus and belt for muscle training
    7.
    发明授权
    Muscle training apparatus and belt for muscle training 有权
    肌肉训练器械和肌肉训练带

    公开(公告)号:US08992397B2

    公开(公告)日:2015-03-31

    申请号:US12674839

    申请日:2008-08-19

    申请人: Yoshiaki Sato

    发明人: Yoshiaki Sato

    摘要: To ensure easy and secure placement of a belt for KAATSU muscle training on a target compressed site near the proximal portion of a limb.A belt 100B has a longer first band-shaped member 110 and a shorter second band-shaped member 120 both of which have a band shape and are connected to a ring-shaped joint member 130 at their respective ends. In order to place the belt 100B on the target compressed site, the limb (right leg in this case) on which the belt 100B is expected to be placed is inserted into a loop of the first band-shaped member 110 formed by passing the end of the first band-shaped member 110 through an opening in the joint member 130, and the belt is moved up to the target compressed site. Then, the first band-shaped member 110 and the second band-shaped member 120 are pulled with both hands in the opposite directions. The belt 100B is placed on the target compressed site with the belt 100B being tensioned appropriately.

    摘要翻译: 为了确保在肢体近端部位附近的目标压缩部位上容易且安全地放置用于KAATSU肌肉训练的腰带。 带100B具有较长的第一带状构件110和较短的第二带状构件120,它们都具有带状并且在它们各自的端部处连接到环形接头构件130。 为了将皮带100B放置在目标压缩部位上,期望将皮带100B放置在其上的肢体(在这种情况下为右腿)被插入到通过使端部形成的第一带状部件110的环中 的第一带状构件110通过接头构件130中的开口,并且带被移动到目标压缩位置。 然后,第一带状构件110和第二带​​状构件120用双手在相反的方向拉动。 皮带100B被放置在目标压缩部位上,带100B被适当张紧。

    Muscle Building Tool and Control Method Thereof
    8.
    发明申请
    Muscle Building Tool and Control Method Thereof 审中-公开
    肌肉建筑工具及其控制方法

    公开(公告)号:US20140324097A1

    公开(公告)日:2014-10-30

    申请号:US14358833

    申请日:2012-02-27

    申请人: Yoshiaki Sato

    发明人: Yoshiaki Sato

    IPC分类号: A61B17/12

    摘要: A muscle building tool 1 is used to build, by applying a predetermined pressure to at least one of a user's four limbs to restrict blood flow, a muscle of the limb, and includes: a belt 10 that is wrapped around the at least one of the four limbs and applies the pressure to the muscle; a fastener 40 that maintains a loop shape of the belt 10 in a state of applying the pressure to the muscle; a tension sensor 60 that measures a tension acting on the belt 10 when wrapping the belt 10; and a pressure sensor that is configured to automatically start an operation when the tension measured by the tension sensor 60 exceeds a predetermined threshold, and measures the pressure applied to the muscle.

    摘要翻译: 肌肉建筑工具1用于通过向用户的四肢中的至少一个施加预定的压力来建立肢体的肌肉,并且包括:围绕所述至少一个 四肢并施加压力到肌肉; 紧固件40,其将皮带10的环形状保持在对肌肉施加压力的状态; 张力传感器60,其测量当缠绕带10时作用在带10上的张力; 以及压力传感器,其被构造成当由张力传感器60测量的张力超过预定阈值时自动开始操作,并且测量施加到肌肉的压力。