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公开(公告)号：US06610893B2
公开(公告)日：2003-08-26
申请号：US10240966
申请日：2002-10-07
IPC分类号： C07C20500
CPC分类号： C07C201/08 , C07C205/22
摘要： A process is provided for preparing 4-hydroxy-3-nitrobiphenyl from 4-hydroxy-biphenyl by nitrating in the position adjacent to the phenolic hydroxyl group in high selectivity and yield, and the nitric acid used as the nitrating reagent is metered into the reaction system in a specific manner.
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2.发明授权Process for preparing 2-alkyl-3-aryl- and -heteroaryloxaziridines and novel 2-alkyl-3-aryloxaziridines 失效2-烷基-3-芳基和 - 杂芳基氮杂环丁烷的制备方法和新的2-烷基-3-芳氧基氮杂公开(公告)号：US07074941B2
公开(公告)日：2006-07-11
申请号：US10830622
申请日：2004-04-23
IPC分类号： C07D273/01
CPC分类号： C07D273/00
摘要： 2-Alkyl-3-aryl- or -heteroaryloxaziridines are prepared in a particularly advantageous manner by oxidizing corresponding N-alkyl-aryl- or -heteroarylaldimines with an aromatic percarboxylic acid or a salt thereof in the presence of water, a water-soluble base, and a water-miscible solvent, at temperatures below 30° C. Using this method, it is also possible to obtain novel 2-alkyl-3-aryloxaziridines.
摘要翻译： 通过在水，水溶性碱的存在下，用芳族过羧酸或其盐氧化相应的N-烷基 - 芳基 - 或 - 杂芳基醛亚胺，以特别有利的方式制备2-烷基-3-芳基 - 或 - 杂芳基氧氮丙啶 ，和水混溶性溶剂，温度低于30℃。使用这种方法，也可以获得新的2-烷基-3-芳氧基氮杂。
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3.发明授权Process for preparing 2-alkyl-3aryl-and-heteroaryloxaziridines and novel 2-alkyl-3-aryloxaziridines 失效2-烷基-3-芳基 - 和杂芳基氮杂环丁烷的制备方法和新的2-烷基-3-芳氧基氮杂公开(公告)号：US06740761B2
公开(公告)日：2004-05-25
申请号：US09899421
申请日：2001-07-05
IPC分类号： C07D27301
CPC分类号： C07D273/00
摘要： 2-Alkyl-3-aryl- or -heteroaryloxaziridines are prepared in a particularly advantageous manner by oxidizing corresponding N-alkyl-aryl- or -heteroarylaldimines with an aromatic percarboxylic acid or a salt thereof in the presence of water, a water-soluble base, and a water-miscible solvent, at temperatures below 30° C. Using this method, it is also possible to obtain novel 2-alkyl-3-aryloxaziridines.
摘要翻译： 通过在水，水溶性碱的存在下，用芳香族过羧酸或其盐氧化相应的N-烷基 - 芳基 - 或 - 杂芳基醛亚胺，以特别有利的方式制备2-烷基-3-芳基 - 或 - 杂芳基氧氮丙啶 ，和水混溶性溶剂，温度低于30℃。使用这种方法，也可以获得新的2-烷基-3-芳氧基氮杂。
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4.发明申请METHOD OF PRODUCING 2-PHENOXYACETALS AND THE CORRESPONDING 2-PHENOXY-CARBALDEHYDES THEREFROM 失效生产2-苯氧基乙酸的方法及其相应的2-苯氧基羰基公开(公告)号：US20100286449A1
公开(公告)日：2010-11-11
申请号：US12665066
申请日：2008-06-11
IPC分类号： C07C45/42 , C07C41/50 , C07C43/315 , C07C47/277
CPC分类号： C07C205/37 , C07B41/04 , C07C45/515 , C07C201/12
摘要： The invention relates to a novel process for preparing 2-phenoxyacetals and the corresponding 2-phenoxycarbaldehydes. These compounds are important intermediates for the preparation of active pharmaceutical ingredients.
摘要翻译： 本发明涉及一种制备2-苯氧基缩醛和相应的2-苯氧基羰基醛的新方法。 这些化合物是制备活性药物成分的重要中间体。
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公开(公告)号：US07276630B2
公开(公告)日：2007-10-02
申请号：US11525281
申请日：2006-09-22
IPC分类号： C07C211/00
CPC分类号： C07C227/18 , C07B37/04 , C07C229/38
摘要： A process is provided for preparing optionally substituted arylated benzylamines from the corresponding optionally substituted aryl halides and optionally substituted benzylamines using a specific solvent mixture, a base and a catalyst comprising a palladium compound and a bisaryldialkylphosphine.
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6.发明授权公开(公告)号：US06956129B2
公开(公告)日：2005-10-18
申请号：US10074180
申请日：2002-02-12
IPC分类号： C07C45/46 , C07C45/62 , C07C49/697 , C07C51/363 , C07C57/60 , C07C51/347 , C07C231/14 , C07C233/00
CPC分类号： C07C57/60 , C07C45/46 , C07C45/62 , C07C49/697 , C07C51/363
摘要： Polyhalogenated cinnamic acids and cinnamic acid derivatives are prepared by reacting diazonium salts accessible from polyhalogenated anilines with acrylic acid or acrylic acid derivatives in the presence of a homogeneous, palladium-containing catalyst at about −5 to about +100° C. Some of the cinnamic acids and cinnamic acid derivatives obtainable in this way are new. Cinnamic acids and cinnamic acid derivatives which can be prepared according to the invention can be used for the preparation of indanones which are precursors for agro- and pharmaceutical chemicals and for substances having liquid-crystalline properties.
摘要翻译： 多卤代肉桂酸和肉桂酸衍生物通过在大约-5至大约+ 100℃的均相的含钯催化剂存在下，将可从多卤代苯胺获得的重氮盐与丙烯酸或丙烯酸衍生物反应来制备。一些肉桂酸 以这种方式获得的酸和肉桂酸衍生物是新的。 可以根据本发明制备的肉桂酸和肉桂酸衍生物可用于制备作为农药和药物化学品的前体的茚满酮和具有液晶性质的物质。
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公开(公告)号：US06559340B2
公开(公告)日：2003-05-06
申请号：US10013203
申请日：2001-12-07
IPC分类号： C07C23910
CPC分类号： C07C239/10
摘要： This invention relates to a process for preparing N-substituted hydroxylamines from N-substituted aryl- or heteroaryloxaziridines by acid hydrolysis and isolation of the N-substituted hydroxylamines in the form of their salts.
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公开(公告)号：US20140128617A1
公开(公告)日：2014-05-08
申请号：US14125475
申请日：2012-06-19
申请人： Wahed Ahmed Moradi , Norbert Lui , Michael Dockner
发明人： Wahed Ahmed Moradi , Norbert Lui , Michael Dockner
IPC分类号： C07D231/14
CPC分类号： C07D231/14 , C07C231/02
摘要： The present invention relates to a simplified process for preparing pyrazolylcarboxanilides by reacting pyrazolylcarboxylic esters with anilines in the presence of a base and removing at least one reaction product.
摘要翻译： 本发明涉及通过吡唑基羧酸酯与苯胺在碱的存在下反应并除去至少一种反应产物来制备吡唑基甲酰苯胺的简化方法。
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公开(公告)号：US08455689B2
公开(公告)日：2013-06-04
申请号：US12991265
申请日：2009-04-24
申请人： Michael Dockner , Heiko Rieck , Wahed Ahmed Moradi , Norbert Lui
发明人： Michael Dockner , Heiko Rieck , Wahed Ahmed Moradi , Norbert Lui
IPC分类号： C07C233/05
CPC分类号： C07C231/12 , C07C233/15
摘要： The present invention relates to a process for preparing substituted biphenylanilides of the formula I wherein R1 is a protected amino group which comprises reacting a compound of formula II in the presence of a base and of a palladium catalyst in a solvent, with an organoboron compound of formula (III)
摘要翻译： 本发明涉及一种制备式I取代的联苯酰苯胺的方法，其中R 1是被保护的氨基，其包括在碱和Pd催化剂存在下，在溶剂中使式Ⅱ化合物与有机硼化合物反应 式（III）
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10.发明申请公开(公告)号：US20100274049A1
公开(公告)日：2010-10-28
申请号：US12809830
申请日：2008-12-16
IPC分类号： C07C229/06
CPC分类号： C07C227/16 , C07C253/30 , C07C229/30 , C07C255/30
摘要： The present invention relates to a process for preparing 2-fluoroacyl-3-aminoacrylic acid derivatives by reacting fluorinated carboxylic acids with dialkylaminoacrylic acid derivatives and acid halides.
摘要翻译： 本发明涉及通过氟化羧酸与二烷基氨基丙烯酸衍生物和酰卤反应制备2-氟酰基-3-氨基丙烯酸衍生物的方法。
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