公开(公告)号：US4968805A

公开(公告)日：1990-11-06

申请号：US310591

申请日：1989-02-15

申请人： Itaru Okada ,  Shigeru Suzuki ,  Shuko Okui ,  Yoji Takahashi ,  Toshiki Fukuchi ,  Tetsuo Nakajima

发明人： Itaru Okada ,  Shigeru Suzuki ,  Shuko Okui ,  Yoji Takahashi ,  Toshiki Fukuchi ,  Tetsuo Nakajima

IPC分类号： A01N43/50 ,  C07D401/12

CPC分类号： C07D401/12

摘要： Disclosed herein are pyrazole derivatives which are represented by the following formula (I): ##STR1## wherein R.sup.1 represents a C.sub.1 -C.sub.4 alkyl group or a benzyl group; R.sup.2 represents a hydrogen atom or a C.sub.1 -C.sub.4 alkyl group; X represents a hydrogen atom, a halogen atom or a C.sub.1 -C.sub.4 alkyl group; R.sup.2 may combine with X to form ##STR2## wherein R.sup.5 represents a hydrogen atom or a C.sub.1 -C.sub.3 alkyl group; R.sup.3 represents a hydrogen atom or a C.sub.1 -C.sub.4 alkyl group; R.sup.4 s independently represent a hydrogen atom, a halogen atom, a C.sub.1 -C.sub.5 alkyl group, a C.sub.1 -C.sub.4 alkoxy group, a C.sub.1 -C.sub.4 alkylthio group, a trifluoromethyl group, a C.sub.1 -C.sub.4 haloalkoxy group, a phenyl group, an alkyl-substituted phenyl group or ##STR3## wherein Y represents an oxygen atom or a sulfur atom, R.sup.6 s independently represent a hydrogen atom, a C.sub.1 -C.sub.4 alkyl group, a C.sub.1 -C.sub.4 alkoxy group, a halogen atom, a nitro group, a cyano group or a trifluoromethyl group and n represents 1 or 2, adjacent R.sup.4 s being able to combine together to form ##STR4## wherein R.sup.7 represents a hydrogen atom or a methyl group; l represents 0 or 1; and m represents 1, 2, or 3. The pyrazole derivatives of the formula (I) show a high activity suitable for active ingredient of insecticidal and miticidal composition as well as fungicidal composition.

公开(公告)号：US4950668A

公开(公告)日：1990-08-21

申请号：US181695

申请日：1988-04-14

申请人： Itaru Okada ,  Shuko Okui ,  Yoji Takahashi ,  Toshiki Fukuchi

发明人： Itaru Okada ,  Shuko Okui ,  Yoji Takahashi ,  Toshiki Fukuchi

IPC分类号： A01N43/56 ,  C07D231/14 ,  C07D231/16 ,  C07D231/38 ,  C07D231/40 ,  C07D405/12

CPC分类号： C07D231/38 ,  A01N43/56 ,  C07D231/14 ,  C07D231/16 ,  C07D231/40 ,  C07D405/12

摘要： A novel pyrazole derivative and an insecticidal or miticidal composition containing the derivative as the effective ingredient are disclosed.The pyrazole derivative of the present invention has an excellent controlling effect also against harmful insects and mites exhibiting resistance to conventional insecticides and does not disturb the ecosystem since it is less toxic and less residual.

公开(公告)号：US4861777A

公开(公告)日：1989-08-29

申请号：US241387

申请日：1988-09-07

申请人： Itaru Okada ,  Shuko Okui ,  Mana Nishimata ,  Yoji Takahashi ,  Toshiki Fukuchi

发明人： Itaru Okada ,  Shuko Okui ,  Mana Nishimata ,  Yoji Takahashi ,  Toshiki Fukuchi

IPC分类号： C07D231/54 ,  C07D231/56

CPC分类号： C07D231/56 ,  C07D231/54

摘要： A novel pyrazole derivative and an insecticidal or miticidal composition containing the derivative as the effective ingredient are disclosed.The pyrazole derivative of the present invention has an excellent controlling effect also against harmful insects and mites exhibiting resistance to conventional insecticides and does not disturb the ecosystem since it is less toxic and less residual.

公开(公告)号：US07153815B2

公开(公告)日：2006-12-26

申请号：US10500925

申请日：2003-01-10

申请人： Shinji Kawata ,  Shuko Okui ,  Shigeru Suzuki ,  Toshiki Fukuchi ,  Akiyuki Suwa

发明人： Shinji Kawata ,  Shuko Okui ,  Shigeru Suzuki ,  Toshiki Fukuchi ,  Akiyuki Suwa

IPC分类号： A01N35/08 ,  A01N43/54 ,  A01N43/58 ,  A01N43/40 ,  A01N43/08 ,  A01N43/10 ,  A01N37/18 ,  A01N37/20 ,  C07C239/22 ,  C07C239/20 ,  C07D333/28 ,  C07D277/10 ,  C07D277/12 ,  C07D213/81 ,  C07D213/82 ,  C07D413/12 ,  C07D239/24

CPC分类号： C07D213/40 ,  A01N37/50 ,  A01N43/08 ,  A01N43/10 ,  A01N43/40 ,  A01N43/54 ,  A01N43/58 ,  A01N43/60 ,  A01N43/78 ,  A01N43/80 ,  C07C251/76 ,  C07D213/61 ,  C07D213/68 ,  C07D213/74 ,  C07D213/75 ,  C07D213/77

摘要： A insecticide characterized by containing as active ingredient a hydrazone derivative of formula (I) wherein A and Q are an aryl or a heterocyclic group, W is oxygen atom, an aminylene, an alkylene group, an oxyalkylene group or an alkyleneoxy, X1 and X2 are hydrogen atom, an alkyl, an alkenyl, an alkynyl, an aryl, a heterocyclic group, formyl, an acyl, an alkoxycarbonyl, an aryloxycarbonyl, a heterocyclic oxycarbonyl, an alkylsulfinyl, an arylsulfinyl, a heterocyclic sulfinyl, an alkylsulfonyl, an arylsulfonyl or a heterocyclic sulfonyl, Y is oxygen atom or sulfur atom, Z is hydrogen atom, a halogen atom, cyano, an alkyl, an alkenyl, an alkynyl, an amino, an alkoxy or an alkylthio, the substituents may be substituted; and novel hydrazon derivatives.

摘要翻译： 一种杀虫剂，其特征在于含有作为活性成分的式（I）腙衍生物，其中A和Q为芳基或杂环基，W为氧原子，亚氨基，亚烷基，氧化烯基或亚烷基氧基，X ^{1和X 2是氢原子，烷基，烯基，炔基，芳基，杂环基，甲酰基，酰基，烷氧基羰基，芳氧基羰基，杂环氧基羰基 ，烷基亚磺酰基，芳基亚磺酰基，杂环亚磺酰基，烷基磺酰基，芳基磺酰基或杂环磺酰基，Y是氧原子或硫原子，Z是氢原子，卤素原子，氰基，烷基，烯基，炔基， 氨基，烷氧基或烷硫基，取代基可以被取代; 和腙衍生物。}

公开(公告)号：US20050203149A1

公开(公告)日：2005-09-15

申请号：US10500925

申请日：2003-01-10

申请人： Shinji Kawata ,  Shuko Okui ,  Shigeru Suzuki ,  Toshiki Fukuchi ,  Akiyuki Suwa

发明人： Shinji Kawata ,  Shuko Okui ,  Shigeru Suzuki ,  Toshiki Fukuchi ,  Akiyuki Suwa

IPC分类号： C07D237/12 ,  A01N37/18 ,  A01N37/50 ,  A01N43/08 ,  A01N43/10 ,  A01N43/40 ,  A01N43/54 ,  A01N43/58 ,  A01N43/60 ,  A01N43/78 ,  A01N43/80 ,  C07C251/76 ,  C07C255/66 ,  C07C257/02 ,  C07C323/41 ,  C07C323/48 ,  C07D213/40 ,  C07D213/61 ,  C07D213/68 ,  C07D213/74 ,  C07D213/75 ,  C07D213/77 ,  C07D239/30 ,  C07D241/12 ,  C07D261/10 ,  C07D277/20 ,  C07D277/30 ,  C07D277/32 ,  C07D277/82 ,  C07D307/16 ,  C07D307/52 ,  C07D333/24 ,  C07D333/28 ,  C07D417/12 ,  A01N37/34 ,  A01N43/36

CPC分类号： C07D213/40 ,  A01N37/50 ,  A01N43/08 ,  A01N43/10 ,  A01N43/40 ,  A01N43/54 ,  A01N43/58 ,  A01N43/60 ,  A01N43/78 ,  A01N43/80 ,  C07C251/76 ,  C07D213/61 ,  C07D213/68 ,  C07D213/74 ,  C07D213/75 ,  C07D213/77

摘要： A insecticide characterized by containing as active ingredient a hydrazone derivative of formula (I) wherein A and Q are an aryl or a heterocyclic group, W is oxygen atom, an aminylene, an alkylene group, an oxyalkylene group or an alkyleneoxy, X1 and X2 are hydrogen atom, an alkyl, an alkenyl, an alkynyl, an aryl, a heterocyclic group, formyl, an acyl, an alkoxycarbonyl, an aryloxycarbonyl, a heterocyclic oxycarbonyl, an alkylsulfinyl, an arylsulfinyl, a heterocyclic sulfinyl, an alkylsulfonyl, an arylsulfonyl or a heterocyclic sulfonyl, Y is oxygen atom or sulfur atom, Z is hydrogen atom, a halogen atom, cyano, an alkyl, an alkenyl, an alkynyl, an amino, an alkoxy or an alkylthio, the substituents may be substituted; and novel hydrazon derivatives.

摘要翻译： 一种杀虫剂，其特征在于含有作为活性成分的式（I）腙衍生物，其中A和Q为芳基或杂环基，W为氧原子，亚氨基，亚烷基，氧化烯基或亚烷基氧基，X ^{1和X 2是氢原子，烷基，烯基，炔基，芳基，杂环基，甲酰基，酰基，烷氧基羰基，芳氧基羰基，杂环氧基羰基 ，烷基亚磺酰基，芳基亚磺酰基，杂环亚磺酰基，烷基磺酰基，芳基磺酰基或杂环磺酰基，Y是氧原子或硫原子，Z是氢原子，卤素原子，氰基，烷基，烯基，炔基， 氨基，烷氧基或烷硫基，取代基可以被取代; 和腙衍生物。}

公开(公告)号：US06849633B2

公开(公告)日：2005-02-01

申请号：US10028786

申请日：2001-12-28

申请人： Shuko Okui ,  Nobuo Kyomura ,  Toshiki Fukuchi ,  Ken Tanaka ,  Manabu Katsurada ,  Kazuya Okano ,  Naoko Sumitani ,  Akiko Miyauchi ,  Akiko Yabe

发明人： Shuko Okui ,  Nobuo Kyomura ,  Toshiki Fukuchi ,  Ken Tanaka ,  Manabu Katsurada ,  Kazuya Okano ,  Naoko Sumitani ,  Akiko Miyauchi ,  Akiko Yabe

IPC分类号： A01N43/56 ,  A01N43/58 ,  A01N43/60 ,  A01N47/02 ,  C07D401/12 ,  C07D403/12 ,  C07D401/14

CPC分类号： C07D401/12 ,  A01N43/56 ,  A01N43/58 ,  A01N43/60 ,  A01N47/02 ,  C07D403/12

摘要： The invention provides a novel pest control agent having a high systemic activity and a high safety with reduced adverse influences on the environment neighboring the place to which the agent is applied, and a process for producing the same.Namely, the present invention relates to a novel 1-aryl-3-cyano-5-heteroarylalkylaminopyrazole derivative represented by the following general formula (1) and a process for producing the same, and a pest control agent containing the same as an active ingredient. (wherein X represents N or C-halogen, R1 represents an alkyl group, an alkenyl group, an alkynyl group, or a haloalkyl group, R2 represents hydrogen atom, an alkyl group, or an acyl group, R3 represents hydrogen atom or an alkyl group, A represents any one of the groups represented by A-1 to A-4, R4 represents hydrogen atom, an alkyl group, a halogen atom, and n represents 0, 1, or 2, provided that R1 is a haloalkyl group except a perhaloalkyl group when A is A-1 and n is 0, and that n is not 0 when A is A-4.).

摘要翻译： 本发明提供了一种具有高体系活性和高安全性的新型有害生物防治剂及其对施用该药剂的地方附近的环境的不良影响，以及其制备方法。本发明涉及一种 由以下通式（1）表示的新颖的1-芳基-3-氰基-5-杂芳基烷基氨基吡唑衍生物及其制备方法和含有该有效成分的害虫控制剂（其中X表示N或C - 卤素，R 1表示烷基，烯基，炔基或卤代烷基，R 2表示氢原子，烷基或酰基，R 3表示氢原子或 烷基，A表示由A-1〜A-4表示的基团中的任一个，R 4表示氢原子，烷基，卤素原子，n表示0,1或2，条件是R 当A是A-1且n是0时，除了全卤代烷基之外的卤代烷基，和tha 当A为A-4时，t n不为0。

公开(公告)号：US06335357B1

公开(公告)日：2002-01-01

申请号：US09402454

申请日：1999-10-07

申请人： Shuko Okui ,  Nobuo Kyomura ,  Toshiki Fukuchi ,  Ken Tanaka

发明人： Shuko Okui ,  Nobuo Kyomura ,  Toshiki Fukuchi ,  Ken Tanaka

IPC分类号： A01N4356

CPC分类号： C07D401/12 ,  A01N43/56 ,  A01N43/78 ,  A01N47/02 ,  C07D231/44 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D417/12

摘要： A 1-aryl-3-cyano-5-(het)arylalkylaminopyrazole derivative represented by the general formula (1): process of making, intermediate thereof and pesticide therewith.

摘要翻译： 由通式（1）表示的1-芳基-3-氰基-5-（het）芳烷基氨基吡唑衍生物：其制备方法，其中间体和农药。

公开(公告)号：US07371768B2

公开(公告)日：2008-05-13

申请号：US10355182

申请日：2003-01-31

申请人： Shuko Okui ,  Nobuo Kyomura ,  Toshiki Fukuchi ,  Kazuya Okano ,  Liangyou He ,  Akiko Miyauchi

发明人： Shuko Okui ,  Nobuo Kyomura ,  Toshiki Fukuchi ,  Kazuya Okano ,  Liangyou He ,  Akiko Miyauchi

IPC分类号： A01N43/56

CPC分类号： C07D401/12 ,  A01N43/56

摘要： The present invention relates to pest control agent having systemic activity and a high safety along with a wide insecticidal spectrum and excellent insecticidal activity, which are 1-aryl-3-cyano-5-pyridylalkylaminopyrazole derivatives represented by formula (1): wherein X represents an N or C-halogen atom; R1 represents a haloalkyl group, excluding a perhaloalkyl group; R2 represents a hydrogen atom or an alkyl group, R3 represents a hydrogen atom, an alkyl group, or an acyl group; and R4 represents a hydrogen atom, a hydroxyl group, an alkyl group, a haloalkyl group, an alkoxy group, a haloalkoxy group, an alkylthio group, an alkylsulfinyl group, an alkylsulfonyl group, a halogen atom, a nitro group, or a cyano group.

摘要翻译： 本发明涉及具有全身活性和高安全性以及广泛的杀虫谱和优异的杀虫活性的害虫防治剂，它是由式（1）表示的1-芳基-3-氰基-5-吡啶基烷基氨基吡唑衍生物：其中X表示 N或C-卤素原子; R 1表示不包括全卤代烷基的卤代烷基; R 2表示氢原子或烷基，R 3表示氢原子，烷基或酰基; R 4表示氢原子，羟基，烷基，卤代烷基，烷氧基，卤代烷氧基，烷硫基，烷基亚磺酰基，烷基磺酰基，卤素原子 ，硝基或氰基。

公开(公告)号：US20050085524A1

公开(公告)日：2005-04-21

申请号：US10474179

申请日：2002-04-02

申请人： Itaru Okada ,  Eiji Takizawa ,  Kazuhiko Kikutake ,  Toshiki Fukuchi

发明人： Itaru Okada ,  Eiji Takizawa ,  Kazuhiko Kikutake ,  Toshiki Fukuchi

IPC分类号： A01N43/56 ,  C07C211/29 ,  C07C217/54 ,  C07C217/58 ,  C07D231/14 ,  C07D231/20 ,  A61K31/415

CPC分类号： C07C217/54 ,  A01N43/56 ,  C07C211/29 ,  C07C217/58 ,  C07D231/14 ,  C07D231/20

摘要： The present invention provides novel compounds with fungicidal and bactericidal activity as well as insecticidal and miticidal activity, which are useful for controlling hazardous biological organisms and belong to pyrazolecarboxamides represented by the following formula (I): wherein R1 represents C1-C5 alkyl; R2 represents C1-C5 alkyl, C1-C5 haloalkyl, or the like; R3 represents hydrogen or C1-C3 alkyl; R4 represents halogen, C1-C5 alkyl or the like; n is an integer of 0 to 4; R5 represents alkyl, haloalkyl, alkoxy, haloalkoxy or the like; n represents an integer of 1 to 5; and X represents hydrogen, C1-C3 alkyl, C1-C3 alkoxy, halogen, C1-C3 haloalkoxy or nitro.

摘要翻译： 本发明提供具有杀真菌和杀菌活性以及杀虫和杀螨活性的新型化合物，其可用于防治有害生物体并属于由下式（I）表示的吡唑酰胺：其中R 1， 表示C 1 -C 5烷基; R 2表示C 1 -C 5烷基，C 1 -C 5烷基，C 1 -C 5烷基，C 1 -C 5烷基，C 1 -C 5烷基， 卤代烷基等; R 3表示氢或C 1 -C 3烷基; R 4表示卤素，C 1 -C 5烷基等; n为0〜4的整数。 R 5表示烷基，卤代烷基，烷氧基，卤代烷氧基等; n表示1〜5的整数， 和X代表氢，C 1 -C 3烷基，C 1 -C 3烷氧基，卤素，C C 1 -C 3卤代烷氧基或硝基。

公开(公告)号：US4722934A

公开(公告)日：1988-02-02

申请号：US026198

申请日：1987-03-16

申请人： Susumu Matsumoto ,  Shigeru Suzuki ,  Hiroki Ohta ,  Yoshiaki Higashino ,  Toshiki Fukuchi

发明人： Susumu Matsumoto ,  Shigeru Suzuki ,  Hiroki Ohta ,  Yoshiaki Higashino ,  Toshiki Fukuchi

IPC分类号： A01N43/82 ,  A01N43/824 ,  C07D285/12 ,  C07D285/125 ,  C07D285/13 ,  C07D285/135 ,  C07D417/12

CPC分类号： C07D285/12 ,  A01N43/82 ,  C07D285/125 ,  C07D285/13 ,  C07D285/135 ,  C07D417/12

摘要： The present invention relates to a thiadiazole derivative of the following general formula (I) and an insecticidal and miticidal composition containing the same as an active ingredient: ##STR1## wherein A represents a group of the formula ##STR2## R.sup.1 and R.sup.2 independently represent a hydrogen atom, a halogen atom, a lower alkyl group, a trifluoromethyl group, a cyano group or a nitro group or jointly represent a methylenedioxy group, R.sup.3 represents a hydrogen atom or a lower alkyl group, R.sup.4 represents a lower alkyl group, a lower alkoxy group, a lower alkylthio group, a monoalkylamino group having a lower alkyl group or a dialkylamino group having lower alkyl group, and n is an integer of from 1 through 3.