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1.发明申请Process for the Preparation of 5-Substituted 3-Aryl-3-(trifluoromethyl)-3,4-dihydro-2H-pyrroles 审中-公开5-取代的3-芳基-3-（三氟甲基）-3,4-二氢-2H-吡咯的制备方法公开(公告)号：US20120029202A1
公开(公告)日：2012-02-02
申请号：US13105613
申请日：2011-05-11
申请人： Koichi ARAKI , Jun Mihara , Norio Sasaki , Peter Bruechner , Kei Domon , Johannes-Rudolf Jansen , Norbert Lui
发明人： Koichi ARAKI , Jun Mihara , Norio Sasaki , Peter Bruechner , Kei Domon , Johannes-Rudolf Jansen , Norbert Lui
IPC分类号： C07D207/20 , C07D403/10
CPC分类号： C07D207/22 , C07C51/353 , C07C69/65 , C07C2601/14 , C07C57/62
摘要： The present invention relates to a process for the manufacturing of 5-substituted 3-aryl-3-(trifluoromethyl)-3,4-dihydro-2H-pyrroles of formula (I) which comprises the following steps: (i) reacting a compound of formula (II) with a isonitrile compound of formula (III) in the presence of a metal catalyst to obtain compounds of formula (IV) (ii) isomerizing compounds of formula (IV) to obtain compounds of formula (V) and (iii) reacting the dihydropyrrole compound of formula (V) under acidic conditions, to obtain the compounds of formula (I), wherein X, n, Z, Y, and T are as defined in the description.
摘要翻译： 本发明涉及制备式（I）的5-取代的3-芳基-3-（三氟甲基）-3,4-二氢-2H-吡咯的方法，其包括以下步骤：（i）使化合物 式（Ⅳ）化合物与式（Ⅳ）的异腈化合物在金属催化剂存在下反应，得到式（Ⅳ）化合物（ⅱ）使式（Ⅳ）化合物异构化得到式（Ⅴ）和（ⅲ）化合物 ）在酸性条件下使式（Ⅴ）的二氢吡咯化合物反应，得到其中X，n，Z，Y和T如说明书中所定义的式（I）化合物。
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公开(公告)号：US09375000B2
公开(公告)日：2016-06-28
申请号：US13818291
申请日：2011-09-13
申请人： Jun Mihara , Mamoru Hatazawa , Daiei Yamazaki , Hidetoshi Kishikawa , Kei Domon , Hidekazu Watanabe , Norio Sasaki , Tetsuya Murata , Koichi Araki , Eiichi Shimojo , Teruyuki Ichihara , Tadashi Ishikawa , Katsuhiko Shibuya , Ulrich Görgens , Peter Bruechner , Reiner Fischer , Johannes-Rudolf Jansen , Tobias Kapferer , Simon Maechling , Michael Maue , Arnd Voerste
发明人： Jun Mihara , Mamoru Hatazawa , Daiei Yamazaki , Hidetoshi Kishikawa , Kei Domon , Hidekazu Watanabe , Norio Sasaki , Tetsuya Murata , Koichi Araki , Eiichi Shimojo , Teruyuki Ichihara , Tadashi Ishikawa , Katsuhiko Shibuya , Ulrich Görgens , Peter Bruechner , Reiner Fischer , Johannes-Rudolf Jansen , Tobias Kapferer , Simon Maechling , Michael Maue , Arnd Voerste
IPC分类号： C07D207/08 , A01N43/36 , C07D207/12 , C07D207/26 , C07D401/04 , C07D403/04 , C07D403/10 , C07D403/14 , C07D409/12 , C07D409/14 , C07D417/04 , A01N43/40 , A01N43/56 , A01N43/653 , A01N43/713
CPC分类号： A01N43/36 , A01N43/40 , A01N43/56 , A01N43/653 , A01N43/713 , C07D207/12 , C07D207/26 , C07D401/04 , C07D403/04 , C07D403/10 , C07D403/14 , C07D409/12 , C07D409/14 , C07D417/04
摘要： Arylpyrrolidines of Formula (I): wherein each substituent is as defined in the specification, and use thereof as pesticides and animal parasite-controlling agents.
摘要翻译： 式（I）的芳基吡咯烷酮：其中每个取代基如说明书中所定义，及其作为农药和动物寄生虫控制剂的用途。
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公开(公告)号：US20140046069A1
公开(公告)日：2014-02-13
申请号：US13818291
申请日：2011-09-13
申请人： Jun Mihara , Mamoru Hatazawa , Daiei Yamazaki , Hidetoshi Kishikawa , Kei Domon , Hidekazu Watanabe , Norio Sasaki , Tetsuya Murata , Koichi Araki , Eiichi Shimojo , Teruyuki Ichihara , Tadashi Ishikawa , Katsuhiko Shibuya , Ulrich Goergens , Peter Bruechner , Reiner Fischer , Johannes-Rudolf Jansen , Tobias Kapferer , Simon Maechling , Michael Maue , Arnd Voerste
发明人： Jun Mihara , Mamoru Hatazawa , Daiei Yamazaki , Hidetoshi Kishikawa , Kei Domon , Hidekazu Watanabe , Norio Sasaki , Tetsuya Murata , Koichi Araki , Eiichi Shimojo , Teruyuki Ichihara , Tadashi Ishikawa , Katsuhiko Shibuya , Ulrich Goergens , Peter Bruechner , Reiner Fischer , Johannes-Rudolf Jansen , Tobias Kapferer , Simon Maechling , Michael Maue , Arnd Voerste
IPC分类号： A01N43/36 , A01N43/713 , A01N43/653 , A01N43/40 , A01N43/56
CPC分类号： A01N43/36 , A01N43/40 , A01N43/56 , A01N43/653 , A01N43/713 , C07D207/12 , C07D207/26 , C07D401/04 , C07D403/04 , C07D403/10 , C07D403/14 , C07D409/12 , C07D409/14 , C07D417/04
摘要： Arylpyrrolidines of Formula (I): wherein each substituent is as defined in the specification, and use thereof as pesticides and animal paracite-controlling agents.
摘要翻译： 式（I）的芳基吡咯烷酮：其中每个取代基如本说明书中所定义，以及其作为农药和动物皂甙控制剂的用途。
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公开(公告)号：US20120129854A1
公开(公告)日：2012-05-24
申请号：US13318131
申请日：2010-04-27
申请人： Jun Mihara , Tetsuya Murata , Daiei Yamazaki , Yasushi Yoneta , Koichi Araki , Norio Sasaki , Kei Domon , Mamoru Hatazawa , Eiichi Shimojo , Teruyuki Ichihara , Masashi Ataka , Katsuhiko Shibuya , Ulrich Görgens
发明人： Jun Mihara , Tetsuya Murata , Daiei Yamazaki , Yasushi Yoneta , Koichi Araki , Norio Sasaki , Kei Domon , Mamoru Hatazawa , Eiichi Shimojo , Teruyuki Ichihara , Masashi Ataka , Katsuhiko Shibuya , Ulrich Görgens
IPC分类号： A01N43/84 , C07D417/04 , C07D401/04 , C07D401/14 , C07D413/14 , C07D405/14 , C07D409/14 , C07D403/04 , A01N43/36 , A01N43/78 , A01N43/42 , A01N43/54 , A61K31/402 , A61K31/428 , A61K31/4709 , A61K31/5377 , A61K31/435 , A61K31/517 , A01P7/04 , A01P7/00 , A01P5/00 , A01P9/00 , A61P33/00 , A61P33/02 , C07D207/08
CPC分类号： C07D207/08 , A01N43/36 , A01N43/42 , A01N43/54 , A01N43/56 , A01N43/78 , C07D401/04 , C07D417/04
摘要： The invention is directed to arylpyrrolidines compounds which exhibit excellent insecticidal efficacy and which may be used as in the agrochemical field or in the yield of veterinary medicine. The compounds are represented by formula (I): wherein the respective substituents are defined in the specification.
摘要翻译： 本发明涉及具有优异杀虫功效的芳基吡咯烷酮化合物，其可以如在农业化学领域中使用或兽医药品的收率使用。 化合物由式（I）表示：其中各个取代基在说明书中定义。
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公开(公告)号：US20100216792A1
公开(公告)日：2010-08-26
申请号：US12588411
申请日：2009-10-14
申请人： Ulrich Görgens , Jun Mihara , Tetsuya Murata , Daiei Yamazaki , Yasushi Yoneta , Koichi Araki , Norio Sasaki , Kei Domon , Mamoru Hatazawa , Eiichi Shimojo , Teruyuki Ichihara , Masashi Ataka , Katsuhiko Shibuya
发明人： Ulrich Görgens , Jun Mihara , Tetsuya Murata , Daiei Yamazaki , Yasushi Yoneta , Koichi Araki , Norio Sasaki , Kei Domon , Mamoru Hatazawa , Eiichi Shimojo , Teruyuki Ichihara , Masashi Ataka , Katsuhiko Shibuya
IPC分类号： A01N43/84 , C07D401/12 , A01N43/40 , C07D403/04 , A01N43/54 , C07D417/04 , A01N43/78 , C07D207/08 , C07D403/12 , A01N43/36 , A01N43/50 , A01N43/56 , A01N43/647 , A01N43/653 , A01N43/713 , C07D403/14 , C07D413/14 , C07D413/12 , A01P7/02 , A01P7/04
CPC分类号： A01N43/84 , A01N43/36 , A01N43/40 , A01N43/54 , A01N43/56 , A01N43/653 , A01N43/713 , A01N43/76 , A01N43/78 , C07D207/08 , C07D207/09 , C07D401/04 , C07D401/12 , C07D401/14 , C07D403/04 , C07D403/12 , C07D403/14 , C07D405/12 , C07D405/14 , C07D409/12 , C07D409/14 , C07D413/12 , C07D417/04 , C07D417/14
摘要： The invention is directed to arylpyrrolidines compounds which exhibit excellent insecticidal efficacy and which may be used as in the agrochemical field or in the field of veterinary medicine. The compounds are represented by formula (I): wherein the respective substituents are defined in the specification.
摘要翻译： 本发明涉及具有优异杀虫功效的芳基吡咯烷化合物，其可以在农药领域或兽医学领域中使用。 化合物由式（I）表示：其中各个取代基在说明书中定义。
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公开(公告)号：US08450483B2
公开(公告)日：2013-05-28
申请号：US12588411
申请日：2009-10-14
申请人： Ulrich Görgens , Jun Mihara , Tetsuya Murata , Daiei Yamazaki , Yasushi Yoneta , Koichi Araki , Norio Sasaki , Kei Domon , Mamoru Hatazawa , Eiichi Shimojo , Teruyuki Ichihara , Masashi Ataka , Katsuhiko Shibuya
发明人： Ulrich Görgens , Jun Mihara , Tetsuya Murata , Daiei Yamazaki , Yasushi Yoneta , Koichi Araki , Norio Sasaki , Kei Domon , Mamoru Hatazawa , Eiichi Shimojo , Teruyuki Ichihara , Masashi Ataka , Katsuhiko Shibuya
IPC分类号： C07D239/28 , A61K31/505
CPC分类号： A01N43/84 , A01N43/36 , A01N43/40 , A01N43/54 , A01N43/56 , A01N43/653 , A01N43/713 , A01N43/76 , A01N43/78 , C07D207/08 , C07D207/09 , C07D401/04 , C07D401/12 , C07D401/14 , C07D403/04 , C07D403/12 , C07D403/14 , C07D405/12 , C07D405/14 , C07D409/12 , C07D409/14 , C07D413/12 , C07D417/04 , C07D417/14
摘要： The invention is directed to arylpyrrolidines compounds which exhibit excellent insecticidal efficacy and which may be used as in the agrochemical field or in the field of veterinary medicine. The compounds are represented by formula (I): wherein the respective substituents are defined in the specification.
摘要翻译： 本发明涉及具有优异杀虫功效的芳基吡咯烷化合物，其可以在农药领域或兽医学领域中使用。 化合物由式（I）表示：其中各个取代基在说明书中定义。
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公开(公告)号：US08410141B2
公开(公告)日：2013-04-02
申请号：US13319287
申请日：2010-05-18
申请人： Tetsuya Murata , Yasushi Yoneta , Hidetoshi Kishikawa , Jun Mihara , Daiei Yamazaki , Mamoru Hatazawa , Norio Sasaki , Kei Domon , Eiichi Shimojo , Teruyuki Ichihara , Katsuhiko Shibuya , Masashi Ataka , Ulrich Görgens
发明人： Tetsuya Murata , Yasushi Yoneta , Hidetoshi Kishikawa , Jun Mihara , Daiei Yamazaki , Mamoru Hatazawa , Norio Sasaki , Kei Domon , Eiichi Shimojo , Teruyuki Ichihara , Katsuhiko Shibuya , Masashi Ataka , Ulrich Görgens
IPC分类号： A61K31/4427 , A61K31/41 , A61K31/415 , A61K31/4164 , A61K31/4192 , A61K31/4196 , C07D401/14 , C07D257/02 , C07D249/04 , C07D249/08 , C07D233/00 , C07D231/00 , C07D207/00
CPC分类号： A01N43/40 , A01N43/36 , A01N43/50 , A01N43/56 , A01N43/647 , A01N43/653 , A01N43/713 , C07D207/20 , C07D401/04 , C07D401/14 , C07D403/04 , C07D403/10 , C07D403/14 , C07D405/14
摘要： The invention relates to novel arylpyrroline compounds of formula (I) which have excellent insecticidal activity and which can thus be used as an insecticide.
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公开(公告)号：US20120108635A1
公开(公告)日：2012-05-03
申请号：US13319287
申请日：2010-05-18
申请人： Tetsuya Murata , Yasushi Yoneta , Hidetoshi Kishikawa , Jun Mihara , Daiei Yamazaki , Mamoru Hatazawa , Norio Sasaki , Kei Domon , Eiichi Shimojo , Teruyuki Ichihara , Katsuhiko Shibuya , Masashi Ataka , Ulrich Görgens
发明人： Tetsuya Murata , Yasushi Yoneta , Hidetoshi Kishikawa , Jun Mihara , Daiei Yamazaki , Mamoru Hatazawa , Norio Sasaki , Kei Domon , Eiichi Shimojo , Teruyuki Ichihara , Katsuhiko Shibuya , Masashi Ataka , Ulrich Görgens
IPC分类号： A01N43/713 , A01N43/653 , C07D401/04 , A01N43/40 , A01P7/04 , C07D405/14 , A01N43/36 , A01N43/56 , A01N43/50 , A01N43/647 , C07D401/14 , C07D403/10
CPC分类号： A01N43/40 , A01N43/36 , A01N43/50 , A01N43/56 , A01N43/647 , A01N43/653 , A01N43/713 , C07D207/20 , C07D401/04 , C07D401/14 , C07D403/04 , C07D403/10 , C07D403/14 , C07D405/14
摘要： The invention relates to novel arylpyrroline compounds of formula (I) which have excellent insecticidal activity and which can thus be used as an insecticide.
摘要翻译： 本发明涉及具有优异杀虫活性并因此可用作杀虫剂的式（I）的新型芳基吡咯啉化合物。
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公开(公告)号：US20100305124A1
公开(公告)日：2010-12-02
申请号：US12753185
申请日：2010-04-02
申请人： Martin FUSSLEIN , Ernst Rudolf Gesing , Markus Heil , Bernd Alig , Eva-Maria Franken , Olga Malsam , Arnd Voerste , Koichi Araki , Norio Sasaki , Sachio Kudo , Eiichi Shimojo , Teruyuki Ichihara , Masashi Ataka , Katsuhiko Shibuya
发明人： Martin FUSSLEIN , Ernst Rudolf Gesing , Markus Heil , Bernd Alig , Eva-Maria Franken , Olga Malsam , Arnd Voerste , Koichi Araki , Norio Sasaki , Sachio Kudo , Eiichi Shimojo , Teruyuki Ichihara , Masashi Ataka , Katsuhiko Shibuya
IPC分类号： A01N43/84 , C07D401/14 , C07D401/12 , C07D413/14 , A01N43/40 , A01N43/54 , A01N43/66 , A01P7/04 , A01P7/02 , A01P5/00 , A01P9/00
CPC分类号： C07D401/12 , A01N43/40 , A01N43/42 , A01N43/54 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/647 , A01N43/653 , A01N43/84 , C07D213/75 , C07D237/20 , C07D401/14
摘要： The present invention relates to aminopyridine and aminopyridazine derivatives of the general formula (I) in which R1, X, W and Q have the definitions given in the description, to a number of processes for preparing them, and to their use as insecticides.
摘要翻译： 本发明涉及通式（I）的氨基吡啶和氨基哒嗪衍生物，其中R1，X，W和Q具有说明书中给出的定义，其制备方法的许多方法及其作为杀虫剂的用途。
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公开(公告)号：US08536201B2
公开(公告)日：2013-09-17
申请号：US13519819
申请日：2010-12-23
申请人： Jun Mihara , Mamoru Hatazawa , Daiei Yamazaki , Norio Sasaki , Tetsuya Murata , Eiichi Shimojo , Teruyuki Ichihara , Masashi Ataka , Katsuhiko Shibuya , Hidetoshi Kishikawa , Ulrich Görgens
发明人： Jun Mihara , Mamoru Hatazawa , Daiei Yamazaki , Norio Sasaki , Tetsuya Murata , Eiichi Shimojo , Teruyuki Ichihara , Masashi Ataka , Katsuhiko Shibuya , Hidetoshi Kishikawa , Ulrich Görgens
IPC分类号： A61K31/4439 , A61K31/40 , A01N43/36 , A01N43/40 , C07D213/44 , C07D207/08
CPC分类号： C07D401/04 , C07D207/08
摘要： The present invention relates to novel pesticidal arylpyrrolidine compounds (arylpyrrolidines) having the general formula (I) wherein A, X1, X2, X3, X4, R1, R2, R3, R4, and G are as defined in the application and their use as pesticide, in particular for combating animal pests which occur in the agricultural and/or the veterinary field, as well as to a preparation methods for preparing such compounds.
摘要翻译： 本发明涉及具有通式（I）的新型农药芳基吡咯烷化合物（芳基吡咯烷），其中A，X 1，X 2，X 3，X 4，R 1，R 2，R 3，R 4和G如本申请中所定义， 杀虫剂，特别是用于对抗在农业和/或兽医领域中发生的动物害虫，以及制备这种化合物的制备方法。
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