Quinoline Derivatives and Their Use as Pesticides
    1.
    发明申请
    Quinoline Derivatives and Their Use as Pesticides 审中-公开
    喹啉衍生物及其作为农药的用途

    公开(公告)号:US20090029855A1

    公开(公告)日:2009-01-29

    申请号:US12282608

    申请日:2007-03-12

    CPC分类号: C07D215/12 C07D215/60

    摘要: This invention relates to quinoline derivatives of formula I wherein R1, R2, R3 are each independently halogen, hydroxy, cyano, amino, nitro, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C7-cycloalkyl, C3-C7-cycloalkyl-C1-C4-alkyl, C1-C6-alkoxy, C2-C6-alkenyloxy, C2-C6-alkynyloxy, C1-C4-alkoxy-C1-C4-alkoxy, C3-C7-cycloalkyl-C1-C4-alkoxy, C(OH)(CF3)2, C1-C6-haloalkyl, C1-C6-haloalkoxy, C1-C6-alkylthio, C1-C6-haloalkylthio, C1-C6-alkylsulfinyl, C1-C6-haloalkylsulfinyl, C1-C6-alkylsulfonyl, C1-C6-haloalkylsulfonyl, C(Ra)═O, C(Ra)═NORb, C(═O)ORx, or C(═O)NRxRy; Ra is hydrogen or C1-C4-alkyl; Rb is hydrogen, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl, C1-C4-haloalkyl, or C2-C4-haloalkenyl; Rx, Ry are each independently hydrogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy-C1-C4-alkyl, C1-C4-thioalkyl-C1-C4-alkyl, C1-C4-alkyl-S(═O)C1-C4-alkyl, C1-C4-alkyl-S(═O)2C1-C4-alkyl, C3-C6-cyloalkyl, C1-C4-alkyl-C3-C6-cycloalkyl, C3-C6-alkenyl, C3-C6-alkinyl; R4, R5, R6, R7 are each independently hydrogen, halogen, cyano, amino, nitro, hydroxy, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-haloalkyl, C1-C6-haloalkoxy, C1-C6-alkylthio, C1-C6-haloalkylthio, C1-C6-alkylsulfinyl, C1-C6-haloalkylsulfinyl, C1-C6-alkylsulfonyl, C1-C6-haloalkylsulfonyl, or C(═O)ORc; Rc is hydrogen, C1-C6-alkyl, C2-C6-alkenyl, or C2-C6-alkinyl; m and n are each independently 1, 2, 3, 4, or 5; p is 0, 1, 2, 3, 4, or 5; and the N-oxides, enantiomers, diastereomers and salts thereof, processes and intermediates for the preparation of compounds I, use of compounds I for combating insects, acarids, or nematodes and a method for treating, controlling, preventing or protecting animals against infestation or infection by parasites using compounds I.

    摘要翻译: 本发明涉及式I的喹啉衍生物,其中R 1,R 2,R 3各自独立地为卤素,羟基,氰基,氨基,硝基,C 1 -C 6烷基,C 2 -C 6 - 烯基,C 2 -C 6炔基,C 3 -C 7 - 环烷基,C 3 -C 7 - 环烷基-C 1 -C 4 - 烷基,C 1 -C 6 - 烷氧基,C 2 -C 6 - 烯氧基,C 2 -C 6 - 炔氧基,C 1 -C 4烷氧基-C 1 -C 4烷氧基,C 3 -C 7 - 环烷基 - C 1 -C 6烷氧基,C(OH)(CF 3)2,C 1 -C 6卤代烷基,C 1 -C 6卤代烷氧基,C 1 -C 6烷硫基,C 1 -C 6卤代烷硫基,C 1 -C 6烷基亚磺酰基, C 1 -C 6烷基磺酰基,C 1 -C 6卤代烷基磺酰基,C(R a)-O,C(R a)-NOR b,C(-O)OR x或C(-O)NR x R y; R a是氢或C 1 -C 4 - 烷基; R b是氢,C 1 -C 4 - 烷基,C 2 -C 4 - 烯基,C 2 -C 4 - 炔基,C 1 -C 4卤代烷基或C 2 -C 4 - 卤代烯基; R x,R y各自独立地为氢,C 1 -C 4 - 烷基,C 1 -C 4 - 卤代烷基,C 1 -C 4 - 烷氧基-C 1 -C 4烷基,C 1 -C 4 - 硫代烷基-C 1 -C 4烷基,C 1 -C 4烷基 - S(-O)C 1 -C 4 - 烷基,C 1 -C 4烷基-S(-O)2 C 1 -C 4烷基,C 3 -C 6 - 环烷基,C 1 -C 4烷基-C 3 -C 6环烷基,C 3 -C 6 - 烯基,C 3 -C 6 - 炔基; R4,R5,R6,R7各自独立地为氢,卤素,氰基,氨基,硝基,羟基,C1-C6-烷基,C1-C6-烷氧基,C1-C6-卤代烷基,C1-C6-卤代烷氧基,C1-C6- C 1 -C 6烷基亚磺酰基,C 1 -C 6烷基磺酰基,C 1 -C 6卤代烷基磺酰基或C(-O)OR c; R c是氢,C 1 -C 6 - 烷基,C 2 -C 6 - 烯基或C 2 -C 6 - 炔基; m和n各自独立地为1,2,3,4或5; p是0,1,2,3,4或5; 及其N-氧化物,对映异构体,非对映异构体及其盐,制备化合物I的方法和中间体,化合物I用于防治昆虫,螨虫或线虫的用途,以及用于治疗,控制,预防或保护动物免受感染或 使用化合物I的寄生虫感染

    Thiophene-Sulphonic Acid Picolyl Amides
    7.
    发明申请
    Thiophene-Sulphonic Acid Picolyl Amides 审中-公开
    噻吩磺酸吡啶基酰胺

    公开(公告)号:US20100222219A1

    公开(公告)日:2010-09-02

    申请号:US12438169

    申请日:2007-08-13

    CPC分类号: A01N43/40 C07D409/12

    摘要: The present invention relates to thiophene-sulfonic acid picolyl amides of the Formula (I), where RI to R7 and n are as defined in the claims and to the N-oxides, the agriculturally acceptable salts and the veterinarily acceptable salts of the compounds (I), with the proviso that if the thiophene ring is bonded to the sulfonyl group via position 2, R6 cannot be at position 5. The invention also relates to a process for preparing these compounds. Furthermore, the invention relates to the use of the compounds I and the N-oxides and the agriculturally acceptable salts thereof for combating phytopathogenic fungi (hereinafter referred to as harmful fungi). Additionally, the compounds (I), their N-oxides and salts can be used for controlling arthropodal pests. Furthermore, the invention relates to seed comprising a compound (I) or an N-oxide or agriculturally acceptable salt thereof.

    摘要翻译: 本发明涉及式(I)的噻吩 - 磺酸吡啶甲酰胺,其中R 1至R 7和n如权利要求中所定义,和N-氧化物,农业上可接受的盐和化合物的兽医学上可接受的盐 I),条件是如果噻吩环通过位置2与磺酰基键合,则R6不能在5位。本发明还涉及制备这些化合物的方法。 此外,本发明涉及化合物I和N-氧化物及其农业上可接受的盐对抗植物病原性真菌(以下称为有害真菌)的用途。 此外,化合物(I),其N-氧化物和盐可用于控制节肢动物害虫。 此外,本发明涉及包含化合物(I)或其N-氧化物或农业上可接受的盐的种子。

    Pyridin-4-ylmethylamides
    8.
    发明申请
    Pyridin-4-ylmethylamides 审中-公开
    吡啶-4-基甲基酰胺

    公开(公告)号:US20090069179A1

    公开(公告)日:2009-03-12

    申请号:US12279117

    申请日:2007-02-13

    CPC分类号: A01N43/40 C07D213/70

    摘要: The present invention relates to pyridin-4-ylmethylamides of the general formula (I), where R1 to R6 and n are as defined in the claims and to the N-oxides and the agriculturally acceptable salts of the compounds I. The invention also relates to a process for preparing these compounds. Furthermore, the invention relates to the use of the compounds I and the N-oxides and the agriculturally acceptable salts thereof for combating phytopathogenic fungi (hereinafter referred to as harmful fungi). Furthermore the compounds I, their N-oxides and salts can be used for controlling arthropodal pests.

    摘要翻译: 本发明涉及通式(I)的吡啶-4-基甲基酰胺,其中R 1至R 6和n如权利要求中所定义,以及化合物I的N-氧化物和农业上可接受的盐。本发明还涉及 涉及制备这些化合物的方法。 此外,本发明涉及化合物I和N-氧化物及其农业上可接受的盐对抗植物病原性真菌(以下称为有害真菌)的用途。 此外,化合物I,其N-氧化物和盐可用于防治节肢动物害虫。