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    Quinoline Derivatives and Their Use as Pesticides
    1.
    发明申请
    Quinoline Derivatives and Their Use as Pesticides 审中-公开
    喹啉衍生物及其作为农药的用途

    公开(公告)号：US20090029855A1

    公开(公告)日：2009-01-29

    申请号：US12282608

    申请日：2007-03-12

    申请人： Michael Puhl ,  Wassilios Grammenos ,  Joachim Rheinheimer ,  Jan Klaas Lohmann ,  Michael Rack ,  Liliana Parra Rapado ,  Christopher Koradin ,  Jurgen Langewald ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Hassan Oloumi-Sadeghi ,  Henry Van Tuyl Cotter ,  David G. Kuhn

    发明人： Michael Puhl ,  Wassilios Grammenos ,  Joachim Rheinheimer ,  Jan Klaas Lohmann ,  Michael Rack ,  Liliana Parra Rapado ,  Christopher Koradin ,  Jurgen Langewald ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Hassan Oloumi-Sadeghi ,  Henry Van Tuyl Cotter ,  David G. Kuhn

    IPC分类号： A01N25/26 ,  C07D215/14 ,  A01N43/42 ,  A01N59/26 ,  A01P5/00 ,  A01P7/04

    CPC分类号： C07D215/12 ,  C07D215/60

    摘要： This invention relates to quinoline derivatives of formula I wherein R1, R2, R3 are each independently halogen, hydroxy, cyano, amino, nitro, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C7-cycloalkyl, C3-C7-cycloalkyl-C1-C4-alkyl, C1-C6-alkoxy, C2-C6-alkenyloxy, C2-C6-alkynyloxy, C1-C4-alkoxy-C1-C4-alkoxy, C3-C7-cycloalkyl-C1-C4-alkoxy, C(OH)(CF3)2, C1-C6-haloalkyl, C1-C6-haloalkoxy, C1-C6-alkylthio, C1-C6-haloalkylthio, C1-C6-alkylsulfinyl, C1-C6-haloalkylsulfinyl, C1-C6-alkylsulfonyl, C1-C6-haloalkylsulfonyl, C(Ra)═O, C(Ra)═NORb, C(═O)ORx, or C(═O)NRxRy; Ra is hydrogen or C1-C4-alkyl; Rb is hydrogen, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl, C1-C4-haloalkyl, or C2-C4-haloalkenyl; Rx, Ry are each independently hydrogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy-C1-C4-alkyl, C1-C4-thioalkyl-C1-C4-alkyl, C1-C4-alkyl-S(═O)C1-C4-alkyl, C1-C4-alkyl-S(═O)2C1-C4-alkyl, C3-C6-cyloalkyl, C1-C4-alkyl-C3-C6-cycloalkyl, C3-C6-alkenyl, C3-C6-alkinyl; R4, R5, R6, R7 are each independently hydrogen, halogen, cyano, amino, nitro, hydroxy, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-haloalkyl, C1-C6-haloalkoxy, C1-C6-alkylthio, C1-C6-haloalkylthio, C1-C6-alkylsulfinyl, C1-C6-haloalkylsulfinyl, C1-C6-alkylsulfonyl, C1-C6-haloalkylsulfonyl, or C(═O)ORc; Rc is hydrogen, C1-C6-alkyl, C2-C6-alkenyl, or C2-C6-alkinyl; m and n are each independently 1, 2, 3, 4, or 5; p is 0, 1, 2, 3, 4, or 5; and the N-oxides, enantiomers, diastereomers and salts thereof, processes and intermediates for the preparation of compounds I, use of compounds I for combating insects, acarids, or nematodes and a method for treating, controlling, preventing or protecting animals against infestation or infection by parasites using compounds I.

    摘要翻译： 本发明涉及式I的喹啉衍生物，其中R 1，R 2，R 3各自独立地为卤素，羟基，氰基，氨基，硝基，C 1 -C 6烷基，C 2 -C 6 - 烯基，C 2 -C 6炔基，C 3 -C 7 - 环烷基，C 3 -C 7 - 环烷基-C 1 -C 4 - 烷基，C 1 -C 6 - 烷氧基，C 2 -C 6 - 烯氧基，C 2 -C 6 - 炔氧基，C 1 -C 4烷氧基-C 1 -C 4烷氧基，C 3 -C 7 - 环烷基 - C 1 -C 6烷氧基，C（OH）（CF 3）2，C 1 -C 6卤代烷基，C 1 -C 6卤代烷氧基，C 1 -C 6烷硫基，C 1 -C 6卤代烷硫基，C 1 -C 6烷基亚磺酰基， C 1 -C 6烷基磺酰基，C 1 -C 6卤代烷基磺酰基，C（R a）-O，C（R a）-NOR b，C（-O）OR x或C（-O）NR x R y; R a是氢或C 1 -C 4 - 烷基; R b是氢，C 1 -C 4 - 烷基，C 2 -C 4 - 烯基，C 2 -C 4 - 炔基，C 1 -C 4卤代烷基或C 2 -C 4 - 卤代烯基; R x，R y各自独立地为氢，C 1 -C 4 - 烷基，C 1 -C 4 - 卤代烷基，C 1 -C 4 - 烷氧基-C 1 -C 4烷基，C 1 -C 4 - 硫代烷基-C 1 -C 4烷基，C 1 -C 4烷基 - S（-O）C 1 -C 4 - 烷基，C 1 -C 4烷基-S（-O）2 C 1 -C 4烷基，C 3 -C 6 - 环烷基，C 1 -C 4烷基-C 3 -C 6环烷基，C 3 -C 6 - 烯基，C 3 -C 6 - 炔基; R4，R5，R6，R7各自独立地为氢，卤素，氰基，氨基，硝基，羟基，C1-C6-烷基，C1-C6-烷氧基，C1-C6-卤代烷基，C1-C6-卤代烷氧基，C1-C6- C 1 -C 6烷基亚磺酰基，C 1 -C 6烷基磺酰基，C 1 -C 6卤代烷基磺酰基或C（-O）OR c; R c是氢，C 1 -C 6 - 烷基，C 2 -C 6 - 烯基或C 2 -C 6 - 炔基; m和n各自独立地为1,2,3,4或5; p是0，1，2，3，4或5; 及其N-氧化物，对映异构体，非对映异构体及其盐，制备化合物I的方法和中间体，化合物I用于防治昆虫，螨虫或线虫的用途，以及用于治疗，控制，预防或保护动物免受感染或 使用化合物I的寄生虫感染

    Method for Preparation of Piperazindione Derivatives
    10.
    发明申请
    Method for Preparation of Piperazindione Derivatives 审中-公开
    哌嗪二酮衍生物的制备方法

    公开(公告)号：US20110144336A1

    公开(公告)日：2011-06-16

    申请号：US13058677

    申请日：2009-07-30

    申请人： Thomas Zierke ,  Eike Hupe ,  Michael Rack ,  Liliana Parra Rapado ,  Timo Frassetto

    发明人： Thomas Zierke ,  Eike Hupe ,  Michael Rack ,  Liliana Parra Rapado ,  Timo Frassetto

    IPC分类号： C07D241/08

    CPC分类号： C07D241/08

    摘要： A process for preparing piperazinedione derivatives of the formula I in which R1 is hydrogen, alkyl, alkenyl, alkynyl and alkylcarbonyl, R2 is hydrogen, alkyl, alkenyl, C3-C4-alkynyl and C(═O)R11, R3, R4 are each hydrogen, alkyl and haloalkyl, where the groups may be substituted, which comprises reacting amines of the formula II H2N—R1  II in which R1 is hydrogen and alkyl which may optionally be substituted with N-acylated amino acid derivatives of the formula III in which X is halogen, Y is halogen, alkoxy or phenyloxy which may be substituted and R2, R3 and R4 are each as defined at the outset, under basic conditions in an aqueous solvent.

    摘要翻译： 其中R 1是氢，烷基，烯基，炔基和烷基羰基，R 2是氢，烷基，烯基，C 3 -C 4炔基和C（= O）R 11，R 3，R 4各自是式I的哌嗪二酮衍生物的方法 氢，烷基和卤代烷基，其中基团可以被取代，其包括使式II的其中R 1是氢的式IIH 2 N-R 1 II的烷基和可以被式III的N-酰化的氨基酸衍生物任选取代的烷基，其中 X是卤素，Y是可以被取代的卤素，烷氧基或苯氧基，R2，R3和R4各自在碱性条件下在水性溶剂中首先定义。