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公开(公告)号:US08445689B2
公开(公告)日:2013-05-21
申请号:US13444286
申请日:2012-04-11
申请人: Nneka T. Breaux , Michael R. Loso , Timothy C. Johnson , Jonathan M. Babcock , Benjamin M. Nugent , Timothy P. Martin , Annette Vitale Brown , Ronald Ross, Jr. , William C. Lo , Matthias S. Ober
发明人: Nneka T. Breaux , Michael R. Loso , Timothy C. Johnson , Jonathan M. Babcock , Benjamin M. Nugent , Timothy P. Martin , Annette Vitale Brown , Ronald Ross, Jr. , William C. Lo , Matthias S. Ober
IPC分类号: C07D213/56 , A61K31/44
CPC分类号: C07C381/10 , A01N43/40 , A01N47/34 , A01N47/36 , A01N47/44 , C07C2601/02 , C07C2601/14 , C07C2603/18 , C07D213/32 , C07D401/12 , C07D405/12 , C07D413/12
摘要: Compounds having the following generic formula are disclosed.
摘要翻译: 公开了具有以下通式的化合物。
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公开(公告)号:US08178685B2
公开(公告)日:2012-05-15
申请号:US12962114
申请日:2010-12-07
申请人: Nneka T. Breaux , Michael R. Loso , Timothy C. Johnson , Jonathan M. Babcock , Benjamin M. Nugent , Timothy P. Martin , Annette Vitale Brown , Ronald Ross, Jr. , William C. Lo , Matthias S. Ober
发明人: Nneka T. Breaux , Michael R. Loso , Timothy C. Johnson , Jonathan M. Babcock , Benjamin M. Nugent , Timothy P. Martin , Annette Vitale Brown , Ronald Ross, Jr. , William C. Lo , Matthias S. Ober
IPC分类号: C07D213/56 , A61K31/44
CPC分类号: C07C381/10 , A01N43/40 , A01N47/34 , A01N47/36 , A01N47/44 , C07C2601/02 , C07C2601/14 , C07C2603/18 , C07D213/32 , C07D401/12 , C07D405/12 , C07D413/12
摘要: Compounds having the following generic formula are disclosed.
摘要翻译: 公开了具有以下通式的化合物。
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公开(公告)号:US08815271B2
公开(公告)日:2014-08-26
申请号:US13285595
申请日:2011-10-31
申请人: Maurice C. H. Yap , Ann M. Buysse , Daniel Knueppel , Yu Zhang , Negar Garizi , Noormohamed M. Niyaz , Christian T. Lowe , Ricky Hunter , Tony K. Trullinger , David A. Demeter , Dan Pernich , Carl Deamicis , Ronald Ross, Jr. , Timothy C. Johnson
发明人: Maurice C. H. Yap , Ann M. Buysse , Daniel Knueppel , Yu Zhang , Negar Garizi , Noormohamed M. Niyaz , Christian T. Lowe , Ricky Hunter , Tony K. Trullinger , David A. Demeter , Dan Pernich , Carl Deamicis , Ronald Ross, Jr. , Timothy C. Johnson
IPC分类号: A01N25/08 , A01N25/28 , A01N25/32 , A01N61/00 , A01N63/00 , A01N43/40 , C07D401/04 , C07D417/14 , A01N43/56 , A01N47/36 , A01N47/18 , C07D401/14 , A61K45/06
CPC分类号: C07D417/14 , A01N25/00 , A01N43/12 , A01N43/56 , A01N43/653 , A01N43/74 , A01N43/76 , A01N43/78 , A01N43/80 , A01N47/18 , A01N47/36 , A01N47/40 , A01N51/00 , A61K31/4439 , A61K31/506 , A61K45/06 , C07D401/04 , C07D401/14 , C07D403/04 , C07D405/14 , C07D409/14 , C07D413/14
摘要: This document discloses molecules having the following formula (“Formula One”): and processes related thereto.
摘要翻译: 该文献公开了具有下式(“一级方程式”)的分子及其相关的方法。
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公开(公告)号:US08350044B2
公开(公告)日:2013-01-08
申请号:US12773062
申请日:2010-05-04
申请人: Tony K. Trullinger , Ricky Hunter , Negar Garizi , Maurice C. H. Yap , Ann M. Buysse , Dan Pernich , Timothy C. Johnson , Kristy Bryan , Carl Deamicis , Yu Zhang , Noormohamed M. Niyaz , CaSandra L. McLeod , Ronald Ross, Jr. , Yuanming Zhu , Peter L. Johnson , Joseph D. Eckelbarger , Marshall H. Parker
发明人: Tony K. Trullinger , Ricky Hunter , Negar Garizi , Maurice C. H. Yap , Ann M. Buysse , Dan Pernich , Timothy C. Johnson , Kristy Bryan , Carl Deamicis , Yu Zhang , Noormohamed M. Niyaz , CaSandra L. McLeod , Ronald Ross, Jr. , Yuanming Zhu , Peter L. Johnson , Joseph D. Eckelbarger , Marshall H. Parker
IPC分类号: C07D417/04 , A01N43/40
CPC分类号: A01N43/78 , A01N43/40 , C07D417/04 , C07D417/14
摘要: This document discloses molecules having the following formula (“Formula I”):
摘要翻译: 该文献公开了具有下式(式I)的分子:
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5.Process for the preparation of 2-substituted-5-(1-alkylthio)alkylpyridines 有权
标题翻译: 2-取代-5-(1-烷硫基)烷基吡啶的制备方法公开(公告)号:US07709650B2
公开(公告)日:2010-05-04
申请号:US12392664
申请日:2009-02-25
IPC分类号: C07D213/00 , C07D213/08
CPC分类号: C07D213/32
摘要: 2-Substituted-5-(1-alkylthio)alkylpyridines are produced efficiently and in high yield from a non-pyridine source by cyclization.
摘要翻译: 2-取代的5-(1-烷硫基)烷基吡啶通过环化从非吡啶源有效且高产率地制备。
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6.Process for the preparation of 2-substituted-5-(1-alkylthio)alkylpyridines 有权
标题翻译: 2-取代-5-(1-烷硫基)烷基吡啶的制备方法公开(公告)号:US08129539B2
公开(公告)日:2012-03-06
申请号:US12722978
申请日:2010-03-12
IPC分类号: C07D213/00
CPC分类号: C07D213/32
摘要: 2-Substituted-5-(1-alkylthio)alkylpyridines are produced efficiently and in high yield from a non-pyridine source by cyclization.
摘要翻译: 2-取代的5-(1-烷硫基)烷基吡啶通过环化从非吡啶源有效且高产率地制备。
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公开(公告)号:US5958426A
公开(公告)日:1999-09-28
申请号:US824646
申请日:1997-03-24
IPC分类号: C12P13/00 , A01N33/08 , A01N37/20 , A01N49/00 , A01N57/12 , A61K31/66 , A61K45/00 , A61P3/08 , A61P3/10 , A61P29/00 , A61P35/00 , A61P43/00 , C07F9/09 , C07F9/113 , C12P13/02 , C12R1/645
CPC分类号: A61K31/661 , A01N33/08 , A01N37/20 , A01N49/00 , A01N57/12 , A61K45/00 , C07F9/091 , C07F9/113 , C12P13/02
摘要: A process for novel sphingolipids and other secondary sphingosine-based compounds is provided which comprises the culturing of an appropriate fungus, harvesting mycelium from the fungus and isolating the sphingolipid from the mycelium. The sphingosine-based materials inhibit protein kinase C, provide an anti-inflammatory effect or provide an anti-tumor effect; furthermore, these sphingosine-based materials provide protection for plants against pathogenic microorganisms.
摘要翻译: 提供新型鞘脂和其它次级鞘氨醇类化合物的方法,其包括培养合适的真菌,从真菌中收获菌丝体并从菌丝体中分离鞘脂。 基于鞘氨醇的物质抑制蛋白激酶C,提供抗炎作用或提供抗肿瘤作用; 此外,这些基于鞘氨醇的材料为防止病原微生物的植物提供保护。
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8.Dihydropyridazinones, pyridazinones and related compounds as fungicides 失效
标题翻译: 二氢哒嗪酮,哒嗪酮和相关化合物作为杀真菌剂公开(公告)号:US5631254A
公开(公告)日:1997-05-20
申请号:US467384
申请日:1995-06-06
IPC分类号: A01N43/40 , A01N43/42 , A01N43/54 , A01N43/58 , A01N43/60 , A01N43/62 , A01N43/653 , A01N43/72 , A01N43/80 , A01N43/82 , A01N43/88 , B27K3/34 , C07D213/64 , C07D213/85 , C07D215/22 , C07D215/227 , C07D237/04 , C07D237/14 , C07D237/18 , C07D237/26 , C07D237/32 , C07D237/36 , C07D239/36 , C07D243/02 , C07D243/04 , C07D273/04 , C07D285/34 , C07D401/04 , C07D403/04 , C07D405/06 , C07D405/10 , C07D407/06 , C07D409/04 , C07D409/06 , C07D413/06 , C07D521/00 , C07F7/08 , A61K31/50 , C07D295/03
CPC分类号: A01N43/40 , A01N43/42 , A01N43/54 , A01N43/58 , A01N43/60 , A01N43/62 , A01N43/653 , A01N43/80 , A01N43/82 , A01N43/88 , C07D213/64 , C07D213/85 , C07D215/227 , C07D231/12 , C07D233/56 , C07D237/04 , C07D237/18 , C07D237/26 , C07D237/32 , C07D237/36 , C07D239/36 , C07D243/02 , C07D249/08 , C07D273/04 , C07D285/34 , C07D401/04 , C07D403/04 , C07D405/06 , C07D405/10 , C07D409/04 , C07D409/06 , C07D413/06 , C07F7/0812
摘要: This invention relates to substituted dihydropyridazinones, pyridazinones and related compounds, of the formula ##STR1## wherein A, Q, D and R1 are as defined within, compositions containing these compounds and methods of controlling agricultural and mammalian fungal diseases.
摘要翻译: 本发明涉及下式的取代二氢哒嗪酮,哒嗪酮和相关化合物,其中A,Q,D和R 1如含有这些化合物的组合物和控制农业和哺乳动物真菌疾病的方法。
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9.2-alkynyl-6-pyridin-2-yl-pyridazinones, 2-alkynyl-6-pyridin-2-yl-dihydropyridazinones, 2-alkynyl-6-pyrimidin-2-yl-pyridazinones and 2-alkynyl-6-pyrimidin-2-yl-dihydropyridazinones and their use as fungicides 失效
标题翻译: 2-炔基-6-吡啶-2-基 - 哒嗪酮,2-炔基-6-吡啶-2-基 - 二氢哒嗪酮,2-炔基-6-嘧啶-2-基 - 哒嗪酮和2-炔基-6-嘧啶-2-基 - 二氢哒嗪酮及其作为杀真菌剂的用途公开(公告)号:US08426412B2
公开(公告)日:2013-04-23
申请号:US12420081
申请日:2009-04-08
申请人: Martha Kelly , Ronald Ross, Jr. , David H. Young
发明人: Martha Kelly , Ronald Ross, Jr. , David H. Young
IPC分类号: C07D401/04 , C07D403/04 , A61K31/501 , A01N63/00
CPC分类号: C07D401/04 , A01N43/58 , C07D403/04
摘要: This invention relates to certain novel 2-alkynyl-6-pyridin-2-yl-pyridazinones, 2-alkynyl-6-pyridin-2-yl-dihydropyridazinones, 2-alkynyl-6-pyrimidin-2-yl-pyridazinones and 2-alkynyl-6-pyrimidin-2-yl-dihydropyridazinones such as those illustrated in Formula I and to the use of these compounds for control of fungal pathogens of plants and mammals.
摘要翻译: 本发明涉及某些新的2-炔基-6-吡啶-2-基 - 哒嗪酮,2-炔基-6-吡啶-2-基 - 二氢哒嗪酮,2-炔基-6-嘧啶-2-基 - 哒嗪酮和2- 炔基-6-嘧啶-2-基 - 二氢哒嗪酮,如式I所示的那些,以及这些化合物用于控制植物和哺乳动物真菌病原体的用途。
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公开(公告)号:US5726176A
公开(公告)日:1998-03-10
申请号:US740546
申请日:1996-10-30
IPC分类号: A01N43/40 , A01N43/42 , A01N43/54 , A01N43/58 , A01N43/60 , A01N43/62 , A01N43/653 , A01N43/72 , A01N43/80 , A01N43/82 , A01N43/88 , B27K3/34 , C07D213/64 , C07D213/85 , C07D215/22 , C07D215/227 , C07D237/04 , C07D237/14 , C07D237/18 , C07D237/26 , C07D237/32 , C07D237/36 , C07D239/36 , C07D243/02 , C07D243/04 , C07D273/04 , C07D285/34 , C07D401/04 , C07D403/04 , C07D405/06 , C07D405/10 , C07D407/06 , C07D409/04 , C07D409/06 , C07D413/06 , C07D521/00 , C07F7/08 , A61K31/50 , C07D295/03
CPC分类号: A01N43/40 , A01N43/42 , A01N43/54 , A01N43/58 , A01N43/60 , A01N43/62 , A01N43/653 , A01N43/80 , A01N43/82 , A01N43/88 , C07D213/64 , C07D213/85 , C07D215/227 , C07D231/12 , C07D233/56 , C07D237/04 , C07D237/18 , C07D237/26 , C07D237/32 , C07D237/36 , C07D239/36 , C07D243/02 , C07D249/08 , C07D273/04 , C07D285/34 , C07D401/04 , C07D403/04 , C07D405/06 , C07D405/10 , C07D409/04 , C07D409/06 , C07D413/06 , C07F7/0812
摘要: This invention relates to substituted dihydropyridazinones, pyridazinones and related compounds, of the formula ##STR1## wherein A, Q, D and R1 are as defined within, compositions containing these compounds and methods of controlling agricultural and mammalian fungal diseases.
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