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公开(公告)号：US3686241A
公开(公告)日：1972-08-22
申请号：US3686241D
申请日：1969-02-03
Applicant: ROUSSEL UCLAF
Inventor： AMIARD GASTON , NOMINE GERARD , TORELLI VESPERTO
IPC: C07B61/00 , C07C59/76 , C07C59/82 , C07C62/38 , C07C69/757 , C07J1/00 , C07J75/00 , C07C69/76 , C09F5/08
CPC classification number: C07J1/00 , C07B61/00 , C07C59/76 , C07C59/82 , C07C62/38 , C07C69/757 , C07J75/00
Abstract: NOVEL 1B-OXY-4-(CARBOXYMETHYL)-5-(P-LOWER ALKOXYPHENYL)-7A-Y-INDANES WHEREIN Y IS AN ALKYL OF 1 TO 18 CARBON ATOMS WHICH ARE USEFUL INTERMEDIATES FOR THE TOTAL SYNTHESIS OF 13B-Y-$1,3,5(10)-GONATRIENES.
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公开(公告)号：US3707540A
公开(公告)日：1972-12-26
申请号：US3707540D
申请日：1966-12-07
Applicant: ROUSSEL UCLAF
Inventor： AMIARD GASTON , HEYMES RENE
IPC: C07D307/60 , C07D501/08 , C07D513/04 , G03C5/39 , C07D93/08 , C07D99/24
CPC classification number: C07D513/04 , C07D307/60 , G03C5/39
Abstract: LACTONES OF 2-(CARBONYL-AMINO-METHYL)-5-HYDROXYMETHYL-3,6-DIHYDRO-2H-1,3-THIAZINE-4 -CARBOXYLIC ACIDS USEFUL AS INTERMEDIATES FOR ANTIBIOTICS OF THE C-CEPHALOSPORINE FAMILY AND THEIR PREPARATION. THE INVENTION RELATES TO NOVEL DIHYDRO-1,3-THIAZINE COMPOUNDS OF THE FORMULA
2-(R-OOC-CH(-Y)-),7-(O=)-1,2,5,7-TETRAHYDRO-4H-FURO(3,4-D)
(3,1)THIAZINE
WHEREIN R IS SELECTED FROM THE GROUP CONSISTING OF ALKYL AND ARALKYL, Y IS SELECTED FROM THE GROUP CONSISTING OF -HN-AC, PHTHALIMIDO AND-NH-R'',R'' IS SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, ALKYL AND ARALKYL AND AC IS THE ACYL RADICAL OF AN ORGANIC CARBOXYLIC ACID OF 1 TO 18 CARBON ATOMS AND TO A NOVEL PROCESS FOR THE PREPARATION OF THE SAID COMPOUNDS.-
公开(公告)号：US3658802A
公开(公告)日：1972-04-25
申请号：US3658802D
申请日：1969-06-26
Applicant: ROUSSEL UCLAF
Inventor： HEYMES RENE , AMIARD GASTON , NOMINE GERARD
IPC: C07D501/46 , A61K31/545 , C07D20060101 , C07D501/04 , C07D501/38 , C07D501/60 , C07D99/24
CPC classification number: C07D501/38
Abstract: THIS INVENTION RELATES TO A CEPHALOSPORINE DERIVATIVE OF THE FORMULA
4-(R1-NH-),8-R2-1,3,4,4A,6,7-HEXAHYDRO-8H-AZETO(2,1-B)-
PYRROLO(3,4-D)(1,3)-THIAZINE
WHEREIN R1 REPRESENTS THE ACYL OF AN ORGANIC ACID AND R2 REPRESENTS A MEMBER SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, ALKYL, SUBSTITUTED ALKYL, ARYL AND SUBSTITUTED ARYL. THESE COMPOUNDS HAVE PARTICULARLY MARKED ANTIBIOTIC PROPERTIES, PARTICULARLY, A REMARKABLE ACTIVITY AGAINST STAPHYLOCOCCI.-
Patent Agency Ranking4.发明授权Racemic and optically active 6h 7h-cis-7-amino-desacetylcephalosporanic acid derivatives and process 失效种间和光活性的6H 7H-CIS-7-氨基 - 脱乙酰壳多糖类衍生物和方法
公开(公告)号：US3642788A
公开(公告)日：1972-02-15
申请号：US3642788D
申请日：1967-03-13
Applicant: ROUSSEL UCLAF
Inventor： HEYMES RENE , AMIARD GASTON
IPC: C07D501/08 , C07D501/18 , C07D513/04 , C07D99/24
CPC classification number: C07D513/04
Abstract: THIS INVENTION RELATES TO A COMPOUND SELECTED FROM THE GROUP CONSISTING OF (1) A RACEMIC 6H,7H-CIS-7-AMINODESACETYLCEPHALOSPORANIC ACID DERIVATIVE OF THE FORMULA
2,3-(-COO-CH2-),7-(R-NH-)-2-CEPHEM
WHEREIN R IS SELECTED FROM THE GROUP CONSISTING OF HYDROGEN AND TRIPHENYLMETHYL, (2) IS OPTICALLY ACTIVE ANTIPODES AND (3) WHEN R IS HYDROGEN THEIR ACID ADDITION SALTS. THE INVENTION ALSO RELATES TO THE PROCESS OF PREPARING THESE COMPOUNDS. THESE COMPOUNDS ARE INTERMEDIATES USEFUL IN THE PREPARATION OF CEPHALOSPORIN ANTIBIOTICS AND THE 7-THIENYLACETYLAMINO DERIVATIVE POSSESSES AN ANTIBIOTIC ACTIVITY.-
5.发明授权Salts of chrysanthemic acid with 1-p-nitrophenyl - 2-n,n - dimethyl-aminopropane-1,3-diols 失效1-N-硝基苯基-2-N，N-二甲基氨基丙基-1,3-二醇的盐酸盐
公开(公告)号：US3590077A
公开(公告)日：1971-06-29
申请号：US3590077D
申请日：1968-07-05
Applicant: ROUSSEL UCLAF
Inventor： MULLER GEORGES , AMIARD GASTON , POITTEVIN ANDRE , TORELLI VESPERTO
IPC: C07D317/72 , C07C91/20
CPC classification number: C07D317/72
Abstract: OPTICAL ISOMERS OF 1-P-NITROPHENYL-2-N,N-DIMETHYLAMINO-PROPANE-1,3-DIOL AND ACID ADDITION SALTS THEREOF, USEFUL FOR THE SEPARATION OF RACEMIC COMPOUNDS AND PREPARATION THEREOF.
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6.发明授权D(_)-and l(+)-threo-1-p-nitrophenyl-2-n,n-dimethylamino-propane 1,3 - diols and the salts thereof 失效D（_） - 和L（+） - THREO-1-P-NITROPHENYL-2-N，N-二甲基氨基丙烷1,3-二醇及其盐
公开(公告)号：US3499929A
公开(公告)日：1970-03-10
申请号：US3499929D
申请日：1967-01-19
Applicant: ROUSSEL UCLAF
Inventor： MULLER GEORGES , AMIARD GASTON , POITTEVIN ANDRE , TORELLI VESPERTO
IPC: C07D317/72 , C07C91/16
CPC classification number: C07D317/72
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公开(公告)号：US3478062A
公开(公告)日：1969-11-11
申请号：US3478062D
申请日：1969-02-03
Applicant: ROUSSEL UCLAF
Inventor： AMIARD GASTON , NOMINE GERARD , TORELLI VESPERTO
IPC: C07B61/00 , C07C59/76 , C07C59/82 , C07C62/38 , C07C69/757 , C07J1/00 , C07J75/00 , C07D5/32 , C07C49/54 , C07C167/02
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公开(公告)号：US3449382A
公开(公告)日：1969-06-10
申请号：US3449382D
申请日：1966-07-27
Applicant: ROUSSEL UCLAF
Inventor： AMIARD GASTON , NOMINE GERARD , TORELLI VESPERTO
IPC: C07B61/00 , C07C59/76 , C07C59/82 , C07C62/38 , C07C69/757 , C07J1/00 , C07J75/00 , C07C167/02 , C07C61/36 , C07C169/08
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