Pesticidal tautomers of 3-aryl-pyrrolidine-2,4-diones and use thereas
    1.
    发明授权
    Pesticidal tautomers of 3-aryl-pyrrolidine-2,4-diones and use thereas 失效
    3-芳基 - 吡咯烷-2,4-二酮的杀虫互变异构体

    公开(公告)号:US5045560A

    公开(公告)日:1991-09-03

    申请号:US460208

    申请日:1990-01-02

    摘要: Insecticidal, acaricidal, herbicidal and antimycotic 3-aryl-pyrrolidine-2,4-diones of the formula ##STR1## in which X represents alkyl, halogen or alkoxy,Y represents hydrogen, alkyl, halogen, alkoxy or halogenoalkyl,Z represents alkyl, halogen or alkoxy,n represents a number from 0-3,R represents hydrogen or represents the groups --CO--R.sup.1 or --CO--O--R.sup.2, in whichR.sup.1 represents alkyl, alkenyl, alkoxyalkyl, alkylthioalkyl, polyalkoxyalkyl or cycloalkyl which can be interrupted by hetero atoms, each of which radicals is optionally substituted by halogen, or represents optionally substituted phenyl, optionally substituted phenylalkyl, substituted hetaryl, substituted phenoxyalkyl or substituted hetaryloxyalkyl, or represents optionally substituted phenyl, optionally substituted phenylalkyl, substituted hetaryl, substituted phenoxyalkyl and substituted hetaryloxyalkyl, andR.sup.2 represents alkyl, alkenyl, alkoxyalkyl, polyalkoxyalkyl or optionally substituted phenyl or cycloalkyl, each of which radicals is optionally substituted by halogen,A represents alkyl, alkenyl, alkinyl, alkoxyalkyl, polyalkoxyalkyl, alkylthioalkyl, or cycloalkyl which is optionally interrupted by a hetero atom, each of which radicals is optionally substituted by halogen, or represents arylalkyl which is optionally substituted by halogen, alkyl, halogenoalkyl, alkoxy or nitro,B and C* independently of one another represent hydrogen, alkyl or alkoxyalkyl.

    摘要翻译: 式(I)的杀虫,杀螨,除草和抗真菌性3-芳基 - 吡咯烷-2,4-二酮其中X代表烷基,卤素或烷氧基,Y代表氢,烷基,卤素,烷氧基或卤代烷基,Z 表示烷基,卤素或烷氧基,n表示0-3的数,R表示氢或表示基团-CO-R1或-CO-O-R2,其中R1表示烷基,烯基,烷氧基烷基,烷硫基烷基,聚烷氧基烷基或环烷基 任何取代的苯基,取代的杂芳基,取代的苯氧基烷基或取代的噻唑烷基,或代表任意取代的苯基,任选取代的苯基烷基,取代的杂芳基, 取代的苯氧基烷基和取代的硫代氧基烷基,R 2表示烷基,链烯基,烷氧基烷基,聚烷氧基烷基或任选取代的苯基或环烷基,各w 任选被卤素取代的基团,A代表烷基,链烯基,炔基,烷氧基烷基,聚烷氧基烷基,烷硫基烷基或环烷基,任选被杂原子间隔,每个基团任选被卤素取代,或表示任选取代的芳基烷基 卤素,烷基,卤代烷基,烷氧基或硝基,B和C *彼此独立地表示氢,烷基或烷氧基烷基。

    Pesticidal 3-aryl-pyrrolidine-2,4-diones
    2.
    发明授权
    Pesticidal 3-aryl-pyrrolidine-2,4-diones 失效
    杀虫剂3-芳基 - 吡咯烷-2,4-二酮

    公开(公告)号:US5186737A

    公开(公告)日:1993-02-16

    申请号:US678479

    申请日:1991-04-01

    摘要: Insecticidal, acaricidal, herbicidal and antimycotic 3-aryl-pyrrolidine-2,4-diones of the formula ##STR1## in which X represents alkyl, halogen or alkoxy,Y represents hydrogen, alkyl, halogen, alkoxy or halogenoalkyl,Z represents alkyl, halogen or alkoxy,n represents a number from 0-3,R represents hydrogen or represents the groups --CO--R.sup.1 or --CO--O--R.sup.2, in whichR.sup.1 represents alkyl, alkenyl, alkoxyalkyl, alkylthioalkyl, polyalkoxyalkyl or cycloalkyl which can be interrupted by hetero atoms, each of which radicals is optionally substituted by halogen, or represents optionally substituted phenyl, optionally substituted phenylalkyl, substituted hetaryl, substituted phenoxyalkyl or substituted hetaryloxyalkyl, or represents optionally substituted phenyl, optionally substituted phenylalkyl, substituted hetaryl, substituted phenoxyalkyl and substituted hetaryloxyalkyl, andR.sup.2 represents alkyl, alkenyl, alkoxyalkyl, polyalkoxyalkyl or optionally substituted phenyl or cycloalkyl, each of which radicals is optionally substituted by halogen,A represents alkyl, alkenyl, alkinyl, alkoxyalkyl, polyalkoxyalkyl, alkylthioalkyl, or cycloalkyl which is optionally interrupted by a hetero atom, each of which radicals is optionally subsituted by halogen, or represents arylalkyl which is optionally substituted by halogen, alkyl, halogenoalkyl, alkoxy or nitro,B and C* independently of one another represent hydrogen, alkyl or alkoxyalkyl.

    摘要翻译: 式(I)的杀虫,杀螨,除草和抗真菌性3-芳基 - 吡咯烷-2,4-二酮其中X代表烷基,卤素或烷氧基,Y代表氢,烷基,卤素,烷氧基或卤代烷基,Z 表示烷基,卤素或烷氧基,n表示0-3的数,R表示氢或表示基团-CO-R1或-CO-O-R2,其中R1表示烷基,烯基,烷氧基烷基,烷硫基烷基,聚烷氧基烷基或环烷基 任何取代的苯基,取代的杂芳基,取代的苯氧基烷基或取代的噻唑烷基,或代表任意取代的苯基,任选取代的苯基烷基,取代的杂芳基, 取代的苯氧基烷基和取代的硫代氧基烷基,R 2表示烷基,链烯基,烷氧基烷基,聚烷氧基烷基或任选取代的苯基或环烷基,各w 任选被卤素取代的基团,A代表烷基,烯基,炔基,烷氧基烷基,聚烷氧基烷基,烷硫基烷基或环烷基,任选被杂原子中断,每个基团任选被卤素取代,或表示任选取代的芳基烷基 卤素,烷基,卤代烷基,烷氧基或硝基,B和C *彼此独立地表示氢,烷基或烷氧基烷基。

    Herbicidal 4-alkoxy- and 4-(substituted)amino-arylpyrrolinone derivatives
    3.
    发明授权
    Herbicidal 4-alkoxy- and 4-(substituted)amino-arylpyrrolinone derivatives 失效
    除草剂4-烷氧基 - 和4-(取代的)氨基 - 吡咯烷酮衍生物

    公开(公告)号:US5191089A

    公开(公告)日:1993-03-02

    申请号:US565536

    申请日:1990-08-09

    CPC分类号: A01N43/36 C07D207/38

    摘要: Herbicidal 4-alkoxy- and 4-(substituted)amino-arylpyrrolinone derivatives of the formula ##STR1## in which X and Y independently of one another represent hydrogen, halogen, alkyl, alkoxy, halogenoalkyl or in each case unsubstituted or substituted aryloxy or arylthio,Z represents halogen, alkyl or alkoxy,n represents the number 0, 1, 2 or 3,A represents in each case unsubstituted or in each case halogen-substituted alkyl, alkenyl, alkynyl, alkoxyalkyl, polyalkoxyalkyl or alkylthioalkyl, cycloalkyl which is optionally interrupted by hetero atoms, arylalkyl which is unsubstituted or substituted by halogen, alkyl, halogenoalkyl, alkoxy and/or nitro, unsubstituted aryl or aryl substituted by a member selected from the group consisting of halogen, alkyl, alkoxy, halogenoalkyl, halogenoalkoxy and phenoxy or phenylthio which are in each case unsubstituted or substituted by halogen, alkyl, alkoxy, halogenoalkyl and/or halogenoalkoxy,B represents hydroxyl, alkoxy, halogenoalkoxy or cycloalkoxy, the cycloalkyl radical being unsubstituted or substituted by halogen and/or alkyl, orB represents the group ##STR2## wherein C and D independently of one another represent hydrogen, alkyl, alkenyl, alkoxyalkyl, alkylthioalkyl or polyalkoxyalkyl, cycloalkyl which is optionally interrupted by hetero atoms or in each case unsubstituted or substituted phenyl, phenylalkyl, phenoxyalkyl, hetaryl or hetarylalkyl, orC and D together with the nitrogen atom to which they are bonded, form a 3- to 9-membered, optionally substituted ring which is optionally interrupted by the further hetero atoms,with the proviso that at least one radical X, Y or Z does not represent chlorine or methyl if B represents hydroxyl and A has a meaning other than optionally substituted aryl.

    摘要翻译: 式(I)的除草4-烷氧基 - 和4-(取代的)氨基 - 芳基吡咯烷酮衍生物,其中X和Y彼此独立地代表氢,卤素,烷基,烷氧基,卤代烷基或在各种情况下是未取代或取代的 芳氧基或芳硫基,Z表示卤素,烷基或烷氧基,n表示数0,1,2或3,A表示各自为未取代的或在各种情况下为卤素取代的烷基,烯基,炔基,烷氧基烷基,聚烷氧基烷基或烷硫基烷基,环烷基 烷基,卤代烷基,烷氧基和/或硝基,未经取代的芳基或被选自卤素,烷基,烷氧基,卤代烷基,卤代烷氧基的成员所取代的芳基, 苯氧基或苯硫基,其各自为未被取代或被卤素,烷基,烷氧基,卤代烷基和/或卤代烷氧基取代,B代表羟基,烷氧基,卤代烷氧基或环 烷氧基,环烷基是未取代的或被卤素和/或烷基取代,或B表示基团,其中C和D彼此独立地表示氢,烷基,烯基,烷氧基烷基,烷硫基烷基或聚烷氧基烷基,任选地中断的环烷基 通过杂原子或在每种情况下未取代或取代的苯基,苯基烷基,苯氧基烷基,杂芳基或杂芳基烷基,或C和D与它们所键合的氮原子一起形成3至9元任选取代的环,其任选地 被另外的杂原子中断,条件是至少一个基团X,Y或Z不表示氯或甲基,如果B表示羟基,并且A具有除任选取代的芳基以外的含义。

    Herbicidal thiazolecarboxamide derivatives
    6.
    发明授权
    Herbicidal thiazolecarboxamide derivatives 失效
    除草噻唑甲酰胺衍生物

    公开(公告)号:US5057142A

    公开(公告)日:1991-10-15

    申请号:US587283

    申请日:1990-09-24

    CPC分类号: C07D277/56 A01N43/78

    摘要: Herbicidal thiazolecarboxamide derivatives of the formula ##STR1## in which n represents the numbers 0 or 1,A represents in each case optionally substituted alkyl, aryl, heteroaryl, arylamino or heteroarylamino,R.sup.1 represents hydrogen, halogen or alkyl,R.sup.2 represents hydrogen, halogen or alkyl,R.sup.3 represents hydrogen, halogen, alkyl or halogenoalkyl,R.sup.4 represents hydrogen, halogen, alkyl or halogenoalkyl,R.sup.5 represents hydrogen, halogen, alkyl, nitro or amino,R.sup.6 represents hydrogen, halogen, alkyl halogenoalkyl, alkoxy, halogenoalkoxy, alkylthio, halogenoalkylthio or alkoxycarbonyl, andR.sup.7 represents hydrogen, halogen, alkyl, nitro or amino

    摘要翻译: 芳基,杂芳基,芳基氨基或杂芳基氨基,R 1表示氢,卤素或烷基,R 2表示氢原子,其中n表示数字0或1, 卤素,烷基或卤代烷基,R 5代表氢,卤素,烷基,硝基或氨基,R 6表示氢,卤素,烷基卤代烷基,烷氧基,卤代烷氧基, 烷硫基,卤代烷硫基或烷氧基羰基,R7表示氢,卤素,烷基,硝基或氨基

    Substituted benzimidazoles
    7.
    发明授权
    Substituted benzimidazoles 失效
    取代的苯并咪唑

    公开(公告)号:US5863933A

    公开(公告)日:1999-01-26

    申请号:US822565

    申请日:1997-03-19

    摘要: The invention relates to new substituted benzimidazole of the general formula (I) ##STR1## in which R.sup.1 represents hydrogen, alkyl, alkoxy or optionally substituted aryl,R.sup.2 represents hydroxyl, cyano or in each case optionally substituted alkyl, alkenyl, alkinyl, alkoxy, alkenyloxy, alkinyloxy, alkylthio, amino, aminocarbonyl, alkylcarbonyl, alkoxycarbonyl, alkoxycarbonyloxy, dialkoxyphosphonyl, (hetero)aryl, (hetero)arylcarbonyl, (hetero)aryloxycarbonyl, (hetero)arylcarbonyloxy or (hetero)arylaminocarbonylaminocarbonyloxy, andR.sup.3 represents fluoroalkyl,X.sup.1, X.sup.2, X.sup.3 and X.sup.4 independently of one another in each case represent hydrogen, halogen, cyano, nitro, in each case optionally substituted alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl or cycloalkyl, optionally substituted, fused dioxyalkylene, or represent hydroxycarbonyl, alkylcarbonyl, alkoxycarbonyl or cycloalkyloxycarbonyl, in each case optionally substituted amino or aminocarbonyl or in each case optionally substituted aryl, aryloxy, arylthio, arylsulphinyl, arylsulphonyl, arylsulphonyloxy, arylcarbonyl, aryloxycarbonyl, arylazo or arylthiomethylsulphonyl, but where at least one of the substituents X.sup.1, X.sup.2, X.sup.3 or X.sup.4 represents halogenoalkyl, with the exception of the chloromethyl radical, halogenoalkoxy, halogenoalkylthio, halogenoalkylsulphinyl, halogenoalkylsulphonyl or alkylsulphonyl, optionally substituted, fused dioxyalkylene, or represent hydroxycarbonyl, alkylcarbonyl, alkoxycarbonyl or cycloalkyloxycarbonyl, in each case optionally substituted amino or aminocarbonyl, or in each case optionally substituted aryl, arylthio, arylsulphinyl, arylsulphonyl, arylsulphonyloxy, arylcarbonyl, aryloxycarbonyl, arylazo or arylthiomethylsulphonyl,their preparation and use as pesticides, and intermediates for their preparation.

    摘要翻译: 本发明涉及通式(I)的新取代的苯并咪唑,其中R 1表示氢,烷基,烷氧基或任选取代的芳基,R 2表示羟基,氰基或在各种情况下任选取代的烷基,烯基,炔基 (杂)芳基羰基,(杂)芳基羰基氧基或(杂)芳基氨基羰基氨基羰基氧基,R3代表氟代烷基,芳基羰氧基, 在各种情况下,X1,X2,X3和X4彼此独立地表示氢,卤素,氰基,硝基,在各种情况下均为任选取代的烷基,烷氧基,烷硫基,烷基亚磺酰基,烷基磺酰基或环烷基,任选取代的稠合二氧亚烷基,或代表羟基羰基 ,烷基羰基,烷氧基羰基或环烷氧基羰基,在每种情况下均为任选取代的氨基或氨基羰基,或在每种情况下任选取代 芳基,芳氧基,芳硫基,芳基亚磺酰基,芳基磺酰基,芳基磺酰氧基,芳基羰基,芳氧基羰基,芳基偶氮或芳基硫代甲基磺酰基,但其中至少一个取代基X1,X2,X3或X4表示卤代烷基,除了氯甲基,卤代烷氧基,卤代烷硫基 ,卤代烷基亚磺酰基,卤代烷基磺酰基或烷基磺酰基,任选取代的稠合的二氧亚烷基,或代表羟基羰基,烷基羰基,烷氧基羰基或环烷氧基羰基,在各种情况下均为任选取代的氨基或氨基羰基,或在每种情况下均为任选取代的芳基,芳硫基,芳基亚磺酰基,芳基磺酰基,芳基磺酰氧基,芳基羰基, 芳氧基羰基,芳基偶氮或芳基硫代甲基磺酰基,它们的制备和用作农药,以及其制备中间体。