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公开(公告)号:US5386034A
公开(公告)日:1995-01-31
申请号:US78001
申请日:1993-06-15
申请人: Said Yous , Isabelle Lesieur , Patrick Depreux , Daniel H. Caignard , Beatrice Guardiola , Gerard Adam , Pierre Renard
发明人: Said Yous , Isabelle Lesieur , Patrick Depreux , Daniel H. Caignard , Beatrice Guardiola , Gerard Adam , Pierre Renard
IPC分类号: A61K31/42 , A61K31/423 , A61K31/425 , A61K31/428 , A61K31/445 , A61K31/495 , A61K31/496 , A61K31/535 , A61K31/536 , A61K31/5377 , A61K31/538 , A61K31/54 , A61K31/5415 , A61P1/14 , A61P25/00 , A61P25/04 , A61P25/08 , A61P25/20 , A61P25/24 , A61P25/26 , A61P25/28 , C07D263/58 , C07D265/36 , C07D277/68 , C07D279/16 , C07D413/12 , C07D417/12
CPC分类号: C07D263/58 , C07D277/68 , C07D413/10 , C07D413/12
摘要: Compounds of general formula (I): ##STR1## where R, X, A, B and p are defined in the description. Medicinal products. Useful for treating sleep disorders comprising the same.
摘要翻译: 通式(I)的化合物:其中R,X,A,B和p在说明书中定义。 药用产品。 用于治疗包含其的睡眠障碍。
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公开(公告)号:US5300507A
公开(公告)日:1994-04-05
申请号:US55665
申请日:1993-04-28
申请人: Said Yous , Isabelle Lesieur , Patrick Depreux , Daniel H. Caignard , Beatrice Guardiola , Gerard Adam , Pierre Renard
发明人: Said Yous , Isabelle Lesieur , Patrick Depreux , Daniel H. Caignard , Beatrice Guardiola , Gerard Adam , Pierre Renard
IPC分类号: A61K31/42 , A61K31/423 , A61K31/425 , A61K31/428 , A61K31/445 , A61K31/495 , A61K31/496 , A61K31/535 , A61K31/536 , A61K31/5377 , A61K31/538 , A61K31/54 , A61K31/5415 , A61P1/14 , A61P25/00 , A61P25/04 , A61P25/08 , A61P25/20 , A61P25/24 , A61P25/26 , A61P25/28 , C07D263/58 , C07D265/36 , C07D277/68 , C07D279/16 , C07D413/12 , C07D417/12 , C07D413/06 , C07D417/06
CPC分类号: C07D263/58 , C07D277/68 , C07D413/10 , C07D413/12
摘要: Compounds of general formula (I): ##STR1## where R, X, A, B and p are defined in the description. Medicinal products useful for treating sleeping disorders comprising the same.
摘要翻译: 通式(I)的化合物:其中R,X,A,B和p在说明书中定义。 用于治疗包含其的睡眠障碍的药用产品。
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公开(公告)号:US5436348A
公开(公告)日:1995-07-25
申请号:US223176
申请日:1994-04-05
申请人: Said Yous , Isabelle Lesieur , Patrick Depreux , Daniel H. Caignard , Beatrice Guardiola , Gerard Adam , Pierre Renard
发明人: Said Yous , Isabelle Lesieur , Patrick Depreux , Daniel H. Caignard , Beatrice Guardiola , Gerard Adam , Pierre Renard
IPC分类号: A61K31/42 , A61K31/423 , A61K31/425 , A61K31/428 , A61K31/445 , A61K31/495 , A61K31/496 , A61K31/535 , A61K31/536 , A61K31/5377 , A61K31/538 , A61K31/54 , A61K31/5415 , A61P1/14 , A61P25/00 , A61P25/04 , A61P25/08 , A61P25/20 , A61P25/24 , A61P25/26 , A61P25/28 , C07D263/58 , C07D265/36 , C07D277/68 , C07D279/16 , C07D413/12 , C07D417/12
CPC分类号: C07D263/58 , C07D277/68 , C07D413/10 , C07D413/12
摘要: Compounds of general formula (I): ##STR1## where R, X, A, B and p are defined in the description. Medicinal products useful for treating sleep disorders comprising the same.
摘要翻译: 通式(I)的化合物:其中R,X,A,B和p在说明书中定义。 可用于治疗包含其的睡眠障碍的药用产品。
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公开(公告)号:US5326775A
公开(公告)日:1994-07-05
申请号:US54604
申请日:1993-04-28
申请人: Said Yous , Isabelle Lesieur , Patrick Depreux , Daniel H. Caignard , Beatrice Guardiola , Gerard Adam , Pierre Renard
发明人: Said Yous , Isabelle Lesieur , Patrick Depreux , Daniel H. Caignard , Beatrice Guardiola , Gerard Adam , Pierre Renard
IPC分类号: A61K31/42 , A61K31/423 , A61K31/425 , A61K31/428 , A61K31/445 , A61K31/495 , A61K31/496 , A61K31/535 , A61K31/536 , A61K31/5377 , A61K31/538 , A61K31/54 , A61K31/5415 , A61P1/14 , A61P25/00 , A61P25/04 , A61P25/08 , A61P25/20 , A61P25/24 , A61P25/26 , A61P25/28 , C07D263/58 , C07D265/36 , C07D277/68 , C07D279/16 , C07D413/12 , C07D417/12
CPC分类号: C07D263/58 , C07D277/68 , C07D413/10 , C07D413/12
摘要: Compounds of general formula (I): ##STR1## where R, X, A, B and p are defined in the description. Medicinal products useful for treating sleep disorders comprising the same.
摘要翻译: 通式(I)的化合物:其中R,X,A,B和p在说明书中定义。 可用于治疗包含其的睡眠障碍的药用产品。
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5.Benzoxazalinonyl and benzothiazolinonyl ethyl isonicotine amides and piperidonamides 失效
标题翻译: 苯并恶唑啉酮和苯并噻唑啉酮乙基异烟碱酰胺和哌啶酮酰胺公开(公告)号:US5322849A
公开(公告)日:1994-06-21
申请号:US54596
申请日:1993-04-28
申请人: Said Yous , Isabelle Lesieur , Patrick Depreux , Daniel H. Caignard , Beatrice Guardiola , Gerard Adam , Pierre Renard
发明人: Said Yous , Isabelle Lesieur , Patrick Depreux , Daniel H. Caignard , Beatrice Guardiola , Gerard Adam , Pierre Renard
IPC分类号: A61K31/42 , A61K31/423 , A61K31/425 , A61K31/428 , A61K31/445 , A61K31/495 , A61K31/496 , A61K31/535 , A61K31/536 , A61K31/5377 , A61K31/538 , A61K31/54 , A61K31/5415 , A61P1/14 , A61P25/00 , A61P25/04 , A61P25/08 , A61P25/20 , A61P25/24 , A61P25/26 , A61P25/28 , C07D263/58 , C07D265/36 , C07D277/68 , C07D279/16 , C07D413/12 , C07D417/12
CPC分类号: C07D263/58 , C07D277/68 , C07D413/10 , C07D413/12
摘要: Compounds of general formula (I): ##STR1## where R, X, A, B and p are defined in the description. Medicinal products useful for treating sleep disorders comprising the same.
摘要翻译: 通式(I)的化合物:其中R,X,A,B和p在说明书中定义。 可用于治疗包含其的睡眠障碍的药用产品。
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6.
公开(公告)号:US5322843A
公开(公告)日:1994-06-21
申请号:US54720
申请日:1993-04-28
申请人: Said Yous , Isabelle Lesieur , Patrick Depreux , Daniel H. Caignard , Beatrice Guardiola , Gerard Adam , Pierre Renard
发明人: Said Yous , Isabelle Lesieur , Patrick Depreux , Daniel H. Caignard , Beatrice Guardiola , Gerard Adam , Pierre Renard
IPC分类号: A61K31/42 , A61K31/423 , A61K31/425 , A61K31/428 , A61K31/445 , A61K31/495 , A61K31/496 , A61K31/535 , A61K31/536 , A61K31/5377 , A61K31/538 , A61K31/54 , A61K31/5415 , A61P1/14 , A61P25/00 , A61P25/04 , A61P25/08 , A61P25/20 , A61P25/24 , A61P25/26 , A61P25/28 , C07D263/58 , C07D265/36 , C07D277/68 , C07D279/16 , C07D413/12 , C07D417/12
CPC分类号: C07D263/58 , C07D277/68 , C07D413/10 , C07D413/12
摘要: Compounds of general formula (I): ##STR1## wherein R, X, A, B and p are defined in the description. Medicinal products useful for treating sleep disorders comprising the same.
摘要翻译: 通式(I)的化合物:其中R,X,A,B和p在说明书中定义。 可用于治疗包含其的睡眠障碍的药用产品。
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公开(公告)号:US5240919A
公开(公告)日:1993-08-31
申请号:US848373
申请日:1992-03-09
申请人: Said Yous , Isabelle Lesieur , Patrick Depreux , Daniel H. Caignard , Beatrice Guardiola , Gerard Adam , Pierre Renard
发明人: Said Yous , Isabelle Lesieur , Patrick Depreux , Daniel H. Caignard , Beatrice Guardiola , Gerard Adam , Pierre Renard
IPC分类号: A61K31/42 , A61K31/423 , A61K31/425 , A61K31/428 , A61K31/445 , A61K31/495 , A61K31/496 , A61K31/535 , A61K31/536 , A61K31/5377 , A61K31/538 , A61K31/54 , A61K31/5415 , A61P1/14 , A61P25/00 , A61P25/04 , A61P25/08 , A61P25/20 , A61P25/24 , A61P25/26 , A61P25/28 , C07D263/58 , C07D265/36 , C07D277/68 , C07D279/16 , C07D413/12 , C07D417/12
CPC分类号: C07D263/58 , C07D277/68 , C07D413/10 , C07D413/12
摘要: Compounds of general formula (I): ##STR1## where R, X, A, B and p are defined in the description. Medicinal products useful for treating sleep disorders comprising the same.
摘要翻译: 通式(I)的化合物:其中R,X,A,B和p在说明书中定义。 可用于治疗包含其的睡眠障碍的药用产品。
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公开(公告)号:US5420158A
公开(公告)日:1995-05-30
申请号:US035936
申请日:1993-03-23
申请人: Said Yous , Daniel Lesieur , Patrick Depreux , Beatrice Guardiola-Lemaitre , Gerard Adam , Pierre Renard , Daniel H. Caignard
发明人: Said Yous , Daniel Lesieur , Patrick Depreux , Beatrice Guardiola-Lemaitre , Gerard Adam , Pierre Renard , Daniel H. Caignard
IPC分类号: A61K31/135 , A61K31/16 , A61K31/215 , A61P17/00 , A61P25/00 , A61P37/00 , A61P43/00 , C07C233/05 , C07C233/58 , C07C233/60 , C07C233/63 , C07C275/24 , C07D295/10 , A01N1/00 , C07C229/34
CPC分类号: C07C233/63 , C07C233/05 , C07C233/58 , C07C233/60 , C07C275/24 , C07C2101/02 , C07C2101/04 , C07C2101/08 , C07C2101/14 , C07C2101/16
摘要: The invention relates to a compound selected from those of general formula (I): ##STR1## in which R, R.sub.1, R.sub.2 and R.sub.3 are as defined in the specification, an optical isomer, and an addition salt thereof with a pharmaceutically-acceptable base.Medicinal product which is useful in the treatment of disorders linked to abnormal melatonin activity.
摘要翻译: 本发明涉及选自通式(I)的化合物:其中R,R 1,R 2和R 3如本说明书中所定义的其中R 1,R 2和R 3如本文所定义的光学异构体及其加成盐与药学上 可接受的基地 可用于治疗与异常褪黑素活性相关的疾病的药用产品。
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公开(公告)号:US5196434A
公开(公告)日:1993-03-23
申请号:US765959
申请日:1991-09-26
申请人: Thierry Taverne , Isabelle Lesieur , Patrick Depreux , Daniel H. Caignard , Beatrice Guardiola , Gerard Adam , Pierre Renard
发明人: Thierry Taverne , Isabelle Lesieur , Patrick Depreux , Daniel H. Caignard , Beatrice Guardiola , Gerard Adam , Pierre Renard
IPC分类号: A61K31/42 , A61K31/423 , A61K31/425 , A61K31/428 , A61K31/44 , A61K31/495 , A61K31/496 , A61K31/505 , A61K31/535 , A61K31/536 , A61K31/5377 , A61K31/538 , A61K31/54 , A61K31/5415 , A61P9/12 , A61P25/04 , A61P25/18 , A61P25/20 , C07D263/58 , C07D265/36 , C07D277/68 , C07D279/16 , C07D413/06 , C07D413/12 , C07D413/14 , C07D417/06 , C07D417/12 , C07D417/14 , C07D491/056
CPC分类号: C07D277/68 , C07D265/36 , C07D279/16 , C07D417/12
摘要: Compound of general formula (I): ##STR1## where R.sub.1, R.sub.2, R.sub.3, n, X and A are defined in the description.Medicinal products.
摘要翻译: 通式(I)的化合物:其中R 1,R 2,R 3,n,X和A在说明书中定义。 药用产品。
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10.Aminoalkyl-benzothiazolinone and -benzoxazolinone compounds having a high 5-HT1A affinity 失效
标题翻译: 具有高5-HT1A亲和力的氨基烷基 - 苯并噻唑啉酮和 - 苯并恶唑啉酮化合物公开(公告)号:US5268381A
公开(公告)日:1993-12-07
申请号:US945492
申请日:1992-09-16
申请人: Thierry Taverne , Isabelle Lesieur , Patrick Depreux , Daniel H. Caignard , Beatrice Guardiola , Gerard Adam , Pierre Renard
发明人: Thierry Taverne , Isabelle Lesieur , Patrick Depreux , Daniel H. Caignard , Beatrice Guardiola , Gerard Adam , Pierre Renard
IPC分类号: C07D265/36 , C07D277/68 , C07D279/16 , C07D417/12 , A61K31/42 , A61K31/425
CPC分类号: C07D277/68 , C07D265/36 , C07D279/16 , C07D417/12
摘要: Compounds of general formula (I): ##STR1## wherein R.sub.1, R.sub.2, R.sub.3, n, X and A are defined in the description. Medicinal products containing the same are useful as antidepressives or anxiolytics due to their 5-HT1A receptor agonist activity.
摘要翻译: 通式(I)的化合物:其中R 1,R 2,R 3,n,X和A在说明书中定义。 含有它们的药物由于其5-HT1A受体激动剂活性而可用作抗抑郁药或抗焦虑药。
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