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公开(公告)号：US4576956A
公开(公告)日：1986-03-18
申请号：US530883
申请日：1983-09-09
申请人： Yasuo Makisumi , Akira Murabayashi , Katsuya Tawara , Yoshihachi Watanabe , Toshio Takahashi , Takao Konishi
发明人： Yasuo Makisumi , Akira Murabayashi , Katsuya Tawara , Yoshihachi Watanabe , Toshio Takahashi , Takao Konishi
IPC分类号： A01N43/80 , A61K31/42 , A61P31/04 , A61P31/10 , A61P33/02 , C07D261/14 , C07D413/04 , C07D413/06 , C07D413/12 , C07D521/00 , A61K31/41 , C07D261/12 , C07D261/20
CPC分类号： C07D231/12 , A01N43/80 , C07D233/56 , C07D249/08 , C07D261/14 , C07D413/04
摘要： New (2-propynylamino)isoxazole and (3-iodo-2-propynylamino)isoxazole derivatives having anti-microbial activity which are used as active ingredients in anti-microbial compositions for medical use, for agricultural use and also for veterinary use.
摘要翻译： 新的（2-丙炔基氨基）异恶唑和具有抗微生物活性的（3-碘-2-丙炔基氨基）异恶唑衍生物，其用作医疗用途，农业用途和兽医用抗微生物组合物中的活性成分。
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公开(公告)号：US4535088A
公开(公告)日：1985-08-13
申请号：US557365
申请日：1983-12-02
IPC分类号： A01N43/78 , A61K31/425 , A61K31/426 , A61K31/428 , A61P31/04 , A61P31/10 , C07D277/20 , C07D277/42 , C07D277/56 , C07D277/82
CPC分类号： C07D277/82 , C07D277/42 , C07D277/56
摘要： New 2-(2-propynylamino)thiazole and 2-(3-iodo-2-propynylamino)thiazole derivatives having anti-microbial activity which are used as an active ingredient in anti-microbial compositions for medical and agricultural use.
摘要翻译： 具有抗微生物活性的新的2-（2-丙炔基氨基）噻唑和2-（3-碘-2-丙炔基氨基）噻唑衍生物用作用于医疗和农业用途的抗微生物组合物中的活性成分。
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公开(公告)号：US4328348A
公开(公告)日：1982-05-04
申请号：US157166
申请日：1980-06-06
IPC分类号： A01N43/50 , C07C53/08 , C07C55/06 , C07C55/10 , C07C59/245 , C07C59/255 , C07C59/265 , C07C65/10 , C07D233/54 , C07D233/56 , C07D233/60 , C07D521/00 , C07D233/96
CPC分类号： C07D233/64 , A01N43/50 , C07C53/08 , C07C55/06 , C07C55/10 , C07C59/245 , C07C59/255 , C07C59/265 , C07C65/10 , C07D231/12 , C07D233/56 , C07D249/08
摘要： Novel benzylimidazole derivatives of the formula: ##STR1## wherein X is halogen, nitro, alkyl, alkoxy, or halobenzyloxy;m is an integer of 0 to 3;Y is oxa, thia or substituted- or unsubstituted-imino;R.sup.1 is alkyl, dialkylaminoalkyl, dibenzylaminoalkyl, 1-pyrrolidinyl, 2-imidazolin-2-yl, or a group of --(CH.sub.2)n--Z--Q(whereinn is an integer of 0 to 4;Z is oxa, thia, or a single bond; andQ is substituted- or unsubstituted-phenyl or thienyl) ##STR2## is methylene, 1-(1-imidazolyl)-1-methylmethylene, 1-(1-imidazolyl)-1-phenylmethylene, 1-phenylmethylene, or substituted or unsubstituted alkylidene;the benzene ring of the above formula being optionally condensed with another benzene ringwith the proviso that when ##STR3## is methylene said benzene ring is condensed with another benzene ring, and acid addition salts thereof which are useful as an antimycotic drug or agricultural fungicide.
摘要翻译： 下式的新型苄基咪唑衍生物：其中X是卤素，硝基，烷基，烷氧基或卤代苄氧基; m为0〜3的整数。 Y是氧杂，硫杂或取代或未取代的亚氨基; R1是烷基，二烷基氨基烷基，二苄基氨基烷基，1-吡咯烷基，2-咪唑啉-2-基或 - （CH2）nZQ（其中n是0-4的整数; Z是氧杂，硫杂或单键） ;和Q是取代或未取代的苯基或噻吩基）是甲亚甲基，1-（1-咪唑基）-1-甲基亚甲基，1-（1-咪唑基）-1-苯基亚甲基，1-苯基亚甲基，或取代或未取代的 未取代的亚烷基; 上式的苯环任选地与另一个苯环稠合，条件是当亚甲基时，苯环与另一个苯环缩合，其酸加成盐可用作抗真菌药物或农药杀真菌剂。
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4.发明授权Bis-imidazolyl-bis-phenylmethane derivatives and their use as fungicides 失效双咪唑基 - 双苯基甲烷衍生物及其作为杀真菌剂的用途
公开(公告)号：US4463011A
公开(公告)日：1984-07-31
申请号：US341634
申请日：1982-01-22
IPC分类号： A01N43/50 , C07C53/08 , C07C55/06 , C07C55/10 , C07C59/245 , C07C59/255 , C07C59/265 , C07C65/10 , C07D233/54 , C07D233/56 , C07D233/60 , C07D521/00 , C07D403/02
CPC分类号： C07D233/64 , A01N43/50 , C07C53/08 , C07C55/06 , C07C55/10 , C07C59/245 , C07C59/255 , C07C59/265 , C07C65/10 , C07D231/12 , C07D233/56 , C07D249/08
摘要： Benzylimidazole derivatives of the formula: ##STR1## wherein X is halogen, nitro, alkyl, alkoxy, or halobenzyloxy;m is an integer of 0 to 3;Y is oxa, thia or substituted- or unsubstituted-imino;R.sup.1 is alkyl, dialkylaminoaklyl, dibenzylaminoalkyl, 1-pyrrolidinyl, 2-imidazolin-2-yl, or a group of --(CH.sub.2)n--Z--Q(wherein n is an integer of 0 to 4; Z is oxa, thia, or a single bond; and Q is substituted- or unsubstituted-phenyl or thienyl) ##STR2## is methylene, 1-(1-imidazolyl)-1-methylmethylene, 1-(1-imidazolyl)-1-phenylmethylene, 1-phenylmethylene, or substituted or unsubstituted alkylidene;the benzene ring of the above formula being optionally condensed with another benzene ringwith the proviso that when ##STR3## is methylene said benzene ring is condensed with another benzene ring, and acid addition salts thereof which are useful as an antimycotic drug or agricultural fungicide.
摘要翻译： 下式的苄基咪唑衍生物：其中X是卤素，硝基，烷基，烷氧基或卤代苄氧基; m为0〜3的整数。 Y是氧杂，噻吩或取代或未取代的亚氨基; R1是烷基，二烷基氨基烷基，二苄基氨基烷基，1-吡咯烷基，2-咪唑啉-2-基或 - （CH2）nZQ（其中n是0-4的整数; Z是氧杂，硫杂或单键 ;和Q是取代或未取代的苯基或噻吩基）是甲亚甲基，1-（1-咪唑基）-1-甲基亚甲基，1-（1-咪唑基）-1-苯基亚甲基，1-苯基亚甲基，或取代或未取代的 未取代的亚烷基; 上式的苯环任选地与另一个苯环稠合，条件是当亚甲基时，苯环与另一个苯环缩合，其酸加成盐可用作抗真菌药物或农药杀真菌剂。
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5.发明授权
公开(公告)号：US4483866A
公开(公告)日：1984-11-20
申请号：US397786
申请日：1982-07-13
IPC分类号： A01N43/50 , C07C53/08 , C07C55/06 , C07C55/10 , C07C59/245 , C07C59/255 , C07C59/265 , C07C65/10 , C07D233/54 , C07D233/56 , C07D233/60 , C07D521/00
CPC分类号： C07D233/64 , A01N43/50 , C07C53/08 , C07C55/06 , C07C55/10 , C07C59/245 , C07C59/255 , C07C59/265 , C07C65/10 , C07D231/12 , C07D233/56 , C07D249/08
摘要： Novel benzylimidazole derivatives of the formula: ##STR1## wherein X is halogen, nitro, alkyl, alkoxy, or halobenzyloxy;m is an integer of 0 to 3;Y is oxa, thia or substituted- or unsubstituted-imino;R.sup.1 is alkyl, dialkylaminoalkyl, dibenzylaminoalkyl, 1-pyrrolidinyl, 2-imidazolin-2-yl, or a group of --(CH.sub.2)n--Z--Q(wherein n is an integer of 0 to 4; Z is oxa, thia, or a single bond; and Q is substituted- or unsubstituted-phenyl or thienyl) ##STR2## is methylene, 1-(1-imidazolyl)-1-methylmethylene, 1-(1-imidazolyl)-1-phenylmethylene, 1-phenylmethylene, or substituted or unsubstituted alkylidene;the benzene ring of the above formula being optionally condensed with another benzene ringwith the proviso that when ##STR3## is methylene said benzene ring is condensed with another benzene ring, and acid addition salts thereof which are useful as an antimycotic drug or agricultural fungicide.
摘要翻译： 下式的新型苄基咪唑衍生物：其中X是卤素，硝基，烷基，烷氧基或卤代苄氧基; m为0〜3的整数。 Y是氧杂，噻吩或取代或未取代的亚氨基; R1是烷基，二烷基氨基烷基，二苄基氨基烷基，1-吡咯烷基，2-咪唑啉-2-基或 - （CH2）nZQ（其中n是0-4的整数; Z是氧杂，硫杂或单键） ;和Q是取代或未取代的苯基或噻吩基）是甲亚甲基，1-（1-咪唑基）-1-甲基亚甲基，1-（1-咪唑基）-1-苯基亚甲基，1-苯基亚甲基，或取代或未取代的 未取代的亚烷基; 上式的苯环任选地与另一个苯环稠合，条件是当亚甲基时，苯环与另一个苯环缩合，其酸加成盐可用作抗真菌药物或农药杀真菌剂。
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公开(公告)号：US4228165A
公开(公告)日：1980-10-14
申请号：US47803
申请日：1979-06-11
IPC分类号： C07D295/18 , A01N47/46 , C07C67/00 , C07C325/00 , C07C331/28 , C07D295/192 , C07D307/14 , A01N43/84 , C07C161/04 , C07D295/12 , C07D307/64
CPC分类号： C07D295/192 , A01N47/46 , C07C331/28
摘要： A compound of the formula: ##STR1## wherein X is oxygen or sulfur;R.sup.1 is hydroxy, C.sub.1 -C.sub.4 alkoxy, phenoxy, amino, C.sub.1 -C.sub.4 alkylamino, C.sub.2 -C.sub.8 dialkylamino, C.sub.6 -C.sub.10 arylamino, tetrahydrofurfurylamino, morpholino or methylpiperazino, but when X is sulfur R.sup.1 must be amino, C.sub.1 -C.sub.4 alkylamino, C.sub.2 -C.sub.8 dialkylamino or morpholino;R.sup.2 is C.sub.1 -C.sub.4 alkoxy or C.sub.2 -C.sub.5 alkoxycarbonyl;R.sup.3 is hydrogen C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.2 -C.sub.8 dialkylamino or halogenand its salts being useful as agricultural fungicides are provided.
摘要翻译： 下式的化合物：其中X是氧或硫; R1是羟基，C1-C4烷氧基，苯氧基，氨基，C1-C4烷基氨基，C2-C8二烷基氨基，C6-C10芳基氨基，四氢糠基氨基，吗啉代或甲基哌嗪基，但是当X是硫时，R1必须是氨基，C1-C4烷基氨基，C2 -C8二烷基氨基或吗啉代; R2是C1-C4烷氧基或C2-C5烷氧基羰基; R3是氢C1-C4烷基，C1-C4烷氧基，C2-C8二烷基氨基或卤素，其盐可用作农业杀真菌剂。
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公开(公告)号：US4248869A
公开(公告)日：1981-02-03
申请号：US946422
申请日：1978-09-25
IPC分类号： C07D295/18 , A01N47/46 , C07C67/00 , C07C325/00 , C07C331/28 , C07D295/192 , C07D307/14 , A01N41/00 , C07C161/04 , C07D265/00 , C07D307/64
CPC分类号： C07D295/192 , A01N47/46 , C07C331/28
摘要： A compound of the formula: ##STR1## wherein X is oxygen or sulfur;R.sup.1 is hydroxy, C.sub.1 -C.sub.4 alkoxy, phenoxy, amino, C.sub.1 -C.sub.4 alkylamino, C.sub.2 -C.sub.8 dialkylamino, C.sub.6 -C.sub.10 arylamino, tetrahydrofurfurylamino, morpholino or methylpiperazino, but when X is sulfur R.sup.1 must be amino, C.sub.1 -C.sub.4 alkylamino, C.sub.2 -C.sub.8 dialkylamino or morpholino;R.sup.2 is C.sub.1 -C.sub.4 alkoxy or C.sub.2 -C.sub.5 alkoxycarbonyl;R.sup.3 is hydrogen C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.2 -C.sub.8 dialkylamino or halogenand its salts being useful as agricultural fungicides are provided.
摘要翻译： 下式的化合物：其中X是氧或硫; R1是羟基，C1-C4烷氧基，苯氧基，氨基，C1-C4烷基氨基，C2-C8二烷基氨基，C6-C10芳基氨基，四氢糠基氨基，吗啉代或甲基哌嗪基，但是当X是硫时，R1必须是氨基，C1-C4烷基氨基，C2 -C8二烷基氨基或吗啉代; R2是C1-C4烷氧基或C2-C5烷氧基羰基; R3是氢C1-C4烷基，C1-C4烷氧基，C2-C8二烷基氨基或卤素，其盐可用作农业杀真菌剂。
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