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    Tetrahydrothiopyrano[2,3-b]indole derivatives
    1.
    发明授权
    Tetrahydrothiopyrano[2,3-b]indole derivatives 失效
    四氢噻喃并[2,3-b]吲哚衍生物

    公开(公告)号：US4256640A

    公开(公告)日：1981-03-17

    申请号：US39382

    申请日：1979-05-15

    申请人： Yasuo Makisumi ,  Susumu Takada ,  Takashi Sasatani ,  Natsuki Ishizuka

    发明人： Yasuo Makisumi ,  Susumu Takada ,  Takashi Sasatani ,  Natsuki Ishizuka

    IPC分类号： A61K31/40 ,  A61K31/445 ,  A61P25/04 ,  A61P29/00 ,  C07D209/30 ,  C07D495/04

    CPC分类号： C07D495/04 ,  C07D209/30

    摘要： Tetrahydrothiopyrano[2,3-b]indole derivative represented by the formula I: ##STR1## wherein R.sup.1 is hydrogen, alkyl, hydroxyalkyl, alkenyl, aralkyl, aryl, --COR.sup.5 (wherein R.sup.5 is alkyl, alkenyl, aryl or alkoxy) or ##STR2## (wherein Y is alkylene, oxoalkylene, hydroxyalkylene and R.sup.6 and R.sup.7 are each hydrogen or alkyl): R.sup.2 is hydrogen or alkyl; R.sup.3 is hydrogen, alkyl, hydroxyalkyl, alkenyl, aralkyl, aryl or dialkylaminoalkyl or ##STR3## is pyrrolidino, piperidino, piperazino, 4-alkylpiperazino, 4-arylpiperazino or morpholino; R.sup.4 is hydrogen or alkyl; A is methylene, alkylmethylene, ethylene, alkylethylene; X is hydrogen or one or two groups selected from the group consisting of halogen, alkyl, alkoxy, hydroxy and halogenoalkyl; and n is an integer of 0 to 2 and its pharmaceutically acceptacle salts; synthesized from 2-propargylthioindole or 2-(4-hydroxy-2-butynylthio)-indole; useful as analgesic and anti-inflammatory agent.

    摘要翻译： 由式I表示的四氢噻喃[2,3-b]吲哚衍生物：其中R 1是氢，烷基，羟烷基，烯基，芳烷基，芳基，-COR 5（其中R 5是烷基，烯基，芳基或烷氧基）或 （其中Y是亚烷基，氧代亚烷基，羟基亚烷基，R 6和R 7各自是氢或烷基）：R 2是氢或烷基; R 3是氢，烷基，羟基烷基，烯基，芳烷基，芳基或二烷基氨基烷基，或者是吡咯烷子基，哌啶子基，哌嗪子基，4-烷基哌嗪基，4-芳基哌嗪基或吗啉代; R4是氢或烷基; A是亚甲基，烷基亚甲基，亚乙基，烷基亚乙基; X是氢或选自卤素，烷基，烷氧基，羟基和卤代烷基的一个或两个基团; n为0〜2的整数及其药学上可接受的盐; 由2-炔丙基硫吲哚或2-（4-羟基-2-丁炔硫基） - 吲哚合成; 用作镇痛和抗炎剂。

    Condensed imidazopyridine derivatives useful as psychotropic agents
    3.
    发明授权
    Condensed imidazopyridine derivatives useful as psychotropic agents 失效
    用作精神药物的缩合咪唑并吡啶衍生物

    公开(公告)号：US4753951A

    公开(公告)日：1988-06-28

    申请号：US920162

    申请日：1986-10-17

    申请人： Susumu Takada ,  Toshio Fujishita ,  Takashi Sasatani ,  Akira Matsushita ,  Masami Eigyo

    发明人： Susumu Takada ,  Toshio Fujishita ,  Takashi Sasatani ,  Akira Matsushita ,  Masami Eigyo

    IPC分类号： C07D471/04 ,  C07D495/14 ,  A61K31/47 ,  C07D471/14

    CPC分类号： C07D471/04 ,  C07D495/14

    摘要： A compound of the formula: ##STR1## (wherein R is phenyl optionally substituted by one or two members selected from the group consisting of trifluoromethyl, C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.5 alkoxy, C.sub.1 -C.sub.5 alkylthio, nitro, amino C.sub.1 -C.sub.5 alkanoylamino and C.sub.1 -C.sub.5 alkoxycarbonyl or 5- or 6-membered heterocyclic group optionally substituted by one or two members selected from the group consisting of halogen, C.sub.1 -C.sub.5 alkyl and C.sub.1 -C.sub.5 alkoxy,Q is hydrogen, C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.10 acyl, C.sub.1 -C.sub.5 alkylsulfonyl or C.sub.6 -C.sub.10 arylsulfonyl, ##STR2## R.sup.1, R.sup.2, R.sup.3, and R.sup.4 each is hydrogen, halogen C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.5 alkoxy or C.sub.1 -C.sub.5 haloalkyl,Q is present on the nitrogen atom of the 1,3 or 5-position, and the dotted line indicates the presence of three double bonds at the position of 2, 3; 3a, 3b; 4, 5 / 1, 3b; 2, 3; 3a, 4 / or 1, 2; 3a, 3b; 4, 5)or its salt, being useful as psychostimulants or anxiolytics, is provided.

    摘要翻译： 下式的化合物：其中R是任选被一个或两个选自三氟甲基，C 1 -C 5烷基，C 1 -C 5烷氧基，C 1 -C 5烷硫基，硝基，氨基， 任选被一个或两个选自卤素，C 1 -C 5烷基和C 1 -C 5烷氧基的成员取代的C 1 -C 5烷酰基氨基和C 1 -C 5烷氧基羰基或5或6元杂环基，Q是氢，C 1 -C 5 烷基，C 1 -C 10酰基，C 1 -C 5烷基磺酰基或C 6 -C 10芳基磺酰基，R 1，R 2，R 3和R 4各自为氢，卤素C 1 -C 5烷基，C 1 -C 5烷氧基或C 1 -C 5烷氧基， C5卤代烷基，Q存在于1,3或5位的氮原子上，虚线表示在2,3,3a，3b; 4,5 / 1,3b的位置存在三个双键 ; 2,3,3a，4 /或1,2; 3a，3b; 4,5）或其盐，可用作精神兴奋剂或抗焦虑剂。

    Method of producing crystalline substrate having concave-convex structure
    7.
    发明授权
    Method of producing crystalline substrate having concave-convex structure 有权
    具有凹凸结构的结晶基板的制造方法

    公开(公告)号：US09306137B2

    公开(公告)日：2016-04-05

    申请号：US14395151

    申请日：2012-08-09

    申请人： Susumu Takada ,  Emi Kuraseko ,  Motoyuki Suzuki

    发明人： Susumu Takada ,  Emi Kuraseko ,  Motoyuki Suzuki

    IPC分类号： H01L33/58 ,  H01L33/22 ,  C30B33/08 ,  B32B37/00 ,  B32B38/10 ,  H01L33/00

    CPC分类号： H01L33/58 ,  B32B37/025 ,  B32B38/10 ,  B32B2310/0831 ,  B32B2323/00 ,  B32B2333/00 ,  B32B2361/00 ,  B32B2379/08 ,  B32B2457/20 ,  C30B33/08 ,  H01L33/005 ,  H01L33/22 ,  H01L2933/0058

    摘要： A method of producing the crystalline substrate having a concave-convex structure includes: (A) forming a transfer film by forming a concave-convex film on a support film on the surface having a concave-convex pattern thereon so that thickness of the residual film of the concave-convex film is 0.01 to 1 μm, the concave-convex pattern of the support film having concave parts with a width of 0.05 to 100 μm, a depth of 0.05 to 10 μm, and a ratio of the depth of the concave part to the width of the concave part of up to 1.5, (B) disposing the transfer film on the crystalline substrate, and transferring the concave-convex film onto the crystalline substrate to produce a crystalline substrate having the concave-convex film thereon, (C) etching the crystalline substrate having the concave-convex film thereon to form a concave-convex structure on the surface of a crystalline substrate.

    摘要翻译： 制造具有凹凸结构的结晶性基板的方法包括：（A）通过在其上具有凹凸图案的表面上的支撑膜上形成凹凸膜形成转印膜，使得残留膜的厚度 所述凹凸膜的凹凸图案为0.01〜1μm，所述支撑膜的凹凸图案的凹部的宽度为0.05〜100μm，深度为0.05〜10μm，所述凹部的深度 （B）将转印膜设置在结晶基板上，将凹凸膜转印到结晶基板上，制作具有凹凸膜的结晶性基板，（ C）蚀刻其上具有凹凸膜的晶体衬底，以在晶体衬底的表面上形成凹凸结构。

    METHOD OF PRODUCING CRYSTALLINE SUBSTRATE HAVING CONCAVE-CONVEX STRUCTURE
    8.
    发明申请
    METHOD OF PRODUCING CRYSTALLINE SUBSTRATE HAVING CONCAVE-CONVEX STRUCTURE 有权
    生产具有凹凸结构的晶体衬底的方法

    公开(公告)号：US20150097204A1

    公开(公告)日：2015-04-09

    申请号：US14395151

    申请日：2012-08-09

    申请人： Susumu Takada ,  Emi Kuraseko ,  Motoyuki Suzuki

    发明人： Susumu Takada ,  Emi Kuraseko ,  Motoyuki Suzuki

    IPC分类号： H01L33/58 ,  B32B38/10 ,  B32B37/00

    CPC分类号： H01L33/58 ,  B32B37/025 ,  B32B38/10 ,  B32B2310/0831 ,  B32B2323/00 ,  B32B2333/00 ,  B32B2361/00 ,  B32B2379/08 ,  B32B2457/20 ,  C30B33/08 ,  H01L33/005 ,  H01L33/22 ,  H01L2933/0058

    摘要： A method of producing the crystalline substrate having a concave-convex structure includes: (A) forming a transfer film by forming a concave-convex film on a support film on the surface having a concave-convex pattern thereon so that thickness of the residual film of the concave-convex film is 0.01 to 1 μm, the concave-convex pattern of the support film having concave parts with a width of 0.05 to 100 μm, a depth of 0.05 to 10 μm, and a ratio of the depth of the concave part to the width of the concave part of up to 1.5, (B) disposing the transfer film on the crystalline substrate, and transferring the concave-convex film onto the crystalline substrate to produce a crystalline substrate having the concave-convex film thereon, (C) etching the crystalline substrate having the concave-convex film thereon to form a concave-convex structure on the surface of a crystalline substrate.

    摘要翻译： 制造具有凹凸结构的结晶性基板的方法包括：（A）通过在其上具有凹凸图案的表面上的支撑膜上形成凹凸膜形成转印膜，使得残留膜的厚度 所述凹凸膜的凹凸图案为0.01〜1μm，所述支撑膜的凹凸图案的凹部的宽度为0.05〜100μm，深度为0.05〜10μm，所述凹部的深度 （B）将转印膜设置在结晶基板上，将凹凸膜转印到结晶基板上，制作具有凹凸膜的结晶性基板，（ C）蚀刻其上具有凹凸膜的晶体衬底，以在晶体衬底的表面上形成凹凸结构。

    Load test machine
    9.
    发明授权
    Load test machine 失效
    负载试验机

    公开(公告)号：US06938494B2

    公开(公告)日：2005-09-06

    申请号：US10750779

    申请日：2004-01-02

    申请人： Susumu Takada ,  Keiichi Furuya

    发明人： Susumu Takada ,  Keiichi Furuya

    IPC分类号： G01N3/02 ,  G01N3/00 ,  G01N3/32 ,  G01N3/34 ,  G01B5/30 ,  G01B7/16 ,  G01L1/00

    CPC分类号： G01N3/32 ,  G01N2203/0005 ,  G01N2203/0048 ,  G01N2203/0073

    摘要： A load test machine includes a base block, at least a pair of posts rising from the base block, a cross head spanning between the pair of posts, and an actuator mounted on the base block or the cross head. The actuator is able to apply a load on a test piece positioned between the cross head and the base block. The cross head is secured to each of the posts via an elastic member, and the elastic member is constructed to be changeable in its jointing position with the cross head or with each of the posts to change a resonance frequency of the test machine.

    摘要翻译： 负载测试机包括基座，至少一对从基座上升的柱，横跨在该对柱之间的十字头，以及安装在基座或十字头上的致动器。 执行器能够将负载施加在位于十字头和基座之间的测试件上。 十字头通过弹性构件固定到每个柱上，并且弹性构件被构造成可以与十字头或每个柱的接合位置改变以改变试验机的共振频率。