Substituted pyrimidine ether compounds and use thereof
    4.
    发明授权
    Substituted pyrimidine ether compounds and use thereof 有权
    取代的嘧啶醚化合物及其用途

    公开(公告)号:US08383640B2

    公开(公告)日:2013-02-26

    申请号:US12597173

    申请日:2008-05-22

    IPC分类号: A61K31/505

    摘要: The invention relates to substituted pyrimidine ether compounds having general formula I: The groups are as defined as specification.The compounds of formula I show high insecticidal activities for imagoes, larvae and nits of harmful acari and insects in the agricultural, civil and zoic fields, especially show excellent insecticidal activities for harmful acari such as Tetranychus cinnabarinus. Good effects can be obtained at very low dose. The compounds also exhibit preferably fungicidal activity. Wherefore, the invention also comprises the uses of compounds of formula I as insecticides, acaricides and/or fungicides in agricultural and other fields.

    摘要翻译: 本发明涉及具有通式I的取代的嘧啶醚化合物:这些基团如规定所定义。 式I化合物在农业,民用和盐酸领域中对于成虫,幼虫和有害螨虫和昆虫的蚊子具有很高的杀虫活性,特别是对有害猕猴桃(Tetranychus cinnabarinus)具有极好的杀虫活性。 在非常低的剂量下可以获得良好的效果。 所述化合物还优选具有杀真菌活性。 因此,本发明还包括在农业和其他领域中式I化合物作为杀虫剂,杀螨剂和/或杀真菌剂的用途。

    Substituted azole compounds and its preparation and use thereof
    5.
    发明授权
    Substituted azole compounds and its preparation and use thereof 有权
    取代的唑化合物及其制备和用途

    公开(公告)号:US07795179B2

    公开(公告)日:2010-09-14

    申请号:US10598033

    申请日:2005-02-17

    摘要: The invention relates to fungicide and insecticide, especifically to the substituted azole compounds and its preparation method and use thereof. The azole compounds of the invention having general formula (I): The compounds of present invention, having broad spectrum fungicidal activity, applied for controlling various disease in plants. For example they have good activity against the diseases such as cucumber downy mildew, cucumber grey mold, cucumber powdery mildew, tomato early blight, tomato late blight, phytophthora blight of pepper, grape downy mildew, grape white rot, apple ring rot, apple alternaria leaf spot, rice sheath blight, rice blast, wheat leaf rust, wheat leaf blotch, wheat powdery mildew, rapesclerotiniose, corn southern leaf blight. Some compounds have good insecticidal or acaricidal activity and can be used to control insects and acacids of various crops. For example they are used to control army worm, diamond backmoth and aphid, and culex mosquito.

    摘要翻译: 本发明涉及杀真菌剂和杀虫剂,特别涉及取代的唑化合物及其制备方法和用途。 具有通式(I)的本发明唑类化合物:具有广谱杀真菌活性的本发明化合物被用于控制植物中的各种疾病。 例如,它们对黄瓜霜霉病,黄瓜灰霉病,黄瓜白粉病,番茄早疫病,番茄晚疫病,胡椒疫霉病,葡萄霜霉病,葡萄白腐病,苹果腐烂,苹果轮虫 叶斑病,水稻纹枯病,稻瘟病,小麦叶锈病,小麦叶斑病,小麦白粉病,rapesclerotiniose,玉米南叶枯病。 一些化合物具有良好的杀虫或杀螨活性,可用于控制各种作物的昆虫和螨类。 例如,它们用于控制军队蠕虫,钻石背蛾和蚜虫,以及库蚊。

    Fluorine-containing diphenyl acrylamide antimicrobial agents
    7.
    发明授权
    Fluorine-containing diphenyl acrylamide antimicrobial agents 失效
    含氟二苯基丙烯酰胺抗菌剂

    公开(公告)号:US6020332A

    公开(公告)日:2000-02-01

    申请号:US20333

    申请日:1998-02-09

    CPC分类号: C07D295/185 A01N37/38

    摘要: Fluorine-containing diphenyl acrylamide of general formula (I) have antimicrobial properties. wherein R.sub.1 and R.sub.2 are independently selected from (C.sub.1 -C.sub.6)alkyl group, alkyl group, (C.sub.1 -C.sub.6)alkoxy group, halo(C.sub.1 -C.sub.6)alkyl group, halo(C.sub.1 -C.sub.6)alkoxy group, (C.sub.1 -C.sub.6)alkoxy(C.sub.1 -C.sub.6)alkyl group, (C.sub.3 -C.sub.6)cycloalkyl group, (C.sub.3 -C.sub.6)cycloalkyl(C.sub.1 -C.sub.4)alkyl group, (C.sub.2 -C.sub.6)alkenyl group, halo(C.sub.2 -C.sub.6)alkenyl group, (C.sub.3 -C.sub.6)alkynyl group, halo(C.sub.3 -C.sub.6)alkynyl group, aryl group, aryloxy(C.sub.1 -C.sub.12)alkyl group, aralkyl group, heterocyclic group;or R.sub.1 and R.sub.2 when taken together may form a 5 or 6-membered ring such that;when R.sub.1 and R.sub.2 are in a 5 membered ring R.sub.1 and R.sub.2 taken together is C(R.sub.6 R.sub.7); andwhen R.sub.1 and R.sub.2 are in a 6 membered ring R.sub.1 and R.sub.2 taken together is CHR.sub.6 -CHR.sub.7 ;where R.sub.6 and R.sub.7 are independently selected from hydrogen, (C.sub.1 -C.sub.6)alkyl group or halogen.

    摘要翻译: 具有通式(I)的含氟二苯基丙烯酰胺具有抗微生物性质。 其中R1和R2独立地选自(C1-C6)烷基,烷基,(C1-C6)烷氧基,卤代(C1-C6)烷基,卤代(C1-C6)烷氧基,(C1-C6) 烷氧基(C1-C6)烷基,(C3-C6)环烷基,(C3-C6)环烷基(C1-C4)烷基,(C2-C6)烯基,卤代(C2-C6)烯基,(C3 -C 6)炔基,卤代(C 3 -C 6)炔基,芳基,芳氧基(C 1 -C 12)烷基,芳烷基,杂环基; 当R 1和R 2一起时可以形成5或6元环,使得 当R 1和R 2为5元环时,R 1和R 2一起为C(R 6 R 7); 当R1和R2为6元环时,R1和R2一起为CHR6-CHR7; 其中R 6和R 7独立地选自氢,(C 1 -C 6)烷基或卤素。

    Substituted pyrimidine ammonia compounds and uses thereof
    9.
    发明授权
    Substituted pyrimidine ammonia compounds and uses thereof 有权
    取代的嘧啶氨化合物及其用途

    公开(公告)号:US09018218B2

    公开(公告)日:2015-04-28

    申请号:US13883920

    申请日:2011-11-18

    摘要: The invention relates to substituted pyrimidine ammonia compounds. The structure of the compounds is represented as the general formula (I): The groups are as defined as specification.The compound represented by formula (I) can be used in the prevention of plants diseases caused by a plurality of pathogenic bacteria such as oomycota, basidiomycota, ascomycota, and fungi imperfecti, and due to these compounds have good bioactivity, which make them have very good effects at very low doses, especially more effective to powdery mildew of wheat. Therefore, the present invention relates to the use of the compounds having general formula I as fungicides, both in agriculture and other fields.

    摘要翻译: 本发明涉及取代的嘧啶氨化合物。 化合物的结构表示为通式(I):这些基团如规定所定义。 由式(I)表示的化合物可用于预防由许多病原菌如卵菌,担子菌纲,子囊菌和真菌不完全引起的植物疾病,并且由于这些化合物具有良好的生物活性,这使得它们具有非常 在非常低的剂量下效果良好,特别是对小麦白粉病更有效。 因此,本发明涉及在农业和其他领域中具有通式I的化合物作为杀真菌剂的用途。