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公开(公告)号：EP3191454B1
公开(公告)日：2018-10-24
申请号：EP15766344.4
申请日：2015-09-08
发明人： SHI, Yan , CHENG, Peter T.W. , WANG, Ying , JUSUF, Sutjano , TAO, Shiwei , ZHANG, Hao , WU, Shung C. , ROBL, Jeffrey A.
IPC分类号： C07D231/12 , C07D207/323 , C07D307/82 , C07C62/34 , C07D277/593 , A61K31/33 , A61K31/185 , A61P3/10
CPC分类号： C07C62/34 , A61K31/192 , A61K31/343 , A61K31/415 , A61K31/426 , A61K31/44 , A61K31/4418 , C07C59/64 , C07C2601/02 , C07D207/323 , C07D213/55 , C07D213/65 , C07D231/12 , C07D277/30 , C07D277/593 , C07D307/79 , C07D307/82
摘要： The present invention provides compounds of Formula (I): or a stereoisomer, or a pharmaceutically acceptable salt thereof, wherein all of the variables are as defined herein. These compounds are GPR120 G protein coupled receptor modulators which may be used as medicaments
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公开(公告)号：EP3191454A1
公开(公告)日：2017-07-19
申请号：EP15766344.4
申请日：2015-09-08
发明人： SHI, Yan , CHENG, Peter T.W. , WANG, Ying , JUSUF, Sutjano , TAO, Shiwei , ZHANG, Hao , WU, Shung C. , ROBL, Jeffrey A.
IPC分类号： C07D231/12 , C07D207/323 , C07D307/82 , C07C62/34 , C07D277/593 , A61K31/33 , A61K31/185 , A61P3/10
CPC分类号： C07C62/34 , A61K31/192 , A61K31/343 , A61K31/415 , A61K31/426 , A61K31/44 , A61K31/4418 , C07C59/64 , C07C2601/02 , C07D207/323 , C07D213/55 , C07D213/65 , C07D231/12 , C07D277/30 , C07D277/593 , C07D307/79 , C07D307/82
摘要： The present invention provides compounds of Formula (I): or a stereoisomer, or a pharmaceutically acceptable salt thereof, wherein all of the variables are as defined herein. These compounds are GPR120 G protein coupled receptor modulators which may be used as medicaments
摘要翻译： 本发明提供式（I）的化合物或其立体异构体或其药学上可接受的盐，其中所有变量如本文所定义。 这些化合物是可以用作药物的GPR120 G蛋白偶联受体调节剂
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公开(公告)号：EP2054368B1
公开(公告)日：2015-09-16
申请号：EP07814376.5
申请日：2007-08-23
IPC分类号： C07C61/39 , C07C61/40 , C07D203/18 , C07D205/04 , C07D205/08 , C07D263/04 , C07D263/30 , C07D317/72 , C07D493/08 , C07D295/18 , C07C62/38 , C07D451/02 , C07C57/00 , C07C59/00 , C07D217/02 , C07D401/12 , C07D403/04 , C07D407/06
CPC分类号： C07C61/40 , C07B2200/07 , C07C57/50 , C07C57/62 , C07C59/54 , C07C59/56 , C07C59/72 , C07C59/88 , C07C61/39 , C07C62/38 , C07C2603/66 , C07C2603/74 , C07D203/18 , C07D205/04 , C07D205/06 , C07D207/12 , C07D207/14 , C07D207/16 , C07D211/42 , C07D211/46 , C07D213/40 , C07D217/02 , C07D241/08 , C07D257/04 , C07D261/02 , C07D261/08 , C07D263/04 , C07D277/04 , C07D277/46 , C07D277/64 , C07D277/82 , C07D285/135 , C07D295/185 , C07D295/205 , C07D401/12 , C07D403/04 , C07D407/06 , C07D413/04 , C07D471/04 , C07D493/08
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公开(公告)号：EP2566860B1
公开(公告)日：2014-09-10
申请号：EP11720256.4
申请日：2011-05-04
发明人： YE, Xiang-Yang , WACKER, Dean A. , ROBL, Jeffrey A. , WANG, Ying
IPC分类号： C07D401/14 , C07D413/14 , C07D417/12 , C07D417/14 , A61K31/506 , A61K31/4545 , A61K31/437 , A61K31/5375 , A61K31/496 , A61P3/10 , A61P3/04
CPC分类号： C07D417/14 , C07D401/14 , C07D413/14 , C07D417/12
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15.发明公开TRIAZOLOPYRIDINE 11-BETA HYDROXYSTEROID DEHYDROGENASE TYPE I INHIBITORS 审中-公开三唑并吡啶作为11-β-羟基TYPE I抑制剂
公开(公告)号：EP2205598A1
公开(公告)日：2010-07-14
申请号：EP08835346.1
申请日：2008-09-19
发明人： LI, Jun , ROBL, Jeffrey A. , LI, James J. , KENNEDY, Lawrence J. , WANG, Haixia , LI, Jie Jack , QIAN, Xinhua , DESHPANDE, Rajendra P. , KOLLA, Laxma R. , CANN, Reginald O. , WEI, Chenkou , GALELLA, Michael
IPC分类号： C07D471/04 , A61K31/437 , A61P3/10 , A61P19/02
CPC分类号： C07D471/04
摘要： Novel compounds are provided which are 11-beta-hydroxysteroid dehydrogenase type I inhibitors. 11-beta-hydroxysteroid dehydrogenase type I inhibitors are useful in treating, preventing, or slowing the progression of diseases requiring 11-beta-hydroxysteroid dehydrogenase type I inhibitor therapy. These novel compounds of formula I: or stereoisomers or pharmaceutically acceptable salts thereof, wherein G, Q, X, Y, R3, R3a, and R3b are defined herein.
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