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公开(公告)号：EP2957342B1
公开(公告)日：2020-07-29
申请号：EP14751107.5
申请日：2014-02-07
IPC分类号： B01J31/22 , C07C201/12 , C07C205/15 , C07C205/16 , C07C205/26 , C07C205/32 , C07B61/00 , C07C205/02 , C07C237/36 , B01J31/02
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公开(公告)号：EP3669977A1
公开(公告)日：2020-06-24
申请号：EP18846150.3
申请日：2018-08-14
IPC分类号： B01J31/02 , B01J31/40 , C07B53/00 , C07B61/00 , C07C231/02 , C07C231/16 , C07C233/11 , C07C233/13 , C07C233/22 , C07C233/29 , C07C269/06 , C07C271/22 , C07D333/38
摘要： A catalyst represented by General Formula (1) below:
where in the General Formula (1), R 1 to R 14 each independently represent a hydrogen atom or a substituent.-
3.发明授权THIOAMIDE COMPOUND, METHOD FOR PRODUCING THIOAMIDE COMPOUND, METHOD FOR PRODUCING [(4R,6R)-6-AMINOETHYL-1,3-DIOXAN-4-YL]ACETATE DERIVATIVE, AND METHOD FOR PRODUCING ATORVASTATIN 有权硫代酰胺化合物，制备硫代酰胺化合物的方法，制备[（4R，6R）-6-氨基乙基-1,3-二氧杂环己烷-4-基]乙酸酯衍生物的方法，以及制备阿托伐他汀的方法
公开(公告)号：EP2679580B1
公开(公告)日：2017-08-09
申请号：EP12750077.5
申请日：2012-02-14
IPC分类号： C07C327/42 , A61K31/40 , A61P3/06 , A61P13/08 , A61P19/10 , A61P25/28 , C07D207/34 , C07F7/18 , C07B61/00
CPC分类号： C07C327/42 , C07B53/00 , C07D207/337 , C07D207/34 , C07F7/1852 , C07F7/1856 , Y02P20/55
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公开(公告)号：EP2792675A1
公开(公告)日：2014-10-22
申请号：EP12856751.8
申请日：2012-11-30
IPC分类号： C07D307/33 , B01J31/24 , C07C323/12 , C07C381/12 , C07D301/02 , C07D303/22 , C07D309/30 , C07B53/00 , C07B61/00
CPC分类号： C07F7/0812 , B01J31/24 , C07B53/00 , C07C323/12 , C07C323/16 , C07C381/12 , C07D215/227 , C07D301/02 , C07D303/22 , C07D307/33 , C07D309/30 , C07D405/12 , C07F7/12 , C07F7/1844 , C07F9/5059 , C07F9/65616 , Y02P20/55
摘要： A compound represented by the following General Formula (1):
where R 1 represents a protective group for a hydroxyl group or a hydrogen atom, and R 2 represents a methyl group or an ethyl group.-
5.发明公开COMPOUND, MANUFACTURING METHOD THEREFOR, AND METHOD FOR MANUFACTURING OPTICALLY ACTIVE -AMINOPHOSPHONATE DERIVATIVE 审中-公开化合物，工艺用于生产光学活性AMINOPHOSPHONATDERIVATS产生与工艺
公开(公告)号：EP3015472A1
公开(公告)日：2016-05-04
申请号：EP13888338.4
申请日：2013-10-08
发明人： SHIBASAKI, Masakatsu , KUMAGAI, Naoya , YIN, Liang , BAO, Youmei
CPC分类号： C07F9/4062 , B01J31/24 , B01J2231/34 , B01J2531/16 , C07F9/36 , C07F9/4009 , C07F9/4015 , C07F9/4056 , C07F9/5054 , C07F9/65683
摘要： A method for producing a compound represented by General Formula (1), the method including:
reacting a compound represented by General Formula (3) and a compound represented by General Formula (4):
where R 1 and R 2 each represent aliphatic group which may have substituent, or aromatic group which may have substituent (with the proviso that R 1 and R 2 are different groups), R 3 represents aromatic group which may have substituent, and R 4 represents aliphatic group which may have substituent, or aromatic group which may have substituent,
where R 1 and R 2 each represent aliphatic group which may have substituent, or aromatic group which may have substituent (with the proviso that R 1 and R 2 are different groups), and R 3 represents aromatic group which may have substituent,
where R 4 represents aliphatic group which may have substituent, or aromatic group which may have substituent.-
6.发明公开CATALYST AND METHOD FOR PRODUCING OPTICALLY ACTIVE ANTI-1,2-NITROALKANOL COMPOUND 审中-公开催化剂及其制备方法光学活性的ANTI-1,2-NITROALKANOLVERBINDUNG
公开(公告)号：EP2957342A1
公开(公告)日：2015-12-23
申请号：EP14751107.5
申请日：2014-02-07
IPC分类号： B01J31/22 , C07C201/12 , C07C205/15 , C07C205/16 , C07C205/26 , C07C205/32 , C07B61/00 , C07C205/02 , C07C237/36
摘要： A catalyst, which is obtained by mixing a compound expressed by the following Structural Formula (1), a nitroalkane compound, a neodymium-containing compound, a sodium-containing compound, and a carbon structure:
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7.发明公开THIOAMIDE COMPOUND, METHOD FOR PRODUCING THIOAMIDE COMPOUND, METHOD FOR PRODUCING [(4R,6R)-6-AMINOETHYL-1,3-DIOXANE-4-YL]ACETATE DERIVATIVE, AND METHOD FOR PRODUCING ATORVASTATIN 有权硫代酰胺，用于生产硫代酰胺，用于生产[（4 R，6 R）] - 6-氨基乙基-1,3-二恶烷-4-基] -ACETATDERIVATEN AND PROCESS FOR PRODUCING阿托伐他汀
公开(公告)号：EP2679580A1
公开(公告)日：2014-01-01
申请号：EP12750077.5
申请日：2012-02-14
IPC分类号： C07C327/42 , A61K31/40 , A61P3/06 , A61P13/08 , A61P19/10 , A61P25/28 , C07D207/34 , C07F7/18 , C07B61/00
CPC分类号： C07C327/42 , C07B53/00 , C07D207/337 , C07D207/34 , C07F7/1852 , C07F7/1856 , Y02P20/55
摘要： A thioamide compound represented by the following general formula (1):
wherein, in the general formula (1), R 1 represents one of -OR 11 and -NR 12 R 13 ; R 2 and R 3 each independently represent one of a protecting group of an amide group and a hydrogen atom; the R 11 represents one of a protecting group of a hydroxyl group and a hydrogen atom; and the R 12 and R 13 each independently represent one of a protecting group of an amino group and a hydrogen atom, where the R 12 and R 13 may together form a protecting group having a cyclic structure.-
8.发明公开
公开(公告)号：EP3381553A1
公开(公告)日：2018-10-03
申请号：EP16868516.2
申请日：2016-11-21
IPC分类号： B01J31/22 , B01J37/04 , C07C201/12 , C07C205/16 , C07C205/32 , C07C205/54 , C07B61/00 , C07C237/04
CPC分类号： B01J31/22 , B01J37/04 , B01J2231/341 , B01J2531/004 , B01J2531/12 , B01J2531/38 , C07B61/00 , C07C201/12 , C07C205/16 , C07C205/32 , C07C205/54 , C07C237/04
摘要： A catalyst including: neodymium; sodium; and a ligand, which is a compound expressed by Structural Formula (1) below, wherein the neodymium and the ligand form a complex at a molar ratio of 1 : 2 (neodymium : ligand):
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公开(公告)号：EP3015472B1
公开(公告)日：2018-08-01
申请号：EP13888338.4
申请日：2013-10-08
发明人： SHIBASAKI, Masakatsu , KUMAGAI, Naoya , YIN, Liang , BAO, Youmei
IPC分类号： C07F9/40 , C07F9/53 , C07B61/00 , C07F9/6568 , C07F9/36
CPC分类号： C07F9/4062 , B01J31/24 , B01J2231/34 , B01J2531/16 , C07F9/36 , C07F9/4009 , C07F9/4015 , C07F9/4056 , C07F9/5054 , C07F9/65683
摘要： A method for producing a compound represented by General Formula (1), the method including: reacting a compound represented by General Formula (3) and a compound represented by General Formula (4): where R 1 and R 2 each represent aliphatic group which may have substituent, or aromatic group which may have substituent (with the proviso that R 1 and R 2 are different groups), R 3 represents aromatic group which may have substituent, and R 4 represents aliphatic group which may have substituent, or aromatic group which may have substituent, where R 1 and R 2 each represent aliphatic group which may have substituent, or aromatic group which may have substituent (with the proviso that R 1 and R 2 are different groups), and R 3 represents aromatic group which may have substituent, where R 4 represents aliphatic group which may have substituent, or aromatic group which may have substituent.
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10.发明公开OPTICALLY ACTIVE -TRIFLUORMETHYL- -AMINO ACID DERIVATIVE PRODUCTION METHOD 审中-公开光学活性 - 三氟甲基 - 氨基酸衍生物生产方法
公开(公告)号：EP3199524A1
公开(公告)日：2017-08-02
申请号：EP15844955.3
申请日：2015-09-18
发明人： SHIBASAKI, Masakatsu , KUMAGAI, Naoya , YIN, Liang
IPC分类号： C07D213/75 , B01J31/22 , C07B53/00 , C07B57/00 , C07C269/06 , C07C271/22 , C07D471/04 , C07B61/00
CPC分类号： C07D471/04 , B01J31/22 , B01J31/2409 , B01J2231/50 , B01J2531/16 , C07B53/00 , C07B57/00 , C07B61/00 , C07B2200/07 , C07C269/06 , C07C271/22 , C07D213/75
摘要： A method for producing an optically active α-trifluoromethyl-β-amino acid derivative, the method including: allowing a compound represented by the following General Formula (1) and a compound represented by the following General Formula (2) to react in the presence of a copper-optically active phosphine complex obtained from a copper compound and an optically active phosphine compound, to thereby obtain an optically active α-trifluoromethyl-β-amino acid derivative represented by the following General Formula (3):
摘要翻译： 一种光学活性α-三氟甲基-β-氨基酸衍生物的制造方法，其特征在于，使下述通式（1）所示的化合物与下述通式（2）所示的化合物在存在下反应 由铜化合物和光学活性膦化合物得到的铜 - 光活性膦配合物，由此获得由以下通式（3）表示的光学活性α-三氟甲基-β-氨基酸衍生物：
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