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    Indanderivatives
    1.
    发明公开
    Indanderivatives 失效
    Indanderivate。

    公开(公告)号：EP0453066A1

    公开(公告)日：1991-10-23

    申请号：EP91300956.9

    申请日：1991-02-06

    申请人： ZENECA LIMITED

    发明人： Chrystal, Ewan James Turner ,  Barton, John Edward Duncan ,  Cartwright, David

    IPC分类号： C07C59/72 ,  C07C69/736 ,  C07C51/00 ,  C07C67/00 ,  C07C235/34 ,  C07C251/32 ,  A01N37/38 ,  A01N37/52

    CPC分类号： C07C251/60 ,  A01N35/10 ,  A01N37/38 ,  C07C45/71 ,  C07C49/755 ,  C07C59/72 ,  C07C69/708 ,  C07C69/736 ,  C07C235/34 ,  C07C251/44 ,  C07C2602/08

    摘要： A compound of formula (I) :

    in which
    Ar is an optionally substituted aryl or heterocyclic ring system;
    W is O or NR¹ where R¹ is hydrogen or lower alkyl;
    A is=CH or >CH₂ and B is=C-R²,
    >
    C=R⁵ such that
    -B-A- is

    where R² is H or CR⁶ R⁷XR⁸; or
    -B-A- is

    where CR³R⁴ is CH-CR⁶R⁷XR⁸, CH-OCR⁶R⁷XR⁸, C(R⁹)OCOR¹⁰, CR⁹R¹⁰, C(R⁹))OCOR¹⁰, C(R⁹)OR¹⁰, C(OR⁹)OR¹⁰, or CH-CH₂(CO₂R¹¹); or
    -B-A- is

    where
    R5 is =CR⁷XR⁸, =NOCR⁶R⁷XR⁸, =NOR¹¹ or =NOCOR¹¹. where X is (CH₂)n, CH=CH, CH(OR²⁰)CH₂, COCH₂; and n is O, 1 or 2;
    R⁶ and R⁷ are independently selected from H, optionally substituted alkyl, alkenyl or alkynyl, halogen, NR⁹R¹⁰, or R⁶ and R⁷ together with the carbon to which they are attached form an optionally substituted alkenyl or cycloalkyl group;
    R⁸ is CO₂R¹², CN, COR¹², CH₂OR¹², CH(OH)R¹², CH(OR¹²)R¹³, CSNH₂, COSR¹², CSOR¹², CONHSO₂R¹², CONR¹⁴R¹⁵, CONHNR¹⁴R¹⁵, CONHN⁺R¹⁴R¹⁵R¹⁶R¹⁷, CO₂⁻⁺R¹⁹⁺ or COON=CR¹⁴R¹⁵;
    R¹⁹⁺ is an agriculturally acceptable cation;
    R¹⁷⁻ is an agriculturally acceptable anion;
    R⁹, R¹⁰, R¹⁴, R¹⁵ and R¹⁶ are independently selected from H or an optionally substituted alkyl, alkenyl, aryl or alkynyl group or any two of R⁹, R¹⁰, R¹⁴ and R¹⁵, R¹⁶ together with the atom to which they are attached form a cycloalkyl or heterocyclic ring, and R¹⁴ and R¹⁵ may additionally be a heterocyclic ring, provided that when B is CR⁹R¹⁰ or C(R⁹)OR¹⁰, R⁹ and R¹⁰ are not both hydrogen.

    摘要翻译： 式（I）化合物：其中Ar为任选取代的芳基或杂环系统; W是O或NR 1，其中R 1是氢或低级烷基; A为= CH或> CH 2且B为= CR 2，CH 2> C = R 5，使得-BA-为CHEM，其中R 2为H或CR 6 R 7 > XR <8>; 或-BA-是，其中CR 3 R 4是CH-CR 6 R 7 XR 8，CH-OCR 6 R 7 XR 8，C（ R 9）OCOR 1，O，C（R 9）OCOR 1，O，C（R 9） C（OR 9）OR 1，或CH-CH 2（CO 2 R 1）1）。 或-BA-是。 其中X是（CH 2）n，CH = CH，CH（OR 2）O 2，COCH 2; 且n为O，1或2; R 6和R 7独立地选自H，任选取代的烷基，烯基或炔基，卤素，NR 9 R 1或R 6和R 7与 它们所连接的碳形成任选取代的烯基或环烷基; R 8是CO 2 R 1，CN，COR 1，CH 2 OR 1，CH（OH）R 1，CH（OR 1） 2）R 1，3，CSNH 2，COSR 1，CSOR 1，CONHSO 2 R 1，CONR 1 R 4 R 5 >，CONHNR 1 <4> R 1 <5>，CONHN + R 1，R 1，R 1，R 1，R 6，R 1， CO 2 = CO 2 = CR 1，R 2，R 3， R 1 <9> <+>是农业上可接受的阳离子; R 1是农业上可接受的阴离子; R 9，R 1，O，R 1，R 1，R 5和R 6独立地选自H或任选取代的烷基，烯基，芳基 或炔基或R 9，R 1，O，R 1和R 5中的任何两个，R 1和它们的原子一起 连接形成环烷基或杂环，并且R 1和R 5还可以是杂环，条件是当B是CR 9 R 1或C （R 9）OR 1 <0>，R 9和R 1不同时为氢。

    Triazolopyridine derivatives
    2.
    发明公开
    Triazolopyridine derivatives 失效
    三唑并吡啶衍生物

    公开(公告)号：EP0453065A1

    公开(公告)日：1991-10-23

    申请号：EP91300955.1

    申请日：1991-02-06

    申请人： ZENECA LIMITED

    发明人： Pearson, David Philip John ,  Barton, John Edward Duncan ,  Cartwright, David ,  Barnett, Susan Patricia

    IPC分类号： C07D471/04 ,  C07D213/74 ,  C07D401/12 ,  A01N43/90

    CPC分类号： C07D213/74 ,  A01N43/90 ,  C07D401/12 ,  C07D471/04

    摘要： A compound of formula (I) :

    in which
    the dotted lines indicate the presence of two double bonds arranged so as to form a fused hetero-aromatic ring system;
    Ar is an optionally substituted aryl or heterocyclic ring;
    W is O or NR¹, where R¹ is hydrogen or lower alkyl;
    X is (CH₂) n , CH=CH, CH(OR⁵)CH₂, COCH₂;
    where n is O, 1 or 2;
    R² and R³ are independently selected from H, optionally substituted alkyl, alkenyl or alkynyl, halogen, NR⁶R⁷ or R² and R³ together with the carbon to which they are attached form an optionally substituted alkenyl or cycloalkyl group;
    R⁴ is CO₂R⁸, CN, COR⁸, CH₂OR⁸, CH(OH)R⁸, CH(OR⁸)R⁹, CSNH₂, COSR⁸, CSOR⁸, CONHSO₂R⁸, CONR¹⁰R¹¹, CONHNR¹⁰R¹¹, CONHN⁺R¹⁰R¹¹R¹²R¹³⁻, CO₂⁻R¹⁴⁺ or COON=CR¹⁰R¹¹;
    R¹⁴⁺ is an agriculturally acceptable cation; and R¹³⁻ is an agriculturally acceptable anion;
    R⁵, R⁸ and R⁹ are independently selected from H or an optionally substituted alkyl, aryl, alkenyl or alkynyl group; and
    R⁶, R⁷, R¹⁰, R¹¹, and R¹² are independently selected from H or an optionally substituted alkyl, alkenyl, aryl or alkynyl group or any two of R⁶, R⁷, R¹⁰, R¹¹ and R¹² together with the atom to which they are attached form a cycloalkyl or heterocyclic ring. Compounds of formula (I) are herbicidal and composition containing them and methods of treatment using them are also described.

    摘要翻译： 式（I）化合物：其中虚线表示存在两个排列的双键以形成稠合的杂芳族环体系; Ar是任选取代的芳基或杂环; W是O或NR 1，其中R 1是氢或低级烷基; X是（CH 2）n，CH = CH，CH（OR 5）CH 2，COCH 2; 其中n是0,1或2; R 2和R 3独立地选自H，任选取代的烷基，烯基或炔基，卤素，NR 6 R 8或R 2和R 3与它们所连接的碳一起形成任选取代的链烯基或环烷基; R 4是CO 2 R 7，CN，COR 8，CH 2 OR 7，CH（OH）R 7，CH（OR 7）R 8，CSNH 2，COSR 6，CSOR 7，CONHSO 2 R 8，CONR 10 R 11，CONHNR 10 R 11，CONHN + R 10 R 11 R 12 R 13 - ，CO -2 R 14+或COON = CR 10 R 11; R 14+是农业上可接受的阳离子; 而R 13是农业上可接受的阴离子; R 5，R 6和R 6独立地选自H或任选取代的烷基，芳基，烯基或炔基; 和R 7，R 9，R 11，R 11和R 12独立地选自H或任意取代的烷基，烯基，芳基或炔基或R 7，R 9，R 10，R 11和R 12中的任何两个与它们所连接的原子一起 形成环烷基或杂环。 式（I）化合物是除草剂，并且还描述了含有它们的组合物和使用它们的治疗方法。

    Benzisoxazole derivatives
    8.
    发明公开
    Benzisoxazole derivatives 失效
    苯并噻唑衍生物

    公开(公告)号：EP0442655A3

    公开(公告)日：1992-07-08

    申请号：EP91300958.5

    申请日：1991-02-06

    申请人： ZENECA LIMITED

    发明人： Chrystal, Ewan James Turner ,  Barton, John Edward Duncan ,  Cartwright, David ,  Mathews, C. J.

    IPC分类号： C07D261/20 ,  A01N43/80 ,  C07C49/84 ,  C07D413/12 ,  C07D311/54

    CPC分类号： C07D413/10 ,  A01N43/80 ,  C07D261/20

    摘要： A herbicidal compound of formula (I) :
    in which
    Ar is an optionally subsitituted aryl or heterocyclic ring system; R 1 and R 2 are independently selected from H, optionally substituted alkyl, alkenyl or alkynyl, halogen, NR a R b , or R 1 and R 2 together with the carbon to which they are attached form an optionally substituted alkenyl or cycloalkyl group; R 3 is C0 2 R 4 , CN, COR 4 , CH 2 0R 4 , CH(OH)R 4 , CH(OR 4 )R S , CH 2 0S0 2 R 4 , CH 2 0S0 3 R 4 , CH 2 0NR 6 R 7 , CSNH 2 , COSR 4 , CSOR 4 , CONHSO 2 R 4 , CONR 6 R 7 , CONHNR 6 R 7 , CONHN + R 6 R 7 R 8 Y-, CO 2 -M + or COON=CR 6 R 7 ; M is an agriculturally acceptable cation; Y- is an agriculturally acceptable anion; R 4 , and R 5 are independently selected from H or an optionally substituted alkyl, aryl, alkenyl or alkynyl group; R 6 , R 7 , R 8 , R 9 , R a and R b are independently selected from H or an optionally substituted alkyl, alkenyl, aryl or alkynyl group or any two of R 6 , R 7 , R 8 , R 9 , R a and R b together with the atom to which they are attached form a cycloalkyl or heterocyclic ring: R 6 and R 7 may also be a heterocyclic ring; W is O or NR 10 where R 10 is H or lower alkyl; X is (CHz) n , CH=CH, CH(OR c )CH 2 , COCH 2 ; where R c is H or an optionally substituted alkyl, aryl, alkynyl or alkynyl group; and n is 0, 1 or 2. Process for the preparation of these compounds and compositions containing them are also described.

    Heterocyclic compounds
    9.
    发明公开
    Heterocyclic compounds 失效
    Heterozyklische Verbindungen。

    公开(公告)号：EP0355049A2

    公开(公告)日：1990-02-21

    申请号：EP89307454.2

    申请日：1989-07-21

    申请人： ZENECA LIMITED

    发明人： Barton, John Edward Duncan

    IPC分类号： C07D249/18 ,  C07D401/12 ,  A01N43/647

    CPC分类号： C07D401/12 ,  A01N43/647 ,  C07C205/38 ,  C07C217/90 ,  C07D249/18

    摘要： A herbicidal compound of formula (I):
    in which R' is independently selected from H, CN, N0 2 , halogen, lower alkyl, lower haloalkyl; m is an integer of from 1 to 4; R 2 is N or CR' where R 1 is as defined above; R 3 is a group of formula (a), (b) or (c):


    or N-oxide or quaternary salt derivatives thereof wherein R 4 is a specified organic group. Processes for the preparation of these compounds and compositions containing them are also described.

    摘要翻译： 式（I）的除草化合物：其中R 1独立地选自H，CN，NO 2，卤素，低级烷基，低级卤代烷基; m为1〜4的整数， R 2是N或CR 1，其中R 1如上定义; R 3是式（a），（b）或（c）的基团：其中R 4是指定的有机基团的或N-氧化物或季盐衍生物。 还描述了制备这些化合物和含有它们的组合物的方法。

    Substituted benzimidazole and indazole derivatives, processes for their preparation and their use as herbicides
    10.
    发明公开
    Substituted benzimidazole and indazole derivatives, processes for their preparation and their use as herbicides 失效
    取代的苯并咪唑和吲唑衍生物，它们的制备方法和它们作为除草剂的用途。

    公开(公告)号：EP0448206A2

    公开(公告)日：1991-09-25

    申请号：EP91300954.4

    申请日：1991-02-06

    申请人： ZENECA LIMITED

    发明人： Barton, John Edward Duncan ,  Cartwright, David ,  McCormack, Derek

    IPC分类号： C07D231/56 ,  C07D235/06 ,  C07D235/10 ,  C07D235/24 ,  C07D401/12 ,  C07D235/08 ,  C07D235/26 ,  C07D235/22 ,  C07C217/90 ,  C07C205/38 ,  C07C255/25

    CPC分类号： C07D235/24 ,  C07C205/38 ,  C07C217/90 ,  C07C255/25 ,  C07D231/56 ,  C07D235/06 ,  C07D235/08 ,  C07D235/10 ,  C07D235/16 ,  C07D401/12

    摘要： A herbicidal compound of formula (I) :
    or N-oxide or quaternised derivative thereof;

    in which the dotted lines indicate the presence of two double bonds arranged so as to form a fused hetero-aromatic ring system;
    Ar is an optionally substituted aryl or heterocyclic ring system;
    W is 0 or NR 1
    where R 1 is H or lower alkyl;
    A, B, D are independently selected from N, NR 2 , N-E, CR 6 , C-E or C(R 6 )E;
    wherein E is:
    provided 2 of A, B and D are N, NR 2 or N-E and at least one of A, B or D carries a group E;
    where R 2 is H, OR 7 , CN, COOR 8 , alkyl or haloalkyl;
    R 3 and R 4 are independently selected from H, optionally substituted alkyl, alkenyl or alkynyl, halogen, NR 9 R 10 , or
    R 3 and R 4 together with the carbon to which they are attached form an optionally substituted alkenyl or cycloalkyl group;
    R 5 is CO 2 R 11 , CN, COR 11 , CH 2 OR 11 , CH(OH)R", CH(OR 11 )R 12 , CSNH 2 , COSR 11 , CSOR", CONHSO 2 R 11 , CONR 13 R 14 , CONHNR 13 R 14 , CONHN + R 13 R 14 R 15 Y-, CO 2 -M + or COON=CR 13 R 14 ;
    X is (CH 2 ) n , CH=CH, CH(OR 16 )CH 2 or COCH z ;
    where n is 0, 1 or 2;
    M is an agriculturally acceptable cation;
    Y- is an agriculturally acceptable anion;
    R 6 is H, halogen, OR 7 , CN, COOR 8 , alkyl or haloalkyl;
    R 7 and R 8 are independently H or lower alkyl;
    R 11 , R 12 and R 16 are independently selected from H or an optionally substituted alkyl, alkenyl, alkynyl or aryl group; and
    R 9 , R 10 , R 13 , R 14 and R 15 are independently selected from H or an optionally substituted alkyl, alkenyl, alkynyl or aryl group or any two of R 9 , R 10 , R 13 , R 14 and R 15 together with the atom to which they are attached form a cycloalkyl or heterocyclic ring providing that the compound is other than 5-(2,4-dichlorophenoxy)indazol-1- ylacetic acid or its methyl ester.

    Process for the preparation of these compounds and compositions containing them are also described.

    摘要翻译： 式的除草化合物（I）：或N-氧化物或季铵化衍生物; 其中虚线表示的两个双键，例如布置为形成稠合的杂芳环体系的存在; Ar是芳基或杂环OPTIONALLY substituiertem环体系; W是O或NR <1>，其中R <1>是H或低级烷基; A，B，D独立地选自N，NR <2>的N- E，CR <6>，C-E或C（R <6>）E组; worin E是：提供A，B和D中的2是N，NR <2>或N-E和A，B或D中的至少一个携带基团E; 其中R <2>为H，OR <7>，CN，COOR <8>，烷基或卤代烷基; [R <3>和R <4>是unabhängig选自H，任选substituiertem烷基，烯基或炔基，卤素，NR选择<9> - [R <1> <0>，或R <3>和R <4>连同 碳它们在OPTIONALLY substituiertem烯基或环烷基连接形式; [R <5>是CO 2 <1> <1>，CN，COR <1> <1>，CH 2 OR <1> <1>，CH（OH）R <1> <1>，CH（OR <1> < 1>）R <1> <2>，CSNH 2，COSR <1> <1>，CSOR <1> <1>，CONHSO2R <1> <1>，CONR <1> <3> [R <1> <4 >，CONHNR <1> <3> [R <1> <4>，CONHN <+> - [R <1> <3> [R <1> <4> - [R <1> <5>ý< - > CO2 < - >中号<+>或COON = CR <1> <3> [R <1> <4>; X是（CH 2）N，CH = CH，CH（OR <1> <6>）CH 2或COCH 2; 其中n是O，1或2; 中号<+>是农业上可接受的阳离子; ÿ< - >是农业上可接受的阴离子; [R <6>为H，卤素，OR <7>，CN，COOR <8>，烷基或卤代烷基; [R <7>和R <8>是unabhängigH或低级烷基; [R <1> <1>，R <1> <2>和R <1> <6>独立地选自H或任选取代的烷基，烯基，炔基或芳基; 且R <9>，R <1> <0> - [R <1> <3>，R <1> <4>和R <1> <5>独立地选自H或任选取代的烷基，烯基， 炔基或芳基或R的<9> - [R <1> <0> - [R <1> <3>，R <1> <4>和R <1> <5>与原子一起任意两个 它们所连接形成环烷基或杂环环提供没有该化合物不是5-（2,4-二氯苯氧基）其他吲唑-1-基乙酸或它的甲基酯。 用于合成的化合物和含它们的组合物的制备过程中是如此描述。