Pyrimidine-2-phenylamino derivatives
    7.
    发明授权
    Pyrimidine-2-phenylamino derivatives 失效
    嘧啶-2-苯基氨基衍生物

    公开(公告)号:US4904778A

    公开(公告)日:1990-02-27

    申请号:US262122

    申请日:1988-10-24

    摘要: The invention relates to ureas having a herbicidal and plant growth-regulating action of the formula ##STR1## in which R.sup.1 and R.sup.2 each represent, independently of the other, hydrogen, halogen, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.4 -haloalkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -haloalkoxy, C.sub.1 -C.sub.4 -alkoxycarbonyl, C.sub.1 -C.sub.4 -alkoxy-(C.sub.1 -C.sub.4)-alkyl, nitro or cyano, andR.sup.3 and R.sup.4 each represents, independently of the other, hydrogen, halogen, cyano, OH, SH, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.4 -haloalkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -haloalkoxy, C.sub.1 -C.sub.4 -alkylthio, C.sub.1 -C.sub.4 -haloalkylthio, amino, mono-C.sub.1 -C.sub.4 -alkylamino, di-C.sub.1 -C.sub.4 -alkylamino, C.sub.1 -C.sub.4 -alkoxycarbonyl or C.sub.1 -C.sub.4 -alkoxy-(C.sub.1 -C.sub.4)-alkyl,processes and intermediates for the preparation thereof, and herbicidal and plant growth-regulating compositions containing a compound of the formula I.

    N-azidophenylsulfonyl-N'-triazinylureas
    8.
    发明授权
    N-azidophenylsulfonyl-N'-triazinylureas 失效
    N-叠氮苯基磺酰基-N'-三嗪基脲

    公开(公告)号:US4589912A

    公开(公告)日:1986-05-20

    申请号:US763175

    申请日:1985-08-07

    CPC分类号: C07D521/00 A01N47/36

    摘要: The invention relates to N-azidophenylsulfonyl-N'-pyrimidinyl- and -N'-triazinylureas of the general formula ##STR1## wherein E is nitrogen or the methine bridge,R.sub.1 is hydrogen, halogen, nitro, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy, C.sub.1 -C.sub.4 alkoxycarbonyl, C.sub.1 -C.sub.4 alkylthio, C.sub.1 -C.sub.4 alkylsulfinyl, C.sub.1 -C.sub.4 alkylsulfonyl or C.sub.2 -C.sub.5 alkoxyalkoxy,R.sub.2 is C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 alkoxy or C.sub.1 -C.sub.3 haloalkoxy,R.sub.3 is hydrogen, halogen, C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 haloalkyl, C.sub.1 -C.sub.3 alkoxy, C.sub.1 -C.sub.3 haloalkoxy, C.sub.2 -C.sub.5 alkoxyalkoxy or --NR.sub.4 R.sub.5, whereinR.sub.4 is hydrogen or methyl andR.sub.5 is hydrogen, methyl, ethyl or methoxyand to the salts thereof with amines, alkali metal hydroxides and alkaline earth metal hydroxides or with quaternary ammonium bases. These compounds have good pre- and postemergence selective herbicidal and growth regulating properties.

    摘要翻译: 本发明涉及通式为“IMAGE”的N-叠氮苯基磺酰基-N'-嘧啶基和-N'-三嗪基脲,其中E为氮或次甲基桥,R1为氢,卤素,硝基,C1-C4烷基,C1-C4卤代烷基 ,C1-C4烷氧基,C1-C4卤代烷氧基,C1-C4烷氧基羰基,C1-C4烷硫基,C1-C4烷基亚磺酰基,C1-C4烷基磺酰基或C2-C5烷氧基烷氧基,R2是C1-C3烷基,C1-C3烷氧基或C1-C3卤代烷氧基,R3是氢, C 3烷基,C 1 -C 3卤代烷基,C 1 -C 3烷氧基,C 1 -C 3卤代烷氧基,C 2 -C 5烷氧基烷氧基或-NR 4 R 5,其中R 4是氢或甲基,R 5是氢,甲基,乙基或甲氧基,其盐与胺,碱金属氢氧化物和 碱土金属氢氧化物或季铵碱。 这些化合物具有良好的芽前和芽后选择性除草和生长调节性质。

    Pyrimidine derivatives having a herbicidal action and an action
regulating plant growth
    9.
    发明授权
    Pyrimidine derivatives having a herbicidal action and an action regulating plant growth 失效
    具有除草作用的嘧啶衍生物和调节植物生长的作用

    公开(公告)号:US4741760A

    公开(公告)日:1988-05-03

    申请号:US938674

    申请日:1986-12-05

    摘要: N-Pyrimidin-4-yl-N'-sulfonylureas of the formula I and the basic addition salts thereof have herbicidal properties and properties for regulating, especially inhibiting, plant growth: ##STR1## the symbols in this formula having the following meanings: Q is halogen, lower alkyl, lower haloalkyl, lower alkoxy, lower haloalkoxy, nitro, amino, lower alkyl or dialkylamino, lower alkoxycarbonyl, formyl, lower alkoxyalkyl, lower alkoxyalkoxy, lower alkylthio, lower alkylsulfinyl or alkylsulfonyl, C.sub.1 -C.sub.4 -alkenyl or C.sub.1 -C.sub.4 -alkynyl,R.sub.1 is hydrogen, halogen, nitro, a ketal radical, a carbonyl radical substituted by allyl, haloalkyl, alkoxy or cycloalkyl, or is an oxime radical, a lower alkoxy, lower alkylthio, lower alkyl, lower alkylsulfinyl or sulfonyl group,R.sub.2 and R.sub.3 independently of one another are each hydrogen, halogen, lower alkyl, lower haloalkyl, lower alkoxy, lower haloalkoxy, lower alkylthio, lower alkoxyalkyl, lower alkoxyalkoxy, amino, lower alkyl- or dialkylamino or cyclopropyl, and R.sub.2 and Q together can also form a 2-4-membered carbon chain, which is optionally interrupted by an oxygen or sulfur atom or by the group --NR.sub.5 --,R.sub.4 is hydrogen, halogen, lower alkyl, methoxy, nitro or trifluoromethyl,R.sub.5 is hydrogen, C.sub.1 -C.sub.4 -alkyl or C.sub.3 -C.sub.4 -alkenyl,X is oxygen, sulfur, --NR.sub.5 --, ##STR2## --CH.dbd.CH-- or an annularly-linked phenyl ring, and Z is oxygen or sulfur.

    摘要翻译: 式I的N-嘧啶-4-基-N'-磺酰脲及其碱式加成盐具有用于调节,特别是抑制植物生长的除草性质和性质:(I)该式中的符号具有以下 含义:Q为卤素,低级烷基,低级卤代烷基,低级烷氧基,低级卤代烷氧基,硝基,氨基,低级烷基或二烷基氨基,低级烷氧基羰基,甲酰基,低级烷氧基烷基,低级烷氧基烷氧基,低级烷硫基,低级烷基亚磺酰基或烷基磺酰基, 烯基或C 1 -C 4炔基,R 1是氢,卤素,硝基,缩酮基,被烯丙基,卤代烷基,烷氧基或环烷基取代的羰基,或是肟基,低级烷氧基,低级烷硫基,低级烷基,低级 烷基亚磺酰基或磺酰基,R 2和R 3彼此独立地各自为氢,卤素,低级烷基,低级卤代烷基,低级烷氧基,低级卤代烷氧基,低级烷硫基,低级烷氧基烷基,低级烷氧基烷氧基,氨基,低级烷基 - 或二烷基氨基或环丙基, d R2和Q一起也可以形成2-4元碳链,其任选地被氧或硫原子间隔或由-NR 5 - ,R 4是氢,卤素,低级烷基,甲氧基,硝基或三氟甲基, R5是氢,C1-C4-烷基或C3-C4-烯基,X是氧,硫,-NR5-,-CH = CH-或环状连接的苯环,Z是氧或硫。

    N-Azidophenylsulfonyl-N'-pyrimidinyl ureas
    10.
    发明授权
    N-Azidophenylsulfonyl-N'-pyrimidinyl ureas 失效
    N-叠氮苯基磺酰基-N'-嘧啶基脲

    公开(公告)号:US4555262A

    公开(公告)日:1985-11-26

    申请号:US525365

    申请日:1983-08-22

    CPC分类号: C07D521/00 A01N47/36

    摘要: The invention relates to N-azidophenylsulfonyl-N'-pyrimidinyl- and -N'-triazinylureas of the general formula ##STR1## wherein E is nitrogen or the methine bridge,R.sub.1 is hydrogen, halogen, nitro, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy, C.sub.1 -C.sub.4 alkoxycarbonyl, C.sub.1 -C.sub.4 alkylthio, C.sub.1 -C.sub.4 alkylsulfinyl, C.sub.1 -C.sub.4 alkylsulfonyl or C.sub.2 -C.sub.5 alkoxyalkoxy,R.sub.2 is C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 alkoxy or C.sub.1 -C.sub.3 haloalkoxy,R.sub.3 is hydrogen, halogen, C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 haloalkyl, C.sub.1 -C.sub.3 alkoxy, C.sub.1 -C.sub.3 haloalkoxy, C.sub.2 -C.sub.5 alkoxyalkoxy or --NR.sub.4 R.sub.5, whereinR.sub.4 is hydrogen or methyl andR.sub.5 is hydrogen, methyl, ethyl or methoxyand to the salts thereof with amines, alkali metal hydroxides and alkaline earth metal hydroxides or with quaternary ammonium bases. These compounds have good pre- and postemergence selective herbicidal and growth regulating properties.

    摘要翻译: 本发明涉及通式为“IMAGE”的N-叠氮苯基磺酰基-N'-嘧啶基和-N'-三嗪基脲,其中E为氮或次甲基桥,R1为氢,卤素,硝基,C1-C4烷基,C1-C4卤代烷基 ,C1-C4烷氧基,C1-C4卤代烷氧基,C1-C4烷氧基羰基,C1-C4烷硫基,C1-C4烷基亚磺酰基,C1-C4烷基磺酰基或C2-C5烷氧基烷氧基,R2是C1-C3烷基,C1-C3烷氧基或C1-C3卤代烷氧基,R3是氢, C 3烷基,C 1 -C 3卤代烷基,C 1 -C 3烷氧基,C 1 -C 3卤代烷氧基,C 2 -C 5烷氧基烷氧基或-NR 4 R 5,其中R 4是氢或甲基,R 5是氢,甲基,乙基或甲氧基,其盐与胺,碱金属氢氧化物和 碱土金属氢氧化物或季铵碱。 这些化合物具有良好的芽前和芽后选择性除草和生长调节性质。