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157 条记录 (耗时 0.024 秒)

    Use of substituted 1,2,4-oxadiazole derivatives for combating endoparasites, new substituted 1,2,4-oxadiazole derivatives, and processes for their preparation
    92.
    发明授权
    Use of substituted 1,2,4-oxadiazole derivatives for combating endoparasites, new substituted 1,2,4-oxadiazole derivatives, and processes for their preparation 失效
    使用取代的1,2,4-恶二唑衍生物对抗内寄生虫，新的取代的1,2,4-恶二唑衍生物及其制备方法

    公开(公告)号：US5428047A

    公开(公告)日：1995-06-27

    申请号：US124909

    申请日：1993-09-21

    申请人： Peter Jeschke ,  Werner Lindner ,  Achim Harder ,  Norbert Mencke

    发明人： Peter Jeschke ,  Werner Lindner ,  Achim Harder ,  Norbert Mencke

    IPC分类号： A01N43/82 ,  A01N43/836 ,  A61K31/41 ,  A61K31/4245 ,  A61P33/00 ,  A61P33/10 ,  C07D271/06 ,  C07D413/06

    CPC分类号： C07D271/06 ,  A01N43/82 ,  A61K31/41

    摘要： The present invention relates to the use of substituted 1,2,4-oxadiazole derivatives of the general formula I ##STR1## in which R.sup.1 represents hydrogen, alkyl which is optionally substituted by halogen, alkoxy, hydroxyl, amino, alkylamino, dialkylamino, cycloalkylamino as well as cycloalkyl, optionally substituted aryl or hetaryl,R.sup.2 represents hydrogen and alkyl,X represents O, S, SO, SO.sub.2 and N-R.sup.3,R.sup.3 represents hydrogen, alkyl, alkylcarbonyl or halogenoalkylcarbonylR.sup.4 represents identical or different radicals from the series comprising hydrogen, halogen, cyano, nitro, isothiocyanato, amino, aminoacyl, alkylamino, dialkylamino, trialkylammonium halide, sulphonylamino, hydroxyl, mercapto, alkyl, aralkyl, halogenoalkyl, alkoxy, aralkoxy, halogenoalkoxy, aryl, aryloxy, arylthio, arylsulphinyl, arylsulphonyl, alkylthio, halogenoalkylthio, alkylsulphinyl, halogenoalkylsulphinyl, alkylsulphonyl, halogenoalkylsulphonyl, alkoxycarbonyl, alkylcarbonyl, alkylcarbonyloxy, alkoxyalkyl, alkoxyalkoxy, hydroxyalkoxy, hetarylmethyleneoxy,for combating endoparasites in medicine and veterinary medicine, and new compounds of the formula (I) and their preparation.

    摘要翻译： 本发明涉及通式Ⅰ的取代的1,2,4-恶二唑衍生物（Ⅰ），其中R1代表氢，任选被卤素，烷氧基，羟基，氨基，烷基氨基， 二烷基氨基，环烷基氨基以及环烷基，任选取代的芳基或杂芳基，R 2表示氢和烷基，X表示O，S，SO，SO 2和N-R 3，R 3表示氢，烷基，烷基羰基或卤代烷基羰基R 4表示相同或不同的基团， 氨基，氨基酰基，烷基氨基，二烷基氨基，三烷基卤化铵，磺酰基氨基，羟基，巯基，烷基，芳烷基，卤代烷基，烷氧基，芳烷氧基，卤代烷氧基，芳基，芳氧基，芳硫基，芳基亚磺酰基， 芳基磺酰基，烷硫基，卤代烷硫基，烷基亚磺酰基，卤代烷基亚磺酰基，烷基磺酰基，卤代烷基磺酰基，烷氧基羰基，烷基羰基，烷基羰基氧基，烷氧基烷基，烷氧基 烷氧基，羟基烷氧基，杂芳基亚甲氧基，用于对抗医药和兽药中的内寄生虫，以及式（I）的新化合物及其制备。

    Catalyst block
    94.
    发明授权
    Catalyst block 失效
    催化剂块

    公开(公告)号：US4760047A

    公开(公告)日：1988-07-26

    申请号：US36443

    申请日：1987-04-09

    申请人： Peter Jeschke ,  Hartmut Kainer ,  Blagoje Levkov

    发明人： Peter Jeschke ,  Hartmut Kainer ,  Blagoje Levkov

    IPC分类号： B01D53/86 ,  B01J35/04 ,  B01J32/00

    CPC分类号： B01J35/04 ,  B01D53/8631

    摘要： A quadrangular catalyst block having a plurality of through-going slots separated by intermediate walls, each of the slots having first and second characterizing dimensions, with one of the characterizing dimensions being significantly greater than the other.

    摘要翻译： 四边形催化剂块具有由中间壁分隔开的多个贯穿槽，每个槽具有第一和第二特征尺寸，其中一个特征尺寸明显大于另一个。

    Block-form detergent free from alkali hydroxides for use in dishwashing machines and a process for its production
    95.
    发明授权
    Block-form detergent free from alkali hydroxides for use in dishwashing machines and a process for its production 失效
    不含用于洗碗机的碱性氢氧化物的块状洗涤剂及其制造方法

    公开(公告)号：US4690770A

    公开(公告)日：1987-09-01

    申请号：US868913

    申请日：1986-05-29

    申请人： Peter Jeschke ,  Theodor Altenschoepfer ,  Jochen Jacobs ,  Klaus Schumann

    发明人： Peter Jeschke ,  Theodor Altenschoepfer ,  Jochen Jacobs ,  Klaus Schumann

    IPC分类号： C11D3/395 ,  C11D17/00 ,  C11D7/18

    CPC分类号： C11D17/0052 ,  C11D3/3958

    摘要： A block-form detergent free of alkali metal hydroxides for use in dishwashing machines which contain from 65 to 85% by weight to a mixture of anhydrous sodium metasilicate and anhydrous pentasodium triphosphate in a ratio of from 1:1 to 1:2 and from 0.2 to 4% by weight of uniformly distributed active chlorine donors which are, for example, trichloroisocyanuric acid. The production process comprises heating sodium metasilicate to 45.degree. to 55.degree. C. to obtain a clear melt and then adding other constituents, the pentasodium triphosphate and the active chlorine donor being added last, and pouring the melt into flexible molds in which it is left to solidify into blocks. The detergents are stable for storage with good dissolving power.

    摘要翻译： 不含碱金属氢氧化物的块状洗涤剂，其用于洗碗机，其含有65至85重量％的无水偏硅酸钠和无水三磷酸三钠的混合物，其比例为1:1至1:2且0.2重量份 至4重量％的均匀分布的活性氯供体，例如三氯异氰脲酸。 生产过程包括将偏硅酸钠加热至45℃至55℃以获得澄清的熔体，然后加入其他成分，最后加入三磷酸五钠和活性氯供体，并将熔体倒入其中留下的柔性模具中 凝固成块。 洗涤剂稳定存放，溶解力好。

    Refractory plate for slide closures of metallurgical vessels
    96.
    发明授权
    Refractory plate for slide closures of metallurgical vessels 失效
    用于冶金容器滑动关闭的耐火板

    公开(公告)号：US4179046A

    公开(公告)日：1979-12-18

    申请号：US893690

    申请日：1978-04-05

    申请人： Peter Jeschke ,  Gunter Gelsdorf

    发明人： Peter Jeschke ,  Gunter Gelsdorf

    IPC分类号： B22D37/00 ,  B22D41/32 ,  B32B18/00

    CPC分类号： B22D41/32

    摘要： A refractory plate for use in slide closures for metallurgical vessels includes a basic plate element adapted to face a liquid metal melt. The basic plate element is formed of a moldable refractory concrete material including 70 to 95% by weight of alumina and 5 to 30% by weight of a cement containing approximately 80% by weight alumina. Alternatively, the 70 to 95% by weight of alumina may be replaced by an alumina-containing raw material containing more than 70% by weight of alumina, for example at least one raw material selected from the group consisting of sintered bauxite, synthetic mullite, corundum, and grinding disk fragments. The basic plate element has embedded therein a ceramic oxide insert having a cold bending strength higher than 300 kp/cm.sup.2, a hot bending strength at 1500.degree. C. higher than 40 kp/cm.sup.2, a cold compressive strength higher than 2000 kp/cm.sup.2, and a permeability to gas lower than 1.0 nanoperm. The basic plate element and the insert have extending therethrough a throughflow opening. The width of the insert, in a direction transverse to the direction of movement of the refractory plate, is from 1.3 to 3.5 times the diameter of the throughflow opening.

    摘要翻译： 用于冶金容器的滑动封闭件的耐火板包括适于面对液态金属熔体的基本板元件。 基本板元件由可模制的耐火混凝土材料形成，其包含70至95重量％的氧化铝和5至30重量％的含有约80重量％氧化铝的水泥。 或者，70〜95重量％的氧化铝可以由含有70重量％以上的氧化铝的含氧化铝原料代替，例如选自烧结铝土矿，合成莫来石， 刚玉和磨盘碎片。 碱性板元件内嵌有冷弯曲强度高于300kp / cm 2，高于40kp / cm 2的1500℃的热弯曲强度，高于2000kp / cm 2的冷抗压强度的陶瓷氧化物嵌件， 气体渗透率低于1.0纳米。 基本的板元件和插入件已经穿过其中穿过通孔。 在横向于耐火板的运动方向的方向上，插入件的宽度是通流开口直径的1.3至3.5倍。

    18-membered nitrobenzyl- and aminobenzyl-substituted cyclohexadepsipeptides for controlling endoparasites and a process for their preparation
    98.
    发明授权
    18-membered nitrobenzyl- and aminobenzyl-substituted cyclohexadepsipeptides for controlling endoparasites and a process for their preparation 失效
    用于控制内寄生虫的18元硝基苄基 - 和氨基苄基取代的环己缩肽及其制备方法

    公开(公告)号：US07645738B2

    公开(公告)日：2010-01-12

    申请号：US10582555

    申请日：2004-12-07

    申请人： Peter Jeschke ,  Achim Harder

    发明人： Peter Jeschke ,  Achim Harder

    IPC分类号： A61K38/00

    CPC分类号： C07K11/02 ,  A61K38/00 ,  C07D273/00

    摘要： The invention relates to cyclic depsipeptides, especially 18-membered cyclohexadepsipeptides of general formula (I) and the salts thereof, wherein R1 represents nitrobenzyl or R′R″N-benzyl—wherein R′ and R″ independently represent hydrogen, optionally substituted C1-C4-alkyl, formyl, C1-C4-alkoxy-C1-C4-alkyl, C1-C4-alkoxycarbonyl, or hydroxy-C1-C2-alkyl-sulfonyl-C1-C2-alkyl, or, together with the nitrogen atom to which they are bound, R′ and R″ form an optionally substituted monocyclic or polycyclic, optionally bridged and/or spirocyclic, saturated or unsaturated heterocycle containing between one and three other heteroatoms from the group of nitrogen, oxygen and sulphur, or R′ and R″ together form C3-C5-alkylene monocarbonyl or an optionally substituted diacyl radical of a C4-C6-dicarboxylic acid—and R2, R3 and R4 independently represent C1-C4-alkyl. The invention also relates to the optical isomers and racemates of said cyclic depsipeptides, to a method for the production thereof, and to the use of the same for controlling endoparasites.

    摘要翻译： 本发明涉及环状缩肽，特别是通式（I）的18元环己缩肽和其盐，其中R1表示硝基苄基或R'R''N-苄基，其中R'和R“独立地表示氢，任选取代 C 1 -C 4烷基，甲酰基，C 1 -C 4 - 烷氧基-C 1 -C 4 - 烷基，C 1 -C 4 - 烷氧基羰基或羟基-C 1 -C 2 - 烷基 - 磺酰基-C 1 -C 2烷基，或与氮原子一起 R'和R“形成任选取代的单环或多环，任选桥连和/或螺环，饱和或不饱和的杂环，其含有来自氮，氧和硫的一个和三个其它杂原子，或R '和R'一起形成C 3 -C 5 - 亚烷基单羰基或C 4 -C 6 - 二羧酸的任选取代的二酰基 - ，并且R 2，R 3和R 4独立地表示C 1 -C 4 - 烷基。 本发明还涉及所述环状缩酚酸酯的光学异构体和外消旋体，其制备方法及其用于控制​​内寄生虫的用途。