公开(公告)号：US20080139581A1

公开(公告)日：2008-06-12

申请号：US11885536

申请日：2006-03-02

申请人： Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Jan Klaas Lohmann ,  Bern Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Michael Rack

发明人： Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Jan Klaas Lohmann ,  Bern Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Michael Rack

IPC分类号： A01N43/90 ,  A01P3/00 ,  C07D487/04

CPC分类号： C07D487/04

摘要： 2-Substituted 7-aminoazolopyrimidines of the formula I in which the substituents are as defined below: R1 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkoxyalkyl, benzyloxyalkyl, alkoxyalkenyl or alkoxyalkynyl; R2 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkoxyalkyl and alkylthioalkyl, where the carbon chains in R1 and/or R2 may be substituted according to the description; R3 is halogen, cyano, NRARB, hydroxyl, mercapto, alkyl, haloalkyl, cycloalkyl, alkoxy, alkylthio, cycloalkoxy, cycloalkylthio, carboxyl, formyl, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, phenyl, phenoxy, phenylthio, benzyloxy, benzylthio, alkyl-S(O)m—; A is N and CRx; Rx is hydrogen or one of the groups mentioned under R3; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 2-取代的式I的7-氨基偶氮嘧啶，其中取代基如下：R 1是氢，卤素，氰基，烷基，卤代烷基，烯基，炔基，环烷基，烷氧基，烷氧基烷基，苄氧基烷基 ，烷氧基烯基或烷氧基炔基; R 2是氢，卤素，氰基，烷基，卤代烷基，烯基，炔基，环烷基，烷氧基，烷氧基烷基和烷硫基烷基，其中R 1和/或R ^{2可以根据描述代替; R 3是卤素，氰基，NR B，B，羟基，巯基，烷基，卤代烷基，环烷基，烷氧基，烷硫基，环烷氧基，环烷硫基 ，羧基，甲酰基，烷基羰基，烷氧基羰基，烯氧基羰基，炔氧基羰基，苯基，苯氧基，苯硫基，苄氧基，苄硫基，烷基-S（O） A是N和CR R x是氢或R 3中提到的基团之一; 制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。}

公开(公告)号：US20090280982A1

公开(公告)日：2009-11-12

申请号：US12440120

申请日：2007-09-11

申请人： Michael Puhl ,  Liliana Parra Rapado ,  Michael Rack ,  Jan Klaas Lohmann ,  Wassilios Grammenos ,  Wolfgang von Deyn ,  Jürgen Langewald ,  Ernst Baumann ,  Hassan Oloumi-Sadeghi ,  Douglas D. Anspaugh ,  Deborah L. Culbertson

发明人： Michael Puhl ,  Liliana Parra Rapado ,  Michael Rack ,  Jan Klaas Lohmann ,  Wassilios Grammenos ,  Wolfgang von Deyn ,  Jürgen Langewald ,  Ernst Baumann ,  Hassan Oloumi-Sadeghi ,  Douglas D. Anspaugh ,  Deborah L. Culbertson

IPC分类号： A01N25/26 ,  C07D215/36 ,  A01N43/42 ,  A01P7/00 ,  A01P7/04 ,  A01P7/02 ,  A01P5/00

CPC分类号： C07D215/12 ,  C07D215/18 ,  C07D215/20

摘要： The present invention relates to novel biphenyl-4-sulfonicacid (quinolin-4-ylmethyl)-amide compounds of formula (I) wherein R1 and R2 are halogen, OH, CN, NH2, NO2, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C7-cycloalkyl, C1-C6-alkoxy, C1-C6-haloalkyl, C1-C6-haloalkoxy, C1-C6-alkylthio, C1-C6-alkyl-sulfinyl, C1-C6-alkylsulfonyl, etc.; R3, R4, R5, R6 are halogen, H, CN, NH2, NO2, OH, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-haloalkyl, C1-C6-haloalkoxy, C1-C6-alkylthio, C1-C6-alkylsulfinyl, C1-C6-alkyl-sulfonyl, etc.; m is 0, 1, 2, 3, 4, or 5; and n is 1 or 2; and the N-oxides and salts thereof, and their use for combating arthropod pests and nematodes, and also to compositions comprising such compounds as active component. The present invention also relates to a method for controlling arthropod pests or nematode pests.

摘要翻译： 本发明涉及式（I）的新型联苯-4-磺酸（喹啉-4-基甲基） - 酰胺化合物，其中R 1和R 2是卤素，OH，CN，NH 2，NO 2，C 1 -C 6烷基，C 2 -C 6 - 烯基，C2-C6-炔基，C3-C7-环烷基，C1-C6-烷氧基，C1-C6-卤代烷基，C1-C6-卤代烷氧基，C1-C6-烷硫基，C1-C6烷基亚磺酰基，C1-C6 - 烷基磺酰基等; R3，R4，R5，R6是卤素，H，CN，NH2，NO2，OH，C1-C6-烷基，C1-C6-烷氧基，C1-C6-卤代烷基，C1-C6-卤代烷氧基，C1-C6-烷硫基， C 1 -C 6烷基亚磺酰基，C 1 -C 6烷基磺酰基等; m为0,1,2,3,4或5; n为1或2; 及其N-氧化物及其盐，以及它们用于防治节肢动物害虫和线虫的用途，以及包含这些化合物作为活性成分的组合物。 本发明还涉及一种防治节肢动物害虫或线虫害虫的方法。

公开(公告)号：US09271501B2

公开(公告)日：2016-03-01

申请号：US14364532

申请日：2012-12-06

申请人： Joachim Rheinheimer ,  Violeta Terteryan ,  Stefan Redlich ,  Doris Kremzow ,  Claudia Rosenbaum ,  Sebastian Georgios Rohrer ,  Wassilios Grammenos ,  Christian Pilger ,  Franz Roehl ,  Markus Gewehr ,  Gerd Stammler ,  Jurith Montag ,  Hubert Sauter

发明人： Joachim Rheinheimer ,  Violeta Terteryan ,  Stefan Redlich ,  Doris Kremzow ,  Claudia Rosenbaum ,  Sebastian Georgios Rohrer ,  Wassilios Grammenos ,  Christian Pilger ,  Franz Roehl ,  Markus Gewehr ,  Gerd Stammler ,  Jurith Montag ,  Hubert Sauter

IPC分类号： A01N47/12 ,  A01N37/50 ,  A01N47/28 ,  A01N47/24 ,  A01N43/08 ,  A01N43/76 ,  A01N43/713 ,  A01N43/80 ,  A01N43/90 ,  A01N43/54 ,  A01N43/653 ,  C07D231/22 ,  C07D249/12 ,  A01N43/56 ,  A01N43/78 ,  A01N43/82 ,  A01N43/88

CPC分类号： A01N43/56 ,  A01N37/50 ,  A01N43/08 ,  A01N43/54 ,  A01N43/653 ,  A01N43/713 ,  A01N43/76 ,  A01N43/78 ,  A01N43/80 ,  A01N43/82 ,  A01N43/88 ,  A01N43/90 ,  A01N47/12 ,  A01N47/24 ,  A01N47/28 ,  C07D231/22 ,  C07D249/12

摘要： The present invention relates to the use of strobilurine type compounds of formula I and the N-oxides and the salts thereof for combating phytopathogenic fungi containing a mutation in the mitochondrial cytochrome b gene conferring resistance to Qo inhibitors, and to methods for combating such fungi. The invention also relates to novel compounds, processes for preparing these compounds, to compositions comprising at least one such compound, to plant health applications, and to seeds coated with at least one such compound.

摘要翻译： 本发明涉及式I的顺风草酸型化合物及其N-氧化物及其盐与抗Qo抑制剂抗性的线粒体细胞色素b基因中含有突变的植物病原性真菌的对抗，以及抗真菌的方法。 本发明还涉及新化合物，制备这些化合物的方法，包含至少一种这样的化合物的组合物，用于植物健康应用，以及用至少一种这样的化合物包被的种子。

公开(公告)号：US20080132522A1

公开(公告)日：2008-06-05

申请号：US11631006

申请日：2005-07-12

申请人： Joachim Rheinheimer ,  Frank Schieweck ,  Thomas Grote ,  Carsten Blettner ,  Anja Schwogler ,  Markus Gewehr ,  Wassilios Grammenos ,  Udo Hunger ,  Bernd Muller ,  Peter Schafer ,  Jochen Dietz ,  John-Bryan Speakman ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Joachim Rheinheimer ,  Frank Schieweck ,  Thomas Grote ,  Carsten Blettner ,  Anja Schwogler ,  Markus Gewehr ,  Wassilios Grammenos ,  Udo Hunger ,  Bernd Muller ,  Peter Schafer ,  Jochen Dietz ,  John-Bryan Speakman ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/54 ,  C07D401/04 ,  A01P3/00 ,  A01P13/00 ,  A01P15/00

CPC分类号： C07D239/34 ,  C07D401/04 ,  C07D403/12

摘要： The invention relates to 2-substituted pyrimidines of the formula I in which the index n and the substituents R1 to R4, B and L are as defined in the description and Y is a group —O— or —S—, and to processes for their preparation, pesticidal compositions and methods for controlling harmful fungi and animal pests using the compounds according to the invention.

摘要翻译： 本发明涉及式I的2-取代嘧啶，其中指数n和取代基R 1至R 4，B和L如说明书中所定义，以及 Y是基团-O-或-S-，并且使用本发明的化合物进行制备，杀虫组合物和控制有害真菌和动物害虫的方法。

公开(公告)号：US20070270311A1

公开(公告)日：2007-11-22

申请号：US11661566

申请日：2005-09-02

申请人： Carsten Blettner ,  Jordi Blasco ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Jochen Dietz ,  John-Bryan Speakman ,  Thorsten Jabs ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

发明人： Carsten Blettner ,  Jordi Blasco ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Jochen Dietz ,  John-Bryan Speakman ,  Thorsten Jabs ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  A01P3/00 ,  C07D487/02

CPC分类号： A01N43/90 ,  A01N47/06 ,  A01N47/12 ,  A01N47/16 ,  C07D487/04

摘要： 6-Phenyl-7-aminotriazolopyrimidines of the formula I in which the substituents are as defined below: R1 is hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle, which comprises one to four heteroatoms from the group consisting of O, N and S, R2 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which comprises one to four heteroatoms from the group consisting of O, N and S, R3,R4,R5,R6,R7 are hydrogen or one of the groups mentioned under R2, R4, together with R3 or R6, may also form a five- or six-membered saturated or unsaturated ring which, in addition to carbon atoms, may comprise one to three further heteroatoms from the group consisting of O, N and S as ring members; R2 with R3, R4 with R5, R6 with R7 may in each case together, with formation of spiro groups, also form a C2-C5-alkylene, or alkenylene or alkynylene chain which may be interrupted by one to three heteroatoms from the group consisting of O, N and S; p is zero or 1; L is halogen, alkyl, haloalkyl, alkoxy, cyano, nitro, amino, alkylamino, dialkylamino, alkylcarbonylamino, C(O)—R, S(O)n—R; where n is zero, 1 or 2; R is hydrogen, alkyl, haloalkyl, alkoxy, alkenyloxy, alkynyloxy, amino, alkylamino, dialkylamino; m is 1, 2, 3, 4 or 5; X is halogen, cyano, alkyl, alkoxy, alkenyloxy, alkynyloxy or haloalkoxy; Y is oxygen or sulfur; Z is hydrogen, alkyl, haloalkyl, cycloalkyl, alkylcarbonyl, cycloalkylcarbonyl, alkenyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl, phenyl, naphthyl, a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which comprises one to four heteroatoms from the group consisting of O, N and S; or Z together with R4 or R6 may also form a five- or six-membered saturated or unsaturated ring which, in addition to carbon atoms and Y, may comprise one or two further heteroatoms from the group consisting of O, N and S as ring members the groups R1 to R7, Z and R may be substituted according to the description; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

公开(公告)号：US20080249113A1

公开(公告)日：2008-10-09

申请号：US11659192

申请日：2005-07-28

申请人： Carsten Blettner ,  Jochen Dietz ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Carsten Blettner ,  Jochen Dietz ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04 ,  A01N25/26 ,  A01P3/00

CPC分类号： A01N43/90 ,  A01N43/653 ,  A01N47/14 ,  A01N43/50 ,  A01N57/12 ,  A01N47/04 ,  A01N37/34 ,  A01N43/40 ,  A01N37/50 ,  A01N37/46 ,  A01N43/84 ,  A01N37/38 ,  A01N43/28 ,  A01N47/38 ,  A01N43/54 ,  A01N43/32 ,  A01N59/20 ,  A01N2300/00

摘要： Fungicidal mixtures, comprising as active components 1) a 5-chloro-6-phenyl-7-heterocyclylaminotriazolopyrimidine of the formula I, in which D together with the nitrogen atom forms a pyrrolidine, piperidine or azepine ring, which rings are unsubstituted or substituted by one or two methyl groups or by an ethyl, propyl or butyl group; and L is methyl, fluorine or chlorine; and 2) at least one active compound II selected from the following groups: A) azoles; B) strobilurins; C) acylalanines; D) amine derivatives; E) anilinopyrimidines; F) dicarboximides; G) cinnamides and analogs; H) antibiotics; K) dithiocarbamates; L) heterocyclic compounds according to the description; M) sulfur and copper fungicides; N) nitrophenyl derivatives; O) phenylpyrroles; P) sulfenic acid derivatives; Q) other fungicides according to the description; or R) growth retardants; in a synergistically effective amount, novel triazolopyrimidines, methods for controlling harmful fungi using compounds or mixtures of a compound I with an active compound of groups A) to R) and the use of the compounds I with the active compounds of groups A) to R) for preparing such mixtures, and also compositions comprising these compounds or mixtures.

摘要翻译： 包含作为活性组分的杀真菌混合物1）式I的5-氯-6-苯基-7-杂环基氨基三唑并嘧啶，其中D与氮原子一起形成吡咯烷，哌啶或氮杂环，该环是未取代的或被 一个或两个甲基或乙基，丙基或丁基; L为甲基，氟或氯; 和2）至少一种选自以下组的活性化合物II：A）唑类; B）嗜球果伞素 C）酰基丙氨酸; D）胺衍生物; E）苯胺嘧啶嘧啶; F）二羧酰亚胺; G）肉桂酸酯类似物; H）抗生素; K）二硫代氨基甲酸盐; L）杂环化合物; M）硫和铜杀菌剂; N）硝基苯基衍生物; O）苯基吡咯; P）亚磺酸衍生物; Q）其他杀菌剂根据说明; 或R）生长阻滞剂; 协同有效量的新型三唑并嘧啶，使用化合物或化合物I与A）至R）的活性化合物的混合物来控制有害真菌的方法以及将化合物I与基团A）至R的活性化合物 ），以及包含这些化合物或混合物的组合物。

公开(公告)号：US5430172A

公开(公告)日：1995-07-04

申请号：US228379

申请日：1994-04-15

申请人： Wassilios Grammenos ,  Wolfgang Siegel ,  Klaus Oberdorf ,  Bernd Mueller ,  Hubert Sauter ,  Reinhard Doetzer

发明人： Wassilios Grammenos ,  Wolfgang Siegel ,  Klaus Oberdorf ,  Bernd Mueller ,  Hubert Sauter ,  Reinhard Doetzer

IPC分类号： C07B61/00 ,  C07C45/46 ,  C07C45/48 ,  C07C49/84 ,  C07C65/40 ,  C07C67/313 ,  C07C69/734 ,  C07C69/736 ,  C07C235/34 ,  C07C235/80 ,  C07C251/48 ,  C07C255/54 ,  C07D213/50 ,  C07C41/48 ,  C07C45/61 ,  C07C231/12 ,  C07C249/12

CPC分类号： C07C251/48 ,  C07C235/34 ,  C07C235/80 ,  C07C65/40 ,  C07C69/736 ,  C07D213/50 ,  C07C2101/02 ,  C07C2101/08 ,  C07C2101/14

摘要： A process for preparing 4-alkanoylaryl benzyl ethers of the general formula I ##STR1## where R is hydrogen, halogen, cyano; alkyl, alkoxy;X is CH.sub.2, CH--CH.sub.3, CH--CH.sub.2 --CH.sub.3, CH--OCH.sub.3 or N--OCH.sub.3 ;Y is oxygen, sulfur, direct linkage or nitrogen;m is 0, 1, 2 or 3;R.sup.1 is hydrogen; alkyl, alkenyl, alkynyl or alkoxy;R.sup.2 is cyano, halogen, alkyl, alkoxy or haloalkyl;R.sup.3 is alkyl; haloalkyl; cycloalkyl; or an unsubstituted or substituted mono- to trinuclear aromatic system,comprises reacting an aryl benzyl ether of the general formula II ##STR2## where X, Y, R, R.sup.1, R.sup.2 and m have the abovementioned meanings, with a carbonyl halide or with a carboxylic anhydride or with a carboxylic sulfonic anhydride in the presence of an acid and in the presence or absence of a diluent.

摘要翻译： 制备通式I的4-烷酰基芳基苄基醚的方法，其中R是氢，卤素，氰基; 烷基，烷氧基; X是CH 2，CH-CH 3，CH-CH 2 -CH 3，CH-OCH 3或N-OCH 3; Y是氧，硫，直接连接或氮; m为0,1,2或3; R1是氢; 烷基，烯基，炔基或烷氧基; R2是氰基，卤素，烷基，烷氧基或卤代烷基; R3是烷基; 卤代烷基 环烷基 或未取代或取代的单 - 三核芳族体系，包括使通式II的芳基苄基醚其中X，Y，R，R 1，R 2和m具有上述含义，与羰基卤或与 羧酸酐或与羧酸磺酸酐在酸的存在下和在存在或不存在稀释剂的情况下。

公开(公告)号：US20110201496A1

公开(公告)日：2011-08-18

申请号：US12293432

申请日：2007-03-26

申请人： Joachim Rheinheimer ,  Thomas Grote ,  Bernd Müller ,  Wassilios Grammenos ,  Sarah Ulmschneider ,  Jens Renner ,  Reinhard Stierl

发明人： Joachim Rheinheimer ,  Thomas Grote ,  Bernd Müller ,  Wassilios Grammenos ,  Sarah Ulmschneider ,  Jens Renner ,  Reinhard Stierl

IPC分类号： A01N43/54 ,  C07D401/04 ,  A01C1/06 ,  A61K31/506 ,  A01P3/00 ,  A61P35/00

CPC分类号： A01N43/54

摘要： The present invention relates to the use of 5-hetaryl-4-aminopyrimidines of the formula I and their salts for controlling plant-damaging fungi. The invention also relates to novel 5-hetaryl-4-aminopyrimidines and to crop protection compositions comprising at least one such compound as active component. Het is an optionally substituted 5- or 6-membered aromatic heterocycle which has 1, 2, 3 or 4 heteroatoms selected from the group consisting of nitrogen, oxygen and sulfur as ring members, where the 5- or 6-membered heteroaromatic radical may have 1, 2, 3 or 4 identical or different substituents L, R1, R2 are inter alia hydrogen, C1-C8-alkyl, C3-C8-cycloalkyl, C5-C10-bicycloalkyl, C2-C8-alkenyl, C4-C10-alkadienyl, C3-C6-cycloalkenyl, C2-C8-alkynyl, phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which has one, two, three or four heteroatoms from the group consisting of O, N or S as ring members; or together form a ring; R3 is inter alia hydrogen, OH, halogen, cyano, NR31R32, C1-C8-alkyl, C1-C8-alkoxy, C1-C8-alkylthio, C1-C8-alkylsulfinyl, C1-C8-alkylsulfonyl, C2-C8-alkenyl or C2-C8-alkynyl, and R4 is halogen, cyano, hydroxyl, mercapto, N3, C1-C6-alkyl, C2-C8-alkenyl, C2-C8-alkynyl, C1-C6-haloalkyl, C1-C6-alkoxy, C3-C8-alkenyloxy, C3-C8-alkynyloxy, C1-C6-haloalkoxy, C1-C6-alkylthio, C3-C8-alkenylthio, C3-C8-alkinylthio, C1-C6-haloalkylthio, or is a radical of the formula C(═Z)OR41, C(═Z)NR42R43, C(═Z)NR44—NR42R43, C(═Z)R45, CR46R47—OR48, CR46R47—NR42R43, ON(═CR49R50), O—C(═Z)R45, NR42R43a, NR51(C(═Z)R45), NR51(C(═Z)OR41), NR51(C(═Z)—NR42R43), NR52a(N═CR49R50), NR52NR42R43, NR52OR41 or C(═N—X—R45)SR41.

公开(公告)号：US07695728B2

公开(公告)日：2010-04-13

申请号：US11630569

申请日：2005-06-18

申请人： Joachim Rheinheimer ,  Frank Schieweck ,  Thomas Grote ,  Carsten Blettner ,  Anja Schwögler ,  Markus Gewehr ,  Wassilios Grammenos ,  Udo Hünger ,  Bernd Müller ,  Peter Schäfer ,  John-Bryan Speakman ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

发明人： Joachim Rheinheimer ,  Frank Schieweck ,  Thomas Grote ,  Carsten Blettner ,  Anja Schwögler ,  Markus Gewehr ,  Wassilios Grammenos ,  Udo Hünger ,  Bernd Müller ,  Peter Schäfer ,  John-Bryan Speakman ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

IPC分类号： C07D401/04 ,  C07D213/61 ,  C07D417/04 ,  C07D213/70 ,  C07D213/86 ,  C07D213/78 ,  A01N43/40

CPC分类号： C07D401/04 ,  A01N43/40 ,  A01N43/54 ,  A01N43/56 ,  A01N43/653 ,  A01N43/78 ,  C07D213/61 ,  C07D213/70 ,  C07D213/74 ,  C07D213/78 ,  C07D213/84 ,  C07D213/86 ,  C07D417/04

摘要： The invention relates to 2-substituted pyridines of the formula I in which the index n and the substituents R1 to R4 and L are as defined in the description and in each case one of the two ring members X1, X2 is N, the other is C—H or C-halogen; Y is a group —CH—R1—, —N—R1—, —O— or —S— and is five- or six-membered hetaryl comprising 1 to 3 heteroatoms selected from the group consisting of O, N and S or is phenyl, and to processes for their preparation, intermediates for their preparation, pesticidal compositions and methods for controlling harmful fungi and animal pests using the compounds according to the invention.

摘要翻译： 本发明涉及式I中的2-取代吡啶，其中指数n和取代基R 1至R 4和L如说明书中所定义，并且在每种情况下，两个环成员X1，X2中的一个为N，另一个为 C-H或C-卤素; Y是基团-CH-R 1，-N-R 1，-O-或-S-，是包含1至3个选自O，N和S的杂原子的五元或六元杂芳基，或者是 苯基，及其制备方法，其制备中间体，杀虫组合物和使用本发明化合物控制有害真菌和动物害虫的方法。

公开(公告)号：US20090177005A1

公开(公告)日：2009-07-09

申请号：US12344631

申请日：2008-12-29

申请人： Guido MAYER ,  Oliver Cullmann ,  Bernd Wolf ,  Michael Keil ,  Wassilios Grammenos

发明人： Guido MAYER ,  Oliver Cullmann ,  Bernd Wolf ,  Michael Keil ,  Wassilios Grammenos

IPC分类号： C07C249/02

CPC分类号： C07C249/12 ,  C07C251/48

摘要： A process for preparing 2-(chloromethyl)phenylacetic acid derivatives of the formula I, where X is C1-C4-alkoxy or methylamino, by ether cleavage of compounds of the formula II, where R is C1-C4-alkyl, C1-C4-alkoxy, C1-C2-haloalkyl, C1-C4-alkylcarbonyl, C1-C4-alkylcarbonyloxy, halogen, nitro or cyano; n is 2 to 5; and X is as defined above comprises carrying out the reaction in the presence of hydrogen chloride and an inert solvent, and adding a catalyst to the reaction mixture selected from the group consisting of iron, indium and halides, oxides and triflates, thereof.

摘要翻译： 通过醚式裂解式II化合物制备式I的2-（氯甲基）苯乙酸衍生物的方法，其中X为C 1 -C 4烷氧基或甲氨基，其中R为C 1 -C 4 - 烷基，C 1 -C 4 - 烷氧基，C 1 -C 2 - 卤代烷基，C 1 -C 4 - 烷基羰基，C 1 -C 4 - 烷基羰基氧基，卤素，硝基或氰基; n为2〜5; 并且X如上所定义，包括在氯化氢和惰性溶剂的存在下进行反应，并向选自铁，铟和卤化物，氧化物和三氟甲磺酸酯的反应混合物中加入催化剂。