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公开(公告)号：US20200085056A1
公开(公告)日：2020-03-19
申请号：US16473184
申请日：2017-12-26
发明人： Ikki Yonemura , Yusuke Sano , Naoto Shimizu , Akihiro Miyasaka , Akiyuki Suwa , Shunpei Fujie , Ryosuke Tanaka
IPC分类号： A01N43/90 , C07D471/04 , C07D519/00
摘要： In crop production in the fields of agriculture, horticulture and the like, the damage caused by insect pests etc. is still immense, and insect pests resistant to existing insecticides have emerged. Under such circumstances, the development of novel agricultural and horticultural insecticides is desired. The present invention provides an agricultural and horticultural insecticide comprising a 4H-pyrrolopyridine compound represented by the general formula (1): {wherein R1 represents a halogen atom, R2 and R3 each represent a haloalkyl group, Q represents Q-A, Q-B or Q-C, X represents a nitrogen atom, R4 and R7 each represent a hydrogen atom, R2 and R3 each represent a halogen atom, a haloalkyl group or a substituted phenyl group, and m represents 2} or a salt thereof as an active ingredient; and a method for using the insecticide.
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公开(公告)号：US20200085054A1
公开(公告)日：2020-03-19
申请号：US16473166
申请日：2017-12-26
发明人： Ikki Yonemura , Yusuke Sano , Akiyuki Suwa , Shunpei Fujie , Ryosuke Tanaka
IPC分类号： A01N43/76 , C07D413/04 , C07D413/14
摘要： In crop production in the fields of agriculture, horticulture and the like, the damage caused by insect pests etc. is still immense, and insect pests resistant to existing insecticides have emerged. The present invention has been made in view of such circumstances, and an object of the present invention is to develop and provide a novel agricultural and horticultural insecticide. The present invention provides an oxime group-containing condensed heterocyclic compound represented by the general formula (1): {wherein R1 represents an alkoxy group, R2 represents a haloalkyl group, R3 represents a haloalkylthio group, A represents an oxygen atom, A1 represents a CH group, m represents 2, and n represents 1}, or a salt thereof; an agricultural and horticultural insecticide comprising the compound or the salt as an active ingredient; and a method for using the insecticide.
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113.发明申请公开(公告)号：US20190174760A1
公开(公告)日：2019-06-13
申请号：US16311139
申请日：2017-06-30
发明人： Yutaka Abe , Chiaki Yamauchi , Yuhji Sakurai , Hirokazu Fujihara , Soichiro Matsuo , Ikki Yonemura , Akiyuki Suwa , Shunpei Fujie , Ryosuke Tanaka
IPC分类号： A01N43/90 , C07D487/04 , C07D471/04 , C07D413/04
摘要： In crop production in the fields of agriculture, horticulture and the like, the damage caused by insect pests etc. is still immense, and insect pests resistant to existing insecticides have emerged. Under such circumstances, the development of novel agricultural and horticultural insecticides is desired. The present invention provides a condensed heterocyclic compound represented by the general formula (1): {wherein R1 represents a (C1-C6) alkyl group, R2 represents a halo (C1-C6) alkyl group, G1, G2, G3, G4, G5, G6, G7 and G8 each represent CH or N, and m represents an integer of 0 to 2} or a salt thereof; an agricultural and horticultural insecticide comprising the compound or the salt as an active ingredient; and a method for using the insecticide.
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公开(公告)号：US20180002347A1
公开(公告)日：2018-01-04
申请号：US15545078
申请日：2016-01-29
发明人： Ikki Yonemura , Akiyuki Suwa , Soichiro Matsuo , Takanori Aoki
IPC分类号： C07D513/04 , C07D471/04 , C07D417/04 , C07D401/04 , A01N43/52 , A01N43/90 , A01N43/78 , A01N43/76 , C07D498/04 , C07D413/04
CPC分类号： C07D513/04 , A01N43/52 , A01N43/54 , A01N43/76 , A01N43/78 , A01N43/90 , C07D401/04 , C07D413/04 , C07D417/04 , C07D471/04 , C07D498/04
摘要： An object of the present invention is to provide and develop novel agricultural and horticultural insecticides in view of the still immense damage caused by insect pests etc. and the emergence of insect pests resistant to existing insecticides in crop production in the fields of agriculture, horticulture and the like.Provided are a condensed heterocyclic compound represented by the general formula (1): {wherein R1 represents an ethyl group, R2 represents a cycloalkyl group, R3 represents a haloalkyl group, A, A2 and A3 each represent a nitrogen atom or a CH group, A1 represents N-Me, m represents 0 or 2, and n represents 1} or a salt thereof; an agricultural and horticultural insecticide comprising the compound or a salt thereof as an active ingredient; and a method for using the insecticide.
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公开(公告)号：US20170037029A1
公开(公告)日：2017-02-09
申请号：US15298910
申请日：2016-10-20
发明人： Kiyoshi Kita , Akiyuki Suwa , Masatsugu Oda , Koji Tanaka
IPC分类号： C07D401/12 , C07D231/14 , C07D239/28 , C07D333/38 , C07D277/56 , C07D307/68 , C07D327/06 , C07D213/82 , C07D241/24
CPC分类号： C07D401/12 , A61K31/381 , A61K31/39 , A61K31/415 , A61K31/426 , A61K31/44 , A61K31/4439 , A61K31/444 , A61K31/4965 , A61K31/497 , A61K31/505 , C07D213/82 , C07D231/14 , C07D239/28 , C07D241/24 , C07D277/56 , C07D307/68 , C07D327/06 , C07D333/38 , C07D401/00
摘要： An object of the present invention is to provide a novel endoparasite control agent as a parasiticide, an antiprotozoal or the like. Provided is an endoparasite control agent comprising a carboxamide derivative represented by the general formula (I): (wherein Het represents a 5- or 6-membered heterocyclic group), or a salt thereof as an active ingredient.
摘要翻译： 本发明的目的是提供一种新型的寄生虫寄生虫寄生虫寄生虫控制剂，抗原虫等。 本发明提供包含由通式（I）表示的羧酰胺衍生物（其中Het表示5-或6-元杂环基）或其盐作为活性成分的内寄生虫控制剂。
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公开(公告)号：US09562034B2
公开(公告)日：2017-02-07
申请号：US14424763
申请日：2013-08-29
发明人： Kiyoshi Kita , Akiyuki Suwa , Masatsugu Oda , Koji Tanaka
IPC分类号： C07D307/68 , C07D241/24 , C07D401/12 , C07D277/56 , C07D327/06 , C07D239/28 , C07D231/14 , C07D213/82 , C07D333/38 , A61K31/381 , A61K31/39 , A61K31/415 , A61K31/426 , A61K31/44 , A61K31/4965 , A61K31/505 , A61K31/4439 , A61K31/444 , A61K31/497 , C07D401/00
CPC分类号： C07D401/12 , A61K31/381 , A61K31/39 , A61K31/415 , A61K31/426 , A61K31/44 , A61K31/4439 , A61K31/444 , A61K31/4965 , A61K31/497 , A61K31/505 , C07D213/82 , C07D231/14 , C07D239/28 , C07D241/24 , C07D277/56 , C07D307/68 , C07D327/06 , C07D333/38 , C07D401/00
摘要： An object of the present invention is to provide a novel endoparasite control agent as a parasiticide, an antiprotozoal or the like. Provided is an endoparasite control agent comprising a carboxamide derivative represented by the general formula (I): (wherein Het represents a 5- or 6-membered heterocyclic group), or a salt thereof as an active ingredient.
摘要翻译： 本发明的目的是提供一种新型的寄生虫寄生虫寄生虫寄生虫控制剂，抗原虫等。 本发明提供含有通式（I）表示的羧酰胺衍生物（其中，Het表示5元或6元杂环基）或其盐作为有效成分的内寄生虫控制剂。
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公开(公告)号：US20160361299A1
公开(公告)日：2016-12-15
申请号：US15247376
申请日：2016-08-25
IPC分类号： A61K31/4178 , A61K9/00 , A61K9/08 , A61K47/10 , A61K47/38
CPC分类号： A61K31/4178 , A61K9/0014 , A61K9/08 , A61K31/385 , A61K31/4164 , A61K47/10 , A61K47/38
摘要： Disclosed is an antifungal agent for external use, which is characterized by containing a compound represented by the general formula (1), 50 to 95 mass % of an alcohol such as ethanol, 0.1 to 35 mass % of water or the like, and 0.01 to 5 mass % of a cellulose thickening agent. X is a halogen or H.
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118.发明申请PHARMACEUTICAL COMPOSITION FOR TREATMENT OF PNEUMONIA ASSOCIATED WITH FUSARIUM FUNGUS 审中-公开用于治疗与FUSARIUM FUNGUS相关的PNEUMONIA的药物组合物公开(公告)号：US20160279101A1
公开(公告)日：2016-09-29
申请号：US15037488
申请日：2014-11-14
发明人： Tsuyoshi Shimamura , Hiroyasu Koga , Yasuko Nanjoh
IPC分类号： A61K31/4178 , C12Q1/68
CPC分类号： A61K31/4178 , C12Q1/6895 , C12Q2600/112
摘要： The present invention aims to provide a pharmaceutical composition for pneumonia associated at least with a Fusarium fungus as a causative microorganism. Provided is a pharmaceutical composition for pneumonia associated at least with a Fusarium fungus as a causative microorganism, which pharmaceutical composition includes as an effective component a compound represented by the General Formula (1) below: (wherein R represents a halogen atom or hydrogen atom, and X represents a halogen atom).
摘要翻译： （其中R表示卤素原子或氢原子，X表示卤素原子）。
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119.发明授权Crystalline form having specific crystal habit and pharmaceutical composition containing this crystalline form as active ingredient 有权具有特定晶体习性的结晶形式和含有该结晶形式作为活性成分的药物组合物公开(公告)号：US09453006B2
公开(公告)日：2016-09-27
申请号：US14388218
申请日：2013-06-24
发明人： Takaaki Masuda , Yoshiyuki Miyata , Hideo Kaneda
IPC分类号： C07D409/06
CPC分类号： C07D409/06
摘要： Means for improving the solubility of luliconazole is provided. A crystal of luliconazole represented by the following formula is provided, wherein the crystal has such a crystal habit that (011) plane is a specific crystal growth plane. The crystal is characterized in that I(011) with respect to a sum total of I(001), I(100), I(10-1), I(011), I(110), I(11-1), I(10-2), I(11-2), I(020), I(021), I(20-2), I(121), I(013), I(11-3), and I(221) is not less than 25%, provided that integrated intensities of diffraction peaks, which correspond to the (001), (100), (10-1), (011), (110), (11-1), (10-2), (11-2), (020), (021), (20-2), (121), (013), (11-3), and (221) planes, are designated as I(001), I(100), I(10-1), I(011), I(110), I(11-1), I(10-2), I(11-2), I(020), I(021), I(20-2), I(121), I(013), I(11-3), and I(221) respectively in relation to the diffraction peaks detected in a range of 2θ=5 to 35° in a powder X-ray diffractometry using CuKα radiation.
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120.发明申请PHARMACEUTICAL COMPOSITION FOR DISEASES CAUSED BY PATHOGENIC MICROORGANISMS SUCH AS ASPERGILLUS 审中-公开致病微生物如ASPERGILLUS引起的疾病药物组合物公开(公告)号：US20150366845A1
公开(公告)日：2015-12-24
申请号：US14760917
申请日：2013-12-27
IPC分类号： A61K31/4178
CPC分类号： A61K31/4178 , A61K9/2866
摘要： An object is to provide means for precisely treating pneumonia caused by intracellular parasite, protozoa, and/or fungus. A pharmaceutical composition for pneumonia, comprising a compound represented by the following general formula (1) as an active ingredient: (In the formula, R represents a halogen atom or a hydrogen atom, and X represents a halogen atom.)
摘要翻译： 目的是提供精确治疗由细胞内寄生虫，原生动物和/或真菌引起的肺炎的手段。 一种肺炎药物组合物，其特征在于，含有下述通式（1）表示的化合物作为有效成分：（式中，R表示卤原子或氢原子，X表示卤素原子）
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