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    Substituted benzoylphenylureas compounds useful as pesticides
    13.
    发明授权
    Substituted benzoylphenylureas compounds useful as pesticides 失效
    用作农药的取代苯甲酰基苯基化合物

    公开(公告)号：US4847258A

    公开(公告)日：1989-07-11

    申请号：US86339

    申请日：1987-08-17

    Applicant: Elmar Sturm ,  Robert W. Lang ,  Odd Kristiansen

    Inventor： Elmar Sturm ,  Robert W. Lang ,  Odd Kristiansen

    IPC: A01N47/34 ,  C07D239/34

    CPC classification number: C07D239/34 ,  A01N47/34

    Abstract: The invention relates to novel N-benzoyl-N,-4-(5-phenylpyrimid-2-yloxy)phenylureas of formula ##STR1## wherein X.sub.1 is hydrogen, halogen, C.sub.1 -C.sub.3 alkoxy or C.sub.1 -C.sub.3 alkylthio,X.sub.2 is halogen, methyl, C.sub.1 -C.sub.3 alkoxy or C.sub.1 -C.sub.3 alkylthio,Y.sub.1, Y.sub.2, Y.sub.3 and Y.sub.4 are each independently hydrogen, halogen, methyl, trifluoromethyl or methoxy,Z is methyl, halomethyl containing 1 to 3 halogen atoms or pentafluoroethyl; andR.sub.1, R.sub.2 and R.sub.3 are each independently hydrogen, halogen, C.sub.1 -C.sub.3 alkyl, trifluoromethyl or C.sub.1 -C.sub.3 alkoxy,to the preparation thereof and to intermediates for the synthesis of these compounds, as well as to compositions containing them for use in pest control, especially for controlling representatives of the order Acarina that attack plants and animals and for controlling insects. The novel compounds exhibit especially pronounced activity against plant-destructive mites.

    Abstract translation: 本发明涉及式（I）其中X 1为氢，卤素，C 1 -C 3烷氧基或C 1 -C 3烷硫基的新的N-苯甲酰基-N，4-（5-苯基嘧啶-2-基氧）苯基脲，X2 是卤素，甲基，C 1 -C 3烷氧基或C 1 -C 3烷硫基，Y 1，Y 2，Y 3和Y 4各自独立地为氢，卤素，甲基，三氟甲基或甲氧基，Z为甲基，含1至3个卤素原子的卤代甲基或五氟乙基; R 1，R 2和R 3各自独立地为氢，卤素，C 1 -C 3烷基，三氟甲基或C 1 -C 3烷氧基，并且用于合成这些化合物的中间体，以及含有它们用于病虫害防治的组合物， 特别是控制攻击植物和动物并控制昆虫的蜱虫的代表。 新型化合物对植物破坏性螨具有特别显着的活性。

    Substituted 2-azabicycloalkanes as selective herbicides
    17.
    发明授权
    Substituted 2-azabicycloalkanes as selective herbicides 失效
    取代的2-氮杂双环烷烃作为选择性除草剂

    公开(公告)号：US3936458A

    公开(公告)日：1976-02-03

    申请号：US417303

    申请日：1973-11-19

    Applicant: Elmar Sturm ,  Christian Vogel

    Inventor： Elmar Sturm ,  Christian Vogel

    IPC: C07D215/08

    CPC classification number: C07D215/08

    Abstract: Compounds of the formula I ##SPC1##wherein R represents alkyl having from 1 to 4 carbon atoms and one of the symbols R.sub.1 and R.sub.2 is methyl and the other is hydrogen possess favorable herbicidal properties for practical purposes when used in crops for controlling their infestation by undesired plant growth.

    Abstract translation: 其中R代表具有1至4个碳原子的烷基和R1和R2之一的烷基是甲基，而另一个是氢的式I化合物，当用于作物控制其不希望的植物生长侵袭时，具有有效的除草性能 。

    5-esters of milbemycins for controlling parasitic pests
    18.
    发明授权
    5-esters of milbemycins for controlling parasitic pests 失效
    用于控制寄生虫害的米尔倍霉素的5-酯

    公开(公告)号：US4778809A

    公开(公告)日：1988-10-18

    申请号：US895979

    申请日：1986-08-13

    Applicant: Peter Maienfisch ,  Elmar Sturm

    Inventor： Peter Maienfisch ,  Elmar Sturm

    IPC: C07D493/22 ,  A01N43/90 ,  A23K20/195 ,  A61K31/365 ,  A61P33/10 ,  C07H19/01

    CPC classification number: C07H19/01 ,  A01N43/90 ,  A23K20/195

    Abstract: The invention relates to ecto- and endoparasitic milbemycins of formula I ##STR1## wherein R is methyl, ethyl, isopropyl or sec-butyl;R.sub.1 is hydrogen, fluorine or C.sub.1 -C.sub.4 alkyl;R.sub.2 is one of the groups ##STR2## in which formulaeis a value from 2 to 6;X is oxygen or sulfur;R.sub.3 is halogen; andR.sub.4 is hydrogen, C.sub.1 -C.sub.12 alkoxy, C.sub.3 -C.sub.7 cycloalkoxy or C.sub.2 -C.sub.6 alkenyloxy; or C.sub.1 -C.sub.18 alkyl which is unsubstituted or substituted by halogen, C.sub.1 -C.sub.4 alkoxy, hydroxy and/or COOG, G being hydrogen, an alkali metal cation or an alkaline earth metal cation; or R.sub.4 is C.sub.3 -C.sub.7 cycloalkyl which is unsubstituted or substituted by halogen and/or C.sub.1 -C.sub.4 alkyl;C.sub.2 -C.sub.18 alkenyl which is unsubstituted or substituted by halogen;C.sub.2 -C.sub.18 alkynyl which is unsubstituted or substituted by halogen;phenyl which is unsubstituted or substituted by halogen, C.sub.1 -C.sub.4 alkyl C.sub.1 -C.sub.4 alkoxy, nitro, cyano and/or C.sub.1 -C.sub.4 haloalkyl; or a 5- or 6-membered unsaturated or saturated heterocyclic ring system which contains one to three hetero atoms selected from the series consisting of nitrogen, oxygen and sulfur and which is unsubstituted or substituted by oxo and/or by one to three substituents selected from halogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy and/or C.sub.1 -C.sub.4 haloalkyl;to the use thereof in agriculture and to the preparation thereof by esterifying the 5-OH-milbemycins on which they are based.

    Abstract translation: 本发明涉及式I的异位和内寄生米尔倍霉素（I），其中R是甲基，乙基，异丙基或仲丁基; R1是氢，氟或C1-C4烷基; R2是其中公式为2至6的值之一之一; X是氧或硫; R3是卤素; 和R 4是氢，C 1 -C 12烷氧基，C 3 -C 7环烷氧基或C 2 -C 6烯氧基; 或未取代或被卤素取代的C 1 -C 18烷基，C 1 -C 4烷氧基，羟基和/或COOG，G为氢，碱金属阳离子或碱土金属阳离子; 或R 4为未被取代或被卤素和/或C 1 -C 4烷基取代的C 3 -C 7环烷基; 未被取代或被卤素取代的C 2 -C 18烯基; 未被取代或被卤素取代的C 2 -C 18炔基; 未被取代或被卤素取代的苯基，C 1 -C 4烷基C 1 -C 4烷氧基，硝基，氰基和/或C 1 -C 4卤代烷基; 或含有一至三个选自氮，氧和硫的杂原子的5-或6-元不饱和或饱和杂环体系，其未被取代或被氧代和/或被1-3个选自以下的取代基取代： 卤素，C 1 -C 4烷基，C 1 -C 4烷氧基和/或C 1 -C 4卤代烷基; 在农业中的用途以及通过酯化其所基于的5-OH- milbemycins来制备它们。

    5-azolylacetoxymilbemycins as ecto- and endoparasites
    19.
    发明授权
    5-azolylacetoxymilbemycins as ecto- and endoparasites 失效
    5-azolylaceoxymilbemycins as ecto-和endoparasites

    公开(公告)号：US4696922A

    公开(公告)日：1987-09-29

    申请号：US799373

    申请日：1985-11-18

    Applicant: Elmar Sturm ,  Peter Maienfisch

    Inventor： Elmar Sturm ,  Peter Maienfisch

    IPC: A01N43/90 ,  A61K31/365 ,  A61P33/10 ,  C07D493/22 ,  C07H19/01 ,  C07D249/08

    CPC classification number: C07H19/01

    Abstract: The present invention relates to milbemycin derivatives of the formula I ##STR1## wherein X is hydrogen or .beta.-halogen, R is methyl, ethyl, isopropyl or sec-butyl and Az is a 5 membered heterocyclic aromatic ring which contains 2-4 nitrogen atoms and is attached in the 1-position and which is unsubstituted or substituted by one or two C.sub.1 -C.sub.6 alkyl groups. These compounds, and the acid addition salts and metal complexes thereof, are effective pesticides for controlling endo-and ectoparasites, especially for controlling neamatodes which are parasites of animals. The may be obtained by appropriate esterification in 5-position of milbemycin derivatives. The selective .beta.-halogenation of 14,15-epoxymilbemycin derivatives can be effected via the intermediate .DELTA..sup.13,14 -15-hydroxymilbemycins with appropriate halogenating agents.

    Abstract translation: 本发明涉及式I（I）的密尔伯霉素衍生物，其中X是氢或β-卤素，R是甲基，乙基，异丙基或仲丁基，而Az是含有2- 4个氮原子并且连接在1-位且未被取代或被一个或两个C 1 -C 6烷基取代。 这些化合物及其酸加成盐和金属络合物是用于控制内寄生虫和外寄生虫的有效农药，特别是用于控制作为动物寄生虫的寄生虫。 可以通过在密尔伯霉素衍生物的5-位合适的酯化获得。 14,15-环氧米尔伯霉素衍生物的选择性β-卤代化可以通过中间体DELTA 13,14-15-羟吗啉霉素与适当的卤化剂进行。

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