Penta-2,4-dienamides and use as pesticides
    14.
    发明授权
    Penta-2,4-dienamides and use as pesticides 失效
    五 - 2,4-二烯酰胺,用作农药

    公开(公告)号:US5459149A

    公开(公告)日:1995-10-17

    申请号:US309430

    申请日:1994-09-20

    摘要: The present Application discloses pesticidally active compounds of formula (I):Q(CH.sub.2).sub.a (O).sub.b Q.sup.1 CR.sup.2 =CR.sup.3 CR.sup.4 =CR.sup.5 CXNR.sup.1 R.sup.xor a salt or propesticide thereof, wherein Q is an optionally substituted aromatic monocyclic or fused bicyclic ring system in which at least one ring is aromatic, or Q is a dihalovinyl group or a group R.sup.6 --C=C--where R.sup.6 is C.sub.1-4 alkyl, tri C.sub.1-4 alkylsilyl, halo or hydrogen; Q.sup.1 is a 1,2-cyclopropyl ring optionally substituted by one or more groups selected from C.sub.1-3 alkyl, halo, C.sub.1-3 haloalkyl, C.sub.2-3 alkynyl, or cyano; or Q.sup.1 is (CH.sub.2).sub.7 ; a=0 or 1; b=0 or 1; R.sup.2, R.sup.3, R.sup.4 and R.sup.5 are the same or different with at least one being hydrogen and the others being independently selected from hydrogen, halo, C.sub.1-4 alkyl or C.sub.1-4 haloalkyl; X is oxygen or sulphur;R.sup.1 is phenyl optionally substituted by 1-5 substituents chosen from: a) C.sub.1-4 alkyl, C.sub.1-4 alkoxy, phenoxy and methylenedioxy, each optionally substituted by 1 to 5 halo; b) halo, cyano, nitro, formyl, C.sub.1-5 acyl; c) C.sub.2-3 alkynyl, C.sub.2-3 alkenyl, each optionally substituted by 1 to 5 halo; d) a group S(O).sub.n R.sup.7 wherein n=0, 1, 2 and R.sup.7 is C.sub.1-4 alkyl, halo or NR.sup.8 R.sup.9 wherein R.sup.8 and R.sup.9 are independently selected from hydrogen, C.sub.1-4 alkyl and C.sub.1-4 acyl; and a group e) NR.sup.8 R.sup.9 where R.sup.8 and R.sup.9 are as defined above; R.sup.X is hydrogen or an optionally substituted C.sub.1-8 alkyl or benzyl group, their preparation, pesticidal compositions containing them and their use against pests.

    摘要翻译: 本申请公开了式(I)的杀虫活性化合物:Q(CH2)a(O)bQ1 CR2 = CR3 CR4 = CR5 CXNR1Rx或其盐或农药,其中Q是任选取代的芳族单环或稠合双环体系 其中至少一个环是芳族的,或Q是二卤代乙烯基或基团R6-C = C-,其中R6是C1-4烷基,三C1-4烷基甲硅烷基,卤素或氢; Q1是任选被一个或多个选自C 1-3烷基,卤素,C 1-3卤代烷基,C 2-3炔基或氰基的基团取代的1,2-环丙基环; 或Q 1为(CH 2)7; a = 0或1; b = 0或1; R 2,R 3,R 4和R 5相同或不同,至少一个为氢,其余独立地选自氢,卤素,C 1-4烷基或C 1-4卤代烷基; X是氧或硫; R1是任选被1-5个选自下列的取代基取代的苯基:a)C 1-4烷基,C 1-4烷氧基,苯氧基和亚甲二氧基,各自任选被1至5个卤素取代; b)卤素,氰基,硝基,甲酰基,C 1-5酰基; c)C2-3炔基,C2-3烯基,各自任选被1至5个卤素取代; d)基团S(O)n R 7,其中n = 0,1,2且R 7是C 1-4烷基,卤素或NR 8 R 9,其中R 8和R 9独立地选自氢,C 1-4烷基和C 1-4酰基; 和基团e)NR 8 R 9,其中R 8和R 9如上所定义; RX是氢或任选取代的C 1-8烷基或苄基,它们的制备方法,含有它们的杀虫组合物及其对害虫的用途。

    Manufacture of printed circuit boards
    15.
    发明授权
    Manufacture of printed circuit boards 失效
    印刷电路板的制造

    公开(公告)号:US4403410A

    公开(公告)日:1983-09-13

    申请号:US225092

    申请日:1981-01-14

    申请人: John E. Robinson

    发明人: John E. Robinson

    摘要: A process for the manufacture of a printed circuit board is disclosed in which, during the process, conductive tracks 6 are tested for defects 8 relating to their conductivity and any detected defect 8 is repaired by securing a conductive bridge-piece 9 across the defect 8 by a reflow soldering operation. The repair is encapsulated with a protective layer 16 and the manufacturing process, which includes the further application of heat to the circuit board, is continued.

    摘要翻译: 公开了一种用于制造印刷电路板的方法,其中在该过程期间,对导电轨道6进行与其导电性有关的缺陷8的测试,并且通过将导电桥接件9固定在缺陷8上来修复任何检测到的缺陷8 通过回流焊接操作。 修复被保护层16封装,并且继续包括进一步向电路板施加热量的制造过程。

    Imidazo[1,2-a]Pyridine Compounds As Receptor Tyrosine Kinase Inhibitors
    16.
    发明申请
    Imidazo[1,2-a]Pyridine Compounds As Receptor Tyrosine Kinase Inhibitors 审中-公开
    咪唑并[1,2-a]吡啶化合物作为受体酪氨酸激酶抑制剂

    公开(公告)号:US20110184013A1

    公开(公告)日:2011-07-28

    申请号:US13122095

    申请日:2009-09-30

    CPC分类号: C07D487/04 C07D471/04

    摘要: Compounds of Formula I and II: I II having the chemical names cis-6-fluoro-8-(3-fluoropiperidin-4-yloxy)-2-(7-(2-methoxyethoxy)imidazo[1,2-a]pyridin-3-yl)quinoline and 6-fluoro-8-(trans-3-fluoropiperidin-4-yloxy)-2-(7-(2-methoxyethoxy)imidazo[1,2-a]pyridin-3-yl)quinoline, respectively, and enantiomers and pharmaceutically acceptable salts thereof, are receptor tyrosine inhibitors useful in the treatment of diseases mediated by class 3 and class 5 receptor tyrosine kinases. The compounds of this invention have also been found to be inhibitors of Pim-1.

    摘要翻译: 具有化学名称的顺式-6-氟-8-(3-氟哌啶-4-基氧基)-2-(7-(2-甲氧基乙氧基)咪唑并[1,2-a]吡啶的式I和II化合物: 吡啶-3-基)喹啉和6-氟-8-(反式-3-氟哌啶-4-基氧基)-2-(7-(2-甲氧基乙氧基)咪唑并[1,2-a]吡啶-3-基)喹啉 和对映异构体及其药学上可接受的盐是可用于治疗由3类和5类受体酪氨酸激酶介导的疾病的受体酪氨酸抑制剂。 本发明化合物也被发现是Pim-1的抑制剂。

    Cue tip chalk retention system
    20.
    发明授权
    Cue tip chalk retention system 失效
    提示笔尖保留系统

    公开(公告)号:US4867446A

    公开(公告)日:1989-09-19

    申请号:US272451

    申请日:1988-11-17

    申请人: John E. Robinson

    发明人: John E. Robinson

    IPC分类号: A63D15/14 A63D15/16

    CPC分类号: A63D15/16 A63D15/14

    摘要: A cue tip chalk retention system wherein openings are formed on cue tip surfaces and chalk is rubbed into the openings. The openings are formed with a penetrating device comprising a housing with a cavity containing multiple outwardly extending pin members. The pin members have a base portion secured to the cavity lower region and a free end portion located in the cavity upper region. The free end portion includes an exposed pointed end which is used to cleanly penetrate the cue tip surfaces and form the desired chalk retention openings.

    摘要翻译: 提示笔尖保留系统,其中在提示头表面上形成开口,并将白垩摩擦到开口中。 开口形成有穿透装置,该穿透装置包括具有包含多个向外延伸的销构件的空腔的壳体。 销构件具有固定到空腔下部区域的基部和位于空腔上部区域中的自由端部。 自由端部包括暴露的尖端,其用于干净地穿透提示尖端表面并形成所需的粉笔保持开口。