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    5-acylaminopyrimidines
    11.
    发明授权
    5-acylaminopyrimidines 失效
    5-酰氨基嘧啶

    公开(公告)号：US4718934A

    公开(公告)日：1988-01-12

    申请号：US853308

    申请日：1986-04-17

    申请人： Helmut Zondler ,  Hans Tobler ,  Urs Muller

    发明人： Helmut Zondler ,  Hans Tobler ,  Urs Muller

    IPC分类号： A01N43/54 ,  C07D239/42 ,  C07D401/12 ,  C07D405/12 ,  C07D409/12 ,  C07D239/50

    CPC分类号： C07D239/42 ,  A01N43/54 ,  C07D401/12 ,  C07D405/12 ,  C07D409/12

    摘要： The invention relates to novel 5-acylaminopyrimidines of the general formula I ##STR1## wherein R.sub.1 is lower alkyl, lower alkoxy, lower alkoxy-lower alkyl, thioalkyl or halogen; phenyl or phenoxy, each unsubstituted or substituted by halogen, halo-lower alkyl, carbalkoxy-lower alkyl, halo-lower alkoxy, lower alkoxy, phenoxy, halophenoxy, halo-lower alkylthio, cyano or nitro; lower alkenyl or lower alkynyl, or unsubstituted or substituted cycloalkylR.sub.2 is lower alkyl which is unsubstituted or substituted by halogen, cyano or lower alkoxy; phenyl or phenyl-lower alkyl, each unsubstituted or substituted; pyridyl, thienyl or furyl, in which the nucleus is unsubstituted or substituted, or is pyranyl, dihydropyranyl, C.sub.3 -C.sub.7 cycloalkyl or C.sub.3 -C.sub.7 alkenyl, andR.sub.3 is hydrogen or C.sub.1 -C.sub.8 alkyl and R.sub.2 and R.sub.3, together with the carbon atom to which they are attached, may form a cycloalkyl radical, which compounds are effective as plant growth regulators. The invention relates further to compositions which contain at least one of these compounds as active ingredient, and to the use thereof, as well as to the corresponding novel 5-aminopyrimidines and, as intermediates, to the novel azomethines from which they are obtained.

    摘要翻译： 本发明涉及通式Ⅰ（I）的新的5-酰氨基嘧啶，其中R1是低级烷基，低级烷氧基，低级烷氧基 - 低级烷基，硫代烷基或卤素; 苯基或苯氧基，各自未被取代或被卤素，卤代低级烷基，烷氧基 - 低级烷基，卤代低级烷氧基，低级烷氧基，苯氧基，卤代苯氧基，卤代低级烷硫基，氰基或硝基取代。 低级烯基或低级炔基，或未取代或取代的环烷基R2是未被取代或被卤素，氰基或低级烷氧基取代的低级烷基; 苯基或苯基 - 低级烷基，各自未取代或取代; 吡啶基，噻吩基或呋喃基，其中核是未取代或取代的，或是吡喃基，二氢吡喃基，C 3 -C 7环烷基或C 3 -C 7链烯基，R 3是氢或C 1 -C 8烷基，R 2和R 3与它们的碳原子一起 可以形成环烷基，该化合物作为植物生长调节剂是有效的。 本发明进一步涉及含有这些化合物中的至少一种作为活性成分的组合物及其用途，以及相应的新的5-氨基嘧啶以及作为中间体获得的新的偶氮甲碱的组合物。

    Snow glider
    12.
    发明授权
    Snow glider 失效
    滑翔机

    公开(公告)号：US4305603A

    公开(公告)日：1981-12-15

    申请号：US100862

    申请日：1979-12-06

    申请人： Marcel Muller ,  Urs Muller

    发明人： Marcel Muller ,  Urs Muller

    IPC分类号： A63C5/00 ,  A63C5/03 ,  A63C5/04

    CPC分类号： A63C5/031 ,  A63C5/03 ,  A63C5/044

    摘要： A snow glider in the form of an elongated glide plate (1), the upper side of which has at least one stand-on area (2, 3) for the feet of the user and the front part of which is bent upwards in the manner of ski tips. The glide plate (1) is wider at the rear than at the front and in the middle, this wider rear part (6) being bent upwards out of the plane of the middle part (5). The snow glider makes free smooth running on snow possible, changes in the direction of running being effected by a corresponding shift of the center of gravity of the body.

    摘要翻译： 呈滑翔板形式的滑翔机（1），其上侧具有用于使用者的脚的至少一个支撑区域（2,3），并且其前部在其中向上弯曲 滑雪技巧的方式。 滑行板（1）在后部比在前部和中部更宽，该较宽的后部（6）向上弯曲到中间部分（5）的平面之外。 滑翔机可以在雪上自由平稳运行，运行方向的变化是通过相应的身体重心的移动来实现的。

    Azinyliminodithietanes and their fungicidal and nematocidal methods of use
    15.
    发明授权
    Azinyliminodithietanes and their fungicidal and nematocidal methods of use 失效
    Azinyl亚基二环己烷及其杀真菌剂和杀线虫剂的使用方法

    公开(公告)号：US5190945A

    公开(公告)日：1993-03-02

    申请号：US794537

    申请日：1991-11-19

    申请人： Wolfgang Eckhardt ,  Urs Muller

    发明人： Wolfgang Eckhardt ,  Urs Muller

    IPC分类号： A01N43/54 ,  A01N43/60 ,  C07D409/12

    CPC分类号： C07D409/12 ,  A01N43/54 ,  A01N43/60

    摘要： 2-(Pyrimidyl or pyrazinyl)-imino-1,3-dithietanes ##STR1## wherein Ar is one of the radicals ##STR2## R is unsubstituted C.sub.1 -C.sub.3 alkyl or C.sub.1 -C.sub.3 alkyl which is substituted by halogen, C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 alkoxy, C.sub.1 -C.sub.3 alkylthio or cyano, independently of one another, or is unsubstituted or halo-substituted C.sub.3 -C.sub.7 alkenyl, unsubstituted or halo-substituted C.sub.3 -C.sub.7 alkynyl, or C.sub.3 -C.sub.5 cycloalkyl, C.sub.1 -C.sub.3 alkoxy, C.sub.1 -C.sub.3 alkylamino, nitro or halogen,n is a number from 0 to 3,X.sub.1 and X.sub.2 independently of each other are hydrogen or halogen, including the addition salts formed with acids of the formula H.sup..sym. X.sup..crclbar. in which the anion X.sup..crclbar. is Cl.sup..crclbar., Br.sup..crclbar., I.sup..crclbar., HSO.sub.4 -, H.sub.2 PO.sub.4 -, H.sub.2 PO.sub.3 -, NO.sub.3 -, CH.sub.3 COO.sup..crclbar., CH.sub.2 ClCOO-, CF.sub.3 COO-, HOCH.sub.2 COO-, CH.sub.3 CH(OH)COO.sup..crclbar., HOOCCOO.sup..crclbar., HOOCCH.sub.2 COO.sup..crclbar., HOOCCH.dbd.CHCOO.sup..crclbar., ##STR3## a process for the preparation of the compounds of formula I, and novel intermediates of the preparation process are described.The compounds of formula I have nematicidal and fungicidal properties. Nematicidal and fungicidal compositions that contain at least one compound of formula I as active ingredient, and also methods of using the compounds and the compositions in the control of nematodes and fungi, are described.

    摘要翻译： 2-（嘧啶基或吡嗪基） - 亚氨基-1,3-二硫代环己基（I）其中Ar是基团之一R是未被取代的C 1 -C 3烷基或被卤素取代的C 1 -C 3烷基， C 1 -C 3烷基，C 1 -C 3烷氧基，C 1 -C 3烷硫基或氰基，彼此独立地是未取代的或卤素取代的C 3 -C 7链烯基，未取代或卤素取代的C 3 -C 7炔基或C 3 -C 5环烷基，C 1 -C 3烷氧基， C 3烷基氨基，硝基或卤素，n为0至3的数，X 1和X 2彼此独立地为氢或卤素，包括与式H（+）X（ - ）的酸形成的加成盐，其中阴离子X （ - ）为Cl（ - ），Br（ - ），I（ - ），HSO4-，H2PO4-，H2PO3-，NO3-，CH3COO（ - ），CH2ClCOO-，CF3COO-，HOCH2COO-，CH3CH （ - ），HOOCCOO（ - ），HOOCCH2COO（ - ），HOOCCH = CHCOO（ - ），制备式I化合物的方法和制备方法的新中间体。 式I的化合物具有杀线虫和杀真菌性质。 描述了含有至少一种式I化合物作为活性成分的杀线虫和杀真菌组合物，以及使用化合物和组合物控制线虫和真菌的方法。

    Novel tricyclic ketones and fragrance compositions containing same
    16.
    发明授权
    Novel tricyclic ketones and fragrance compositions containing same 失效
    新颖的三环酮和含有它们的香料组合物

    公开(公告)号：US4947002A

    公开(公告)日：1990-08-07

    申请号：US266036

    申请日：1988-11-02

    申请人： Georg Frater ,  Urs Muller

    发明人： Georg Frater ,  Urs Muller

    IPC分类号： A61K8/35 ,  A61L9/01 ,  A61Q13/00 ,  C07C27/00 ,  C07C29/56 ,  C07C35/37 ,  C07C45/00 ,  C07C49/417 ,  C07C49/453 ,  C07C67/00 ,  C07C69/00 ,  C07C69/08 ,  C07C69/16 ,  C11B9/00

    CPC分类号： C07C69/00 ,  C07C35/37 ,  C07C49/453 ,  C11B9/0042 ,  C07C2103/00

    摘要： Novel compounds of the formula ##STR1## wherein: the symbols R.sup.1, R.sup.2, R.sup.4, R.sup.5 and R.sup.6 represent hydrogen or methyl, with the proviso that only one of R.sup.1, R.sup.2 and R.sup.4 represents methyl, and, when either or both R.sup.5 and R.sup.6 represent methyl, then R.sup.1, R.sup.2 and R.sup.4 represent hydrogen; and,either the symbol (.dbd.O) on the carbon designated by the number 1 or the symbol (.dbd.O) on the carbon designated by the number 3, represents a keto group, such that when the group is present on carbon 1, then carbon 3 may contain a methyl group.and their use as odorants are described.

    摘要翻译： 新颖的下式化合物其中：符号R1，R2，R4，R5和R6表示氢或甲基，条件是R1，R2和R4中只有一个表示甲基，当R5和 R6表示甲基，则R1，R2和R4表示氢; 并且由数字1表示的碳上的符号（= O）或由数字3表示的碳上的符号（= O）表示酮基，使得当基团存在于碳1上时，则 碳3可以含有甲基。 并描述它们作为气味剂的用途。

    Process for the preparation of cyclohexanedionecarboxylic acid derivatives
    17.
    发明授权
    Process for the preparation of cyclohexanedionecarboxylic acid derivatives 失效
    环己二酸羧酸衍生物的制备方法

    公开(公告)号：US4803268A

    公开(公告)日：1989-02-07

    申请号：US008445

    申请日：1987-01-29

    申请人： Hans-Georg Brunner ,  Urs Muller

    发明人： Hans-Georg Brunner ,  Urs Muller

    IPC分类号： A01N37/42 ,  C07C51/00 ,  C07C51/347 ,  C07C62/00 ,  C07C62/38 ,  C07C67/00 ,  C07C67/22 ,  C07C69/757 ,  C07C201/00 ,  C07C205/43 ,  C07C231/00 ,  C07C231/12 ,  C07C233/12 ,  C07C235/82 ,  C07C253/00 ,  C07C255/55 ,  C07C255/60 ,  C07C313/00 ,  C07C323/12 ,  C07C323/40 ,  C07D295/18 ,  C07D295/185 ,  C07D279/10

    CPC分类号： C07D295/185 ,  C07C323/00 ,  C07C51/347

    摘要： The present invention relates to a novel, optimized process for the preparation of cyclohexanedionecarboxylic acid derivatives of formula I which can be carried out in a single vessel affording a very good yield, which process comprises heating a reactive carboxylic acid derivative of formula III ##STR1## wherein X is a halide, an alkylsulfonic or arylsulfonic acid radical or the molecular radical ##STR2## which is necessary to form an anhydride and R.sub.1 is alkyl or cycloalkyl, with an alkali metal cyanide or copper cyanide, in an inert organic solvent, to give a mixture, then adding in succession to said mixture, at a temperature in the range from 0.degree. C. to room temperature, zinc chloride, an equimolar amount, with respect to the carboxylic acid derivative of formula III, of a 3,5-cyclohexanedione-1-carboxylic acid derivative of formula II ##STR3## wherein A is an ester or amide radical, and, dropwise, an amine, and, after acidifying the reaction mixture with an aqueous acid, isolating the resultant 4-acyl-3,5-cyclohexanedione-1-carboxylic acid derivative of formula I ##STR4## by extraction. Said cyclohexanedionecarboxylic acid derivatives have herbicidal and plant growth regulating properties.

    摘要翻译： 本发明涉及一种用于制备式I的环己二酸羧酸衍生物的新型优化方法，其可以在单一容器中进行，提供非常好的产率，该方法包括加热式III的反应性羧酸衍生物 （III）其中X是卤化物，烷基磺酸或芳基磺酸基团或在惰性有机溶剂中与碱金属氰化物或氰化铜形成酸酐而R1是烷基或环烷基所必需的分子基团 ，得到混合物，然后在0℃至室温的温度下连续加入所述混合物，相对于式III的羧酸衍生物，等摩尔量的氯化锌为3 （II）的5-环己二酮-1-羧酸衍生物其中A是酯或酰胺基，并逐滴加入胺，并且在用酸水溶液酸化反应混合物后， 通过萃取分离得到式I的所得4-酰基-3,5-环己二酮-1-羧酸衍生物（I）图像+ TR图像。 所述环己二酸羧酸衍生物具有除草和植物生长调节性质。

    Microbicidal and growth-regulating compositions
    18.
    发明授权
    Microbicidal and growth-regulating compositions 失效
    杀菌和生长调节组合物

    公开(公告)号：US4758670A

    公开(公告)日：1988-07-19

    申请号：US567998

    申请日：1984-01-04

    申请人： Urs Muller ,  Hermann Rempfler ,  Hans Tobler

    发明人： Urs Muller ,  Hermann Rempfler ,  Hans Tobler

    IPC分类号： A01N43/50 ,  A01N43/653 ,  C07D233/60 ,  C07D249/08 ,  C07D405/06 ,  C07D521/00 ,  A01N43/64

    CPC分类号： C07D231/12 ,  A01N43/50 ,  A01N43/653 ,  C07D233/56 ,  C07D249/08

    摘要： Fluoroazolylpropane derivatives of the formula I ##STR1## are described, in which Az is imidazolyl or triazolyl, R.sup.1 is hydrogen, alkyl or aralkyl which is unsubstituted or substituted by halogen, alkyl, alkoxy, halogenoalkyl, nitro, cyano, carboxyl or alkoxycarbonyl, R.sup.2 is C.sub.1 -C.sub.10 -alkyl which is unsubstituted or substituted by alkoxy, aralkoxy or phenyl, it being possible for the aromatic nuclei of aralkoxy and phenyl in turn to be unsubstituted or substituted by halogen, alkyl, alkoxy, halogenoalkyl, cyano, carboxyl or alkoxycarbonyl, R.sup.3 is hydrogen, alkyl, alkylcarbonyl or aralkyl which is unsubstituted or substituted by halogen, alkoxy, alkyl, halogenoalkyl, cyano, carboxyl or alkoxycarbonyl, R.sup.5 is an unsubstituted or monosubstituted or polysubstituted radical selected from the series comprising C.sub.1 -C.sub.8 -alkyl, C.sub.3 -C.sub.8 -cycloalkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, phenyl, naphthyl, biphenyl, benzylphenyl, benzyloxyphenyl, phenoxyphenyl and aralkyl, and X is oxygen or sulfur; including the acid addition salts, quaternary azolium salts and metal complexes.Methods of preparing these products are also disclosed, as are agrochemical compositions containing one of these compounds as the active substance. A process for controlling phytopathogenic microorganisms and/or for regulating plant growth by means of these substances is also described.

    摘要翻译： 描述了式I的氟唑基丙烷衍生物，其中Az是咪唑基或三唑基，R1是氢，未被取代或被卤素，烷基，烷氧基，卤代烷基，硝基，氰基，羧基或烷氧基羰基取代的烷基或芳烷基，R2 是未被取代或被烷氧基，芳烷氧基或苯基取代的C 1 -C 10 - 烷基，芳烷氧基和苯基的芳族核可能是未被取代的或被卤素，烷基，烷氧基，卤代烷基，氰基，羧基或烷氧基羰基 R 3是未取代的或被卤素，烷氧基，烷基，卤代烷基，氰基，羧基或烷氧基羰基取代的烷基，烷基，烷基羰基或芳烷基，R 5是未取代的或单取代的或多取代的基团，其选自包括C 1 -C 8烷基， C 3 -C 8 - 环烷基，C 3 -C 6 - 烯基，C 3 -C 6炔基，苯基，萘基，联苯基，苄基苯基，苄氧基苯基，苯氧基苯基和芳烷基，X是氧或硫; 包括酸加成盐，季铵盐和金属络合物。 还公开了制备这些产物的方法，以及含有这些化合物之一作为活性物质的农药组合物。 还描述了通过这些物质控制植物病原微生物和/或调节植物生长的方法。

    DEVICE FOR THE AUTOMATED OPENING OF FLIP TUBES
    19.
    发明申请
    DEVICE FOR THE AUTOMATED OPENING OF FLIP TUBES 有权
    用于自动打开卷管的装置

    公开(公告)号：US20130118118A1

    公开(公告)日：2013-05-16

    申请号：US13698554

    申请日：2011-05-18

    申请人： Walter Kubler ,  Rainer Beckbissinger ,  Urs Muller

    发明人： Walter Kubler ,  Rainer Beckbissinger ,  Urs Muller

    IPC分类号： B65B69/00

    CPC分类号： B65B69/00 ,  B01L3/50825 ,  B01L2300/043 ,  G01N35/04 ,  G01N2035/0405

    摘要： A tool device for the automated opening of flip tubes including an actuating plunger which is provided and configured to move the actuating portion at least in open direction and thereby to exert an opening moment on the lid portion, and wherein the device further includes a damping means which is configured to exert a damping moment on the container lid at least during a period of the actuation of the actuating portion by the actuating plunger, which damping moment is less in amount and is in an opposite direction compared to the opening moment.

    摘要翻译： 一种用于自动打开翻盖管的工具装置，包括致动柱塞，其致动柱塞被设置和构造成至少沿打开方向移动致动部分，从而在盖部分上施加开启力矩，并且其中该装置还包括阻尼装置 其构造成至少在通过致动柱塞致动部分的致动周期期间在容器盖上施加阻尼力矩，该阻尼力矩较少，并且与开启力矩相反。