Aryl imidazoles and their use as anti-cancer agents
    11.
    发明申请
    Aryl imidazoles and their use as anti-cancer agents 有权
    芳基咪唑及其作为抗癌剂的用途

    公开(公告)号:US20080262015A9

    公开(公告)日:2008-10-23

    申请号:US10579149

    申请日:2004-11-15

    Abstract: Therapeutically effective 2,4,5-trisubstituted imidazole compounds are provided. Also provided are methods -of preparing the compounds and pharmaceutical compositions comprising the compounds alone or in combination with other agents. The present invention further provides for the use of the compounds as anti-cancer agents; wherein: R1 is aryl, substituted aryl, heterocycle, substituted heterocycle, heteroaryl, substituted heteroaryl or amino; R2 and R3 are independently aryl, substituted aryl, heterocycle, heteroaryl, substituted heterocycle, or substituted heteroaryl or R2 and R3 when taken together along with the carbon atoms they are attached to, form aryl or substituted aryl, and R4 is hydrogen, halogen, hydroxyl, thiol, lower alkyl, substituted lower alkyl, lower alkenyl, substituted lower alkenyl, lower alkynyl, substituted lower alkynyl, alkylalkenyl, alkyl alkynyl, alkoxy, alkylthio, aryl, aryloxy, amino, amido, carboxyl, aryl, substituted aryl, heterocycle, heteroaryl, substituted heterocycle, heteroalkyl, cycloalkyl, substituted cycloalkyl, alkylcycloalkyl, alkylcycloheteroalkyl, nitro, cyano or —S(O)o.2R wherein R is alkyl, substituted alkyl, aryl, substituted aryl, heterocycle, heteroaryl, substituted heterocycle, or substituted heteroaryl.

    Abstract translation: 提供了治疗上有效的2,4,5-三取代的咪唑化合物。 还提供了制备化合物和药物组合物的方法,所述药物组合物包含单独的化合物或与其它药剂组合。 本发明还提供了化合物作为抗癌剂的用途; 其中:R1是芳基,取代的芳基,杂环,取代的杂环,杂芳基,取代的杂芳基或氨基; R2和R3独立地是芳基,取代的芳基,杂环,杂芳基,取代的杂环或取代的杂芳基,或者当R 2和R 3与它们连接的碳原子一起形成时,R 2和R 3,形成芳基或取代的芳基,且R 4是氢,卤素, 羟基,硫醇,低级烷基,取代的低级烷基,低级烯基,取代的低级烯基,低级炔基,取代的低级炔基,烷基烯基,烷基炔基,烷氧基,烷硫基,芳基,芳氧基,氨基,酰胺基,羧基,芳基,取代的芳基,杂环 ,杂芳基,取代的杂环,杂烷基,环烷基,取代的环烷基,烷基环烷基,烷基环杂烷基,硝基,氰基或-S(O)o2R其中R是烷基,取代的烷基,芳基,取代的芳基,杂环,杂芳基,取代的杂环或 取代的杂芳基。

    Aryl imidazoles and their use as anti-cancer agents
    12.
    发明申请
    Aryl imidazoles and their use as anti-cancer agents 有权
    芳基咪唑及其作为抗癌剂的用途

    公开(公告)号:US20070123553A1

    公开(公告)日:2007-05-31

    申请号:US10579149

    申请日:2004-11-15

    Abstract: Therapeutically effective 2,4,5-trisubstituted imidazole compounds are provided. Also provided are methods -of preparing the compounds and pharmaceutical compositions comprising the compounds alone or in combination with other agents. The present invention further provides for the use of the compounds as anti-cancer agents; wherein: R1 is aryl, substituted aryl, heterocycle, substituted heterocycle, heteroaryl, substituted heteroaryl or amino; R2 and R3 are independently aryl, substituted aryl, heterocycle, heteroaryl, substituted heterocycle, or substituted heteroaryl or R2 and R3 when taken together along with the carbon atoms they are attached to, form aryl or substituted aryl, and R4 is hydrogen, halogen, hydroxyl, thiol, lower alkyl, substituted lower alkyl, lower alkenyl, substituted lower alkenyl, lower alkynyl, substituted lower alkynyl, alkylalkenyl, alkyl alkynyl, alkoxy, alkylthio, aryl, aryloxy, amino, amido, carboxyl, aryl, substituted aryl, heterocycle, heteroaryl, substituted heterocycle, heteroalkyl, cycloalkyl, substituted cycloalkyl, alkylcycloalkyl, alkylcycloheteroalkyl, nitro, cyano or —S(O)o.2R wherein R is alkyl, substituted alkyl, aryl, substituted aryl, heterocycle, heteroaryl, substituted heterocycle, or substituted heteroaryl.

    Abstract translation: 提供了治疗上有效的2,4,5-三取代的咪唑化合物。 还提供了制备化合物和药物组合物的方法,所述药物组合物包含单独的化合物或与其它药剂组合。 本发明还提供了化合物作为抗癌剂的用途; 其中:R1是芳基,取代的芳基,杂环,取代的杂环,杂芳基,取代的杂芳基或氨基; R2和R3独立地是芳基,取代的芳基,杂环,杂芳基,取代的杂环或取代的杂芳基,或者当R 2和R 3与它们连接的碳原子一起形成时,R 2和R 3,形成芳基或取代的芳基,且R 4是氢,卤素, 羟基,硫醇,低级烷基,取代的低级烷基,低级烯基,取代的低级烯基,低级炔基,取代的低级炔基,烷基烯基,烷基炔基,烷氧基,烷硫基,芳基,芳氧基,氨基,酰胺基,羧基,芳基,取代的芳基,杂环 ,杂芳基,取代的杂环,杂烷基,环烷基,取代的环烷基,烷基环烷基,烷基环杂烷基,硝基,氰基或-S(O)o2R其中R是烷基,取代的烷基,芳基,取代的芳基,杂环,杂芳基,取代的杂环或 取代的杂芳基。

    Oil separator for air conditioners
    13.
    发明申请
    Oil separator for air conditioners 有权
    空调油分离器

    公开(公告)号:US20060107687A1

    公开(公告)日:2006-05-25

    申请号:US11285112

    申请日:2005-11-23

    CPC classification number: F25B43/02 F25B2400/02

    Abstract: Disclosed herein is an oil separator for air conditioners that is capable of separating oil from refrigerant. The oil separator comprises a shell having a cylindrical space defined therein, a refrigerant introduction pipe for introducing refrigerant into the shell, a refrigerant discharge pipe for discharging the refrigerant out of the shell, and oil-drop growth accelerating member for accelerating growth of oil drops contained in the refrigerant flowing in the shell.

    Abstract translation: 本文公开了一种能够从制冷剂中分离油的空调用油分离器。 油分离器包括壳体,其中限定有圆柱形空间,用于将制冷剂引入壳体的制冷剂引入管,用于将制冷剂从壳体排出的制冷剂排出管和用于加速油滴生长的油滴生长促进构件 包含在流过壳体的制冷剂中。

    Air conditioner
    14.
    发明申请
    Air conditioner 审中-公开
    冷气机

    公开(公告)号:US20060080990A1

    公开(公告)日:2006-04-20

    申请号:US11249706

    申请日:2005-10-14

    Abstract: Disclosed is an air conditioner. The air conditioner a main compressor for compressing a refrigerant; a four-way valve disposed at a discharge side of the main compressor and switching a fluid path; an outdoor heat exchanger having one side connected with the four-way valve; an indoor heat exchanger having one side connected with the outdoor heat exchanger and the other side connected with the four-way valve; an expansion valve disposed between the outdoor heat exchanger and the indoor heat exchanger; and an auxiliary compression unit for reducing the load on the main compressor. Accordingly, since the load on the main compressor decreases, efficiency and reliability of the main compressor are enhanced and noises are reduced. In addition, an instrumental part such as a bearing inside the main compressor is not subject to abrasion and high heat damage to a motor unit is prevented.

    Abstract translation: 公开了一种空调。 空调机是用于压缩制冷剂的主压缩机; 四通阀,设置在主压缩机的排出侧并切换流体路径; 一侧与四通阀连接的室外热交换器; 室内热交换器,其一侧与室外热交换器连接,另一侧与四通阀连接; 设置在室外热交换器和室内热交换器之间的膨胀阀; 以及用于减小主压缩机上的负载的辅助压缩单元。 因此,由于主压缩机上的负载下降,主压缩机的效率和可靠性提高,噪音降低。 此外,诸如主压缩机内部的轴承的工具部件不会磨损,并且防止对电动机单元的高热损坏。

    Abutment of dental implant and aesthetic surface treatment method of the same
    15.
    发明申请
    Abutment of dental implant and aesthetic surface treatment method of the same 审中-公开
    牙根植入物的基台和美观表面处理方法相同

    公开(公告)号:US20050181330A1

    公开(公告)日:2005-08-18

    申请号:US10919173

    申请日:2004-08-16

    Applicant: Soo Kim Yoon Lee

    Inventor: Soo Kim Yoon Lee

    CPC classification number: A61C8/005 A61C8/0069

    Abstract: The present invention discloses an abutment of a dental implant consisting of an abutment screw and a shoulder surface. The upper structure of a crown or bridge abutment, i.e., the abutment screw is made of titanium alloy, and surface-treated in brown color by an anodizing process, and the connecting structure thereof, i.e., the shoulder surface is made of ceramic material containing zirconia of a white color, thereby providing an adequate mechanical strength, while maintaining the natural color of human teeth and light permeability. Further, the present invention discloses a method of aesthetically surface-treating the abutment screw of a dental implant abutment by using the anodizing process, and a method of fabricating the shoulder surface of a dental implant abutment.

    Abstract translation: 本发明公开了一种由基牙螺钉和肩部表面构成的牙科植入物的支座。 顶部或桥接台座的上部结构,即基台螺钉由钛合金制成,并通过阳极氧化处理以棕色进行表面处理,其连接结构即肩部表面由含有 氧化锆白色,从而提供足够的机械强度,同时保持人牙的自然色泽和透光性。 此外,本发明公开了一种通过使用阳极氧化处理来美观地表面处理牙科植入物邻接的基台螺钉的方法,以及一种制造牙科植入物基台的肩表面的方法。

    Image forming apparatus and method of controlling the same
    18.
    发明授权
    Image forming apparatus and method of controlling the same 有权
    图像形成装置及其控制方法

    公开(公告)号:US08094328B2

    公开(公告)日:2012-01-10

    申请号:US11954047

    申请日:2007-12-11

    Abstract: An image forming apparatus and a method to control the same. The image forming apparatus determines whether the object to be printed is real money. If the object is real money, the image forming apparatus prints a variety of counterfeit money discrimination information (e.g., the counterfeit money preventing pattern, the warning message, or the unique number of the image forming apparatus used for printing the money) on the back side of the copy of the money, and prints the original image of the money on the front side of the copy of the money without any change. Therefore, the image forming apparatus can color-print the original image of the money without any change, and can prevent the copied money from being used as counterfeit money.

    Abstract translation: 一种图像形成装置及其控制方法。 图像形成装置确定要打印的对象是否是真实货币。 如果对象是实际货币,则图像形成装置在背面打印各种假币鉴别信息(例如,伪钞防止图案,警告信息或用于打印货币的图像形成装置的唯一号码) 副本的一面,并在货币副本的正面打印货币的原始图像,而不做任何改变。 因此,图像形成装置可以在没有任何变化的情况下对原始图像进行彩色打印,并且可以防止被复制的货币被用作伪造货币。

    IMAGE FORMING APPARATUS AND BOGUS NOTE MANAGING SYSTEM INCLUDING THE SAME
    20.
    发明申请
    IMAGE FORMING APPARATUS AND BOGUS NOTE MANAGING SYSTEM INCLUDING THE SAME 审中-公开
    图像形成装置和BOGUS注释管理系统,包括它们

    公开(公告)号:US20080135373A1

    公开(公告)日:2008-06-12

    申请号:US11850228

    申请日:2007-09-05

    Abstract: An image forming apparatus, a bogus note managing system including the same, and a bogus note managing method that are capable of accurately and efficiently managing a bogus note such that the bogus note cannot be used for a bad purpose, the image forming apparatus including: a read unit to determine whether an object to be read is money; a storage unit to store money registration information including identification information of the money; a comparison unit to compare money identification information, which is received so as to identify the money, with the identification information stored in the storage unit when the object to be read is the money; and a control unit to control history information of the money to be stored in the storage unit when the money identification information is identical to the identification information.

    Abstract translation: 一种图像形成装置,包括该图像形成装置的虚假票据管理系统以及能够准确且有效地管理虚假票据的虚假票据管理方法,使得虚假票据不能用于不良目的,该图像形成装置包括: 一个阅读单元来确定一个要读取的对象是否是金钱; 存储单元,用于存储包括货币的识别信息的货币登记信息; 比较单元,用于当要读取的对象是货币时,将存储在存储单元中的识别信息与用于识别货币的接收的货币识别信息进行比较; 以及控制单元,用于当货币识别信息与识别信息相同时,控制要存储在存储单元中的货币的历史信息。

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