3-(Pyridin-2-Yl)-[1,2,4]-Triazines as Fungicides
    35.
    发明申请
    3-(Pyridin-2-Yl)-[1,2,4]-Triazines as Fungicides 审中-公开
    3-(吡啶-2-基) - [1,2,4] - 三嗪作为杀真菌剂

    公开(公告)号:US20090111692A1

    公开(公告)日:2009-04-30

    申请号:US12226026

    申请日:2007-04-11

    摘要: The invention relates to 3-(pyridin-2-yl)-[1,2,4]-triazines of formula (I) and their use in the control of parasitic fungi and to herbicides that contain said compounds as an effective ingredient thereof. In formula (I), R1, R2 independently represent OH, halogen, NO2, NH2, C1-C8 alkyl, C1-C8 alkoxy, C1-C8 halogenalkyl, C1-C8 halogenalkoxy, C1-C8 alkylamino or di(C1-C8 alkyl)amino, or they form, together with the C atoms to which they are bound, a saturated five-, six- or seven-membered carbocycle or heterocycle, which, in addition to the carbon ring members, has one or two heteroatoms selected from oxygen or sulfur as the ring members, the carbocycle and the heterocycle being unsubstituted or having 1, 2, 3 or 4 C1-C4 alkyl groups as the substituents; R3 represents hydrogen, C1-C4 alkyl, C1-C4 alkoxy, C1-C4 halogenalkyl, C1-C4 halogenalkoxy, C3-C6 cycloalkyl, C3-C6 cycloalkylmethyl, or halogen; R4 represents hydrogen, C1-C4 alkyl, C1-C4 alkoxy, C1-C4 halogenalkyl, C1-C4 halogenalkoxy or halogen; R5 represents C1-C8 alkyl, C1-C8 halogenalkyl, C1-C8 alkoxy, C1-C8 halogenalkoxy, C3-C8 cycloalkyl, C3-C8 cycloalkyloxy, five- or six-membered heteroaryl, phenyl, phenoxy, benzyl, benzyloxy, five- or six-membered heteroarylmethyl or five- or six-membered heteroaryloxy, said cyclic groups being unsubstituted or having 1, 2, 3, 4 or 5 groups Ra.

    摘要翻译: 本发明涉及式(I)的3-(吡啶-2-基) - [1,2,4] - 三嗪及其在控制寄生真菌中的用途以及含有所述化合物作为其有效成分的除草剂。 在式(I)中,R 1,R 2独立地表示OH,卤素,NO 2,NH 2,C 1 -C 8烷基,C 1 -C 8烷氧基,C 1 -C 8卤代烷基,C 1 -C 8卤代烷氧基,C 1 -C 8烷基氨基或二 )氨基,或者它们与它们所键合的C原子一起形成饱和的五元,六元或七元碳环或杂环,其除了碳环成员之外还具有一个或两个选自以下的杂原子: 氧或硫作为环成员,碳环和杂环是未取代的或具有1,2,3或4个C 1 -C 4烷基作为取代基; R 3表示氢,C 1 -C 4烷基,C 1 -C 4烷氧基,C 1 -C 4卤代烷基,C 1 -C 4卤代烷氧基,C 3 -C 6环烷基,C 3 -C 6环烷基甲基或卤素; R4表示氢,C1-C4烷基,C1-C4烷氧基,C1-C4卤代烷基,C1-C4卤代烷氧基或卤素; R5表示C1-C8烷基,C1-C8卤代烷基,C1-C8烷氧基,C1-C8卤代烷氧基,C3-C8环烷基,C3-C8环烷氧基,五元或六元杂芳基,苯基,苯氧基,苄基,苄氧基, 或六元杂芳基甲基或五元或六元杂芳氧基,所述环状基团是未取代的或具有1,2,3,4或5个基团Ra。

    2-(Pyridin-2-Yl)-Pyrimidines for Use as Fungicides
    36.
    发明申请
    2-(Pyridin-2-Yl)-Pyrimidines for Use as Fungicides 审中-公开
    2-(吡啶-2-基) - 嘧啶用作杀真菌剂

    公开(公告)号:US20090105072A1

    公开(公告)日:2009-04-23

    申请号:US12225862

    申请日:2007-04-11

    摘要: The present invention relates to 2-(pyridin-2-yl)pyrimidines and their use for controlling harmful fungi, and also to crop protection compositions comprising such compounds as effective component. in which: Q is a fused saturated 5-, 6- or 7-membered carbocycle or a 5-, 6- or 7-membered heterocycle which, in addition to the carbon ring members, has one or two heteroatoms selected from the group consisting of oxygen and sulfur as ring members, where the carbocycle and the heterocycle are unsubstituted or have 1, 2, 3 or 4 C1-C4-alkyl groups as substituents; R1 is hydrogen, OH, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy or halogen; R2 is hydrogen, NO2, halogen, C1-C6-alkyl, C3-C6-cycloalkyl, C1-C6-alkoxy, C1-C6-haloalkyl or C1-C6-haloalkoxy; R3 is hydrogen, halogen, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, or C1-C4-haloalkoxy; R4 is phenyl, 5-membered heteroaryl which has 1, 2, 3 or 4 nitrogen atoms or 1 heteroatom selected from the group consisting of oxygen and sulfur and optionally 1, 2 or 3 nitrogen atoms as ring atoms, or 6-membered hetaryl which has 1, 2, 3 or 4 nitrogen atoms as ring members, where phenyl and 5- and 6-membered hetaryl may have 1, 2, 3 or 4 substituents Ra.

    摘要翻译: 本发明涉及2-(吡啶-2-基)嘧啶及其用于控制​​有害真菌的用途,还涉及包含有效成分的化合物的作物保护组合物。 其中:Q是稠合的饱和的5-,6-或7-元碳环或5-,6-或7-元杂环,其除了碳环成员之外还具有一个或两个选自以下的杂原子: 的氧和硫作为环成员,其中碳环和杂环是未取代的或具有1,2,3或4个C 1 -C 4 - 烷基作为取代基; R 1是氢,OH,C 1 -C 4 - 烷基,C 1 -C 4 - 烷氧基,C 1 -C 4卤代烷基,C 1 -C 4卤代烷氧基或卤素; R2是氢,NO2,卤素,C1-C6-烷基,C3-C6-环烷基,C1-C6-烷氧基,C1-C6卤代烷基或C1-C6-卤代烷氧基; R 3是氢,卤素,C 1 -C 4 - 烷基,C 1 -C 4 - 烷氧基,C 1 -C 4卤代烷基或C 1 -C 4卤代烷氧基; R4是苯基,具有1,2,3或4个氮原子的5元杂芳基或选自氧和硫以及任选的1,2或3个氮原子作为环原子的1个杂原子,或6元杂芳基, 具有1,2,3或4个氮原子作为环成员,其中苯基和5-和6-元杂芳基可以具有1,2,3或4个取代基R a。

    Azolylmethyloxiranes, Their Use for Controlling Phytopathogenic Fungi and Agents Containing Said Compounds
    40.
    发明申请
    Azolylmethyloxiranes, Their Use for Controlling Phytopathogenic Fungi and Agents Containing Said Compounds 审中-公开
    唑基甲基环氧乙烷,它们用于控制植物病原真菌和含有所述化合物的试剂

    公开(公告)号:US20090197929A1

    公开(公告)日:2009-08-06

    申请号:US12306339

    申请日:2007-06-25

    IPC分类号: A01N43/64 C07D249/08 A01P3/00

    摘要: The present invention relates to azolylmethyloxiranes of the general formula I in which A or B is a 5-membered heteroaryl selected from the group consisting of thienyl, furyl, pyrrolyl, pyrazolyl, imidazolyl, oxazolyl, thiazolyl, isoxazolyl and isothiazolyl which is substituted by one to three of the following substituents: halogen, NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, and the respective other substituent A or B is phenyl which is optionally substituted by one to three of the following substituents: halogen, NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, and to the plant-compatible acid addition salts or metal salts thereof, to the use of the compounds of the formula I for controlling phytopathogenic fungi and to compositions comprising these compounds.

    摘要翻译: 本发明涉及通式I的唑基甲基环氧乙烷,其中A或B是选自噻吩基,呋喃基,吡咯基,吡唑基,咪唑基,恶唑基,噻唑基,异恶唑基和被一个取代基的异噻唑基的5元杂芳基 至三个以下取代基:卤素,NO 2,氨基,C 1 -C 4 - 烷基,C 1 -C 4 - 烷氧基,C 1 -C 4 - 卤代烷基,C 1 -C 4 - 卤代烷氧基,C 1 -C 4烷基氨基,C 1 -C 4二烷基氨基,硫代 或其它取代基A或B为任选被一至三个以下取代基取代的苯基:卤素,NO 2,氨基,C 1 -C 4 - 烷基,C 1 -C 4 - 烷氧基,C 1 -C 4 - 烷硫基, C 4-卤代烷基,C 1 -C 4卤代烷氧基,C 1 -C 4 - 烷基氨基,C 1 -C 4 - 二烷基氨基,硫代或C 1 -C 4 - 烷硫基,以及与植物相容的酸加成盐或其金属盐, 用于控制植物病原真菌的式I化合物和包含这些化合物的组合物。