Isoxazole(isothiazole)-5-carboxamides
    42.
    发明授权
    Isoxazole(isothiazole)-5-carboxamides 失效
    异佛唑(异噻唑)-5-羧酰胺

    公开(公告)号:US5080708A

    公开(公告)日:1992-01-14

    申请号:US337640

    申请日:1989-04-13

    摘要: Isoxazole(isothiazole)-5-carboxamides of the formula ##STR1## where X is oxygen or sulfur,R.sup.1 is hydrogen, substituted or unsubstituted alkyl, alkoxy, substituted or unsubstituted cycloalkyl, a 5- or 6-membered heterocyclic radical having one or two heteroatoms selected from the group consisting of oxygen, sulfur and nitrogen, and which may be substituted, or substituted or unsubstituted phenyl, orR.sup.2 is formyl, 4,5-dihydrooxazol-2-yl or a radical of the formula COYR.sup.5 or CONR.sup.6 R.sup.7, whereY is oxygen or sulfur,R.sup.5 ishydrogen, substituted or unsubstituted alkyl, substituted or unsubstituted alkenyl, haloalkenyl, substituted or unsubstituted alkynyl,cycloalkyl,cycloalkenyl,substituted or unsubstituted phenyl,a 5- or 6-membered heterocyclic radical having one or two heteroatoms selected from the group consisting of oxygen, sulfur and nitrogen,cycloalkanimino, phthalimido, succinimido, or a radical ##STR2## R.sup.3 and R.sup.4 have the meanings defined herein, or their agriculturally acceptable salts possess herbicidal activity.

    摘要翻译: 其中X是氧或硫,R 1是氢,取代或未取代的烷基,烷氧基,取代或未取代的环烷基,具有一个或两个的5-或6-元杂环基的异噻唑(异噻唑)-5-甲酰胺, 选自氧,硫和氮的杂原子,并且其可以被取代,或取代或未取代的苯基,或R 2是甲酰基,4,5-二氢恶唑-2-基或式COYR 5或CONR 6 R 7的基团,其中 Y是氧或硫,R5是氢,取代或未取代的烷基,取代或未取代的烯基,卤代烯基,取代或未取代的炔基,环烷基,环烯基,取代或未取代的苯基,具有一个或两个杂原子的5-或6-元杂环基 选自氧,硫和氮,环亚烷基亚氨基,邻苯二甲酰亚氨基,琥珀酰亚胺基或自由基,CH 2 CH(OH)CH 2(OH)等,R 3和R 4具有本文定义的含义或其农业 超可接受的盐具有除草活性。

    N-((6-trifluoromethyl
pyrimidin-2-yl)-aminocarbonyl)-2-carboalkoxybenzenesulfonamides
    44.
    发明授权
    N-((6-trifluoromethyl pyrimidin-2-yl)-aminocarbonyl)-2-carboalkoxybenzenesulfonamides 失效
    N - ((6-三氟甲基吡啶-2-基) - 氨基羰基)-2-羧酸甲苯磺酰胺

    公开(公告)号:US5069710A

    公开(公告)日:1991-12-03

    申请号:US337866

    申请日:1989-04-14

    IPC分类号: A01N47/36 C07D521/00

    CPC分类号: C07D521/00 A01N47/36

    摘要: N-((6-Trifluoromethylpyrimidin-2-yl)- aminocarbonyl)-2-carboalkoxybenzenesulfonamides of the general formula Ia ##STR1## where the substituents have the following meanings: R.sup.1 is hydrogen or halogen;R.sup.2 is hydrogen, C.sub.1 -C.sub.5 -alkyl, C.sub.3 -C.sub.4 -alkenyl, C.sub.3 -C.sub.4 -alkynyl, C.sub.1 -C.sub.5 -haloalkyl, C.sub.3 -C.sub.5 -alkoxyalkyl, C.sub.3 -C.sub.5 -haloalkoxyalkyl or C.sub.5 -C.sub.6 -cycloalkyl,R.sup.3 is hydrogen, C.sub.1 -C.sub.2 -alkyl, allyl, propargyl or C.sub.1 -C.sub.5 -alkoxy,R.sup.4 is halogen, C.sub.1 -C.sub.2 -alkyl, C.sub.1 -C.sub.3 -alkylthio or C.sub.1 -C.sub.3 -alkylamino,R.sup.3 not denoting hydrogen or C.sub.1 -C.sub.2 -alkyl when R.sup.4 is C.sub.1 -C.sub.2 -alkyl, and their environmentally tolerated salts, processes for their manufacture, and their use.

    摘要翻译: 具有通式Ia的N - ((6-三氟甲基嘧啶-2-基) - 氨基羰基)-2-烷氧羰基苯磺酰胺其中取代基具有以下含义:R 1是氢或卤素; R2是氢,C1-C5-烷基,C3-C4-烯基,C3-C4-炔基,C1-C5-卤代烷基,C3-C5-烷氧基烷基,C3-C5-卤代烷氧基烷基或C5-C6-环烷基,R3是氢, C 1 -C 2 - 烷基,烯丙基,炔丙基或C 1 -C 5 - 烷氧基,R 4是卤素,C 1 -C 2烷基,C 1 -C 3 - 烷硫基或C 1 -C 3烷基氨基,R 3不表示氢或C 1 -C 2烷基 是C 1 -C 2烷基,及其环境耐受的盐,其制备方法及其用途。

    Aromatic carboxylic acid derivatives and the use thereof for controlling
undesirable plant growth
    46.
    发明授权
    Aromatic carboxylic acid derivatives and the use thereof for controlling undesirable plant growth 失效
    芳族羧酸衍生物及其用于控制​​不期望的植物生长的用途

    公开(公告)号:US5015285A

    公开(公告)日:1991-05-14

    申请号:US409408

    申请日:1989-09-19

    摘要: Aromatic carboxylic acid derivatives of the formula ##STR1## in which the radical ##STR2## is a substituted or unsubstituted quinoline, naphthalene, benzofuran, thiophene or pyridine radical,R.sup.1 is hydrogen, alkylidenaminoxy, unsubstituted or substituted cycloalkylidenaminoxy, succinyliminoxy, unsubstituted or substituted alkenyloxy, alkynyloxy, azolyl, alkylsulfonylamino, alkoxycarbonylalkyloxy, N-azolylalkyloxy, unsubstituted or substituted alkoxy, unsubstituted or substituted phenylalkoxy, hydroxyl or the radical O.sup..crclbar. M.sup..sym., M.sup..sym. being one equivalent of an alkali metal, alkaline earth metal or organic ammonium ion,R.sup.2 and R.sup.3 are alkyl, haloalkyl, alkoxy, haloalkoxy or alkylthio,X is oxygen or sulfur,Y and Z are nitrogen or the methine group, andR.sup.4 and R.sup.5 are hydrogen, halogen, alkyl, haloalkyl, nitro, alkoxy, unsubstituted or substituted alkenyloxy, acylamino, alkylamino, dialkylamino or arylamino, and their use for controlling the growth of unwanted plants.

    摘要翻译: 式(Ⅰ)的芳族羧酸衍生物,其中基团是取代或未取代的喹啉,萘,苯并呋喃,噻吩或吡啶基,R1是氢,亚烷基氨基氧基,未取代的或取代的环烷基氨基氧基,琥珀酰亚氨基,未取代的 或取代的烯氧基,炔氧基,唑基,烷基磺酰基氨基,烷氧羰基烷氧基,N-吡唑烷基氧基,未取代或取代的烷氧基,未取代或取代的苯基烷氧基,羟基或O( - )M(+),M(+ ,碱土金属或有机铵离子,R2和R3是烷基,卤代烷基,烷氧基,卤代烷氧基或烷硫基,X是氧或硫,Y和Z是氮或次甲基,R4和R5是氢,卤素,烷基, 卤代烷基,硝基,烷氧基,未取代或取代的烯氧基,酰氨基,烷基氨基,二烷基氨基或芳基氨基,以及它们用于控制不想要的植物生长的用途。

    5-(N-3,4,5,6-tetrahydrophthalimido)cinnamic acid derivatives
    47.
    发明授权
    5-(N-3,4,5,6-tetrahydrophthalimido)cinnamic acid derivatives 失效
    5-(N-3,4,5,6-四氢邻苯二甲酰亚氨基)肉桂酸衍生物

    公开(公告)号:US5009701A

    公开(公告)日:1991-04-23

    申请号:US403382

    申请日:1989-09-06

    CPC分类号: C07D209/48 A01N37/46

    摘要: 5-(N-3,4,5,6-Tetrahydrophthalimido)-cinnamic acid derivatives of the formula Ib ##STR1## where the substituents have the following meanings: Y is chlorine, bromine or C.sub.1 -C.sub.4 -alkyl;R.sup.1 is hydrogen, C.sub.1 -C.sub.8 -alkyl, substituted or unsubstituted C.sub.2 -C.sub.4 alkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, or substituted or unsubstituted phenyl or benzyl,R.sup.2 is C.sub.5 -C.sub.8 -alkyl, substituted or unsubstituted C.sub.2 -C.sub.4 -alkyl, C.sub.1 -C.sub.6 -alkoxy, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkenyloxy, C.sub.3 -C.sub.6 -alkynyl, C.sub.3 -C.sub.6 -alkynyloxy, or substituted or unsubstituted phenyl, phenoxy, benzyl or benzyloxy,R.sub.3 C.sub.1 -C.sub.6 -alkyl, or substituted or unsubstituted C.sub.2 -C.sub.6 -alkyl,methods of manufacturing these compounds, and their use as herbicides.

    摘要翻译: 式Ib Ib的5-(N-3,4,5,6-四氢邻苯二甲酰亚氨基) - 肉桂酸衍生物,其中取代基具有以下含义:Y是氯,溴或C 1 -C 4 - 烷基; R 1是氢,C 1 -C 8 - 烷基,取代或未取代的C 2 -C 4烷基,C 3 -C 6 - 烯基,C 3 -C 6炔基或取代或未取代的苯基或苄基,R 2是C 5 -C 8 - 烷基,取代或未取代的C 2- C 1 -C 6 - 烷基,C 1 -C 6 - 烷氧基,C 3 -C 6 - 烯基,C 3 -C 6 - 烯氧基,C 3 -C 6 - 炔基,C 3 -C 6 - 炔氧基或取代或未取代的苯基,苯氧基,苄基或苄氧基, - 烷基或取代或未取代的C 2 -C 6 - 烷基,制备这些化合物的方法及其作为除草剂的用途。

    Cyanoquinoline compounds
    49.
    发明授权
    Cyanoquinoline compounds 失效
    氰基喹啉化合物

    公开(公告)号:US5565408A

    公开(公告)日:1996-10-15

    申请号:US423325

    申请日:1995-04-17

    摘要: Cyanoquinoline compounds Ia or Ib ##STR1## where R.sup.1 is CH.dbd.C(CN).sub.2 ; CH.dbd.N--N.dbd.CH--(5-quinolyl); methylsulfonyl; CH.dbd.NOH; halogen; hydroxyl; nitro; cyano; unsubstituted or substituted C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxy or C.sub.1 -C.sub.4 -alkylthio, pyrrolidinyl; piperidinyl; morpholinyl; thiomorpholinyl; unsubstituted or substituted phenyl, phenoxy, phenylthio, phenyldithiolyl, phenylsulfonyl or pyrrolyl;m is 0, 1, 2 or 3;R.sup.2 is hydrogen; hydroxyl; halogen; C.sub.1 -C.sub.4 -alkoxy; --NR.sup.3 R.sup.4 ; --NR.sup.5 --CXR.sup.6 or --N.dbd.CR.sup.7 R.sup.8 ;R.sup.3 is hydrogen or unsubstituted or substituted C.sub.1 -C.sub.4 -alkyl;R.sup.4 is a radical R.sup.3 ; C.sub.1 -C.sub.4 -alkylamino; di-C.sub.1 -C.sub.4 -alkylamino; substituted C.sub.1 -C.sub.4 -alkyl; CH.dbd.N--(3-cyano-2-quinolinyl); or R.sup.3 and R.sup.4 together form C.sub.4 - or C.sub.3 -alkylene which may be interrupted by a hetero atom, or unsubstituted or substituted 1,3-butadienyl;R.sup.5 and R.sup.7 are each hydrogen or C.sub.1 -C.sub.4 -alkyl;R.sup.6 and R.sup.8 are each a radical R.sup.5 ; substituted C.sub.1 -C.sub.4 -alkyl; C.sub.3 -C.sub.7 -cycloalkyl; C.sub.1 -C.sub.4 -alkoxycarbonyl; unsubstituted or substituted phenyl or unsubstituted or substituted amino, andX is oxygen or sulfur,processes for their preparation and herbicides which contain them.

    摘要翻译: 氰基喹啉化合物Ia或Ib其中R 1是CH = C(CN)2; CH = N-N = CH-(5-喹啉基); 甲基磺酰基; CH = NOH; 卤素; 羟; 硝基 氰基; 未取代或取代的C 1 -C 4 - 烷基,C 1 -C 4 - 烷氧基或C 1 -C 4 - 烷硫基,吡咯烷基; 哌啶基; 吗啉基 硫代吗啉基; 未取代或取代的苯基,苯氧基,苯硫基,苯基二硫代基,苯基磺酰基或吡咯基; m为0,1,2或3; R2是氢; 羟; 卤素; C1-C4-烷氧基; -NR3R4; -NR5-CXR6或-N = CR7R8; R3是氢或未取代的或取代的C1-C4-烷基; R4是一个基团R3; C 1 -C 4烷基氨基; 二-C 1 -C 4烷基氨基; 取代的C 1 -C 4 - 烷基; CH = N-(3-氰基-2-喹啉基); 或者R 3和R 4一起形成可以被杂原子间隔的C4-或C3-亚烷基,或未取代或取代的1,3-丁二烯基; R5和R7各自为氢或C1-C4-烷基; R6和R8各自为基团R5; 取代的C 1 -C 4 - 烷基; C 3 -C 7 - 环烷基; C 1 -C 4烷氧基羰基; 未取代或取代的苯基或未取代或取代的氨基,X为氧或硫,其制备方法和含有它们的除草剂。