Substituted 1,8-naphthyridines, their preparation and their use as
antidotes
    7.
    发明授权
    Substituted 1,8-naphthyridines, their preparation and their use as antidotes 失效
    取代的1,8-萘啶,其制备及其用作解毒剂

    公开(公告)号:US5258356A

    公开(公告)日:1993-11-02

    申请号:US13202

    申请日:1993-02-01

    IPC分类号: A01N25/32 C07D471/04

    CPC分类号: C07D471/04 A01N25/32

    摘要: A combination of a variety of herbicides with safening agents which are substituted 1,8-naphthyridines of the formula ##STR1## where R.sup.1 is mercapto, hydroxyl, halogen, benzylthio, amino or NR.sup.2 R.sup.3, whereR.sup.2 is a group ##STR2## where A is C.sub.1 -C.sub.8 -alkyl, R.sup.3 is hydrogen, XR.sup.4, where X is oxygen or sulfur and R.sup.4 is C.sub.1 -C.sub.12 -alkyl,R.sup.5 and R.sup.7 are each hydrogen, C.sub.1 -C.sub.12 -alkyl, hydroxyl, halogen, mercapto, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -alkylthio, dialkylamino where each alkyl is of 1 to 6 carbon atoms, phenoxy or phenylthio, halo-(C.sub.1 -C.sub.3)-alkyl, C.sub.1 -C.sub.4 -alkoxy-(C.sub.1 -C.sub.3)-alkyl, andR.sup.6 is hydrogen, C.sub.1 -C.sub.12 -alkyl, carboxyl or C.sub.1 -C.sub.4 -alkoxycarbonyl or the plant-tolerated salts thereof.

    摘要翻译: 各种除草剂与安全剂的组合,其为R1为巯基,羟基,卤素,苄硫基,氨基或NR2R3的式VIII取代的1,8-萘啶,其中R2为基团,其中A 是C 1 -C 8 - 烷基,R 3是氢,XR 4,其中X是氧或硫,R 4是C 1 -C 12烷基,R 5和R 7各自是氢,C 1 -C 12烷基,羟基,卤素,巯基,C 1 -C 4 - 烷氧基,C 1 -C 4烷氧基 - (C 1 -C 3) - 烷基,和C 1 -C 4 - 烷氧基 - (C 1 -C 3) - 烷基, R6是氢,C1-C12-烷基,羧基或C1-C4-烷氧基羰基或其植物耐受的盐。

    Thiophene-2-carboxylic acid derivatives, their preparation and their use
for controlling undesirable plant growth
    8.
    发明授权
    Thiophene-2-carboxylic acid derivatives, their preparation and their use for controlling undesirable plant growth 失效
    噻吩-2-羧酸衍生物,其制备及其用于控制​​不期望的植物生长的用途

    公开(公告)号:US5034049A

    公开(公告)日:1991-07-23

    申请号:US463163

    申请日:1990-01-09

    CPC分类号: C07D333/38 A01N43/10

    摘要: Thiophene-2-carboxylic acid derivatives of the general formula I ##STR1## where R.sup.1 to R.sup.3 are each hydrogen, halogen, branched or straight-chain C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.8 -alkoxy, C.sub.1 -C.sub.6 -haloalkyl, C.sub.1 -C.sub.6 -haloalkoxy, nitro, cyano, unsubstituted phenyl or phenyl which is mono- to trisubstituted by C.sub.1 -C.sub.4 -alkyl, halogen, C.sub.1 -C.sub.5 -haloalkyl, C.sub.1 -C.sub.4 -alkoxy or C.sub.1 -C.sub.5 -haloalkoxy;X is --OR.sup.4 or --NH--OR.sup.5,R.sup.4 being branched or straight-chain C.sub.3 -C.sub.10 -alkynylalkyl which is unsubstituted or substituted by halogen; andR.sup.5 being branched or straight-chain C.sub.1 -C.sub.5 -alkyl which is unsubstituted or substituted by halogen, or branched or straight-chain C.sub.3 -C.sub.10 -alkynylalkyl which is unsubstituted or substituted by halogen;with the proviso that R.sup.4 is not propargyl when R.sup.2 and R.sup.3 are both hydrogen or when R.sup.2 is halogen or R.sup.3 is chlorine, methyl or methoxy.The compounds I are suitable for combating the growth of unwanted plants.

    摘要翻译: 通式I的噻吩-2-羧酸衍生物其中R 1至R 3各自为氢,卤素,支链或直链C 1 -C 6 - 烷基,C 1 -C 8 - 烷氧基,C 1 -C 6 - 卤代烷基,C 1 C 1-6卤代烷氧基,硝基,氰基,未取代的苯基或被C 1 -C 4 - 烷基,卤素,C 1 -C 5 - 卤代烷基,C 1 -C 4 - 烷氧基或C 1 -C 5 - 卤代烷氧基单 - X为-OR4或-NH-OR5,R4为未取代或被卤素取代的支链或直链C 3 -C 10 - 炔基烷基; 并且R 5是未被取代或被卤素取代的支链或直链C 1 -C 5 - 烷基,或未被取代或被卤素取代的支链或直链C 3 -C 10 - 炔基烷基; 条件是当R 2和R 3均为氢时或R 2为卤素或R 3为氯,甲基或甲氧基时,R 4不是炔丙基。 化合物I适用于对抗不想要的植物的生长。

    Pyrimido(5,4-e)-as-triazine-5,7(6H,8H)-diones
    9.
    发明授权
    Pyrimido(5,4-e)-as-triazine-5,7(6H,8H)-diones 失效
    嘧啶并(5,4-e)-as-三嗪-5,7(6H,8H) - 二酮

    公开(公告)号:US5069708A

    公开(公告)日:1991-12-03

    申请号:US547160

    申请日:1990-07-03

    IPC分类号: A01N43/90 C07D487/04

    CPC分类号: A01N43/90

    摘要: Herbicidal agents containing a pyrimido[5,4-e]-as-triazine-5,7-(6H,8H)-dione Ia ##STR1## (R.sup.1, R.sup.2 .dbd.H, C.sub.1 -C.sub.6 -alkyl, C.sub.3 -C.sub.6 -cycloalkyl, C.sub.2 -C.sub.8 -alkenyl, phenyl or benzyl, R.sup.3 .dbd.H, halogen, nitro, C.sub.1 -C.sub.8 -alkyl which may carry up to three further substituents, C.sub.2 -C.sub.6 -alkenyl, phenyl-C.sub.2 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -cycloalkyl which may carry up to 3 C.sub.1 -C.sub.4 -alkyl substituents, a 5- or 6-membered heterocyclic structure where up to 2 of the ring members are O, S or NR.sup.4 ; --CO--R.sup.4 or --CO--O--R.sup.4 ; phenyl or hetaryl, which may carry up to 3 further substituents; or ZR.sup.6 ; R.sup.4 .dbd.H, C.sub.1 -C.sub.6 -alkyl; Z.dbd.O, S or --N(R.sup.7)--; R.sup.6 .dbd.H, C.sub.1 -C.sub.6 -alkyl, phenyl or benzyl, which may carry up to 3 further substituents; R.sup.7 .dbd.H, C.sub.1 -C.sub.6 -alkyl or R.sup.6 and R.sup.7 together with nitrogen form a 5- or 6-membered ring which may contain O; n=0 or 1) or a salt of Ia with a mineral acid.

    摘要翻译: 含有嘧啶并[5,4-e] -as-三嗪-5,7-(6H,8H) - 二酮Ia(Ia)(R1,R2 = H,C1-C6-烷基,C3- C 2 -C 6环烷基,C 2 -C 8 - 烯基,苯基或苄基,R 3 = H,卤素,硝基,可带有至多三个其它取代基的C 1 -C 8烷基,C 2 -C 6 - 链烯基,苯基-C 2 -C 6 - 烯基, 可含有3个C 1 -C 4烷基取代基的C 3 -C 6环烷基,其中至多2个环成员为O,S或NR 4的5或6元杂环结构; -CO-R 4或-CO- R 4 = H,C 1 -C 6 - 烷基; Z = O,S或-N(R 7) - ; R 6 = H,C 1 -C 6烷基; - 烷基,苯基或苄基,其可以带有多达3个其它取代基; R 7 = H,C 1 -C 6 - 烷基或者R 6和R 7与氮一起形成5-或6-元环,其可以含有O; n = 0或 1)或Ia与无机酸的盐。