2-substituted pyrimidines
    52.
    发明授权
    2-substituted pyrimidines 失效
    2-取代的嘧啶

    公开(公告)号:US07488732B2

    公开(公告)日:2009-02-10

    申请号:US10549936

    申请日:2004-03-30

    摘要: 2-Substituted pyrimidines of the formula I in which the index n and the substituents L, Ra, Rb, Rc, Rz, Ru, Rv, A′, A″ and A′″ are as defined in the description and: R1 is C3-C10-alkyl, C3-C10-alkenyl, C3-C10-alkynyl, C3-C12-cycloalkyl, C3-C10-cycloalkenyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via carbon and contains one to four heteroatoms from the group consisting of O, N and S, R2 is halogen, cyano, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl, C1-C4-alkoxy, C3-C4-alkenyloxy or C3-C4-alkynyloxy, where the alkyl, alkenyl and alkynyl radicals of R2 may be substituted by halogen, cyano, nitro, C1-C2-alkoxy or C1-C4-alkoxycarbonyl, and R3 is cyano, CO2Ra, C(═O)NRzRb, C(═O)—N—ORb, C(═S)—NRaRb, C(═NORa)NRzRb, C(═NRa)NRzRb, C(═O)NRa—NRzRb, C(═N—NRzRc)NRaRb, C(═O)Ra, C(═NORb)Ra, C(═N—NRzRb)Ra, CRaRb—ORz, CRaRb—NRzRc, ON(═CRaRb), O—C(═O)Ra, NRaRb′, NRa(C(═O)Rb), NRa(C(═O)ORb), NRa(C(═O)—NRzRb), NRa(C(═NRc)Rb), NRa(N═CRcRb), NRa—NRzRb, NRz—ORa, NRa(C(═NRc)—NRzRb), NRa(C(═NORc)Rb), processes for preparing these compounds, compositions comprising these compounds and their pesticidal use are described.

    摘要翻译: 其中指数n和取代基L,Ra,Rb,Rc,Rz,Ru,Rv,A',A“和A”'如说明书中所定义的式I的2-取代的嘧啶:R1 C 3 -C 10 - 烷基,C 3 -C 10 - 烯基,C 3 -C 10 - 炔基,C 3 -C 12 - 环烷基,C 3 -C 10 - 环烯基或五至十元饱和的部分不饱和或芳族杂环,其通过碳 并且含有一至四个由O,N和S组成的组的杂原子,R2是卤素,氰基,C1-C4-烷基,C2-C4-烯基,C2-C4-炔基,C1-C4-烷氧基,C3-C4 - 烯氧基或C 3 -C 4 - 炔氧基,其中R 2的烷基,烯基和炔基可以被卤素,氰基,硝基,C 1 -C 2 - 烷氧基或C 1 -C 4 - 烷氧基羰基取代,并且R 3是氰基,CO 2 R a,C( -O)NR z R b,C(-O)-N-OR b,C(-S)-NR a R b,C(-NOR a)NR z R b,C(-NR a)NR z R b,C(O)NR a -NR b R b,C -NRaRb,C(-O)Ra,C(-NORb)Ra,C(-N-NRzRb)Ra,CRaRb-ORz,CRaRb-NRzRc,ON(-CRaRb),OC(-O)Ra,NRaRb ,NR a(C(-O)R b),NR a(C(-O)R b),NR a(C(-O)OR b) NRa-N RzRb,NRz-ORa,NRa(C(-NRc)-NRzRb),NRa(C(-NORc)Rb),制备这些化合物的方法,包含这些化合物的组合物及其杀虫剂用途。

    (Hetero)Cyclyl(Thio) Carboxylic Acid Anilides For Controlling Pathogenic Fungi
    58.
    发明申请
    (Hetero)Cyclyl(Thio) Carboxylic Acid Anilides For Controlling Pathogenic Fungi 审中-公开
    (异构)环状(硫代)羧酸酰苯胺用于控制致病真菌

    公开(公告)号:US20070299115A1

    公开(公告)日:2007-12-27

    申请号:US11661679

    申请日:2005-09-05

    摘要: The invention relates to (hetero)cyclyl(thio)carboxylic acid anilides of general formula (I) and to salts of said anilides that can be used for agricultural purposes for controlling pathogenic fungi. In said formula, the variables are defined as follows: A represents a phenyl or at least a monounsaturated 5- or 6-membered heterocycle comprising 1, 2 or 3 heteroatoms, selected from N, O, S, S(═O) and S(═O)2 as ring members, whereby phenyl and the monounsaturated 5- or 6-membered heterocycle can be unsubstituted or can be substituted according to the description; B represents a group of general formula (II), in which the variables R3, R4, R5 and the index m are defined as cited in the claims and the description; Y represents oxygen or sulphur, R1 represents H, OH, alkyl, cycloalkyl, alkoxy, haloalkyl, halocycloalkyl or haloalkoxy; R2 represents halogen, nitro, CN, alkyl, cycloalkyl, alkenyl, alkynyl, alkoxy, haloalkyl, halocycloalkyl, haloalkenyl, haloalkynyl or haloalkoxy; and n represents 0, 1, 2, 3 or 4; and salts that can be used for agricultural purposes. The invention also relates to the use of the (hetero)cyclyl(thio)carboxylic acid anilides of general formula (I), to a method for controlling pathogenic fungi and to a crop protection agent containing at least one compound of general formula (I) and/or an agriculturally compatible salt of said compound.

    摘要翻译: 本发明涉及通式(I)的(杂)环(硫代)羧酸酰苯胺和可用于农业目的的用于控制致病真菌的所述酰苯胺的盐。 在所述式中,变量定义如下:A表示苯基或至少一个单不饱和的5-或6-元杂环,其包含1,2或3个选自N,O,S,S(-O)和S (-O)2,作为环成员,由此苯基和单不饱和的5-或6-元杂环可以是未取代的或可以根据描述被取代; B表示通式(II)的基团,其中定义了变量R 3,R 4,R 5和指数m, 如权利要求和说明书所引用的; Y表示氧或硫,R 1表示H,OH,烷基,环烷基,烷氧基,卤代烷基,卤代环烷基或卤代烷氧基; R 2表示卤素,硝基,CN,烷基,环烷基,烯基,炔基,烷氧基,卤代烷基,卤代环烷基,卤代烯基,卤代炔基或卤代烷氧基。 并且n表示0,1,2,3或4; 和可用于农业目的的盐。 本发明还涉及通式(I)的(杂)环(硫代)羧酸二酰苯胺用于控制致病真菌的方法和含有至少一种通式(I)的化合物的作物保护剂, 和/或所述化合物的农业上相容的盐。